Kristoffer Sahlholm - Related publications

Affiliations: 
Karolinska Institute, Stockholm, Sweden 
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50 most relevant papers in past 60 days:
Year Citation  Score
2020 Yarur HE, González MP, Verbel-Vergara D, Andrés ME, Gysling K. Crosstalk between dopamine D1 and corticotropin releasing factor type 2 receptors leads to occlusion of their ERK1/2 signaling. Journal of Neurochemistry. PMID 32215915 DOI: 10.1111/jnc.15016   
2020 Wilding TJ, Huettner JE. Cadmium activates AMPA and NMDA receptors with M3 helix cysteine substitutions. The Journal of General Physiology. 152. PMID 32342094 DOI: 10.1085/jgp.201912537   
2020 Gao J, Chang Z, Tian R, Li P, Ahmad F, Jia X, Liang Q, Zhao X. Reversible and site-specific immobilization of β-adrenergic receptor by aptamer-directed method for receptor-drug interaction analysis. Journal of Chromatography. A. 461091. PMID 32376022 DOI: 10.1016/j.chroma.2020.461091   
2020 Liu C, Xia L, Fu K, Cao X, Yan W, Cheng J, Roux T, Peletier LA, Yin X, Guo D. Revisit ligand-receptor interaction at the human vasopressin V receptor: A kinetic perspective. European Journal of Pharmacology. 173157. PMID 32360346 DOI: 10.1016/j.ejphar.2020.173157   
2020 Christie AE, Hull JJ, Dickinson PS. Assessment and comparison of putative amine receptor complement/diversity in the brain and eyestalk ganglia of the lobster, Homarus americanus. Invertebrate Neuroscience : In. 20: 7. PMID 32215729 DOI: 10.1007/s10158-020-0239-5   
2020 Fernandez TJ, De Maria M, Lobingier BT. A cellular perspective of bias at G protein-coupled receptors. Protein Science : a Publication of the Protein Society. PMID 32297394 DOI: 10.1002/pro.3872   
2020 Wang Y, Joseph J, Gao Y, Hu B, Geng X, Wu D, Wang J, Zhang F. Revealing the Interaction Modes of 5-HT2A Receptor Antagonists and the Structure-Based Virtual Screening from FDA and TCMNP Database. Journal of Biomolecular Structure & Dynamics. 1-20. PMID 32406337 DOI: 10.1080/07391102.2020.1768900   
2020 Pandey S, Maharana J, Li XX, Woodruff TM, Shukla AK. Emerging Insights into the Structure and Function of Complement C5a Receptors. Trends in Biochemical Sciences. PMID 32402749 DOI: 10.1016/j.tibs.2020.04.004   
2020 Gingell JJ, Rees TA, Hendrikse ER, Siow A, Rennison D, Scotter J, Harris PWR, Brimble MA, Walker CS, Hay DL. Distinct Patterns of Internalization of Different Calcitonin Gene-Related Peptide Receptors. Acs Pharmacology & Translational Science. 3: 296-304. PMID 32296769 DOI: 10.1021/acsptsci.9b00089   
2020 Baldwin MW, Ko MC. Functional evolution of vertebrate sensory receptors. Hormones and Behavior. 104771. PMID 32437717 DOI: 10.1016/j.yhbeh.2020.104771   
2020 Hendrikse ER, Liew LP, Bower RL, Bonnet M, Jamaluddin MA, Prodan N, Richards KD, Walker CS, Pairaudeau G, Smith DM, Rujan RM, Sudra R, Reynolds CA, Booe JM, Pioszak AA, et al. Identification of Small-Molecule Positive Modulators of Calcitonin-like Receptor-Based Receptors. Acs Pharmacology & Translational Science. 3: 305-320. PMID 32296770 DOI: 10.1021/acsptsci.9b00108   
2020 Zhu Z, Yi F, Epplin MP, Liu D, Summer SL, Mizu R, Shaulsky G, XiangWei W, Tang W, Burger PB, Menaldino DS, Myers SJ, Liotta DC, Hansen KB, Yuan H, et al. Negative allosteric modulation of GluN1/GluN3 NMDA receptors. Neuropharmacology. 108117. PMID 32389749 DOI: 10.1016/j.neuropharm.2020.108117   
2020 Sadanandan SM, Kreko-Pierce T, Khatri SN, Pugh JR. Cannabinoid type 2 receptors inhibit GABAA receptor-mediated currents in cerebellar Purkinje cells of juvenile mice. Plos One. 15: e0233020. PMID 32437355 DOI: 10.1371/journal.pone.0233020   
