Nicholas Griggs

University of Michigan, Ann Arbor, Ann Arbor, MI 
"Nicholas Griggs"
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Montgomery D, Anand JP, Griggs N, et al. (2019) Novel Dimethyltyrosine-Tetrahydroisoquinoline Peptidomimetics with Aromatic Tetrahydroisoquinoline Substitutions Show In Vitro Kappa and Mu Opioid Receptor Agonism. Acs Chemical Neuroscience
Henry S, Fernandez TM, Anand JP, et al. (2019) Structural Simplification of a Tetrahydroquinoline Core Peptidomimetic µ-Opioid-Receptor (MOR) Agonist/ δ-Opioid Receptor (DOR) Antagonist Produces Improved Metabolic Stability  . Journal of Medicinal Chemistry
Nastase AF, Anand JP, Bender AM, et al. (2019) Dual Pharmacophores Explored via Structure-Activity Relationship (SAR) Matrix: Insights into Potent, Bifunctional Opioid Ligand Design. Journal of Medicinal Chemistry
Nastase AF, Griggs NW, Anand JP, et al. (2018) Synthesis and pharmacological evaluation of novel C-8 substituted tetrahydroquinolines as balanced-affinity mu/delta opioid ligands for the treatment of pain. Acs Chemical Neuroscience
Anand JP, Kochan KE, Nastase AF, et al. (2018) In Vivo Effects of μ Opioid Receptor Agonist/δ Opioid Receptor Antagonist Peptidomimetics Following Acute and Repeated Administration. British Journal of Pharmacology
Harland AA, Pogozheva ID, Griggs NW, et al. (2017) Placement of hydroxy moiety on pendant of peptidomimetic scaffold modulates mu and kappa opioid receptor efficacy. Acs Chemical Neuroscience
Healy JR, Bezawada P, Griggs NW, et al. (2016) Benzylideneoxymorphone: A new lead for development of bifunctional mu/delta opioid receptor ligands. Bioorganic & Medicinal Chemistry Letters
Harland AA, Bender AM, Griggs NW, et al. (2016) Effects of N-Substitutions on the Tetrahydroquinoline (THQ) core of Mixed-Efficacy μ-Opioid Receptor (MOR)/ δ-Opioid Receptor (DOR) Ligands. Journal of Medicinal Chemistry
Bender AM, Griggs NW, Gao C, et al. (2015) Rapid Synthesis of Boc-2',6'-dimethyl-l-tyrosine and Derivatives and Incorporation into Opioid Peptidomimetics. Acs Medicinal Chemistry Letters. 6: 1199-203
Yao XQ, Malik R, Griggs NW, et al. (2015) Dynamic coupling and allosteric networks in the alpha subunit of heterotrimeric G proteins. The Journal of Biological Chemistry
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