| Year |
Citation |
Score |
| 2021 |
Sahani RL, Diana-Rivero R, Vernekar SKV, Wang L, Du H, Zhang H, Castaner AE, Casey MC, Kirby KA, Tedbury PR, Xie J, Sarafianos SG, Wang Z. Design, Synthesis and Characterization of HIV-1 CA-Targeting Small Molecules: Conformational Restriction of PF74. Viruses. 13. PMID 33804121 DOI: 10.3390/v13030479 |
0.583 |
|
| 2021 |
Wang L, Casey MC, Vernekar SKV, Sahani RL, Kirby KA, Du H, Zhang H, Tedbury PR, Xie J, Sarafianos SG, Wang Z. Novel PF74-like small molecules targeting the HIV-1 capsid protein: Balance of potency and metabolic stability. Acta Pharmaceutica Sinica. B. 11: 810-822. PMID 33777683 DOI: 10.1016/J.Apsb.2020.07.016 |
0.57 |
|
| 2020 |
Wang L, Casey MC, Vernekar SKV, Sahani RL, Kankanala J, Kirby KA, Du H, Hachiya A, Zhang H, Tedbury PR, Xie J, Sarafianos SG, Wang Z. Novel HIV-1 capsid-targeting small molecules of the PF74 binding site. European Journal of Medicinal Chemistry. 204: 112626. PMID 32814250 DOI: 10.1016/J.Ejmech.2020.112626 |
0.568 |
|
| 2020 |
Wang L, Casey MC, Vernekar SKV, Do HT, Sahani RL, Kirby KA, Du H, Hachiya A, Zhang H, Tedbury PR, Xie J, Sarafianos SG, Wang Z. Chemical profiling of HIV-1 capsid-targeting antiviral PF74. European Journal of Medicinal Chemistry. 200: 112427. PMID 32438252 DOI: 10.1016/J.Ejmech.2020.112427 |
0.545 |
|
| 2020 |
Vernekar SKV, Sahani RL, Casey MC, Kankanala J, Wang L, Kirby KA, Du H, Zhang H, Tedbury PR, Xie J, Sarafianos SG, Wang Z. Toward Structurally Novel and Metabolically Stable HIV-1 Capsid-Targeting Small Molecules. Viruses. 12. PMID 32316297 DOI: 10.3390/V12040452 |
0.607 |
|
| 2017 |
Vernekar SKV, Tang J, Wu B, Huber AD, Casey MC, Myshakina NS, Wilson DJ, Kankanala J, Kirby KA, Parniak MA, Sarafianos SG, Wang Z. Double-winged 3-Hydroxypyrimidine-2,4-diones: Potent and Selective Inhibition against HIV-1 RNase H with Significant Antiviral Activity. Journal of Medicinal Chemistry. PMID 28525279 DOI: 10.1021/Acs.Jmedchem.7B00440 |
0.554 |
|
| 2017 |
Tang J, Vernekar SK, Chen YL, Miller L, Huber AD, Myshakina N, Sarafianos SG, Parniak MA, Wang Z. Synthesis, biological evaluation and molecular modeling of 2-Hydroxyisoquinoline-1,3-dione analogues as inhibitors of HIV reverse transcriptase associated ribonuclease H and polymerase. European Journal of Medicinal Chemistry. 133: 85-96. PMID 28384548 DOI: 10.1016/J.Ejmech.2017.03.059 |
0.555 |
|
| 2015 |
Vernekar SK, Qiu L, Zhang J, Kankanala J, Li H, Geraghty RJ, Wang Z. 5'-Silylated 3'-1,2,3-triazolyl Thymidine Analogues as Inhibitors of West Nile Virus and Dengue Virus. Journal of Medicinal Chemistry. 58: 4016-28. PMID 25909386 DOI: 10.1021/Acs.Jmedchem.5B00327 |
0.537 |
|
| 2015 |
Vernekar SK, Liu Z, Nagy E, Miller L, Kirby KA, Wilson DJ, Kankanala J, Sarafianos SG, Parniak MA, Wang Z. Design, synthesis, biochemical, and antiviral evaluations of C6 benzyl and C6 biarylmethyl substituted 2-hydroxylisoquinoline-1,3-diones: dual inhibition against HIV reverse transcriptase-associated RNase H and polymerase with antiviral activities. Journal of Medicinal Chemistry. 58: 651-64. PMID 25522204 DOI: 10.1021/Jm501132S |
0.538 |
|
| 2014 |
Vernekar SKV, Qiu L, Zacharias J, Geraghty RJ, Wang Z. Synthesis and antiviral evaluation of 4′-(1,2,3-triazol-1-yl) thymidines Medchemcomm. 5: 603-608. DOI: 10.1039/C4Md00039K |
0.56 |
|
| 2013 |
Sirivolu VR, Vernekar SK, Ilina T, Myshakina NS, Parniak MA, Wang Z. Clicking 3'-azidothymidine into novel potent inhibitors of human immunodeficiency virus. Journal of Medicinal Chemistry. 56: 8765-80. PMID 24102161 DOI: 10.1021/Jm401232V |
0.579 |
|
| 2012 |
Sirivolu VR, Vernekar SK, Marchand C, Naumova A, Chergui A, Renaud A, Stephen AG, Chen F, Sham YY, Pommier Y, Wang Z. 5-Arylidenethioxothiazolidinones as inhibitors of tyrosyl-DNA phosphodiesterase I. Journal of Medicinal Chemistry. 55: 8671-84. PMID 23006064 DOI: 10.1021/Jm3008773 |
0.446 |
|
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