Year |
Citation |
Score |
2014 |
Ghisaidoobe AT, van den Berg RJ, Butt SS, Strijland A, Donker-Koopman WE, Scheij S, van den Nieuwendijk AM, Koomen GJ, van Loevezijn A, Leemhuis M, Wennekes T, van der Stelt M, van der Marel GA, van Boeckel CA, Aerts JM, et al. Identification and development of biphenyl substituted iminosugars as improved dual glucosylceramide synthase/neutral glucosylceramidase inhibitors. Journal of Medicinal Chemistry. 57: 9096-104. PMID 25250725 DOI: 10.1021/jm501181z |
0.462 |
|
2001 |
Burm BEA, Blokker P, Jongmans E, Van Kampen E, Wanner MJ, Koomen GJ. Synthesis of xestomanzamines a and b Heterocycles. 55: 495-503. DOI: 10.3987/Com-00-9107 |
0.364 |
|
2000 |
Deghati PYF, Wanner MJ, Koomen GJ. Regioselective nitration of purine nucleosides: Synthesis of 2- nitroadenosine and 2-nitroinosine Tetrahedron Letters. 41: 1291-1295. DOI: 10.1016/S0040-4039(99)02271-6 |
0.334 |
|
1999 |
Madre M, Panchenko N, Golbraikh A, Zhuk R, Pandit UK, Geenevasen J, Koomen GJ. Purine nucleoside analogues. 11. An alternative synthesis of N- and O-alkyl derivatives of 9- and 7-[(2-acetoxyethoxy)methyl]-N2-acetylguanine Collection of Czechoslovak Chemical Communications. 64: 685-695. DOI: 10.1135/Cccc19990685 |
0.56 |
|
1999 |
Barends J, Van Der Linden JB, Van Delft FL, Koomen GJ. Palladium-catalyzed amination of 6-chloropurine. Synthesis of N6- substituted adenosine analogues Nucleosides and Nucleotides. 18: 2121-2126. |
0.364 |
|
1998 |
Overkleeft HS, Renkema GH, Neele J, Vianello P, Hung IO, Strijland A, van der Burg AM, Koomen GJ, Pandit UK, Aerts JM. Generation of specific deoxynojirimycin-type inhibitors of the non-lysosomal glucosylceramidase. The Journal of Biological Chemistry. 273: 26522-7. PMID 9756888 DOI: 10.1074/jbc.273.41.26522 |
0.567 |
|
1998 |
Burm BEA, Meijler MM, Korver J, Wanner MJ, Koomen GJ. Synthesis of the brominated marine alkaloids (±)-arborescidine A, B and C Tetrahedron. 54: 6135-6146. DOI: 10.1016/S0040-4020(98)00306-8 |
0.307 |
|
1997 |
Wanner MJ, Koomen GJ. Biomimetic synthesis of racemic alkaloids Pharmacochemistry Library. 28: 179-187. DOI: 10.1016/S0165-7208(97)80064-5 |
0.317 |
|
1997 |
Wanner MJ, Koomen GJ. Biomimetic Synthesis of Nitraria Alkaloids, based on Tetrahydropyridine Synthons Journal of the Indian Chemical Society. 74: 891-895. |
0.302 |
|
1996 |
Petra DGI, De Boer RF, Koomen GJ, Meeuwenoord NJ, Kuyl-Yeheskiely E, Van Der Marel GA, Van Boom JH. Synthesis and properties of a fluorescent nucleotide derivative Recueil Des Travaux Chimiques Des Pays-Bas-Journal of the Royal Netherlands. 115: 99-102. DOI: 10.1002/Recl.19961150117 |
0.39 |
|
1995 |
Madre M, Geita L, Zhuk R, Koomen GJ. Purine nucleoside analogues. 7. 9-[2-(Alkylthio)ethoxymethyl] derivatives of adenine, hypoxanthine and guanine Chinese Pharmaceutical Journal. 47: 469-481. |
