| Year |
Citation |
Score |
| 2020 |
Guillon C, Vetrano AM, Saxena J, Hunter A, Verderone G, Finetti TM, Wisnoski J, DeMatteo PW, Rapp RD, Heindel ND, Joseph LB, Heck DE, Laskin JD. Derivatives of 1,2,4-triazole imines acting as dual iNOS and tumor cell growth inhibitors. Bioorganic Chemistry. 103: 104128. PMID 32745761 DOI: 10.1016/J.Bioorg.2020.104128 |
0.331 |
|
| 2019 |
Guillon C, Jan YH, Heck DE, Mariano TM, Rapp RD, Jetter M, Kardos K, Whittemore M, Akyea E, Jabin I, Laskin JD, Heindel ND. Phototoxicity of 7-oxycoumarins with keratinocytes in culture. Bioorganic Chemistry. 89: 103014. PMID 31170642 DOI: 10.1016/J.Bioorg.2019.103014 |
0.343 |
|
| 2018 |
Laskin JD, Jan YH, Jetter MM, Guillon CD, Mariano TM, Heck DE, Heindel ND. Identification of a Pyranocoumarin Photosensitizer that is a Potent Inhibitor of Keratinocyte Growth. Photochemistry and Photobiology. PMID 29315592 DOI: 10.1111/Php.12882 |
0.378 |
|
| 2016 |
Szilagyi JT, Mishin V, Heck DE, Jan YH, Aleksunes LM, Richardson JR, Heindel ND, Laskin DL, Laskin JD. Selective Targeting of Heme Protein in Cytochrome P450 and Nitric Oxide Synthase by Diphenyleneiodonium. Toxicological Sciences : An Official Journal of the Society of Toxicology. PMID 26880746 DOI: 10.1093/Toxsci/Kfw031 |
0.301 |
|
| 2015 |
Yang S, Jan YH, Mishin V, Richardson JR, Hossain MM, Heindel ND, Heck DE, Laskin DL, Laskin JD. Sulfa drugs inhibit sepiapterin reduction and chemical redox cycling by sepiapterin reductase. The Journal of Pharmacology and Experimental Therapeutics. 352: 529-40. PMID 25550200 DOI: 10.1124/Jpet.114.221572 |
0.312 |
|
| 2012 |
Fabio K, Guillon C, Lacey CJ, Lu SF, Heindel ND, Ferris CF, Placzek M, Jones G, Brownstein MJ, Simon NG. Synthesis and evaluation of potent and selective human V1a receptor antagonists as potential ligands for PET or SPECT imaging. Bioorganic & Medicinal Chemistry. 20: 1337-45. PMID 22249122 DOI: 10.1016/J.Bmc.2011.12.013 |
0.3 |
|
| 2012 |
Young SC, Fabio KM, Huang MT, Saxena J, Harman MP, Guillon CD, Vetrano AM, Heck DE, Flowers RA, Heindel ND, Laskin JD. Investigation of anticholinergic and non-steroidal anti-inflammatory prodrugs which reduce chemically induced skin inflammation. Journal of Applied Toxicology : Jat. 32: 135-41. PMID 21319177 DOI: 10.1002/Jat.1645 |
0.304 |
|
| 2005 |
Martey CA, Vetrano AM, Whittemore MS, Mariano TM, Heck DE, Laskin DL, Heindel ND, Laskin JD. Inhibition of interferon-gamma signaling by a mercurio-substituted dihydropsoralen in murine keratinocytes. Biochemical Pharmacology. 70: 1726-34. PMID 16259964 DOI: 10.1016/J.Bcp.2005.10.001 |
0.686 |
|
| 2002 |
Martey CA, Vetrano AM, Whittemore MS, Mariano TM, Gentile SL, Heck DE, Laskin DL, Heindel ND, Laskin JD. Mechanisms of growth inhibition in keratinocytes by mercurio-substituted 4',5'-dihydropsoralens. Biochemical Pharmacology. 63: 2001-9. PMID 12093477 DOI: 10.1016/S0006-2952(02)00992-9 |
