Stacy Markison

Affiliations: 
Crinetics Pharmaceuticals 
Area:
Behavioral Pharmacology & Toxicology
Google:
"Stacy Markison"
Mean distance: 17.13 (cluster 19)
 
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Publications

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Lanier MC, Moorjani M, Luo Z, et al. (2009) N-[6-amino-2-(heteroaryl)pyrimidin-4-yl]acetamides as A2A receptor antagonists with improved drug like properties and in vivo efficacy. Journal of Medicinal Chemistry. 52: 709-17
Zhang X, Tellew JE, Luo Z, et al. (2008) Lead optimization of 4-acetylamino-2-(3,5-dimethylpyrazol-1-yl)-6-pyridylpyrimidines as A2A adenosine receptor antagonists for the treatment of Parkinson's disease. Journal of Medicinal Chemistry. 51: 7099-110
Chen C, Tucci FC, Jiang W, et al. (2008) Pharmacological and pharmacokinetic characterization of 2-piperazine-alpha-isopropyl benzylamine derivatives as melanocortin-4 receptor antagonists. Bioorganic & Medicinal Chemistry. 16: 5606-18
Zhang X, Rueter JK, Chen Y, et al. (2008) Synthesis of N-pyrimidinyl-2-phenoxyacetamides as adenosine A2A receptor antagonists. Bioorganic & Medicinal Chemistry Letters. 18: 1778-83
Slee DH, Moorjani M, Zhang X, et al. (2008) 2-Amino-N-pyrimidin-4-ylacetamides as A2A receptor antagonists: 2. Reduction of hERG activity, observed species selectivity, and structure-activity relationships. Journal of Medicinal Chemistry. 51: 1730-9
Slee DH, Chen Y, Zhang X, et al. (2008) 2-Amino-N-pyrimidin-4-ylacetamides as A2A receptor antagonists: 1. Structure-activity relationships and optimization of heterocyclic substituents. Journal of Medicinal Chemistry. 51: 1719-29
Slee DH, Zhang X, Moorjani M, et al. (2008) Identification of novel, water-soluble, 2-amino-N-pyrimidin-4-yl acetamides as A2A receptor antagonists with in vivo efficacy. Journal of Medicinal Chemistry. 51: 400-6
Chen C, Jiang W, Tran JA, et al. (2008) Identification and characterization of pyrrolidine diastereoisomers as potent functional agonists and antagonists of the human melanocortin-4 receptor Bioorganic and Medicinal Chemistry Letters. 18: 129-136
Tran JA, Jiang W, Tucci FC, et al. (2007) Design, synthesis, in vitro, and in vivo characterization of phenylpiperazines and pyridinylpiperazines as potent and selective antagonists of the melanocortin-4 receptor Journal of Medicinal Chemistry. 50: 6356-6366
Jiang W, Tran JA, Tucci FC, et al. (2007) Synthesis and characterization of pyrrolidine derivatives as potent agonists of the human melanocortin-4 receptor Bioorganic and Medicinal Chemistry Letters. 17: 6546-6552
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