0.308 |
|
1995 |
Wanner MJ, Koomen GJ. Biomimetic synthesis of nitraramine The Journal of Organic Chemistry. 60: 5634-5637. |
0.301 |
|
1994 |
Wanner MJ, Koomen GJ. Biomimetic synthesis of nazlinin and nitrarine Pure and Applied Chemistry. 66: 2239-2242. DOI: 10.1351/pac199466102239 |
0.301 |
|
1994 |
Boogaard AT, Pandit UK, Koomen GJ. Ring D modifications of ellipticine. Part 2. Chlorination of ellipticine via its N-oxide and synthesis and selective acetylation of 5,6,11-trimethyl-5H-benzo[b]carbazole. Tetrahedron. 50: 4811-4828. DOI: 10.1016/S0040-4020(01)85018-3 |
0.539 |
|
1992 |
Hartgers WA, De Boer RF, Wanner MJ, Koomen GJ. A potential suicide inhibitor of adenylosuccinate lyase Nucleosides and Nucleotides. 11: 1325-1332. DOI: 10.1080/07328319208021176 |
0.319 |
|
1992 |
Koomen GJ, Provoost LM, Van Maarschalkerwaart DAH, Willard NP. Synthesis of an acyclic analogue of azidothymidine Nucleosides and Nucleotides. 11: 1297-1303. DOI: 10.1080/07328319208021174 |
0.337 |
|
1992 |
Plug JPM, Koomen GJ, Pandit UK. An expedient synthesis of 9-hydroxyellipticine Synthesis. 1221-1222. DOI: 10.1055/S-1992-26342 |
0.517 |
|
1992 |
Vloon WJ, van den Bos JC, Koomen GJ, Pandit UK. Synthesis of ring C modified sesbanimide analogues Tetrahedron. 48: 8317-8328. DOI: 10.1016/S0040-4020(01)80499-3 |
0.537 |
|
1992 |
Plug JPM, Koomen GJ, Pandit UK. Sythesis of novel annulated ellipticines via Claisen rearrangement reactions Tetrahedron Letters. 33: 2179-2182. DOI: 10.1016/0040-4039(92)88171-Z |
0.577 |
|
1991 |
Wanner MJ, Koomen GJ. Biomimetic synthesis of quinolizidine alkaloids Tetrahedron. 47: 8431-8442. DOI: 10.1016/S0040-4020(01)96184-8 |
0.314 |
|
1991 |
van den Bos JC, Vloon WJ, Koomen GJ, Pandit UK. Synthesis of acyclic analogues of sesbanimides A and B Tetrahedron. 47: 6787-6794. DOI: 10.1016/S0040-4020(01)82330-9 |
0.562 |
|
1990 |
Van Maarschalkerwaart DAH, Willard NP, Koomen GJ. Carbocyclic nucleoside analogues. Synthesis and properties of 1-(4-hydroxymethyl-2-cyclopenten-1-yl)-thymine Nucleosides and Nucleotides. 9: 787-791. DOI: 10.1080/15257779008043144 |
0.321 |
|
1989 |
Langendoen A, Plug JPM, Koomen GJ, Pandit UK. Regiospecific C-9 substitution of ellipticine derivatives Tetrahedron. 45: 1759-1762. DOI: 10.1016/S0040-4020(01)80040-5 |
0.514 |
|
1988 |
Wanner MJ, Koomen GJ. 2-Substituted Glutarimides via Preformed Wittig Reagents Synthesis. 1988: 325-327. DOI: 10.1055/S-1988-27558 |
0.304 |
|
1988 |
Langendoen A, Koomen GJ, Pandit UK. An approach to novel ellipticine glycosides Tetrahedron. 44: 3627-3631. DOI: 10.1016/S0040-4020(01)85992-5 |
0.546 |
|
1988 |
WANNER MJ, KOOMEN G. ChemInform Abstract: 2-Substituted Glutarimides via Preformed Wittig Reagents. Cheminform. 19. DOI: 10.1002/CHIN.198833239 |
0.303 |
|
1987 |