0.697 |
|
| 2002 |
Mariano TM, Vetrano AM, Gentile SL, Heck DE, Whittemore MS, Guillon CD, Jabin I, Rapp RD, Heindel ND, Laskin JD. Cell-impermeant pyridinium derivatives of psoralens as inhibitors of keratinocyte growth. Biochemical Pharmacology. 63: 31-9. PMID 11754871 DOI: 10.1016/S0006-2952(01)00855-3 |
0.359 |
|
| 2001 |
Whittemore MS, Heindel ND, Jabin I, Guillon C, Mcneel TE, Rapp RD, Heck DE, Laskin JD. Synthetic approaches to 4,8-dimethyl-5′-(N-pyridiniummethyl)- 4′,5′-dihydropsoralens and 4,8-dimethyl-5′- (N-aminomethyl)- 4′,5′-dihydropsoralens†‡ Journal of Heterocyclic Chemistry. 38: 909-916. DOI: 10.1002/Jhet.5570380415 |
0.317 |
|
| 2000 |
Jabin I, Heindel ND, Rapp RD, Laskin JD. Synthetic approaches to 3-substituted-5′-(N-pyridiniummethyl)-4′,5′-dihydropsoralen † Journal of Heterocyclic Chemistry. 37: 31-39. DOI: 10.1002/Jhet.5570370106 |
0.321 |
|
| 1992 |
Stephont RL, Niedbala RS, Schrayt KJ, Heindel ND. Synthesis of 4-trans-[1-[4-[2-(5-chloro-2-methoxybenzamido)ethyl] benzenesulfonyl]ureido]cyclohexanol hemisuccinate ester Organic Preparations and Procedures International. 24: 339-342. DOI: 10.1080/00304949209355897 |
0.332 |
|
| 1991 |
Heindel ND, Van Dongen JMAM, Sachais BS, Phillips JH, Gallo MA, Laskin JD. Syntheses of psoralen analogues and evaluation of their inhibition of epidermal growth factor binding Journal of Pharmaceutical Sciences. 80: 686-689. PMID 1941569 DOI: 10.1002/Jps.2600800715 |
0.345 |
|
| 1990 |
Jetter MM, Heindel ND, Laskin JD. Novel synthesis of dihydroxanthyletin and dihydroseselin derivatives Journal of Heterocyclic Chemistry. 27: 995-997. DOI: 10.1002/Jhet.5570270433 |
0.318 |
|
| 1986 |
Heindel ND, Foster N, Varkey T. Nitrations of 4',5'-dihydropsoralens: A route to radiopharmaceutical precursors Journal of Heterocyclic Chemistry. 23: 1579-1582. DOI: 10.1002/Jhet.5570230564 |
0.307 |
|
| 1985 |
Heindel ND, Van Dort M, Cahn M. The 1,3,4-oxadiazole moiety, a protective synthon for indirect radioiodination Journal of Heterocyclic Chemistry. 22: 209-210. DOI: 10.1002/Jhet.5570220149 |
0.347 |
|
| 1985 |
Heindel ND, Choudhuri M, Ressner J, Foster N. Aminomethyl psoralens. Electrophilic substitutions of hydroxymethylphthamide on linear furocoumarins Journal of Heterocyclic Chemistry. 22: 73-76. DOI: 10.1002/Jhet.5570220119 |
0.335 |
|
| 1983 |
Heindel ND, Conley RA, Minatelli JA, Boschelli DH. Benzylidene-thiolactone rearrangement: Synthesis and rearrangement of 5-substituted 3-benzylidene-4-thiolen-2-ones Journal of Organic Chemistry. 48: 3051-3053. DOI: 10.1021/Jo00166A023 |
0.304 |
|
| 1981 |
