Year |
Citation |
Score |
2015 |
Arai K, Buonamici S, Chan B, Corson L, Endo A, Gerard B, Hao M, Karr C, Kira K, Lee L, Liu X, Lowe JT, Luo T, Marcaurelle LA, Mizui Y, et al. Abstract 5564: Total synthesis of 6-deoxypladienolide D and assessment of splicing inhibitory activity in a mutant SF3B1 cancer cell line Cancer Research. 75: 5564-5564. DOI: 10.1158/1538-7445.Am2015-5564 |
0.326 |
|
2014 |
Arai K, Buonamici S, Chan B, Corson L, Endo A, Gerard B, Hao MH, Karr C, Kira K, Lee L, Liu X, Lowe JT, Luo T, Marcaurelle LA, Mizui Y, et al. Total synthesis of 6-deoxypladienolide D and Assessment of Splicing Inhibitory Activity in a Mutant SF3B1 cancer cell line. Organic Letters. 16: 5560-3. PMID 25376106 DOI: 10.1021/Ol502556C |
0.333 |
|
2013 |
Gerard B, Lee MD, Dandapani S, Duvall JR, Fitzgerald ME, Kesavan S, Lowe JT, Marié JC, Pandya BA, Suh BC, O'Shea MW, Dombrowski M, Hamann D, Lemercier B, Murillo T, ... ... Marcaurelle LA, et al. Synthesis of stereochemically and skeletally diverse fused ring systems from functionalized C-glycosides. The Journal of Organic Chemistry. 78: 5160-71. PMID 23692141 DOI: 10.1021/Jo4000916 |
0.425 |
|
2013 |
Kesavan S, Marcaurelle LA. Translational synthetic chemistry. Nature Chemical Biology. 9: 210-3. PMID 23508175 DOI: 10.1038/Nchembio.1207 |
0.329 |
|
2013 |
Gerard B, O’Shea MW, Donckele E, Kesavan S, Akella LB, Xu H, Jacobsen EN, Marcaurelle LA. Correction to Application of a Catalytic Asymmetric Povarov Reaction using Chiral Ureas to the Synthesis of a Tetrahydroquinoline Library Acs Combinatorial Science. 16: 46-46. DOI: 10.1021/Co400123X |
0.377 |
|
2012 |
Gerard B, O'Shea MW, Donckele E, Kesavan S, Akella LB, Xu H, Jacobsen EN, Marcaurelle LA. Application of a catalytic asymmetric Povarov reaction using chiral ureas to the synthesis of a tetrahydroquinoline library. Acs Combinatorial Science. 14: 621-30. PMID 23088641 DOI: 10.1021/Co300098V |
0.429 |
|
2012 |
Lowe JT, Lee MD, Akella LB, Davoine E, Donckele EJ, Durak L, Duvall JR, Gerard B, Holson EB, Joliton A, Kesavan S, Lemercier BC, Liu H, Marié JC, Mulrooney CA, ... ... Marcaurelle LA, et al. Synthesis and profiling of a diverse collection of azetidine-based scaffolds for the development of CNS-focused lead-like libraries. The Journal of Organic Chemistry. 77: 7187-211. PMID 22853001 DOI: 10.1021/Jo300974J |
0.438 |
|
2012 |
Heidebrecht RW, Mulrooney C, Austin CP, Barker RH, Beaudoin JA, Cheng KC, Comer E, Dandapani S, Dick J, Duvall JR, Ekland EH, Fidock DA, Fitzgerald ME, Foley M, Guha R, ... ... Marcaurelle LA, et al. Diversity-Oriented Synthesis Yields a Novel Lead for the Treatment of Malaria. Acs Medicinal Chemistry Letters. 3: 112-117. PMID 22328964 DOI: 10.1021/Ml200244K |
0.34 |
|
2012 |
Fitzgerald ME, Mulrooney CA, Duvall JR, Wei J, Suh BC, Akella LB, Vrcic A, Marcaurelle LA. Build/couple/pair strategy for the synthesis of stereochemically diverse macrolactams via head-to-tail cyclization. Acs Combinatorial Science. 14: 89-96. PMID 22252910 DOI: 10.1021/Co200161Z |
0.396 |
|
2011 |
Chou DH, Duvall JR, Gerard B, Liu H, Pandya BA, Suh BC, Forbeck EM, Faloon P, Wagner BK, Marcaurelle LA. Synthesis of a novel suppressor of beta-cell apoptosis via diversity-oriented synthesis. Acs Medicinal Chemistry Letters. 2: 698-702. PMID 21927648 DOI: 10.1021/Ml200120M |
0.396 |