Langendoen A, Koomen GJ, Pandit UK. A new approach to C-9 hydroxylation of N(6)-substituted ellipticine Heterocycles. 26: 91-94. DOI: 10.3987/R-1987-01-0091 |
0.495 |
|
1987 |
Langendoen A, Koomen GJ, Pandit UK. Side-chain substitution of 6-methylellipticine approach to a new class of ellipticine derivatives Heterocycles. 26: 69-73. DOI: 10.3987/R-1987-01-0069 |
0.468 |
|
1987 |
Wanner MJ, Willard NP, Koomen GJ, Pandit UK. Stereospecific synthesis of (+)- and (-)-sesbanimide A Tetrahedron. 43: 2549-2556. DOI: 10.1016/S0040-4020(01)81662-8 |
0.541 |
|
1986 |
Wijsmuller WFA, Wanner MJ, Koomen GJ, Pandit UK. Pyridocarbazole alkaloids. Synthesis of olivacine and ellipticine analogues Heterocycles. 24: 1795-1797. DOI: 10.1002/Chin.198647359 |
0.566 |
|
1986 |
Koomen GJ, Wolschrijn H, van Rhijn JBM, Wanner MJ, Pandit UK. Synthesis of 5-fluoro-3-(2-tetrahydrofuryl)-6-vinyluracil. Design of a 5-fu-derivative with extended conjugation Heterocycles. 24: 939-941. DOI: 10.1002/Chin.198642214 |
0.519 |
|
1986 |
Wanner MJ, Willard NP, Koomen GJ, Pandit UK. Synthesis of (7R,8S,9R,10S,11S)-sesbanimide A Journal of the Chemical Society - Series Chemical Communications. 396-397. DOI: 10.1002/Chin.198634331 |
0.418 |
|
1985 |
Koomen GJ, van Rhijn JBMv, Pandit UK. Non-glycosidic derivatives of 5-fluorouracil Nucleosides and Nucleotides. 4: 215-216. DOI: 10.1080/07328318508077858 |
0.476 |
|
1985 |
Odijk WM, Koomen GJ. Fluorescent nucleoside analogues. Synthesis of fluorescent pyrido[2,1-i]purines, and their corresponding ribosides Tetrahedron. 41: 1893-1904. DOI: 10.1016/S0040-4020(01)96552-4 |
0.443 |
|
1984 |
WANNER MJ, KOOMEN G, PANDIT UK. ChemInform Abstract: STUDIES IN THE STEREOSPECIFIC SYNTHESIS OF SESBANIMIDE. SYNTHESIS OF 4-SACCHARIDALGLUTARIMIDES Chemischer Informationsdienst. 15. DOI: 10.1002/Chin.198448332 |
0.557 |
|
1983 |
Wanner MJ, Koomen GJ, Pandit UK. Inter- and intramolecular addition of ester anions to nicotinium salts. A facile approach to nauclefine and ellipticine derivatives Tetrahedron. 39: 3673-3681. DOI: 10.1016/S0040-4020(01)88606-3 |
0.62 |
|
1983 |
WANNER MJ, KOOMEN G, PANDIT UK. ChemInform Abstract: A CONVENIENT SYNTHESIS OF 6-METHYLELLIPTICINE AND 6-METHYLOLIVACINE Chemischer Informationsdienst. 14. DOI: 10.1002/Chin.198322343 |
0.559 |
|
1982 |
Wanner MJ, Koomen GJ, Pandit UK. Synthesis of polynuclear heterocycles via the reaction of α-ester carbanions with quaternized nicotinamide salts. A facile stereoselective synthesis of sesbanine Tetrahedron. 38: 2741-2748. DOI: 10.1016/0040-4020(82)80032-X |
0.615 |
|
1982 |
WANNER MJ, KOOMEN G, PANDIT UK. ChemInform Abstract: A New Approach to Ellipticine Analogues; Synthesis of 11-Hydroxy-5,6-dimethyl-pyrido[4,3-b]carbazole. Chemischer Informationsdienst. 13. DOI: 10.1002/Chin.198233202 |
0.542 |
|
1980 |