2020 Del Rosario JS, Yudin Y, Su S, Hartle CM, Mirshahi T, Rohacs T. Gi-coupled receptor activation potentiates Piezo2 currents via Gβγ. Embo Reports. e49124. PMID 32227462 DOI: 10.15252/embr.201949124   
2020 Lü S, Jiang M, Tian X, Hong S, Zhang J, Zhang Y. Characterization of an A-Type Muscarinic Acetylcholine Receptor and Its Possible Non-neuronal Role in the Oriental Armyworm, Walker (Lepidoptera: Noctuidae). Frontiers in Physiology. 11: 400. PMID 32425811 DOI: 10.3389/fphys.2020.00400   
2020 Grimes L, Griffiths J, Pasqualetto G, Brancale A, Kemp PJ, Young MT, van der Goes van Naters W. Drosophila taste neurons as an agonist-screening platform for P2X receptors. Scientific Reports. 10: 8292. PMID 32427920 DOI: 10.1038/s41598-020-65169-9   
2020 Liang YL, Belousoff MJ, Fletcher MM, Zhang X, Khoshouei M, Deganutti G, Koole C, Furness SGB, Miller LJ, Hay DL, Christopoulos A, Reynolds CA, Danev R, Wootten D, Sexton PM. Structure and Dynamics of Adrenomedullin Receptors AM and AM Reveal Key Mechanisms in the Control of Receptor Phenotype by Receptor Activity-Modifying Proteins. Acs Pharmacology & Translational Science. 3: 263-284. PMID 32296767 DOI: 10.1021/acsptsci.9b00080   
2020 Albrecht C, Appert-Collin A, Bagnard D, Blaise S, Romier-Crouzet B, Efremov RG, Sartelet H, Duca L, Maurice P, Bennasroune A. Transmembrane Peptides as Inhibitors of Protein-Protein Interactions: An Efficient Strategy to Target Cancer Cells? Frontiers in Oncology. 10: 519. PMID 32351895 DOI: 10.3389/fonc.2020.00519   
2020 Park J, Langmead CJ, Riddy DM. New Advances in Targeting the Resolution of Inflammation: Implications for Specialized Pro-Resolving Mediator GPCR Drug Discovery. Acs Pharmacology & Translational Science. 3: 88-106. PMID 32259091 DOI: 10.1021/acsptsci.9b00075   
2020 Wang X, Jespers W, Bongers BJ, Habben Jansen MCC, Stangenberger CM, Dilweg MA, Gutiérrez-de-Terán H, IJzerman AP, Heitman LH, van Westen GJP. Characterization of cancer-related somatic mutations in the adenosine A receptor. European Journal of Pharmacology. 173126. PMID 32348778 DOI: 10.1016/j.ejphar.2020.173126   
2020 Schupp M, Park SH, Qian B, Yu W. Electrophysiological Studies of GABA Receptors Using QPatch II, the Next Generation of Automated Patch-Clamp Instruments. Current Protocols in Pharmacology. 89: e75. PMID 32271492 DOI: 10.1002/cpph.75   
2020 Ruland JG, Kirchhofer SB, Klindert S, Bailey CP, Bünemann M. Voltage modulates the effect of μ receptor activation in a ligand-dependent manner. British Journal of Pharmacology. PMID 32297669 DOI: 10.1111/bph.15070   
2020 Schihada H, Ma X, Zabel U, Vischer HF, Schulte G, Leurs R, Pockes S, Lohse MJ. Development of a conformational histamine H receptor biosensor for the synchronous screening of agonists and inverse agonists. Acs Sensors. PMID 32397705 DOI: 10.1021/acssensors.0c00397   
2020 Luo S, Hou Y, Zhang Y, Ma T, Shao W, Xiao C. Adenosine A Receptor Agonist PSB-0777 Modulates Synaptic Proteins and AMPA Receptor Expression in A Dose- and Time-Dependent Manner in Rat Primary Cortical Neurons. Biological & Pharmaceutical Bulletin. PMID 32448843 DOI: 10.1248/bpb.b19-01007   
2020 Abbas H, Borde P, Willars GB, Ferry DR, Safrany ST. Hazards of Using When Performing Ligand Binding Assays: Lessons From the Sigma-1 and Sigma-2 Receptors. Frontiers in Pharmacology. 11: 309. PMID 32231573 DOI: 10.3389/fphar.2020.00309   
2020 Rahman MM, Teng J, Worrell BT, Noviello CM, Lee M, Karlin A, Stowell MHB, Hibbs RE. Structure of the Native Muscle-type Nicotinic Receptor and Inhibition by Snake Venom Toxins. Neuron. PMID 32275860 DOI: 10.1016/j.neuron.2020.03.012   
