| Year |
Citation |
Score |
| 2004 |
Jiang X, Zhao B, Britton R, Lim LY, Leong D, Sanghera JS, Zhou BB, Piers E, Andersen RJ, Roberge M. Inhibition of Chk1 by the G2 DNA damage checkpoint inhibitor isogranulatimide. Molecular Cancer Therapeutics. 3: 1221-7. PMID 15486189 |
0.395 |
|
| 2004 |
Britton RA, Piers E, Patrick BO. Total synthesis of (+/-)-13-methoxy-15-oxozoapatlin, a rearranged kaurane diterpenoid. The Journal of Organic Chemistry. 69: 3068-75. PMID 15104445 DOI: 10.1002/CHIN.200435177 |
0.542 |
|
| 2001 |
Piers E, Harrison CL, Zetina-Rocha C. Intramolecular conjugate addition of alkenyl and aryl functions to enones initiated by lithium-iodine exchange. Organic Letters. 3: 3245-7. PMID 11594805 DOI: 10.1021/ol016288u |
0.655 |
|
| 2000 |
Piers E, Caillé S, Chen G. A formal total synthesis of the sesterterpenoid (+/-)-dysidiolide and approaches to the syntheses of (+/-)-6-epi-, (+/-)-15-epi-, and (+/-)-6,15-bisepidysidiolide. Organic Letters. 2: 2483-6. PMID 10956527 |
0.306 |
|
| 2000 |
Piers E, Yee JG, Gladstone PL. CuCl-mediated intramolecular oxidative coupling of aryl- and alkenyltrimethylstannane functions Organic Letters. 2: 481-4. PMID 10814356 |
0.687 |
|
| 2000 |
Piers E, Britton R, Andersen RJ. Improved synthesis of isogranulatimide, a G2 checkpoint inhibitor. Syntheses Of didemnimide C, isodidemnimide A, neodidemnimide A, 17-methylgranulatimide, and isogranulatimides A-C. The Journal of Organic Chemistry. 65: 530-5. PMID 10813968 DOI: 10.1021/Jo9914723 |
0.476 |
|
| 2000 |
Piers E, Walker SD, Armbrust R. A new cycloheptenone annulation method: Use of the bifunctional reagent (Z)-5-iodo-l-tributylstannyIpent-l-ene in organic synthesis Journal of the Chemical Society, Perkin Transactions 1. 635-637. DOI: 10.1039/A909922K |
0.519 |
|
| 2000 |
Piers E, McEachern EJ, Burns PA. Cu(I)-mediated intramolecular conjugate addition of alkenyltrimethylstannane functions to α,β-unsaturated ketones: A convenient preparation of functionalized cis-fused bicyclo[4.3.0]non-8-en-3-ones and Bicyclo[3.3.0]oct-6-en-3-ones Tetrahedron. 56: 2753-2765. DOI: 10.1016/S0040-4020(00)00131-9 |
0.326 |
|
| 1999 |
Piers E, Skupinska KA, Wallace DJ. CuCN-mediated intramolecular conjugate additions. Syntheses of functionalized, cis-fused bicyclo[6.3.0]undecanes, bicyclo[6.4.0]dodecanes, and bicyclo[7.4.0]tridecanes Synlett. 1867-1870. |
0.654 |
|
| 1998 |
Roberge M, Berlinck RG, Xu L, Anderson HJ, Lim LY, Curman D, Stringer CM, Friend SH, Davies P, Vincent I, Haggarty SJ, Kelly MT, Britton R, Piers E, Andersen RJ. High-throughput assay for G2 checkpoint inhibitors and identification of the structurally novel compound isogranulatimide. Cancer Research. 58: 5701-6. PMID 9865726 |
0.422 |
|
| 1998 |
Piers E, Boehringer EM, Yee JGK. Novel synthesis of functionalized cyclobutane derivatives via intramolecular conjugate addition of alkenyltrimethylstannane functions to α,β-alkynic esters mediated by copper(I) chloride Journal of Organic Chemistry. 63: 8642-8643. DOI: 10.1021/jo981803w |
0.382 |
|
| 1998 |
Berlmck RGS, Britton R, Piers E, Lim L, Roberge M, Rosana Moreira Da Rocha, Andersen RJ. Granulatimide and isogranulatimide, aromatic alkaloids with G2 checkpoint inhibition activity isolated from the Brazilian ascidian Didemnum granulatum: Structure elucidation and synthesis Journal of Organic Chemistry. 63: 9850-9856. DOI: 10.1021/Jo981607P |
0.459 |
|
| 1996 |
Piers E, McEachern EJ, Romero MA. Intermolecular copper(I) chloride-mediated coupling of alkenyltrialkylstannane functions: A convenient synthesis of conjugated diene systems Tetrahedron Letters. 37: 1173-1176. DOI: 10.1016/0040-4039(95)02403-4 |
0.325 |
|
| 1996 |
Piers E, Coish PDG. Butyllithium mediated cyclization of substituted cis-1-(alk-4-ynyl)-2-hydroxymethyl-1-iodocyclopropanes: Synthesis of functionalized spiro[2.4]heptanes Synthesis. 502-506. |
0.425 |
|
| 1996 |
Piers E, McEachern EJ. Trifunctional Reagents in Organic Synthesis: Sequential, Chemoselective Reactions Leading to the Preparation of Structurally Novel Tricycles Synlett. 1996: 1087-1090. |
0.308 |
|
| 1995 |
