Year |
Citation |
Score |
2021 |
La Cruz TE, González-Bobes F, Eastgate MD, Sfouggatakis C, Zheng B, Kopp N, Xiao Y, Fan Y, Galindo KA, Pathirana C, Galella MA, Deerberg J. Scalable Asymmetric Synthesis of the All Triamino Cyclohexane Core of BMS-813160. The Journal of Organic Chemistry. PMID 34355895 DOI: 10.1021/acs.joc.1c01162 |
0.48 |
|
2018 |
Maity P, Reddy VVR, Mohan J, Korapati S, Narayana H, Cherupally N, Chandrasekaran S, Ramachandran R, Sfouggatakis C, Eastgate MD, Simmons EM, Vaidyanathan R. Development of a Scalable Synthesis of BMS-978587 Featuring a Stereospecific Suzuki Coupling of a Cyclopropane Carboxylic Acid Organic Process Research & Development. 22: 888-897. DOI: 10.1021/Acs.Oprd.8B00171 |
0.459 |
|
2017 |
Smith MJ, Lawler MJ, Kopp N, Mcleod DD, Davulcu AH, Lin D, Katipally K, Sfouggatakis C. Development of a Concise Multikilogram Synthesis of LPA-1 Antagonist BMS-986020 via a Tandem Borylation–Suzuki Procedure Organic Process Research & Development. 21: 1859-1863. DOI: 10.1021/acs.oprd.7b00301 |
0.658 |
|
2015 |
Ortiz A, Benkovics T, Beutner GL, Shi Z, Bultman M, Nye J, Sfouggatakis C, Kronenthal DR. Scalable Synthesis of the Potent HIV Inhibitor BMS-986001 by Non-Enzymatic Dynamic Kinetic Asymmetric Transformation (DYKAT). Angewandte Chemie (International Ed. in English). 54: 7185-8. PMID 25925234 DOI: 10.1002/Anie.201502290 |
0.445 |
|
2009 |
Smith AB, Sfouggatakis C, Risatti CA, Sperry JB, Zhu W, Doughty VA, Tomioka T, Gotchev DB, Bennett CS, Sakamoto S, Atasoylu O, Shirakami S, Bauer D, Takeuchi M, Koyanagi J, et al. Spongipyran Synthetic Studies. Evolution of a Scalable Total Synthesis of (+)-Spongistatin 1. Tetrahedron. 65: 6489-6509. PMID 20640040 DOI: 10.1016/J.Tet.2009.04.003 |
0.636 |
|
2009 |
Smith AB, Doughty VA, Sfouggatakis C, Bennett CS, Koyanagi J, Takeuchi M. Spongistatin synthetic studies. An efficient, second-generation construction of an advanced ABCD intermediate (Organic Letters (2002) 4) Organic Letters. 11: 785. |
0.633 |
|
2008 |
Smith AB, Tomioka T, Risatti CA, Sperry JB, Sfouggatakis C. Gram-scale synthesis of (+)-spongistatin 1: development of an improved, scalable synthesis of the F-ring subunit, fragment union, and final elaboration. Organic Letters. 10: 4359-62. PMID 18754594 DOI: 10.1021/ol801792k |
0.569 |
|
2004 |
Smith AB, Sfouggatakis C, Gotchev DB, Shirakami S, Bauer D, Zhu W, Doughty VA. Spongistatin synthetic studies. evolution of a scalable synthesis for the EF fragment of (+)-Spongistatin 1 exploiting a Petasis-Ferrier union/rearrangement tactic. Organic Letters. 6: 3637-40. PMID 15387567 DOI: 10.1021/ol048418f |
0.685 |
|
2003 |
Smith AB, Pitram SM, Boldi AM, Gaunt MJ, Sfouggatakis C, Moser WH. Multicomponent linchpin couplings. Reaction of dithiane anions with terminal epoxides, epichlorohydrin, and vinyl epoxides: efficient, rapid, and stereocontrolled assembly of advanced fragments for complex molecule synthesis. Journal of the American Chemical Society. 125: 14435-45. PMID 14624591 DOI: 10.1021/ja0376238 |
0.657 |
|
2003 |
Smith AB, Zhu W, Shirakami S, Sfouggatakis C, Doughty VA, Bennett CS, Sakamoto Y. Total synthesis of (+)-spongistatin 1. An effective second-generation construction of an advanced EF Wittig salt, fragment union, and final elaboration. Organic Letters. 5: 761-4. PMID 12605509 DOI: 10.1021/Ol034037A |
0.724 |
|
2002 |
Smith AB, Doughty VA, Sfouggatakis C, Bennett CS, Koyanagi J, Takeuchi M. Spongistatin synthetic studies. An efficient, second-generation construction of an advanced ABCD intermediate. Organic Letters. 4: 783-6. PMID 11869127 DOI: 10.1021/Ol017273Z |
0.721 |
|
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