Wanner MJ, Hageman JJ, Koomen GJ, Pandit UK. Potential carcinostatics. 4. Synthesis and biological properties of erythro- and threo-beta-fluoroaspartic acid and erythro-beta-fluoroasparagine. Journal of Medicinal Chemistry. 23: 85-7. PMID 7359517 DOI: 10.1021/Jm00175A017 |
0.548 |
|
1980 |
Wanner MJ, Van Wijk EM, Koomen GJ, Pandit UK. Potential carcinostatics. V. Synthesis and properties of potential inhibitors of the adenylosuccinate synthetase and adenylosuccinate lyase system Recueil Des Travaux Chimiques Des Pays Bas. 99: 20-23. DOI: 10.1002/Recl.19780970711 |
0.609 |
|
1980 |
Wanner MJ, Hageman JJM, Koomen GJ, Pandit UK. POTENTIAL CARCINOSTATICS. 4. SYNTHESIS AND BIOLOGICAL PROPERTIES OF ERYTHRO- AND THREO-β-FLUOROASPARTIC ACID AND ERYTHRO-β-FLUOROASPARAGINE Cheminform. 11. DOI: 10.1002/Chin.198024111 |
0.503 |
|
1979 |
ODIJK WM, WANNER MJ, KOOMEN GJ, PANDIT UK. ChemInform Abstract: POTENTIAL CARCINOSTATIC AGENTS. PART III. PSEUDO-GLYCOSIDIC DERIVATIVES OF 5-FLUOROURACIL Chemischer Informationsdienst. 10. DOI: 10.1002/Chin.197909223 |
0.515 |
|
1978 |
Wanner MJ, Hageman JJM, Koomen GJ, Pandit UK. Potential Carcinostatics. Part Ii. Synthesis And Properties Of Potential Inhibitors Of The Adenylosuccinate Synthetase And Adenylosuccinate Lyase Systems Cheminform. 11. DOI: 10.1002/Chin.197843246 |
0.521 |
|
1978 |
HAGEMAN JJM, WANNER MJ, KOOMEN GJ, PANDIT UK. ChemInform Abstract: POTENTIAL CARCINOSTATICS. SYNTHESIS AND BIOLOGICAL PROPERTIES OF D- AND L-β,β-DIFLUOROASPARTIC ACID AND β,β-DIFLUOROASPARAGINE Chemischer Informationsdienst. 9. DOI: 10.1002/Chin.197816128 |
0.489 |
|
1978 |
THIELLIER HPM, KOOMEN GJ, PANDIT UK. ChemInform Abstract: UNCONVENTIONAL NUCLEOTIDE ANALOGS. XVIII. RING EXPANSION OF URIDINE HALOCARBENE ADDUCTS. SYNTHESIS OF DIAZEPINE NUCLEOSIDES Chemischer Informationsdienst. 9. DOI: 10.1002/chin.197802343 |
0.341 |
|
1978 |
Wanner MJ, Hageman JJM, Koomen GJ, Pandit UK. Potential carcinostatics. Synthesis and properties of potential inhibitors of the adenylosuccinate synthetase and adenylosuccinate lyase systems Recueil Des Travaux Chimiques Des Pays Bas. 97: 211-214. |
0.479 |
|
1977 |
Hageman JJ, Wanner MJ, Koomen GJ, Pandit UK. Potential carcinostatics. Synthesis and biological properties of d- and 1-beta,beta-difluoroaspartic acid and beta,beta-difluoroasparagine. Journal of Medicinal Chemistry. 20: 1677-9. PMID 592334 DOI: 10.1021/Jm00222A029 |
0.471 |
|
1977 |
Thiellier HPM, Koomen GJ, Pandit UK. Unconventional nucleotide analogues1 1 Part XV. H.P.M Thiellier, G.J. Koomen and U.K. Pandit, Heterocycles 5, 19 (1976). Reaction of carbenes with uracil and uridine derivatives Tetrahedron. 33: 1493-1500. DOI: 10.1016/0040-4020(77)88011-3 |
0.587 |
|
1977 |
