| Year |
Citation |
Score |
| 2010 |
Bressi JC, Jennings AJ, Skene R, Wu Y, Melkus R, De Jong R, O'Connell S, Grimshaw CE, Navre M, Gangloff AR. Exploration of the HDAC2 foot pocket: Synthesis and SAR of substituted N-(2-aminophenyl)benzamides. Bioorganic & Medicinal Chemistry Letters. 20: 3142-5. PMID 20392638 DOI: 10.1016/j.bmcl.2010.03.091 |
0.477 |
|
| 2002 |
Verlinde C, Bressi J, Choe J, Suresh S, Buckner F, Voorhis WV, Michels P, Gelb M, Hol W. Protein structure-based design of anti-protozoal drugs Journal of the Brazilian Chemical Society. 13: 843-844. DOI: 10.1590/S0103-50532002000600018 |
0.379 |
|
| 2002 |
Verlinde CLMJ, Bressi JC, Choe J, Suresh S, Buckner FS, Van Voorhis WC, Michels PAM, Gelb MH, Hol WGJ. Protein structure-based design of anti-protozoal drugs Journal of the Brazilian Chemical Society. 13: 843-848. |
0.432 |
|
| 2001 |
Bressi JC, Verlinde CL, Aronov AM, Shaw ML, Shin SS, Nguyen LN, Suresh S, Buckner FS, Van Voorhis WC, Kuntz ID, Hol WG, Gelb MH. Adenosine analogues as selective inhibitors of glyceraldehyde-3-phosphate dehydrogenase of Trypanosomatidae via structure-based drug design. Journal of Medicinal Chemistry. 44: 2080-93. PMID 11405646 DOI: 10.1021/Jm000472O |
0.585 |
|
| 2001 |
Suresh S, Bressi JC, Kennedy KJ, Verlinde CL, Gelb MH, Hol WG. Conformational changes in Leishmania mexicana glyceraldehyde-3-phosphate dehydrogenase induced by designed inhibitors. Journal of Molecular Biology. 309: 423-35. PMID 11371162 DOI: 10.1006/Jmbi.2001.4588 |
0.592 |
|
| 2001 |
Kennedy KJ, Bressi JC, Gelb MH. A disubstituted NAD+ analogue is a nanomolar inhibitor of trypanosomal glyceraldehyde-3-phosphate dehydrogenase. Bioorganic & Medicinal Chemistry Letters. 11: 95-8. PMID 11206479 DOI: 10.1016/S0960-894X(00)00608-9 |
0.57 |
|
| 2000 |
Bressi JC, Choe J, Hough MT, Buckner FS, Van Voorhis WC, Verlinde CL, Hol WG, Gelb MH. Adenosine analogues as inhibitors of Trypanosoma brucei phosphoglycerate kinase: elucidation of a novel binding mode for a 2-amino-N(6)-substituted adenosine. Journal of Medicinal Chemistry. 43: 4135-50. PMID 11063610 DOI: 10.1021/Jm000287A |
0.588 |
|
| 2000 |
Golisade A, Bressi JC, Van Calenbergh S, Gelb MH, Link A. Polymer-assisted solution-phase synthesis of 2'-amido-2'-deoxyadenosine derivatives targeted at the NAD(+)-binding sites of parasite enzymes. Journal of Combinatorial Chemistry. 2: 537-44. PMID 11029179 DOI: 10.1021/Cc0000343 |
0.488 |
|
| 1998 |
Bernstein BE, Williams DM, Bressi JC, Kuhn P, Gelb MH, Blackburn GM, Hol WG. A bisubstrate analog induces unexpected conformational changes in phosphoglycerate kinase from Trypanosoma brucei. Journal of Molecular Biology. 279: 1137-48. PMID 9642090 DOI: 10.1006/Jmbi.1998.1835 |
0.562 |
|
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