2020 Lombardi JP, Kinzlmaier DA, Jacob TC. Visualizing GABA A Receptor Trafficking Dynamics with Fluorogenic Protein Labeling. Current Protocols in Neuroscience. 92: e97. PMID 32364672 DOI: 10.1002/cpns.97   
2020 Giri R, Alberts I, Harding WW. Synthesis, pharmacological evaluations, and molecular docking studies on a new 1,3,4,11b-tetrahydro-1H-fluoreno[9,1-cd]azepine framework: Rigidification of D receptor selective 1-phenylbenzazepines and discovery of a new 5-HT receptor scaffold. Chemical Biology & Drug Design. PMID 32279445 DOI: 10.1111/cbdd.13691   
2020 Changeux JP. Discovery of the First Neurotransmitter Receptor: The Acetylcholine Nicotinic Receptor. Biomolecules. 10. PMID 32260196 DOI: 10.3390/biom10040547   
2020 Matyśniak D, Nowak N, Pomorski P. P2X7 receptor activity landscape in rat and human glioma cell lines. Acta Biochimica Polonica. 67: 7-14. PMID 32187491 DOI: 10.18388/abp.2020_2848   
2020 Soto P, Gaete PS, Fuentes C, Lozano B, Naulin PA, Figueroa XF, Barrera NP. Function of P2X4 Receptors Is Directly Modulated by a 1:1 Stoichiometric Interaction With 5-HTA Receptors. Frontiers in Cellular Neuroscience. 14: 106. PMID 32431598 DOI: 10.3389/fncel.2020.00106   
2020 Ziffert I, Kaiser A, Babilon S, Mörl K, Beck-Sickinger AG. Unusually persistent Gα-signaling of the neuropeptide Y receptor depletes cellular G pools and leads to a G-refractory state. Cell Communication and Signaling : Ccs. 18: 49. PMID 32223755 DOI: 10.1186/s12964-020-00537-6   
2020 Zhu X, Finlay DB, Glass M, Duffull SB. Evaluation of the profiles of CB cannabinoid receptor signalling bias using joint kinetic modelling. British Journal of Pharmacology. PMID 32293708 DOI: 10.1111/bph.15066   
2020 Blankenbach KV, Bruno G, Wondra E, Spohner AK, Aster NJ, Vienken H, Trautmann S, Ferreirós N, Wieland T, Bruni P, Meyer Zu Heringdorf D. The WD40 repeat protein, WDR36, orchestrates sphingosine kinase-1 recruitment and phospholipase C-β activation by G-coupled receptors. Biochimica Et Biophysica Acta. Molecular and Cell Biology of Lipids. 158704. PMID 32244061 DOI: 10.1016/j.bbalip.2020.158704   
2020 Tian M, Abdelrahman A, Baqi Y, Fuentes E, Azazna D, Spanier C, Densborn S, Hinz S, Schmid R, Müller CE. Discovery and structure-relationships of salicylanilide derivatives as potent, non-acidic P2X1 receptor antagonists. Journal of Medicinal Chemistry. PMID 32345019 DOI: 10.1021/acs.jmedchem.0c00435   
2020 Vieira G, Cavalli J, Gonçalves ECD, Braga SFP, Ferreira RS, Santos ARS, Cola M, Raposo NRB, Capasso R, Dutra RC. Antidepressant-Like Effect of Terpineol in an Inflammatory Model of Depression: Involvement of the Cannabinoid System and D2 Dopamine Receptor. Biomolecules. 10. PMID 32443870 DOI: 10.3390/biom10050792   
2020 Verweij EWE, Al Araaj B, Prabhata WR, Prihandoko R, Nijmeijer S, Tobin AB, Leurs R, Vischer HF. Differential Role of Serines and Threonines in Intracellular Loop 3 and C-Terminal Tail of the Histamine H Receptor in β-Arrestin and G Protein-Coupled Receptor Kinase Interaction, Internalization, and Signaling. Acs Pharmacology & Translational Science. 3: 321-333. PMID 32296771 DOI: 10.1021/acsptsci.0c00008   
2020 Bennett KA, Christopher JA, Tehan BG. Structure-based discovery and development of metabotropic glutamate receptor 5 negative allosteric modulators. Advances in Pharmacology (San Diego, Calif.). 88: 35-58. PMID 32416871 DOI: 10.1016/bs.apha.2020.03.001   
