Hans-Georg Breitinger, Ph.D. - Related publications

Affiliations: 
German University of Cairo 
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50 most relevant papers in past 60 days:
Year Citation  Score
2020 Olander ER, Janzen D, Villmann C, Jensen AA. Comparison of biophysical properties of α1β2 and α3β2 GABAA receptors in whole-cell patch-clamp electrophysiological recordings. Plos One. 15: e0234080. PMID 32479525 DOI: 10.1371/journal.pone.0234080   
2020 Breitinger U, Breitinger HG. Modulators of the inhibitory glycine receptor. Acs Chemical Neuroscience. PMID 32391682 DOI: 10.1021/acschemneuro.0c00054   
2020 Wilding TJ, Huettner JE. Cadmium activates AMPA and NMDA receptors with M3 helix cysteine substitutions. The Journal of General Physiology. 152. PMID 32342094 DOI: 10.1085/jgp.201912537   
2020 Perszyk RE, Myers SJ, Yuan H, Gibb AJ, Furukawa H, Sobolevsky AI, Traynelis SF. Hodgkin-huxley-katz prize lecture: genetic and pharmacological control of glutamate receptor channel through a highly conserved gating motif. The Journal of Physiology. PMID 32468591 DOI: 10.1113/JP278086   
2020 Salazar H, Mischke S, Plested AJR. Measurements of the Timescale and Conformational Space of AMPA Receptor Desensitization. Biophysical Journal. PMID 32559412 DOI: 10.1016/j.bpj.2020.05.029   
2020 Baldwin MW, Ko MC. Functional evolution of vertebrate sensory receptors. Hormones and Behavior. 104771. PMID 32437717 DOI: 10.1016/j.yhbeh.2020.104771   
2020 Zhu Z, Yi F, Epplin MP, Liu D, Summer SL, Mizu R, Shaulsky G, XiangWei W, Tang W, Burger PB, Menaldino DS, Myers SJ, Liotta DC, Hansen KB, Yuan H, et al. Negative allosteric modulation of GluN1/GluN3 NMDA receptors. Neuropharmacology. 108117. PMID 32389749 DOI: 10.1016/j.neuropharm.2020.108117   
2020 Liu C, Xia L, Fu K, Cao X, Yan W, Cheng J, Roux T, Peletier LA, Yin X, Guo D. Revisit ligand-receptor interaction at the human vasopressin V receptor: A kinetic perspective. European Journal of Pharmacology. 173157. PMID 32360346 DOI: 10.1016/j.ejphar.2020.173157   
2020 Gao J, Chang Z, Tian R, Li P, Ahmad F, Jia X, Liang Q, Zhao X. Reversible and site-specific immobilization of β-adrenergic receptor by aptamer-directed method for receptor-drug interaction analysis. Journal of Chromatography. A. 461091. PMID 32376022 DOI: 10.1016/j.chroma.2020.461091   
2020 Ladurner A, Linder T, Wang L, Hiebl V, Schuster D, Schnürch M, Mihovilovic MD, Atanasov AG, Dirsch VM. Characterization of a Structural Leoligin Analog as Farnesoid X Receptor Agonist and Modulator of Cholesterol Transport. Planta Medica. PMID 32485752 DOI: 10.1055/a-1171-8357   
2020 Falk-Petersen CB, Tsonkov TM, Nielsen MS, Harpsøe K, Bundgaard C, Frølund B, Kristiansen U, Gloriam DE, Wellendorph P. Discovery of a new class of orthosteric antagonists with nanomolar potency at extrasynaptic GABA receptors. Scientific Reports. 10: 10078. PMID 32572053 DOI: 10.1038/s41598-020-66821-0   
2020 Bennett KA, Christopher JA, Tehan BG. Structure-based discovery and development of metabotropic glutamate receptor 5 negative allosteric modulators. Advances in Pharmacology (San Diego, Calif.). 88: 35-58. PMID 32416871 DOI: 10.1016/bs.apha.2020.03.001   
