Year |
Citation |
Score |
2005 |
Esslinger CS, Agarwal S, Gerdes J, Wilson PA, Davis ES, Awes AN, O'Brien E, Mavencamp T, Koch HP, Poulsen DJ, Rhoderick JF, Chamberlin AR, Kavanaugh MP, Bridges RJ. The substituted aspartate analogue L-beta-threo-benzyl-aspartate preferentially inhibits the neuronal excitatory amino acid transporter EAAT3. Neuropharmacology. 49: 850-61. PMID 16183084 DOI: 10.1016/J.Neuropharm.2005.08.009 |
0.852 |
|
2005 |
Bridges RJ, Esslinger CS. The excitatory amino acid transporters: pharmacological insights on substrate and inhibitor specificity of the EAAT subtypes. Pharmacology & Therapeutics. 107: 271-85. PMID 16112332 DOI: 10.1016/j.pharmthera.2005.01.002 |
0.512 |
|
2005 |
Esslinger CS, Cybulski KA, Rhoderick JF. Ngamma-aryl glutamine analogues as probes of the ASCT2 neutral amino acid transporter binding site. Bioorganic & Medicinal Chemistry. 13: 1111-8. PMID 15670919 DOI: 10.1016/j.bmc.2004.11.028 |
0.329 |
|
2002 |
Carrigan CN, Bartlett RD, Esslinger CS, Cybulski KA, Tongcharoensirikul P, Bridges RJ, Thompson CM. Synthesis and in vitro pharmacology of substituted quinoline-2,4-dicarboxylic acids as inhibitors of vesicular glutamate transport. Journal of Medicinal Chemistry. 45: 2260-76. PMID 12014964 DOI: 10.1021/Jm010261Z |
0.512 |
|
1999 |
Koch HP, Kavanaugh MP, Esslinger CS, Zerangue N, Humphrey JM, Amara SG, Chamberlin AR, Bridges RJ. Differentiation of substrate and nonsubstrate inhibitors of the high-affinity, sodium-dependent glutamate transporters. Molecular Pharmacology. 56: 1095-104. PMID 10570036 |
0.571 |
|
1999 |
Carrigan CN, Esslinger CS, Bartlett RD, Bridges RJ, Thompson CM. Quinoline-2,4-dicarboxylic acids: synthesis and evaluation as inhibitors of the glutamate vesicular transport system. Bioorganic & Medicinal Chemistry Letters. 9: 2607-12. PMID 10498218 DOI: 10.1016/S0960-894X(99)00444-8 |
0.503 |
|
1998 |
Esslinger CS, Koch HP, Kavanaugh MP, Philips DP, Chamberlin AR, Thompson CM, Bridges RJ. Structural determinants of substrates and inhibitors: probing glutamate transporters with 2,4-methanopyrrolidine-2,4-dicarboxylate. Bioorganic & Medicinal Chemistry Letters. 8: 3101-6. PMID 9873684 DOI: 10.1016/S0960-894X(98)00560-5 |
0.521 |
|
1998 |
Bartlett RD, Esslinger CS, Thompson CM, Bridges RJ. Substituted quinolines as inhibitors of L-glutamate transport into synaptic vesicles. Neuropharmacology. 37: 839-46. PMID 9776380 DOI: 10.1016/S0028-3908(98)00080-X |
0.624 |
|
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