|
2011 |
Dandapani S, Lowe JT, Comer E, Marcaurelle LA. Diversity-oriented synthesis of 13- to 18-membered macrolactams via ring-closing metathesis. The Journal of Organic Chemistry. 76: 8042-8. PMID 21875084 DOI: 10.1021/Jo2011957 |
0.398 |
|
2011 |
Pandya BA, Dandapani S, Duvall JR, Rowley A, Mulrooney CA, Ryba T, Dombrowski M, Harton M, Young DW, Marcaurelle LA. Practical asymmetric synthesis of β-hydroxy γ-amino acids via complimentary aldol reactions. Tetrahedron. 67: 6131-6137. PMID 21822337 DOI: 10.1016/J.Tet.2011.06.043 |
0.38 |
|
2011 |
Akella LB, Marcaurelle LA. Application of a sparse matrix design strategy to the synthesis of dos libraries. Acs Combinatorial Science. 13: 357-64. PMID 21526822 DOI: 10.1021/Co200020J |
0.394 |
|
2011 |
Gerard B, Duvall JR, Lowe JT, Murillo T, Wei J, Akella LB, Marcaurelle LA. Synthesis of a stereochemically diverse library of medium-sized lactams and sultams via S(N)Ar cycloetherification. Acs Combinatorial Science. 13: 365-74. PMID 21526820 DOI: 10.1021/Co2000218 |
0.418 |
|
2011 |
Comer E, Liu H, Joliton A, Clabaut A, Johnson C, Akella LB, Marcaurelle LA. Fragment-based domain shuffling approach for the synthesis of pyran-based macrocycles. Proceedings of the National Academy of Sciences of the United States of America. 108: 6751-6. PMID 21383141 DOI: 10.1073/Pnas.1015255108 |
0.434 |
|
2011 |
Gerard B, Marié JC, Pandya BA, Lee MD, Liu H, Marcaurelle LA. Large-scale synthesis of all stereoisomers of a 2,3-unsaturated C-glycoside scaffold. The Journal of Organic Chemistry. 76: 1898-901. PMID 21341742 DOI: 10.1021/Jo1022926 |
0.38 |
|
2010 |
Duvall JR, Vrcic A, Marcaurelle LA. Small-Molecule Library Synthesis on Silicon-Functionalized SynPhase Lanterns. Current Protocols in Chemical Biology. 2: 135-151. PMID 22679566 DOI: 10.1002/9780470559277.Ch100038 |
0.433 |
|
2010 |
Marcaurelle LA, Comer E, Dandapani S, Duvall JR, Gerard B, Kesavan S, Lee MD, Liu H, Lowe JT, Marie JC, Mulrooney CA, Pandya BA, Rowley A, Ryba TD, Suh BC, et al. An aldol-based build/couple/pair strategy for the synthesis of medium- and large-sized rings: discovery of macrocyclic histone deacetylase inhibitors. Journal of the American Chemical Society. 132: 16962-76. PMID 21067169 DOI: 10.1021/Ja105119R |
0.43 |
|
2010 |
Dandapani S, Marcaurelle LA. Current strategies for diversity-oriented synthesis. Current Opinion in Chemical Biology. 14: 362-70. PMID 20409744 DOI: 10.1016/J.Cbpa.2010.03.018 |
0.44 |
|
2009 |
Kelly AR, Wei J, Kesavan S, Marié JC, Windmon N, Young DW, Marcaurelle LA. Accessing skeletal diversity using catalyst control: formation of n and n + 1 macrocyclic triazole rings. Organic Letters. 11: 2257-60. PMID 19473044 DOI: 10.1021/Ol900562U |
0.349 |
|
2009 |
Marcaurelle LA, Johannes C, Yohannes D, Tillotson BP, Mann D. Diversity-oriented synthesis of a cytisine-inspired pyridone library leading to the discovery of novel inhibitors of Bcl-2. Bioorganic & Medicinal Chemistry Letters. 19: 2500-3. PMID 19329314 DOI: 10.1016/J.Bmcl.2009.03.037 |
0.414 |
|
2009 |
Ryba TD, Depew KM, Marcaurelle LA. Large scale preparation of silicon-functionalized SynPhase Polystyrene lanterns for solid-phase synthesis. Journal of Combinatorial Chemistry. 11: 110-6. PMID 19049425 DOI: 10.1021/Cc8000986 |
0.389 |
|
2008 |