2020 Wang Y, Joseph J, Gao Y, Hu B, Geng X, Wu D, Wang J, Zhang F. Revealing the Interaction Modes of 5-HT2A Receptor Antagonists and the Structure-Based Virtual Screening from FDA and TCMNP Database. Journal of Biomolecular Structure & Dynamics. 1-20. PMID 32406337 DOI: 10.1080/07391102.2020.1768900   
2020 Lombardi JP, Kinzlmaier DA, Jacob TC. Visualizing GABA A Receptor Trafficking Dynamics with Fluorogenic Protein Labeling. Current Protocols in Neuroscience. 92: e97. PMID 32364672 DOI: 10.1002/cpns.97   
2020 da Costa Couto ARGM, Price KL, Mesoy S, Capes E, Lummis SCR. The M4 Helix Is Involved in α7 nACh Receptor Function. Acs Chemical Neuroscience. PMID 32364364 DOI: 10.1021/acschemneuro.0c00027   
2020 Mattedi G, Acosta-Gutiérrez S, Clark T, Gervasio FL. A combined activation mechanism for the glucagon receptor. Proceedings of the National Academy of Sciences of the United States of America. PMID 32571939 DOI: 10.1073/pnas.1921851117   
2020 Sadanandan SM, Kreko-Pierce T, Khatri SN, Pugh JR. Cannabinoid type 2 receptors inhibit GABAA receptor-mediated currents in cerebellar Purkinje cells of juvenile mice. Plos One. 15: e0233020. PMID 32437355 DOI: 10.1371/journal.pone.0233020   
2020 Zaccor NW, Sumner CJ, Snyder SH. The nonselective cation channel TRPV4 inhibits angiotensin II receptors. The Journal of Biological Chemistry. PMID 32493776 DOI: 10.1074/jbc.RA120.014325   
2020 Dalby NO, Falk-Petersen CB, Leurs U, Scholze P, Krall J, Frølund B, Wellendorph P. Silencing of spontaneous activity at α4β1/3δ GABA receptors in hippocampal granule cells reveals different ligand pharmacology. British Journal of Pharmacology. PMID 32484592 DOI: 10.1111/bph.15146   
2020 Lindemann M, Moldovan RP, Hinz S, Deuther-Conrad W, Gündel D, Dukic-Stefanovic S, Toussaint M, Teodoro R, Juhl C, Steinbach J, Brust P, Müller CE, Wenzel B. Development of a Radiofluorinated Adenosine A Receptor Antagonist as Potential Ligand for PET Imaging. International Journal of Molecular Sciences. 21. PMID 32366046 DOI: 10.3390/ijms21093197   
2020 Pandey S, Maharana J, Li XX, Woodruff TM, Shukla AK. Emerging Insights into the Structure and Function of Complement C5a Receptors. Trends in Biochemical Sciences. PMID 32402749 DOI: 10.1016/j.tibs.2020.04.004   
2020 Park J, Fu Z, Frangaj A, Liu J, Mosyak L, Shen T, Slavkovich VN, Ray KM, Taura J, Cao B, Geng Y, Zuo H, Kou Y, Grassucci R, Chen S, et al. Structure of human GABA receptor in an inactive state. Nature. PMID 32581365 DOI: 10.1038/s41586-020-2452-0   
2020 Burada AP, Vinnakota R, Kumar J. The Architecture of GluD2 Ionotropic Delta Glutamate Receptor Elucidated by cryo-EM. Journal of Structural Biology. 107546. PMID 32512155 DOI: 10.1016/j.jsb.2020.107546   
2020 Wang A, Zhang Y, Chu H, Liao C, Zhang Z, Li G. Higher Accuracy Achieved for Protein-Ligand Binding Pose Prediction by Elastic Network Model Based Ensemble Docking. Journal of Chemical Information and Modeling. PMID 32383873 DOI: 10.1021/acs.jcim.9b01168   
2020 Soto P, Gaete PS, Fuentes C, Lozano B, Naulin PA, Figueroa XF, Barrera NP. Function of P2X4 Receptors Is Directly Modulated by a 1:1 Stoichiometric Interaction With 5-HTA Receptors. Frontiers in Cellular Neuroscience. 14: 106. PMID 32431598 DOI: 10.3389/fncel.2020.00106   
2020 Gillet C, Kurth S, Kuenzel T. Muscarinic modulation of M and h currents in gerbil spherical bushy cells. Plos One. 15: e0226954. PMID 31940388 DOI: 10.1371/journal.pone.0226954   
