Year |
Citation |
Score |
2019 |
Liang SH, Wang L, Stephenson NA, Rotstein BH, Vasdev N. Facile F labeling of non-activated arenes via a spirocyclic iodonium(III) ylide method and its application in the synthesis of the mGluR PET radiopharmaceutical [F]FPEB. Nature Protocols. PMID 30980032 DOI: 10.1038/S41596-019-0149-3 |
0.345 |
|
2017 |
Pekošak A, Rotstein BH, Collier TL, Windhorst AD, Vasdev N, Poot AJ. Stereoselective11C Labeling of a “Native” Tetrapeptide by Using Asymmetric Phase-Transfer Catalyzed Alkylation Reactions European Journal of Organic Chemistry. 2017: 1019-1024. DOI: 10.1002/Ejoc.201601641 |
0.48 |
|
2016 |
Yuan G, Wang F, Stephenson NA, Wang L, Rotstein BH, Vasdev N, Tang P, Liang SH. Metal-free (18)F-labeling of aryl-CF2H via nucleophilic radiofluorination and oxidative C-H activation. Chemical Communications (Cambridge, England). PMID 27917423 DOI: 10.1039/C6Cc07913J |
0.307 |
|
2016 |
Rotstein BH, Wang L, Liu RY, Patteson J, Kwan EE, Vasdev N, Liang SH. Mechanistic Studies and Radiofluorination of Structurally Diverse Pharmaceuticals with Spirocyclic Iodonium(III) Ylides. Chemical Science. 7: 4407-4417. PMID 27540460 DOI: 10.1039/C6Sc00197A |
0.355 |
|
2016 |
Wang L, Mori W, Cheng R, Yui J, Hatori A, Ma L, Zhang Y, Rotstein BH, Fujinaga M, Shimoda Y, Yamasaki T, Xie L, Nagai Y, Minamimoto T, Higuchi M, et al. Synthesis and Preclinical Evaluation of Sulfonamido-based [(11)C-Carbonyl]-Carbamates and Ureas for Imaging Monoacylglycerol Lipase. Theranostics. 6: 1145-59. PMID 27279908 DOI: 10.7150/Thno.15257 |
0.328 |
|
2016 |
Rotstein BH, Liang SH, Placzek MS, Hooker JM, Gee AD, Dollé F, Wilson AA, Vasdev N. (11)C[double bond, length as m-dash]O bonds made easily for positron emission tomography radiopharmaceuticals. Chemical Society Reviews. PMID 27276357 DOI: 10.1039/C6Cs00310A |
0.316 |
|
2015 |
Wang L, Yui J, Wang Q, Zhang Y, Mori W, Shimoda Y, Fujinaga M, Kumata K, Yamasak TI, Hatori A, Rotstein BH, Collier TL, Ran C, Vasdev N, Zhang MR, et al. Synthesis and preliminary PET imaging studies of a FAAH radiotracer ([(11)C]MPPO) based on α-ketoheterocyclic scaffold. Acs Chemical Neuroscience. PMID 26505525 DOI: 10.1021/Acschemneuro.5B00248 |
0.328 |
|
2015 |
Wang L, Jacobson O, Avdic D, Rotstein BH, Weiss ID, Collier L, Chen X, Vasdev N, Liang SH. Ortho-Stabilized (18) F-Azido Click Agents and their Application in PET Imaging with Single-Stranded DNA Aptamers. Angewandte Chemie (International Ed. in English). PMID 26308650 DOI: 10.1002/Anie.201505927 |
0.348 |
|
2015 |
Liang SH, Holland JP, Stephenson NA, Kassenbrock A, Rotstein BH, Daignault CP, Lewis R, Collier L, Hooker JM, Vasdev N. PET neuroimaging studies of [(18)F]CABS13 in a double transgenic mouse model of Alzheimer's disease and nonhuman primates. Acs Chemical Neuroscience. 6: 535-41. PMID 25776827 DOI: 10.1021/Acschemneuro.5B00055 |
0.302 |
|
2014 |
Belding L, Zaretsky S, Rotstein BH, Yudin AK, Dudding T. Shifting the energy landscape of multicomponent reactions using aziridine aldehyde dimers: a mechanistic study. The Journal of Organic Chemistry. 79: 9465-71. PMID 25264960 DOI: 10.1021/Jo501242R |