Thiellier HPM, Koomen GJ, Pandit UK. Unconventional nucleotide analogues-XVIII1 1 Part XVII. H.P.M. Thiellier, G.J. Koomen and U.K. Pandit, Tetrahedron 33, 2603 (1977). Ring expansion of uridine halocarbene adducts. Synthesis of diazepine nucleosides Tetrahedron. 33: 2609-2612. DOI: 10.1016/0040-4020(77)80087-2 |
0.603 |
|
1977 |
Thiellier HPM, Koomen GJ, Pandit UK. Unconventional nucleotide analogues-XVII1 1 Part XVI. H.P.M. Thiellier, G.J. Koomen and U.K. Pandit, Tetrahedron 33, 1493 (1977). Ring-transformations of uracil dihalocarbene adducts Tetrahedron. 33: 2603-2607. DOI: 10.1016/0040-4020(77)80086-0 |
0.585 |
|
1977 |
THIELLIER HPM, KOOMEN GJ, PANDIT UK. ChemInform Abstract: UNCONVENTIONAL NUCLEOTIDE ANALOGS. XV. NOVEL BASE-MODIFIED NUCLEOSIDES Chemischer Informationsdienst. 8: no-no. DOI: 10.1002/Chin.197717341 |
0.539 |
|
1976 |
THIELLIER HPM, KOOMEN GJ, PANDIT UK. ChemInform Abstract: TRANSFORMATIONS OF 1,3-DISUBSTITUTED URACIL-CARBENE ADDUCTS. RING EXPANSION TO 1,3-DIAZEPINE DERIVATIVES Chemischer Informationsdienst. 7: no-no. DOI: 10.1002/Chin.197603227 |
0.559 |
|
1974 |
THIELLIER HPM, BURG AMVD, KOOMEN GJ, PANDIT UK. ChemInform Abstract: REACTION OF CARBENES WITH 1,3-DISUBSTITUTED URACIL DERIVATIVES Chemischer Informationsdienst. 5: no-no. DOI: 10.1002/Chin.197451349 |
0.55 |
|
1973 |
Koomen GJ, Pandit UK. Unconventional nucleotide analogues. IX. N-substituted 3-(pyrimidin-1-yl) pyrrolidin-2-ones. Journal of the Chemical Society. Perkin Transactions 1. 17: 1929-33. PMID 4799178 DOI: 10.1039/P19730001929 |
0.57 |
|
1973 |
Koomen GJ, Kroon AP, Mas Cabré FR, Goores AP, Peereboom R, Pandit UK. Unconventional nucleotide analogues. Part X. Synthesis of N-substituted 3-(Adenin-9-yl)pyrrolidin-2-ones Journal of the Chemical Society, Perkin Transactions 1. 1934-1940. PMID 4363162 DOI: 10.1039/P19730001934 |
0.599 |
|
1973 |
KOOMEN GJ, PANDIT UK. ChemInform Abstract: UNCONVENTIONAL NUCLEOTIDE ANALOGUES PART 9, N-SUBSTITUTED 3-(PYRIMIDIN-1-YL)-PYRROLIDIN-2-ONES Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/chin.197349468 |
0.546 |
|
1971 |
Koomen GJ, Kroon AP, Goores AP, Pandit UK. Non-Sacccfaridal Nucleoside and Hucleotide Analocuses Synthetic Communications. 1: 41-45. DOI: 10.1080/00397917108081615 |
0.421 |
|
1971 |
KOOMEN GJ, KROON AP, GOORES AP, PANDIT UK. ChemInform Abstract: ZUCKERFREIE NUCLEOSID- UND NUCLEOTID-ANALOGA Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/Chin.197139334 |
0.519 |
|
1969 |
Nollet AJH, Koomen GJ, Grose WFA, Pandit UK. Application of NMR spectroscopy in distinguishing between N1- and N3-substituted 2,4-dioxo-1,2,3,4,-tetrahydropyrimidines. Tetrahedron Letters. 10: 4607-4608. DOI: 10.1016/S0040-4039(01)88762-1 |
0.467 |
|
1967 |
Pandit UK, de Jonge K, Koomen GJ, Huisman HO. Heterocyclic steroids IX. A Convenient Synthesis of 14-Aza-11-Keto Steroids Tetrahedron Letters. 8: 3529-3533. |
0.688 |
|
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