Sarah L. Gilliland - Related publications

Affiliations: 
JRH Biosciences, Lenexa, KS, United States 
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50 most relevant papers in past 60 days:
Year Citation  Score
2020 Roche J, Hergalant S, Depp A, Ben Ammar I, Lafont AG, Policar T, Fontaine P, Milla S. First identification of dopamine receptors in pikeperch, Sander lucioperca, during the pre-ovulatory period. Comparative Biochemistry and Physiology. Part D, Genomics & Proteomics. 36: 100747. PMID 32987329 DOI: 10.1016/j.cbd.2020.100747   
2020 Pieterse L, van der Walt MM, Terre'Blanche G. C2-substituted quinazolinone derivatives exhibit A and/or A adenosine receptor affinities in the low micromolar range. Bioorganic & Medicinal Chemistry Letters. 30: 127274. PMID 32631506 DOI: 10.1016/j.bmcl.2020.127274   
2020 Kukkonen JP. Allosteric interactions via the orthosteric ligand binding sites in a constitutive G-protein-coupled receptor homodimer. Pharmacological Research. 105116. PMID 32783977 DOI: 10.1016/j.phrs.2020.105116   
2020 Yang JF, Williams AH, Penthala NR, Prather PL, Crooks PA, Zhan CG. Binding Modes and Selectivity of Cannabinoid 1 (CB1) and Cannabinoid 2 (CB2) Receptor Ligands. Acs Chemical Neuroscience. PMID 32997485 DOI: 10.1021/acschemneuro.0c00551   
2020 Jakubík J, Randáková A, Chetverikov N, El-Fakahany EE, Doležal V. The operational model of allosteric modulation of pharmacological agonism. Scientific Reports. 10: 14421. PMID 32879329 DOI: 10.1038/s41598-020-71228-y   
2020 Hino N, Marumo T, Kotani M, Shimazaki T, Kaku-Fukumoto A, Hikichi H, Karasawa JI, Tomishima Y, Komiyama H, Tatsuda E, Nozawa D, Nakamura T, Chaki S. A Novel Potent and Selective Histamine H3 Receptor Antagonist Enerisant: In Vitro Profiles, In Vivo Receptor Occupancy, Wake-Promoting and Pro-cognitive Effects in Rodents. The Journal of Pharmacology and Experimental Therapeutics. PMID 32862143 DOI: 10.1124/jpet.120.000185   
2020 Moritz AE, Bonifazi A, Guerrero AM, Kumar V, Free RB, Lane JR, Verma RK, Shi L, Newman AH, Sibley DR. Evidence for a stereoselective mechanism for bitopic activity by extended-length antagonists of the D3 dopamine receptor. Acs Chemical Neuroscience. PMID 32969645 DOI: 10.1021/acschemneuro.0c00425   
2020 Siamashvili M, Davis S. Late phase completed clinical trials investigating bromocriptine mesylate quick release as treatment of type 2 diabetes mellitus. Expert Opinion On Pharmacotherapy. 1-7. PMID 33030357 DOI: 10.1080/14656566.2020.1825683   
2020 Cerda-Cavieres C, Quiroz G, Iturriaga-Vásquez P, Rodríguez-Lavado J, Alarcón-Espósito J, Saitz C, Pessoa-Mahana CD, Chung H, Araya-Maturana R, Mella-Raipán J, Cabezas D, Ojeda-Gómez C, Reyes-Parada M, Pessoa-Mahana H. Synthesis, Docking, 3-D-Qsar, and Biological Assays of Novel Indole Derivatives Targeting Serotonin Transporter, Dopamine D2 Receptor, and Mao-A Enzyme: In the Pursuit for Potential Multitarget Directed Ligands. Molecules (Basel, Switzerland). 25. PMID 33050524 DOI: 10.3390/molecules25204614   
2020 Carlson HN, Murphy C, Pratt WE. Shifting motivational states: The effects of nucleus accumbens dopamine and opioid receptor activation on a modified effort-based choice task. Behavioural Brain Research. 112999. PMID 33161034 DOI: 10.1016/j.bbr.2020.112999   
2020 Del Castillo RM, Ramos E, Martínez A. Interaction of graphene with antipsychotic drugs: Is there any charge transfer process? Journal of Computational Chemistry. PMID 33048373 DOI: 10.1002/jcc.26433   
2020 Yang LK, Tao YX. Alanine Scanning Mutagenesis of the DRYxxI Motif and Intracellular Loop 2 of Human Melanocortin-4 Receptor. International Journal of Molecular Sciences. 21. PMID 33076233 DOI: 10.3390/ijms21207611   