0.597 |
|
2014 |
Zaretsky S, Adachi S, Rotstein BH, Hickey JL, Scully CC, St Denis JD, Courtemanche R, Yu JC, Chung BK, Yudin AK. Stereocontrolled disruption of the Ugi reaction toward the production of chiral piperazinones: substrate scope and process development. The Journal of Organic Chemistry. 79: 9948-57. PMID 25254948 DOI: 10.1021/Jo5018316 |
0.569 |
|
2014 |
Rotstein BH, Zaretsky S, Rai V, Yudin AK. Small heterocycles in multicomponent reactions. Chemical Reviews. 114: 8323-59. PMID 25032909 DOI: 10.1021/Cr400615V |
0.617 |
|
2014 |
Rotstein BH, Stephenson NA, Vasdev N, Liang SH. Spirocyclic hypervalent iodine(III)-mediated radiofluorination of non-activated and hindered aromatics. Nature Communications. 5: 4365. PMID 25007318 DOI: 10.1038/Ncomms5365 |
0.387 |
|
2014 |
Rotstein BH, Wey HY, Shoup TM, Wilson AA, Liang SH, Hooker JM, Vasdev N. PET imaging of fatty acid amide hydrolase with [(18)F]DOPP in nonhuman primates. Molecular Pharmaceutics. 11: 3832-8. PMID 25004399 DOI: 10.1021/Mp500316H |
0.303 |
|
2014 |
Rotstein BH, Hooker JM, Woo J, Collier TL, Brady TJ, Liang SH, Vasdev N. Synthesis of [(11)C]Bexarotene by Cu-Mediated [(11)C]Carbon Dioxide Fixation and Preliminary PET Imaging. Acs Medicinal Chemistry Letters. 5: 668-72. PMID 24944741 DOI: 10.1021/Ml500065Q |
0.342 |
|
2013 |
Liang SH, Collier TL, Rotstein BH, Lewis R, Steck M, Vasdev N. Rapid microfluidic flow hydrogenation for reduction or deprotection of 18F-labeled compounds. Chemical Communications (Cambridge, England). 49: 8755-7. PMID 23948863 DOI: 10.1039/C3Cc45166F |
0.307 |
|
2012 |
Roxin Ã, Chen J, Scully CC, Rotstein BH, Yudin AK, Zheng G. Conformational modulation of in vitro activity of cyclic RGD peptides via aziridine aldehyde-driven macrocyclization chemistry. Bioconjugate Chemistry. 23: 1387-95. PMID 22709546 DOI: 10.1021/Bc300239A |
0.577 |
|
2012 |
Rotstein BH, Winternheimer DJ, Yin LM, Deber CM, Yudin AK. Thioester-isocyanides: versatile reagents for the synthesis of cycle-tail peptides. Chemical Communications (Cambridge, England). 48: 3775-7. PMID 22430393 DOI: 10.1039/C2Cc16027G |
0.577 |
|
2012 |
Rotstein BH, Yudin AK. Aziridine-2-carboxaldehyde dimers undergo homo-Ugi 4-component-5-center reactions Synthesis (Germany). 44: 2851-2858. DOI: 10.1055/S-0030-1260261 |
0.555 |
|
2011 |
Rotstein BH, Mourtada R, Kelley SO, Yudin AK. Solvatochromic reagents for multicomponent reactions and their utility in the development of cell-permeable macrocyclic peptide vectors. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 12257-61. PMID 21932287 DOI: 10.1002/Chem.201102096 |
0.609 |
|
2010 |
Rotstein BH, Rai V, Hili R, Yudin AK. Synthesis of peptide macrocycles using unprotected amino aldehydes. Nature Protocols. 5: 1813-22. PMID 21030956 DOI: 10.1038/Nprot.2010.127 |
0.634 |
|
2007 |
Garabatos-Perera JR, Rotstein BH, Thompson A. Comparison of benzene, nitrobenzene, and dinitrobenzene 2-arylsulfenylpyrroles. The Journal of Organic Chemistry. 72: 7382-5. PMID 17705533 DOI: 10.1021/Jo070493R |
0.36 |
|
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