Year |
Citation |
Score |
2020 |
Newton AS, Faver JC, Micevic G, Muthusamy V, Kudalkar SN, Bertoletti N, Anderson KS, Bosenberg MW, Jorgensen WL. Structure-Guided Identification of DNMT3B Inhibitors. Acs Medicinal Chemistry Letters. 11: 971-976. PMID 32435413 DOI: 10.1021/Acsmedchemlett.0C00011 |
0.352 |
|
2019 |
Sasaki T, Gannam ZTK, Kudalkar SN, Frey KM, Lee WG, Spasov KA, Jorgensen WL, Anderson KS. Molecular and cellular studies evaluating a potent 2-cyanoindolizine catechol diether NNRTI targeting wildtype and Y181C mutant HIV-1 reverse transcriptase. Bioorganic & Medicinal Chemistry Letters. PMID 31281023 DOI: 10.1016/J.Bmcl.2019.06.047 |
0.413 |
|
2019 |
Kudalkar SN, Ullah I, Bertoletti N, Mandl HK, Cisneros JA, Beloor J, Chan AH, Quijano E, Saltzman WM, Jorgensen WL, Kumar P, Anderson KS. Structural and pharmacological evaluation of a novel non-nucleoside reverse transcriptase inhibitor as a promising long acting nanoformulation for treating HIV. Antiviral Research. PMID 31034849 DOI: 10.1016/J.Antiviral.2019.04.010 |
0.322 |
|
2018 |
Sasaki T, Kudalkar SN, Bertoletti N, Anderson KS. DRONE: Direct Tracking of DNA Cytidine Deamination and Other DNA Modifying Activities. Analytical Chemistry. PMID 30256094 DOI: 10.1021/Acs.Analchem.8B01405 |
0.304 |
|
2018 |
Liu Y, Ji L, Eno M, Kudalkar S, Li A, Schimpgen M, Benchama O, Morales P, Xu S, Hurst DP, Wu S, Mohammad KA, Wood JT, Zvonok N, Papahatjis D, et al. (R)-N-(1-Methyl-2-hydroxyethyl)-13-(S)-methyl-arachidonamide (AMG315): A Novel Chiral Potent Endocannabinoid Ligand with Stability to Metabolizing Enzymes. Journal of Medicinal Chemistry. PMID 30196704 DOI: 10.1021/Acs.Jmedchem.8B00611 |
0.303 |
|
2017 |
Kudalkar SN, Beloor J, Quijano E, Spasov KA, Lee WG, Cisneros JA, Saltzman WM, Kumar P, Jorgensen WL, Anderson KS. From in silico hit to long-acting late-stage preclinical candidate to combat HIV-1 infection. Proceedings of the National Academy of Sciences of the United States of America. PMID 29279368 DOI: 10.1073/Pnas.1717932115 |
0.316 |
|
2017 |
Chan AH, Lee WG, Spasov KA, Cisneros JA, Kudalkar SN, Petrova ZO, Buckingham AB, Anderson KS, Jorgensen WL. Covalent inhibitors for eradication of drug-resistant HIV-1 reverse transcriptase: From design to protein crystallography. Proceedings of the National Academy of Sciences of the United States of America. PMID 28827354 DOI: 10.1073/Pnas.1711463114 |
0.342 |
|
2017 |
Kudalkar SN, Beloor J, Chan AH, Lee WG, Jorgensen WL, Kumar P, Anderson KS. Structural and Preclinical Studies of Computationally-Designed Non-nucleoside Reverse Transcriptase Inhibitors for Treating HIV infection. Molecular Pharmacology. PMID 28167742 DOI: 10.1124/Mol.116.107755 |
0.396 |
|
2016 |
Kudalkar SN, Kingsley PJ, Marnett LJ. Assay of Endocannabinoid Oxidation by Cyclooxygenase-2. Methods in Molecular Biology (Clifton, N.J.). 1412: 205-15. PMID 27245906 DOI: 10.1007/978-1-4939-3539-0_21 |
0.324 |
|
2015 |
Blobaum AL, Xu S, Rowlinson SW, Duggan KC, Banerjee S, Kudalkar SN, Birmingham WR, Ghebreselasie K, Marnett LJ. Action at a distance: mutations of peripheral residues transform rapid reversible inhibitors to slow, tight binders of cyclooxygenase-2. The Journal of Biological Chemistry. 290: 12793-803. PMID 25825493 DOI: 10.1074/Jbc.M114.635987 |
0.377 |
|
2015 |
Kudalkar SN, Njuma OJ, Li Y, Muldowney M, Fuanta NR, Goodwin DC. A role for catalase-peroxidase large loop 2 revealed by deletion mutagenesis: control of active site water and ferric enzyme reactivity. Biochemistry. 54: 1648-62. PMID 25674665 DOI: 10.1021/Bi501221A |
0.625 |
|
2015 |
Kudalkar SN, Nikas SP, Kingsley PJ, Xu S, Galligan JJ, Rouzer CA, Banerjee S, Ji L, Eno MR, Makriyannis A, Marnett LJ. 13-Methylarachidonic acid is a positive allosteric modulator of endocannabinoid oxygenation by cyclooxygenase. The Journal of Biological Chemistry. 290: 7897-909. PMID 25648895 DOI: 10.1074/Jbc.M114.634014 |
0.358 |
|
2012 |
Kudalkar SN, Campbell RA, Li Y, Varnado CL, Prescott C, Goodwin DC. Enhancing the peroxidatic activity of KatG by deletion mutagenesis Journal of Inorganic Biochemistry. 116: 106-115. PMID 23018273 DOI: 10.1016/J.Jinorgbio.2012.08.002 |
0.454 |
|
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