Piers E, Lemieux R. Reaction of (trimethylgermyl)copper(I)-dimethyl sulfide with acyl chlorides: Efficient syntheses of functionalized acyltrimethylgermanes Organometallics. 14: 5011-5012. |
0.306 |
|
| 1995 |
Piers E, Lemieux R. Platinum-catalysed addition of trimethylgermane to 1-trimethylsilylalk-1- ynes: A convenient synthesis of functionalised 2-trimethylgermylalk-1-enes Journal of the Chemical Society, Perkin Transactions 1. 3-5. |
0.397 |
|
| 1995 |
Piers E, McEachern EJ, Burns PA. Intramolecular Michael additions: Copper(I) chloride-mediated conjugate addition of vinyltrimethylstannane functions to α,β-unsaturated ketones Journal of Organic Chemistry. 60: 2322-2323. |
0.302 |
|
| 1995 |
Piers E, Coish PD. Preparation and cyclopropanation of 2- and 3-iodoalk-2-en-1-ols: Synthesis of functionalized, stereodefined iodocyclopropanes Synthesis. 47-55. |
0.405 |
|
| 1993 |
Piers E, Fleming FF. Palladium(0)-catalyzed conversion of vinyl trifluoromethanesulfonates into α,β-unsaturated nitriles Canadian Journal of Chemistry. 71: 1867-1872. |
0.498 |
|
| 1989 |
Piers E, Fleming FF. Total synthesis of the trans-clerodane diterpenoid (±)-stephalic acid Journal of the Chemical Society, Chemical Communications. 1665-1667. DOI: 10.1039/C39890001665 |
0.491 |
|
| 1989 |
Piers E, Fleming FF. Conversion of enol trifluoromethanesulphonates into α,β- unsaturated nitriles Journal of the Chemical Society, Chemical Communications. 756-757. DOI: 10.1039/C39890000756 |
0.467 |
|
| 1989 |
Piers E, Chong JM, Morton HE. Reaction of (trimethylstanyl)copper(I) reagents with α,β-acettylenic esters. Stereocontrolled synthesis of alkyl (E)- and (Z)-3-tribethylstannyl-2-alkenoates Tetrahedron. 45: 363-380. DOI: 10.1016/0040-4020(89)80065-1 |
0.571 |
|
| 1988 |
Piers E, Lu YF. Deconjugation-alkylation of ethyl 3-(trimethylstannyl)-2-alkenoates. Stereocontrolled synthesis of ethyl 2-alkylidene-3-methylenecyclobutanecarboxylates Journal of Organic Chemistry. 53: 926-927. |
0.401 |
|
| 1987 |
Piers E, Jung GL, Ruediger EH. Synthesis of functionalized bicyclo[3.2.1]octa-2,6dienes by thermal rearrangement of substituted 6-exo(1-alkenyl) bicyclo[3.1.0]hex-2-ene systems Canadian Journal of Chemistry. 65: 670-682. DOI: 10.1139/v87-115 |
0.302 |
|
| 1987 |
Piers E, Skerlj RT. Synthesis of functionalized, stereochemically defined tetrasubstituted alkenes Journal of Organic Chemistry. 52: 4421-4423. |
0.4 |
|
| 1987 |
Piers E, Morton HE, Chong JM. (Trialkylstannyl)copper(I) reagents: Preparation and reaction with α,β-unsaturated carbonyl systems. Preparation of β-trialkylstannyl α,β-unsaturated ketones Canadian Journal of Chemistry. 65: 78-87. |
0.512 |
|
| 1970 |
Kutney JP, Abdurahman N, Gletsos C, Le Quesne P, Piers E, Vlattas I. Total synthesis of indole and dihydroindole alkaloids. V. The total synthesis of dl-quebrachamine and dl-aspidospermidine. A general entry into the aspidosperma alkaloids. Journal of the American Chemical Society. 92: 1727-35. PMID 5418453 DOI: 10.1021/Ja00709A052 |
0.693 |
|
| 1970 |
Kutney JP, Cretney WJ, Le Quesne P, McKague B, Piers E. Total synthesis of indole and dihydroindole alkaloids. IV. The total synthesis of dl-dihydrocleavamine, dl-carbomethoxydihydrocleavamine, dl-coronaridine, dl-dihydrocatharanthine, and dl-ibogamine. A general entry into the iboga and vinca alkaloids. Journal of the American Chemical Society. 92: 1712-26. PMID 5418452 DOI: 10.1021/Ja00709A051 |
0.557 |
|
| 1970 |
Kutney JP, Brown RT, Piers E, Hadfield JR. Total synthesis of indole and dihydroindole alkaloids. 3. The transannular cyclization of carbomethoxydihydrocleavamine and carbomethoxycleavamine derivatives. An approach to vinca and iboga alkaloids. Journal of the American Chemical Society. 92: 1708-12. PMID 5418451 DOI: 10.1021/Ja00709A050 |
0.558 |
|
| 1970 |
Kutney JP, Piers E, Brown RT. Total synthesis of indole and dihydroindole alkaloids. I. Introduction and the transannular cyclization appraoch. Journal of the American Chemical Society. 92: 1700-4. PMID 5418449 DOI: 10.1021/Ja00709A048 |
0.598 |
|
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