Heindel ND, Minatelli JA. Synthesis and antibacterial and anticancer evaluations of α-methylene-γ-butyrolactones Journal of Pharmaceutical Sciences. 70: 84-86. PMID 7229935 DOI: 10.1002/Jps.2600700117 |
0.312 |
|
| 1981 |
Miller GA, Heindel ND, Minatelli JA. Improved Synthesis Of 3‐Aralkylidene‐5‐Arylthiophen‐2‐(3H)Ones Journal of Heterocyclic Chemistry. 13: 1253-1254. DOI: 10.1002/Jhet.5570180638 |
0.342 |
|
| 1980 |
Heindel ND, Reid JR. 7H-[1,2,4]triazolo[5,1-b][1,3]thiazin-7-ones by deamination cyclization of S-acrylates of 4-amino-3(3H)-1,2,4-triazolethiones Journal of Organic Chemistry. 45: 2479-2482. DOI: 10.1021/Jo01300A043 |
0.3 |
|
| 1980 |
Heindel ND, Reid JR. 4-Amino-3-mercapto-4H-1,2,4-triazoles and propargyl aldehydes: A new route to 3-R-8-aryl-1,2,4-triazolo[3,4-b]1,3,4-thiadiazepines Journal of Heterocyclic Chemistry. 17: 1087-1088. DOI: 10.1002/Jhet.5570170547 |
0.305 |
|
| 1980 |
Heindel ND, Friedrich G, Tsai MC. Thiohydrazides and acetylene esters, A new route to 1,3,4-thiadiazoles Journal of Heterocyclic Chemistry. 17: 191-193. DOI: 10.1002/Jhet.5570170138 |
0.302 |
|
| 1979 |
Heindel ND, Corley EG. Cyclization-hydrolysis of a 1,2,4-benzothiadiazine 1,1-dioxide through a diazonium intermediate Journal of the Chemical Society, Chemical Communications. 1008-1009. DOI: 10.1002/Chin.198011245 |
0.302 |
|
| 1978 |
Leiby RW, Corley EG, Heindel ND. A unique ring contraction of 1,4-dihydro-5H-1,3,4-benzotriazepin-5-ones to 1-methyl-2-(methylamino)-4(1H)-quinazolinones via an intermediate Dimroth rearrangement Journal of Organic Chemistry. 43: 3427-3429. DOI: 10.1021/Jo00411A050 |
0.304 |
|
| 1977 |
Leiby RW, Heindel ND. New compounds: synthesis of 2 amino 5H 1,3,4 benzotriazepin 5 ones Journal of Pharmaceutical Sciences. 66: 605-606. PMID 853376 DOI: 10.1002/Jps.2600660444 |
0.362 |
|
| 1977 |
Heindel ND, Fives WP, Carrano RA. New synthesis of 1,4,2-dioxazoles and their pharmacological properties. Journal of Pharmaceutical Sciences. 66: 772-5. PMID 301562 DOI: 10.1002/Chin.197742188 |
0.34 |
|
| 1977 |
Beam CF, Park CA, Heindel ND, Fives WP. The Synthesis of 2-Carbomethoxy-2-carbomethoxymethyl-2,3-dihydro-4(1H)quinazolinones Journal of Heterocyclic Chemistry. 14: 703-704. DOI: 10.1002/Jhet.5570140439 |
0.328 |
|
| 1977 |
Leiby RW, Heindel ND. New Compounds- Synthesis Of 2-Amino-5H-1,3,4-Benzotriazepin-5-Ones Cheminform. 8. DOI: 10.1002/Chin.197744273 |
0.353 |
|
| 1976 |
Leibv RW, Heindel ND. Substituted 2-aminobenzoyl derivatives of methylhydrazine Synthetic Communications. 6: 295-297. DOI: 10.1080/00397917608063525 |
0.329 |
|
| 1976 |
Conley RA, Heindel ND. Thianaphthen-2-one chemistry. 2. The benzylidene thiolactone rearrangement: Synthesis of 2-arylthianaphthene-3-carboxylic acids and esters Journal of Organic Chemistry. 41: 3743-3746. DOI: 10.1021/Jo00885A020 |