Marcaurelle LA, Johannes CW. Application of natural product-inspired diversity-oriented synthesis to drug discovery. Progress in Drug Research. Fortschritte Der Arzneimittelforschung. ProgrèS Des Recherches Pharmaceutiques. 66: 187, 189-216. PMID 18416306 DOI: 10.1007/978-3-7643-8595-8_3 |
0.376 |
|
2003 |
Marcaurelle LA, Pratt MR, Bertozzi CR. Synthesis of thioether-linked analogues of the 2,3-sialyl-TF and MECA-79 antigens: mucin-type glycopeptides associated with cancer and inflammation. Chembiochem : a European Journal of Chemical Biology. 4: 224-8. PMID 12616638 DOI: 10.1002/Cbic.200390036 |
0.599 |
|
2002 |
Bosse F, Marcaurelle LA, Seeberger PH. Linear synthesis of the tumor-associated carbohydrate antigens Globo-H, SSEA-3, and Gb3. The Journal of Organic Chemistry. 67: 6659-70. PMID 12227795 DOI: 10.1021/Jo025834+ |
0.374 |
|
2002 |
Marcaurelle LA, Bertozzi CR. Recent advances in the chemical synthesis of mucin-like glycoproteins. Glycobiology. 12: 69R-77R. PMID 12107076 DOI: 10.1093/Glycob/. |
0.515 |
|
2002 |
Grogan MJ, Pratt MR, Marcaurelle LA, Bertozzi CR. Homogeneous glycopeptides and glycoproteins for biological investigation. Annual Review of Biochemistry. 71: 593-634. PMID 12045107 DOI: 10.1146/Annurev.Biochem.71.110601.135334 |
0.619 |
|
2002 |
Marcaurelle LA, Seeberger PH. Combinatorial carbohydrate chemistry. Current Opinion in Chemical Biology. 6: 289-96. PMID 12023107 DOI: 10.1016/S1367-5931(02)00322-8 |
0.416 |
|
2001 |
Marcaurelle LA, Shin Y, Goon S, Bertozzi CR. Synthesis of oxime-linked mucin mimics containing the tumor-related T(N) and sialyl T(N) antigens. Organic Letters. 3: 3691-4. PMID 11700114 DOI: 10.1021/Ol0166247 |
0.641 |
|
2001 |
Marcaurelle LA, Bertozzi CR. Chemoselective elaboration of O-linked glycopeptide mimetics by alkylation of 3-thioGalNAc. Journal of the American Chemical Society. 123: 1587-95. PMID 11456757 DOI: 10.1021/Ja003713Q |
0.535 |
|
2001 |
Marcaurelle LA, Mizoue LS, Wilken J, Oldham L, Kent SB, Handel TM, Bertozzi CR. Chemical synthesis of lymphotactin: a glycosylated chemokine with a C-terminal mucin-like domain. Chemistry (Weinheim An Der Bergstrasse, Germany). 7: 1129-32. PMID 11303872 DOI: 10.1002/1521-3765(20010302)7:5<1129::Aid-Chem1129>3.0.Co;2-W |
0.534 |
|
1999 |
Marcaurelle LA, Bertozzi CR. New directions in the synthesis of glycopeptide mimetics Chemistry - a European Journal. 5: 1384-1390. DOI: 10.1002/(Sici)1521-3765(19990503)5:5<1384::Aid-Chem1384>3.0.Co;2-X |
0.518 |
|
1998 |
Rodriguez EC, Marcaurelle LA, Bertozzi CR. Aminooxy-, Hydrazide-, and Thiosemicarbazide-Functionalized Saccharides: Versatile Reagents for Glycoconjugate Synthesis. The Journal of Organic Chemistry. 63: 7134-7135. PMID 11672350 DOI: 10.1021/Jo981351N |
0.54 |
|
1998 |
Marcaurelle LA, Rodriguez EC, Bertozzi CR. Synthesis of an oxime-linked neoglycopeptide with glycosylation- dependent activity similar to its native counterpart Tetrahedron Letters. 39: 8417-8420. DOI: 10.1016/S0040-4039(98)01831-0 |
0.508 |
|
1998 |
Marcaurelle LA, Bertozzi CR. Direct incorporation of unprotected ketone groups into peptides during solid-phase synthesis: Application to the one-step modification of peptides with two different biophysical probes for FRET Tetrahedron Letters. 39: 7279-7282. DOI: 10.1016/S0040-4039(98)01588-3 |
0.51 |
|
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