2020 Halpern AL, Kohtz PD, White AM, Houk AK, Rehring JF, Hanson L, McCarter MD, Joshi M, Meng X, Fullerton DA, Weyant MJ. Secretory Phospholipase A2 IIa Mediates Expression of Growth Factor Receptors in Esophageal Adenocarcinoma. Digestive Diseases and Sciences. PMID 32277371 DOI: 10.1007/s10620-020-06241-2   
2020 Moritz AE, Free RB, Weiner WS, Akano EO, Gandhi D, Abramyan A, Keck TM, Ferrer M, Hu X, Southall N, Steiner J, Aubé J, Shi L, Frankowski KJ, Sibley DR. Discovery, Optimization and Characterization of ML417: A Novel and Highly Selective D3 Dopamine Receptor Agonist. Journal of Medicinal Chemistry. PMID 32342685 DOI: 10.1021/acs.jmedchem.0c00424   
2020 Yue S, Zhang T, Shen Q, Song Q, Ji C, Chen Y, Mao M, Kong Y, Chen D, Liu J, Sun Z, Zhao M. Assessment of endocrine-disrupting effects of emerging polyhalogenated carbazoles (PHCZs): In vitro, in silico, and in vivo evidence. Environment International. 140: 105729. PMID 32344252 DOI: 10.1016/j.envint.2020.105729   
2020 Yu J, Gimenez LE, Hernandez CC, Wu Y, Wein AH, Han GW, McClary K, Mittal SR, Burdsall K, Stauch B, Wu L, Stevens SN, Peisley A, Williams SY, Chen V, et al. Determination of the melanocortin-4 receptor structure identifies Ca as a cofactor for ligand binding. Science (New York, N.Y.). 368: 428-433. PMID 32327598 DOI: 10.1126/science.aaz8995   
2020 Malik N, Wahlbeck KA, Thompson LK. Strategies for identifying dynamic regions in protein complexes: Flexibility changes accompany methylation in chemotaxis receptor signaling states. Biochimica Et Biophysica Acta. Biomembranes. 183312. PMID 32304758 DOI: 10.1016/j.bbamem.2020.183312   
2020 Jiang L, Cui J, Zhang C, Xie J, Zhang S, Fu D, Duo W. Sigma-1 receptor is involved in diminished ovarian reserve possibly by influencing endoplasmic reticulum stress-mediated granulosa cells apoptosis. Aging. 12. PMID 32409627 DOI: 10.18632/aging.103166   
2020 Wang A, Zhang Y, Chu H, Liao C, Zhang Z, Li G. Higher Accuracy Achieved for Protein-Ligand Binding Pose Prediction by Elastic Network Model Based Ensemble Docking. Journal of Chemical Information and Modeling. PMID 32383873 DOI: 10.1021/acs.jcim.9b01168   
2020 Hanna GJ, Bae JE, Lorch JH, Haddad RI, Jo VY, Schoenfeld JD, Margalit DN, Tishler RB, Goguen LA, Annino DJ, Chau NG. The Benefits of Adjuvant Trastuzumab for HER-2-Positive Salivary Gland Cancers. The Oncologist. PMID 32310325 DOI: 10.1634/theoncologist.2019-0841   
2020 Antunes GF, Gouveia FV, Rezende FS, Seno MDJ, de Carvalho MC, de Oliveira CC, Dos Santos LCT, de Castro MC, Kuroki MA, Teixeira MJ, Otoch JP, Brandao ML, Fonoff ET, Martinez RCR. Dopamine modulates individual differences in avoidance behavior: A pharmacological, immunohistochemical, neurochemical and volumetric investigation. Neurobiology of Stress. 12: 100219. PMID 32435668 DOI: 10.1016/j.ynstr.2020.100219   
2020 Ngo T, Stephens BS, Gustavsson M, Holden LG, Abagyan R, Handel TM, Kufareva I. Crosslinking-guided geometry of a complete CXC receptor-chemokine complex and the basis of chemokine subfamily selectivity. Plos Biology. 18: e3000656. PMID 32271748 DOI: 10.1371/journal.pbio.3000656   
2020 Koblan KS, Kent J, Hopkins SC, Krystal JH, Cheng H, Goldman R, Loebel A. A Non-D2-Receptor-Binding Drug for the Treatment of Schizophrenia. The New England Journal of Medicine. 382: 1497-1506. PMID 32294346 DOI: 10.1056/NEJMoa1911772   
2020 Pottie E, Tosh DK, Gao ZG, Jacobson KA, Stove CP. Assessment of biased agonism at the A adenosine receptor using β-arrestin and miniGα recruitment assays. Biochemical Pharmacology. 113934. PMID 32224136 DOI: 10.1016/j.bcp.2020.113934