2020 Mielnik CA, Sugamori KS, Finlay DB, Thorpe HHA, Schapira M, Sivananthan N, Li CK, Lam VM, Harrington S, Abdelrahman MH, Trembleau LA, McIntyre Burnham W, Khokhar JY, Salahpour A, Ramsey AJ, et al. A novel allosteric modulator of the cannabinoid CB receptor ameliorates hyperdopaminergia endophenotypes in rodent models. Neuropsychopharmacology : Official Publication of the American College of Neuropsychopharmacology. PMID 33036015 DOI: 10.1038/s41386-020-00876-5   
2020 Bhanu P, Kumar NH, Kumar SH, Relekar M, Anand DA, Kumar J. Comparative molecular docking analysis of the SARS CoV-2 Spike glycoprotein with the human ACE-2 receptors and thrombin. Bioinformation. 16: 532-538. PMID 32994678 DOI: 10.6026/97320630016532   
2020 Reeh K, Summers PA, Gould IR, Woscholski R, Vilar R. Design, synthesis and evaluation of a tripodal receptor for phosphatidylinositol phosphates. Scientific Reports. 10: 18450. PMID 33116198 DOI: 10.1038/s41598-020-75484-w   
2020 Pressly B, Lee RD, Barnych B, Hammock BD, Wulff H. Identification of the Functional Binding Site for the Convulsant Tetramethylenedisulfotetramine in the Pore of the α2β3γ2 GABA-A Receptor. Molecular Pharmacology. PMID 33109687 DOI: 10.1124/molpharm.120.000090   
2020 Gunera J, Baker JG, van Hilten N, Rosenbaum DM, Kolb P. Structure-Based Discovery of Novel Ligands for the Orexin 2 Receptor. Journal of Medicinal Chemistry. PMID 32977721 DOI: 10.1021/acs.jmedchem.0c00964   
2020 Xie XY, Li YY, Ma WH, Chen AF, Sun YT, Lee JY, Riad A, Xu DH, Mach RH, Huang YS. Synthesis, binding, and functional properties of tetrahydroisoquinolino-2-alkyl phenones as selective σR/TMEM97 ligands. European Journal of Medicinal Chemistry. 209: 112906. PMID 33049607 DOI: 10.1016/j.ejmech.2020.112906   
2020 Garrido-Gil P, Rodriguez-Perez AI, Lage L, Labandeira-Garcia JL. Estrogen deficiency and colonic function: surgical menopause and sex differences in angiotensin and dopamine receptor interaction. The Journals of Gerontology. Series a, Biological Sciences and Medical Sciences. PMID 32991714 DOI: 10.1093/gerona/glaa244   
2020 Masih A, Agnihotri AK, Srivastava JK, Pandey N, Bhat HR, Singh UP. Discovery of novel 1,3,5-triazine as adenosine A receptor antagonist for benefit in Parkinson's disease. Journal of Biochemical and Molecular Toxicology. e22659. PMID 33156955 DOI: 10.1002/jbt.22659   
2020 Norel X, Sugimoto Y, Ozen G, Abdelazeem H, Amgoud Y, Bouhadoun A, Bassiouni W, Goepp M, Mani S, Manikpurage HD, Senbel A, Longrois D, Heinemann A, Yao C, Clapp LH. International Union of Basic and Clinical Pharmacology. CIX. Differences and Similarities between Human and Rodent Prostaglandin E Receptors (EP1-4) and Prostacyclin Receptor (IP): Specific Roles in Pathophysiologic Conditions. Pharmacological Reviews. 72: 910-968. PMID 32962984 DOI: 10.1124/pr.120.019331   
2020 Shehroz M, Zaheer T, Hussain T. Computer-aided drug design against spike glycoprotein of SARS-CoV-2 to aid COVID-19 treatment. Heliyon. 6: e05278. PMID 33083627 DOI: 10.1016/j.heliyon.2020.e05278   
2020 da Rocha-Azevedo B, Lee S, Dasgupta A, Vega AR, de Oliveira LR, Kim T, Kittisopikul M, Malik ZA, Jaqaman K. Heterogeneity in VEGF Receptor-2 Mobility and Organization on the Endothelial Cell Surface Leads to Diverse Models of Activation by VEGF. Cell Reports. 32: 108187. PMID 32997988 DOI: 10.1016/j.celrep.2020.108187   
2020 Li Y, Coons LA, Houtman R, Carlson KE, Martin TA, Mayne CG, Melchers D, Jefferson TB, Ramsey JT, Katzenellenbogen JA, Korach KS. A mutant form of ERα associated with estrogen insensitivity affects the coupling between ligand binding and coactivator recruitment. Science Signaling. 13. PMID 32963012 DOI: 10.1126/scisignal.aaw4653   