2020 Grimes L, Griffiths J, Pasqualetto G, Brancale A, Kemp PJ, Young MT, van der Goes van Naters W. Drosophila taste neurons as an agonist-screening platform for P2X receptors. Scientific Reports. 10: 8292. PMID 32427920 DOI: 10.1038/s41598-020-65169-9   
2020 Luo S, Hou Y, Zhang Y, Ma T, Shao W, Xiao C. Adenosine A Receptor Agonist PSB-0777 Modulates Synaptic Proteins and AMPA Receptor Expression in A Dose- and Time-Dependent Manner in Rat Primary Cortical Neurons. Biological & Pharmaceutical Bulletin. PMID 32448843 DOI: 10.1248/bpb.b19-01007   
2020 Burnat G, Brański P, Solich J, Kolasa M, Chruścicka B, Dziedzicka-Wasylewska M, Pilc A. The functional cooperation of 5-HT and mGlu4R in HEK-293 cell line. Pharmacological Reports : Pr. PMID 32472388 DOI: 10.1007/s43440-020-00114-1   
2020 Brimson JM, Akula KK, Abbas H, Ferry DR, Kulkarni SK, Russell ST, Tisdale MJ, Tencomnao T, Safrany ST. Simple ammonium salts acting on sigma-1 receptors yield potential treatments for cancer and depression. Scientific Reports. 10: 9251. PMID 32514120 DOI: 10.1038/s41598-020-65849-6   
2020 Kim HR, Xu J, Maeda S, Duc NM, Ahn D, Du Y, Chung KY. Structural mechanism underlying primary and secondary coupling between GPCRs and the Gi/o family. Nature Communications. 11: 3160. PMID 32572026 DOI: 10.1038/s41467-020-16975-2   
2020 Lü S, Jiang M, Tian X, Hong S, Zhang J, Zhang Y. Characterization of an A-Type Muscarinic Acetylcholine Receptor and Its Possible Non-neuronal Role in the Oriental Armyworm, Walker (Lepidoptera: Noctuidae). Frontiers in Physiology. 11: 400. PMID 32425811 DOI: 10.3389/fphys.2020.00400   
2020 Kniazeff J. The different aspects of the GABA receptor allosteric modulation. Advances in Pharmacology (San Diego, Calif.). 88: 83-113. PMID 32416873 DOI: 10.1016/bs.apha.2020.02.003   
2020 Dripps IJ, Chen R, Shafer AM, Livingston KE, Disney A, Husbands SM, Traynor JR, Rice KC, Jutkiewicz EM. Pharmacological Properties of Delta Opioid Receptor-Mediated Behaviors: Agonist Efficacy and Receptor Reserve. The Journal of Pharmacology and Experimental Therapeutics. PMID 32467352 DOI: 10.1124/jpet.119.262717   
2020 Amata E, Dichiara M, Gentile D, Marrazzo A, Turnaturi R, Arena E, La Mantia A, Tomasello BR, Acquaviva R, Di Giacomo C, Rescifina A, Prezzavento O. Sigma Receptor Ligands Carrying a Nitric Oxide Donor Nitrate Moiety: Synthesis, In Silico, and Biological Evaluation. Acs Medicinal Chemistry Letters. 11: 889-894. PMID 32435401 DOI: 10.1021/acsmedchemlett.9b00661   
2020 Perpina-Viciano C, Isbilir A, Zarca A, Caspar B, Kilpatrick LE, Hill SJ, Smit MJ, Lohse MJ, Hoffmann C. Kinetic analysis of the early signaling steps of the human chemokine receptor CXCR4. Molecular Pharmacology. PMID 32474443 DOI: 10.1124/mol.119.118448   
2020 Schihada H, Ma X, Zabel U, Vischer HF, Schulte G, Leurs R, Pockes S, Lohse MJ. Development of a conformational histamine H receptor biosensor for the synchronous screening of agonists and inverse agonists. Acs Sensors. PMID 32397705 DOI: 10.1021/acssensors.0c00397   
2020 Liu W, Jiang X, Zu Y, Yang Y, Liu Y, Sun X, Xu Z, Ding H, Zhao Q. A comprehensive description of GluN2B-selective N-methyl-D-aspartate (NMDA) receptor antagonists. European Journal of Medicinal Chemistry. 200: 112447. PMID 32450321 DOI: 10.1016/j.ejmech.2020.112447   
