Year |
Citation |
Score |
2017 |
Scannevin RH, Alexander R, Mezzasalma Haarlander T, Burke SL, Singer M, Hou C, Zhang YM, Maguire D, Spurlino J, Deckman I, Carroll KI, Lewandowski F, Devine E, Dzordzorme K, Tounge B, ... ... Rhodes KJ, et al. Discovery of a highly selective chemical inhibitor of matrix metalloproteinase-9 (MMP-9) that allosterically inhibits zymogen activation. The Journal of Biological Chemistry. PMID 28860188 DOI: 10.1074/Jbc.M117.806075 |
0.397 |
|
2011 |
Wilson LJ, Wang B, Yang SM, Scannevin RH, Burke SL, Karnachi P, Rhodes KJ, Murray WV. Discovery of novel Cobactin-T based matrix metalloproteinase inhibitors via a ring closing metathesis strategy. Bioorganic & Medicinal Chemistry Letters. 21: 6485-90. PMID 21925881 DOI: 10.1016/j.bmcl.2011.08.068 |
0.346 |
|
2008 |
Yang SM, Scannevin RH, Wang B, Burke SL, Wilson LJ, Karnachi P, Rhodes KJ, Lagu B, Murray WV. beta-N-Biaryl ether sulfonamide hydroxamates as potent gelatinase inhibitors: part 1. Design, synthesis, and lead identification. Bioorganic & Medicinal Chemistry Letters. 18: 1135-9. PMID 18086526 DOI: 10.1016/j.bmcl.2007.11.119 |
0.372 |
|
2008 |
Yang SM, Scannevin RH, Wang B, Burke SL, Huang Z, Karnachi P, Wilson LJ, Rhodes KJ, Lagu B, Murray WV. beta-N-Biaryl ether sulfonamide hydroxamates as potent gelatinase inhibitors: part 2. Optimization of alpha-amino substituents. Bioorganic & Medicinal Chemistry Letters. 18: 1140-5. PMID 18083558 DOI: 10.1016/j.bmcl.2007.11.129 |
0.301 |
|
2008 |
Zhang YM, Fan X, Chakaravarty D, Xiang B, Scannevin RH, Huang Z, Ma J, Burke SL, Karnachi P, Rhodes KJ, Jackson PF. 1-Hydroxy-2-pyridinone-based MMP inhibitors: synthesis and biological evaluation for the treatment of ischemic stroke. Bioorganic & Medicinal Chemistry Letters. 18: 409-13. PMID 17981034 DOI: 10.1016/j.bmcl.2007.10.045 |
0.452 |
|
2008 |
Zhang YM, Fan X, Yang SM, Scannevin RH, Burke SL, Rhodes KJ, Jackson PF. Syntheses and in vitro evaluation of arylsulfone-based MMP inhibitors with heterocycle-derived zinc-binding groups (ZBGs). Bioorganic & Medicinal Chemistry Letters. 18: 405-8. PMID 17980583 DOI: 10.1016/j.bmcl.2007.10.049 |
0.459 |
|
2006 |
Zhang YM, Fan X, Xiang B, Chakravarty D, Scannevin R, Burke S, Karnachi P, Rhodes K, Jackson P. Synthesis and SAR of alpha-sulfonylcarboxylic acids as potent matrix metalloproteinase inhibitors. Bioorganic & Medicinal Chemistry Letters. 16: 3096-100. PMID 16632358 DOI: 10.1002/chin.200637084 |
0.47 |
|
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