2020 McMullan M, Kelly B, Mihigo HB, Keogh AP, Rodriguez F, Brocos-Mosquera I, García-Bea A, Miranda-Azpiazu P, Callado LF, Rozas I. Di-aryl guanidinium derivatives: Towards improved α2-Adrenergic affinity and antagonist activity. European Journal of Medicinal Chemistry. 112947. PMID 33139112 DOI: 10.1016/j.ejmech.2020.112947   
2020 Igawa T, Kishikawa S, Abe Y, Tsuda M, Inoue K, Ueda T. Analysis of binding residues in monoclonal antibody with high affinity for the head domain of the rat P2X4 receptor. Journal of Biochemistry. PMID 33169129 DOI: 10.1093/jb/mvaa124   
2020 Isaacs DP, Leman RP, Everett TJ, Lopez-Beltran H, Hamilton LR, Oleson EB. Buprenorphine is a weak dopamine releaser relative to heroin, but its pretreatment attenuates heroin-evoked dopamine release in rats. Neuropsychopharmacology Reports. PMID 32935483 DOI: 10.1002/npr2.12139   
2020 Lyons EL, Leone-Kabler S, Kovach AL, Thomas BF, Howlett AC. Cannabinoid receptor subtype influence on neuritogenesis in human SH-SY5Y cells. Molecular and Cellular Neurosciences. 103566. PMID 33049367 DOI: 10.1016/j.mcn.2020.103566   
2020 Sarkar A, Adamska-Bartlomiejczyk A, Piekielna-Ciesielska J, Wtorek K, Kluczyk A, Borics A, Janecka A. Design, Synthesis and Functional Analysis of Cyclic Opioid Peptides with Dmt-Tic Pharmacophore. Molecules (Basel, Switzerland). 25. PMID 32957550 DOI: 10.3390/molecules25184260   
2020 Sałaciak K, Głuch-Lutwin M, Siwek A, Szafarz M, Kazek G, Bednarski M, Nowiński L, Mitchell E, Jastrzębska-Więsek M, Partyka A, Wesołowska A, Kołaczkowski M, Szkaradek N, Marona H, Sapa J, et al. The antidepressant-like activity of chiral xanthone derivatives may be mediated by 5-HT1A receptor and β-arrestin signalling. Journal of Psychopharmacology (Oxford, England). 269881120959605. PMID 33103555 DOI: 10.1177/0269881120959605   
2020 Navarro G, Gonzalez A, Campanacci S, Rivas-Santisteban R, Reyes-Resina I, Casajuana-Martin N, Cordomí A, Pardo L, Franco R. Experimental and computational analysis of biased agonism on full-length and a C-terminally truncated adenosine A receptor. Computational and Structural Biotechnology Journal. 18: 2723-2732. PMID 33101610 DOI: 10.1016/j.csbj.2020.09.028   
2020 Gasperotti AF, Karina Herrera Seitz M, Balmaceda RS, Prosa LM, Jung K, Studdert CA. Direct binding of benzoate derivatives to two chemoreceptors with Cache sensor domains in Halomonas titanicae KHS3. Molecular Microbiology. PMID 33098326 DOI: 10.1111/mmi.14630   
2020 Ametovski A, Macdonald C, Manning JJ, Haneef SAS, Santiago M, Martin L, Sparkes E, Reckers A, Gerona RR, Connor M, Glass M, Banister SD. Exploring Stereochemical and Conformational Requirements at Cannabinoid Receptors for Synthetic Cannabinoids Related to SDB-006, 5F-SDB-006, CUMYL-PICA, and 5F-CUMYL-PICA. Acs Chemical Neuroscience. PMID 33054155 DOI: 10.1021/acschemneuro.0c00591   
2020 Turk LS, Mitchell D, Comoletti D. Purification of a heterodimeric Reelin construct to investigate binding stoichiometry. European Biophysics Journal : Ebj. PMID 33057791 DOI: 10.1007/s00249-020-01465-6   
2020 Watanabe H, Ishida K, Yamamoto M, Horiguchi M, Isobe Y. Synthesis and pharmacological evaluation of 11-(1,6-dimethyl-1,2,3,6-tetrahydropyridin-4-yl)-5H-dibenzo[b,e][1,4]diazepines with clozapine-like receptor occupancy at dopamine D/D receptor. Bioorganic & Medicinal Chemistry Letters. 30: 127563. PMID 32976928 DOI: 10.1016/j.bmcl.2020.127563   
2020 Grachev ID, Meyer PM, Becker GA, Bronzel M, Marsteller D, Pastino G, Voges O, Rabinovich L, Knebel H, Zientek F, Rullmann M, Sattler B, Patt M, Gerhards T, Strauss M, et al. Sigma-1 and dopamine D2/D3 receptor occupancy of pridopidine in healthy volunteers and patients with Huntington disease: a [F] fluspidine and [F] fallypride PET study. European Journal of Nuclear Medicine and Molecular Imaging. PMID 32995944 DOI: 10.1007/s00259-020-05030-3   