0.306 |
|
| 1976 |
Reid JR, Heindel ND. Improved syntheses of 5-substituted-4-amino-3-mercapto-(4H)-1,2,4-triazoles Journal of Heterocyclic Chemistry. 13: 925-926. DOI: 10.1002/Jhet.5570130450 |
0.343 |
|
| 1975 |
Conley RA, Heindel ND. Thianaphthen-2-one chemistry. I. Synthesis of 6H-benzothieno[3,2-c][1]benzopyran-6-ones (11-thiacoumestans) Journal of Organic Chemistry. 40: 3169-3173. DOI: 10.1021/Jo00910A002 |
0.325 |
|
| 1972 |
Lemke TF, Snady HW, Heindel ND. Synthesis and mass spectra of some 2-carbomethoxy-2-carbomethoxymethyl-2,3-dihydro-4(1H)-quinazolinones Journal of Organic Chemistry. 37: 2337-2340. DOI: 10.1021/Jo00979A028 |
0.309 |
|
| 1971 |
Heindel ND, Fives WP, Lemke TF, Carrano RA. Synthesis and selected pharmacology of anthranilamides. Journal of Pharmaceutical Sciences. 60: 703-7. PMID 5125768 DOI: 10.1002/Jps.2600600509 |
0.314 |
|
| 1970 |
Heindel ND, Molnar J. Synthesis and antimalarial activity of amodiaquine analogs Journal of Medicinal Chemistry. 13: 156-157. PMID 5412100 DOI: 10.1021/Jm00295A051 |
0.324 |
|
| 1970 |
Heindel ND, Kennewell PD, Pfau M. Imine-enamine tautomers from hydrazine and aryl hydrazine additions to acetylenedicarboxylate Journal of Organic Chemistry. 35: 80-83. DOI: 10.1021/Jo00826A019 |
0.314 |
|
| 1969 |
Heindel ND, Kennewell PD, Fish VB. Enamine formation from anilines and methyl propiolate. The synthesis of 4(1h)-quinolones Journal of Heterocyclic Chemistry. 6: 77-81. DOI: 10.1002/Jhet.5570060113 |
0.323 |
|
| 1968 |
Heindel ND, Bechara IS, Kennewell PD, Molnar J, Ohnmacht CJ, Lemke SM, Lemke TF. Cyclization of Aniline-acetylenedicarboxylate adducts. A modified Conrad-Limpach method for the synthesis of potential aritimalarials Journal of Medicinal Chemistry. 11: 1218-1221. PMID 5680041 DOI: 10.1021/Jm00312A025 |
0.303 |
|
| 1968 |
Heindel ND, Fish VB, Lemke TF. Cyclization of anthranilamide-acetylenedicarboxylate adducts. A facile synthesis of 1,4-benzodiazepine-3,5-diones Journal of Organic Chemistry. 33: 3997-4004. DOI: 10.1021/Jo01275A001 |
0.338 |
|
| 1967 |
Heindel ND, Bechara IS, Lemke TF, Fish VB. Cyclization of aniline-acetylenedicarboxylate adducts. An improved synthesis of 8-nitro-2-carbomethoxy-4(1H)-quinolones Journal of Organic Chemistry. 32: 4155-4157. DOI: 10.1021/Jo01287A127 |
0.336 |
|
| 1967 |
Heindel ND, Fish VB, Ryan MF, Lepley AR. Heterocyclic syntheses involving acetylenedicarboxylate adducts of thiosalicylic acid derivatives Journal of Organic Chemistry. 32: 2678-2681. DOI: 10.1021/Jo01284A006 |
0.317 |
|
| 1967 |
Taylor EC, Heindel ND. A convenient synthesis of dimethyl 4-phenylacridinates Journal of Organic Chemistry. 32: 1666-1667. DOI: 10.1021/Jo01280A105 |
0.318 |
|
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