Year |
Citation |
Score |
2022 |
Choi PJ, Tomek P, Tercel M, Reynisson J, Park TIH, Cooper EA, Denny WA, Jose J, Leung E. Conjugation of Palbociclib with MHI-148 Has an Increased Cytotoxic Effect for Breast Cancer Cells and an Altered Mechanism of Action. Molecules (Basel, Switzerland). 27. PMID 35164144 DOI: 10.3390/molecules27030880 |
0.313 |
|
2020 |
Choi PJ, Park TI, Cooper E, Dragunow M, Denny WA, Jose J. Heptamethine cyanine dye mediated drug delivery: Hype or Hope. Bioconjugate Chemistry. PMID 32530288 DOI: 10.1021/Acs.Bioconjchem.0C00302 |
0.341 |
|
2020 |
Choi PJ, Cooper E, Schweder P, Mee E, Turner C, Faull R, Denny WA, Dragunow M, Park TI, Jose J. PARP inhibitor cyanine dye conjugate with enhanced cytotoxic and antiproliferative activity in patient derived glioblastoma cell lines. Bioorganic & Medicinal Chemistry Letters. 30: 127252. PMID 32527552 DOI: 10.1016/J.Bmcl.2020.127252 |
0.379 |
|
2019 |
Choi PJ, Cooper E, Schweder P, Mee E, Faull R, Denny WA, Dragunow M, Park TI, Jose J. The synthesis of a novel Crizotinib heptamethine cyanine dye conjugate that potentiates the cytostatic and cytotoxic effects of Crizotinib in patient-derived glioblastoma cell lines. Bioorganic & Medicinal Chemistry Letters. PMID 31378572 DOI: 10.1016/J.Bmcl.2019.07.051 |
0.392 |
|
2018 |
Choi P, Noguchi K, Ishiyama M, Denny WA, Jose J. A mitochondria-selective near-infrared-emitting fluorescent dye for cellular imaging studies. Bioorganic & Medicinal Chemistry Letters. PMID 29731365 DOI: 10.1016/J.Bmcl.2018.05.001 |
0.315 |
|
2017 |
Jose J, Tavares CDJ, Ebelt ND, Lodi A, Edupuganti R, Xie X, Devkota AK, Kaoud TS, Van Den Berg CL, Anslyn EV, Tiziani S, Bartholomeusz C, Dalby KN. Serotonin Analogues as Inhibitors of Breast Cancer Cell Growth. Acs Medicinal Chemistry Letters. 8: 1072-1076. PMID 29057053 DOI: 10.1021/Acsmedchemlett.7B00282 |
0.739 |
|
2017 |
Spicer JA, Miller CK, O'Connor PD, Jose J, Huttunen KM, Jaiswal JK, Denny WA, Akhlaghi H, Browne KA, Trapani JA. Substituted arylsulphonamides as inhibitors of perforin-mediated lysis. European Journal of Medicinal Chemistry. 137: 139-155. PMID 28582670 DOI: 10.1016/J.Ejmech.2017.05.048 |
0.362 |
|
2016 |
Spicer JA, Miller CK, O'Connor PD, Jose J, Huttunen KM, Jaiswal JK, Denny WA, Akhlaghi H, Browne KA, Trapani JA. Benzenesulphonamide inhibitors of the cytolytic protein perforin. Bioorganic & Medicinal Chemistry Letters. PMID 28110869 DOI: 10.1016/J.Bmcl.2016.12.057 |
0.35 |
|
2016 |
Ebelt ND, Taveres CDJ, Xie X, Naguib YW, Jose J, Ruwona TB, Devkota AK, Park J, Kaoud TS, Anslyn EV, Chang JT, Cui Z, Bartholomeusz C, Dalby KN. Abstract 3774: KD06 is a novel anti-cancer drug that causes cell death in triple-negative breast cancer cell lines and tumor xenografts Cancer Research. 76: 3774-3774. DOI: 10.1158/1538-7445.Am2016-3774 |
0.777 |
|
2015 |
Gozzi GJ, Bouaziz Z, Winter E, Daflon-Yunes N, Honorat M, Guragossian N, Marminon C, Valdameri G, Bollacke A, Guillon J, Pinaud N, Marchivie M, Cadena SM, Jose J, Le Borgne M, et al. Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity. Drug Design, Development and Therapy. 9: 3481-95. PMID 26170632 DOI: 10.2147/Dddt.S84982 |
0.313 |
|
2015 |
Jabor Gozzi G, Bouaziz Z, Winter E, Daflon-Yunes N, Aichele D, Nacereddine A, Marminon C, Valdameri G, Zeinyeh W, Bollacke A, Guillon J, Lacoudre A, Pinaud N, Cadena SM, Jose J, et al. Converting potent indeno[1,2-b]indole inhibitors of protein kinase CK2 into selective inhibitors of the breast cancer resistance protein ABCG2. Journal of Medicinal Chemistry. 58: 265-77. PMID 25272055 DOI: 10.1021/Jm500943Z |
0.33 |
|
2014 |
