| Year |
Citation |
Score |
| 2019 |
Chen S, Kapilashrami K, Senevirathne C, Wang Z, Wang J, Linscott JA, Luo M. Substrate-differentiated Transition States of SET7/9-catalyzed Lysine Methylation. Journal of the American Chemical Society. PMID 31034218 DOI: 10.1021/Jacs.9B02553 |
0.365 |
|
| 2016 |
Linscott JA, Kapilashrami K, Wang Z, Senevirathne C, Bothwell IR, Blum G, Luo M. Kinetic isotope effects reveal early transition state of protein lysine methyltransferase SET8. Proceedings of the National Academy of Sciences of the United States of America. PMID 27940912 DOI: 10.1073/Pnas.1609032114 |
0.35 |
|
| 2016 |
Daryaee F, Chang A, Schiebel J, Lu Y, Zhang Z, Kapilashrami K, Walker SG, Kisker C, Sotriffer CA, Fisher SL, Tonge PJ. Correlating Drug-Target Kinetics and In vivo Pharmacodynamics: Long Residence Time Inhibitors of the FabI Enoyl-ACP Reductase. Chemical Science. 7: 5945-5954. PMID 27547299 DOI: 10.1039/C6Sc01000H |
0.515 |
|
| 2016 |
Warrier T, Kapilashrami K, Argyrou A, Ioerger TR, Little D, Murphy KC, Nandakumar M, Park S, Gold B, Mi J, Zhang T, Meiler E, Rees M, Somersan-Karakaya S, Porras-De Francisco E, et al. N-methylation of a bactericidal compound as a resistance mechanism in Mycobacterium tuberculosis. Proceedings of the National Academy of Sciences of the United States of America. PMID 27432954 DOI: 10.1073/Pnas.1606590113 |
0.404 |
|
| 2016 |
Cai XC, Kapilashrami K, Luo M. Synthesis and Assays of Inhibitors of Methyltransferases. Methods in Enzymology. 574: 245-308. PMID 27423865 DOI: 10.1016/Bs.Mie.2016.01.009 |
0.431 |
|
| 2016 |
Bommineni GR, Kapilashrami K, Cummings JE, Lu Y, Knudson SE, Gu C, Walker SG, Slayden RA, Tonge PJ. Thiolactomycin-based inhibitors of bacterial β-ketoacyl-ACP synthases with in vivo activity. Journal of Medicinal Chemistry. PMID 27187871 DOI: 10.1021/Acs.Jmedchem.6B00236 |
0.56 |
|
| 2016 |
Cai XC, Kapilashrami K, Luo M. Synthesis and Assays of Inhibitors of Methyltransferases Methods in Enzymology. DOI: 10.1016/bs.mie.2016.01.009 |
0.355 |
|
| 2015 |
Torres A, Luke JD, Kullas AL, Kapilashrami K, Botbol Y, Koller A, Tonge PJ, Chen EI, Macian F, van der Velden AW. Asparagine deprivation mediated by Salmonella asparaginase causes suppression of activation-induced T cell metabolic reprogramming. Journal of Leukocyte Biology. PMID 26497246 DOI: 10.1189/Jlb.4A0615-252R |
0.47 |
|
| 2015 |
Aldawsari FS, Aguayo-Ortiz R, Kapilashrami K, Yoo J, Luo M, Medina-Franco JL, Velázquez-Martínez CA. Resveratrol-salicylate derivatives as selective DNMT3 inhibitors and anticancer agents. Journal of Enzyme Inhibition and Medicinal Chemistry. 1-9. PMID 26118420 DOI: 10.3109/14756366.2015.1058256 |
0.466 |
|
| 2013 |
Schiebel J, Kapilashrami K, Fekete A, Bommineni GR, Schaefer CM, Mueller MJ, Tonge PJ, Kisker C. Structural basis for the recognition of mycolic acid precursors by KasA, a condensing enzyme and drug target from Mycobacterium tuberculosis. The Journal of Biological Chemistry. 288: 34190-204. PMID 24108128 DOI: 10.1074/Jbc.M113.511436 |
0.556 |
|
| 2013 |
Kapilashrami K, Bommineni GR, Machutta CA, Kim P, Lai CT, Simmerling C, Picart F, Tonge PJ. Thiolactomycin-based β-ketoacyl-AcpM synthase A (KasA) inhibitors: fragment-based inhibitor discovery using transient one-dimensional nuclear overhauser effect NMR spectroscopy. The Journal of Biological Chemistry. 288: 6045-52. PMID 23306195 DOI: 10.1074/Jbc.M112.414516 |
0.566 |
|
| 2010 |
Machutta CA, Bommineni GR, Luckner SR, Kapilashrami K, Ruzsicska B, Simmerling C, Kisker C, Tonge PJ. Slow onset inhibition of bacterial beta-ketoacyl-acyl carrier protein synthases by thiolactomycin. The Journal of Biological Chemistry. 285: 6161-9. PMID 20018879 DOI: 10.1074/Jbc.M109.077909 |
0.581 |
|
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