2020 Bernhard M, Laube B. Thermophoretic analysis of ligand-specific conformational states of the inhibitory glycine receptor embedded in copolymer nanodiscs. Scientific Reports. 10: 16569. PMID 33024136 DOI: 10.1038/s41598-020-73157-2   
2020 Moya B, Tontini C, Santos A. IgE sialylation: unravelling a key anaphylactic mediator. Allergy. PMID 33147354 DOI: 10.1111/all.14649   
2020 Prada JP, Wangorsch G, Kucka K, Lang I, Dandekar T, Wajant H. A systems-biology model of the tumor necrosis factor (TNF) interactions with TNF receptor 1 and 2. Bioinformatics (Oxford, England). PMID 32991680 DOI: 10.1093/bioinformatics/btaa844   
2020 Barrett JA, Choi J, Lakshmikanthan S, Kim YY, Greene D, Kolli P, Song TH, Choi IY, Kim YH, Lebel F. Eflapegrastim Enhanced Efficacy Compared to Pegfilgrastim in Neutropenic Rats Supports Potential for Same-Day Dosing. Experimental Hematology. PMID 33002567 DOI: 10.1016/j.exphem.2020.09.199   
2020 Boutin JA, Witt-Enderby PA, Sotriffer C, Zlotos DP. Melatonin receptor ligands: A pharmaco-chemical perspective. Journal of Pineal Research. 69: e12672. PMID 32531076 DOI: 10.1111/jpi.12672   
2020 Akhoon BA, Choudhary S, Tiwari H, Kumar A, Barik MR, Rathor L, Pandey R, Nargotra A. Discovery of a new donepezil-like acetylcholinesterase inhibitor for targeting Alzheimer's disease: computational studies with biological validation. Journal of Chemical Information and Modeling. PMID 32955256 DOI: 10.1021/acs.jcim.0c00496   
2020 Işbilir A, Möller J, Arimont M, Bobkov V, Perpiñá-Viciano C, Hoffmann C, Inoue A, Heukers R, de Graaf C, Smit MJ, Annibale P, Lohse MJ. Advanced fluorescence microscopy reveals disruption of dynamic CXCR4 dimerization by subpocket-specific inverse agonists. Proceedings of the National Academy of Sciences of the United States of America. PMID 33148803 DOI: 10.1073/pnas.2013319117   
2020 Li M, Huang C, Wu X, Ding F, Hu Z, Zhu Y, Zhao L, Hou L, Chen H, Wang H, Xu J, Tang D. The optimization of a novel selective antagonist for human M muscarinic acetylcholine receptor. Bioorganic & Medicinal Chemistry Letters. 30: 127632. PMID 33132116 DOI: 10.1016/j.bmcl.2020.127632   
2020 Zhang L, Li S, Liu X, Wang Z, Jiang M, Wang R, Xie L, Liu Q, Xie X, Shang D, Li M, Wei Z, Wang Y, Fan C, Luo ZQ, et al. Sensing of autoinducer-2 by functionally distinct receptors in prokaryotes. Nature Communications. 11: 5371. PMID 33097715 DOI: 10.1038/s41467-020-19243-5   
2020 Leung SW. The vascular impact of IP-TP receptor interactions. Acta Physiologica (Oxford, England). e13577. PMID 33135294 DOI: 10.1111/apha.13577   
2020 Bhattarai A, Pawnikar S, Miao Y. Mechanism of ligand recognition by human ACE2 receptor. Biorxiv : the Preprint Server For Biology. PMID 33140043 DOI: 10.1101/2020.10.30.362749   
2020 Mercer SE, Chaturvedula PV, Conway CM, Cook DA, Davis CD, Pin SS, Macci R, Schartman R, Signor LJ, Widmann KA, Whiterock VJ, Chen P, Xu C, Herbst JJ, Kostich WA, et al. Azepino-indazoles as calcitonin gene-related peptide (CGRP) receptor antagonists. Bioorganic & Medicinal Chemistry Letters. 127624. PMID 33096162 DOI: 10.1016/j.bmcl.2020.127624   
2020 Davies JR, Masuyer G, Stenmark P. Structural and Biochemical Characterization of Botulinum Neurotoxin Subtype B2 Binding to Its Receptors. Toxins. 12. PMID 32957706 DOI: 10.3390/toxins12090603   
2020 Ricart-Ortega M, Berizzi AE, Pereira V, Malhaire F, Catena J, Font J, Gómez-Santacana X, Muñoz L, Zussy C, Serra C, Rovira X, Goudet C, Llebaria A. Mechanistic Insights into Light-Driven Allosteric Control of GPCR Biological Activity. Acs Pharmacology & Translational Science. 3: 883-895. PMID 33073188 DOI: 10.1021/acsptsci.0c00054