Zamora-Olivares D, Kaoud TS, Jose J, Ellington A, Dalby KN, Anslyn EV. Differential sensing of MAP kinases using SOX-peptides. Angewandte Chemie (International Ed. in English). 53: 14064-8. PMID 25319433 DOI: 10.1002/Anie.201408256 |
0.718 |
|
2014 |
Devkota AK, Edupuganti R, Yan C, Shi Y, Jose J, Wang Q, Kaoud TS, Cho EJ, Ren P, Dalby KN. Reversible covalent inhibition of eEF-2K by carbonitriles. Chembiochem : a European Journal of Chemical Biology. 15: 2435-42. PMID 25224652 DOI: 10.1002/Cbic.201402321 |
0.738 |
|
2014 |
Tavares CDJ, Jose J, Devkota AK, Park J, Kaoud TS, Anslyn EV, Dalby KN. Abstract 5462: Antiproliferative and cytotoxic activities of 5-(nonyloxy)tryptamine derivatives in breast cancer cells Cancer Research. 74: 5462-5462. DOI: 10.1158/1538-7445.Am2014-5462 |
0.747 |
|
2012 |
Kaoud TS, Yan C, Mitra S, Tseng CC, Jose J, Taliaferro JM, Tuohetahuntila M, Devkota A, Sammons R, Park J, Park H, Shi Y, Hong J, Ren P, Dalby KN. From in Silico Discovery to intra-Cellular Activity: Targeting JNK-Protein Interactions with Small Molecules. Acs Medicinal Chemistry Letters. 3: 721-725. PMID 23002419 DOI: 10.1021/Ml300129B |
0.721 |
|
2012 |
Kaoud TS, Park H, Mitra S, Yan C, Tseng CC, Shi Y, Jose J, Taliaferro JM, Lee K, Ren P, Hong J, Dalby KN. Manipulating JNK signaling with (--)-zuonin A. Acs Chemical Biology. 7: 1873-83. PMID 22916726 DOI: 10.1021/Cb300261E |
0.77 |
|
2012 |
Kaoud TS, Yan C, Tseng C, Jose J, Devkota AK, Taliaferro J, Ren P, Dalby K. Abstract 4776: From in-silico screening to anti-cancer activity: The discovery of a potent inhibitor targeting the JNK-JIP interaction Cancer Research. 72: 4776-4776. DOI: 10.1158/1538-7445.Am2012-4776 |
0.769 |
|
2011 |
Jose J, Loudet A, Ueno Y, Wu L, Chen HY, Son DH, Barhoumi R, Burghardt R, Burgess K. Energy transfer cassettes in silica nanoparticles target intracellular organelles. Organic & Biomolecular Chemistry. 9: 3871-7. PMID 21455504 DOI: 10.1039/C0Ob00967A |
0.746 |
|
2011 |
Loudet A, Ueno Y, Wu L, Jose J, Barhoumi R, Burghardt R, Burgess K. Organelle-selective energy transfer: a fluorescent indicator of intracellular environment. Bioorganic & Medicinal Chemistry Letters. 21: 1849-51. PMID 21316231 DOI: 10.1016/J.Bmcl.2011.01.040 |
0.747 |
|
2011 |
Ueno Y, Jose J, Loudet A, Pérez-Bolívar C, Anzenbacher P, Burgess K. Encapsulated energy-transfer cassettes with extremely well resolved fluorescent outputs. Journal of the American Chemical Society. 133: 51-5. PMID 21105708 DOI: 10.1021/Ja107193J |
0.756 |
|
2010 |
Jose J, Loudet A, Ueno Y, Barhoumi R, Burghardt RC, Burgess K. Intracellular imaging of organelles with new water-soluble benzophenoxazine dyes. Organic & Biomolecular Chemistry. 8: 2052-9. PMID 20401381 DOI: 10.1039/B925845K |
0.748 |
|
2009 |
Jose J, Ueno Y, Castro JC, Li L, Burgess K. Energy transfer dyads based on Nile Red. Tetrahedron Letters. 50: 6442-6445. PMID 20160911 DOI: 10.1016/J.Tetlet.2009.08.130 |
0.613 |
|
2009 |
Jose J, Ueno Y, Burgess K. Water-soluble Nile Blue derivatives: syntheses and photophysical properties. Chemistry (Weinheim An Der Bergstrasse, Germany). 15: 418-23. PMID 19025740 DOI: 10.1002/Chem.200801104 |
0.633 |
|
2007 |
Han J, Jose J, Mei E, Burgess K. Chemiluminescent energy-transfer cassettes based on fluorescein and nile red. Angewandte Chemie (International Ed. in English). 46: 1684-7. PMID 17397078 DOI: 10.1002/Anie.200603307 |
0.565 |
|
2006 |
Jose J, Burgess K. Syntheses and properties of water-soluble Nile Red derivatives. The Journal of Organic Chemistry. 71: 7835-9. PMID 16995693 DOI: 10.1021/Jo061369V |
0.497 |
|
2006 |
Jose J, Burgess K. Benzophenoxazine-based fluorescent dyes for labeling biomolecules Tetrahedron. 62: 11021-11037. DOI: 10.1016/J.Tet.2006.08.056 |
0.473 |
|
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