2020 Fuller PJ, Yao YZ, Yang J, Young MJ. Structural determinants of activation of the mineralocorticoid receptor: an evolutionary perspective. Journal of Human Hypertension. PMID 32467588 DOI: 10.1038/s41371-020-0360-2   
2020 Ledderose C, Bromberger S, Slubowski CJ, Sueyoshi K, Junger WG. Frontline Science: P2Y11 receptors support T cell activation by directing mitochondrial trafficking to the immune synapse. Journal of Leukocyte Biology. PMID 32531829 DOI: 10.1002/JLB.2HI0520-191R   
2020 Hellyer SD, Aggarwal S, Chen AN, Leach K, Lapinsky DJ, Gregory KJ. Development of Clickable Photoaffinity Ligands for Metabotropic Glutamate Receptor 2 Based on Two Positive Allosteric Modulator Chemotypes. Acs Chemical Neuroscience. PMID 32396330 DOI: 10.1021/acschemneuro.0c00009   
2020 Arsova A, Møller TC, Vedel L, Hansen JL, Foster SR, Gregory KJ, Bräuner-Osborne H. Detailed in vitro pharmacological characterization of clinically tested negative allosteric modulators of the metabotropic glutamate receptor 5 (mGlu5). Molecular Pharmacology. PMID 32358164 DOI: 10.1124/mol.119.119032   
2020 Ghali MGZ, Arborelius UP, Yaşargil MG. β-Adrenergic receptor structure and function: molecular insights guiding the development of novel therapeutic strategies to treat malignancy. Journal of Receptor and Signal Transduction Research. 1-15. PMID 32456520 DOI: 10.1080/10799893.2020.1759091   
2020 Yuan S, Roos PM, Larsson SC. IL-1 Receptor Antagonist, IL-2 Receptor Alpha Subunit and Amyotrophic Lateral Sclerosis. European Journal of Neurology. PMID 32441415 DOI: 10.1111/ene.14338   
2020 Ma YP, Yang Y, Jiang SM, Liu L, Zhang Z, Wang YN, Zou GM, Li WG. Angiotensin II type 1 receptor blockers favorably affect renal angiotensin II and MAS receptor expression in patients with diabetic nephropathy. Journal of the Renin-Angiotensin-Aldosterone System : Jraas. 21: 1470320320919607. PMID 32370637 DOI: 10.1177/1470320320919607   
2020 Zhang X, Meng R, Wang H, Xing J. Differential Effects of Components in Artemisia annua Extract on the Induction of Drug-Metabolizing Enzyme Expression Mediated by Nuclear Receptors. Planta Medica. PMID 32557519 DOI: 10.1055/a-1178-0852   
2020 Möller J, Isbilir A, Sungkaworn T, Osberg B, Karathanasis C, Sunkara V, Grushevskyi EO, Bock A, Annibale P, Heilemann M, Schütte C, Lohse MJ. Single-molecule analysis reveals agonist-specific dimer formation of µ-opioid receptors. Nature Chemical Biology. PMID 32541966 DOI: 10.1038/s41589-020-0566-1   
2020 Georges GJ, Dengl S, Bujotzek A, Hesse F, Fischer JAA, Gärtner A, Benz J, Lauer ME, Ringler P, Stahlberg H, Plath F, Brinkmann U, Imhof-Jung S. The Contorsbody, an antibody format for agonism: Design, structure, and function. Computational and Structural Biotechnology Journal. 18: 1210-1220. PMID 32542107 DOI: 10.1016/j.csbj.2020.05.007   
2020 Gurevich VV, Gurevich EV. Biased GPCR signaling: Possible mechanisms and inherent limitations. Pharmacology & Therapeutics. 107540. PMID 32201315 DOI: 10.1016/j.pharmthera.2020.107540   
2020 Rogers MA, Fantauzzo KA. The emerging complexity of PDGFRs: activation, internalization and signal attenuation. Biochemical Society Transactions. PMID 32369556 DOI: 10.1042/BST20200004