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22 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 McNamara N, Rahmani R, Sykes ML, Avery VM, Baell J. Hit-to-lead optimization of novel benzimidazole phenylacetamides as broad spectrum trypanosomacides. Rsc Medicinal Chemistry. 11: 685-695. PMID 33479668 DOI: 10.1039/d0md00058b  0.664
2020 Varghese S, Rahmani R, Drew DR, Beeson JG, Baum J, Smith BJ, Baell J. Structure activity studies of truncated latrunculin analogues with anti-malarial activity. Chemmedchem. PMID 32929894 DOI: 10.1002/Cmdc.202000399  0.631
2020 Varghese S, Rahmani R, Russell S, Deora GS, Ferrins L, Toynton A, Jones A, Sykes M, Kessler A, Eufrásio A, Cordeiro AT, Sherman J, Rodriguez A, Avery VM, Piggott MJ, et al. Discovery of Potent -Ethylurea Pyrazole Derivatives as Dual Inhibitors of and . Acs Medicinal Chemistry Letters. 11: 278-285. PMID 32184957 DOI: 10.1021/Acsmedchemlett.9B00218  0.752
2019 Vuckovic Z, Gentry PR, Berizzi AE, Hirata K, Varghese S, Thompson G, van der Westhuizen ET, Burger WAC, Rahmani R, Valant C, Langmead CJ, Lindsley CW, Baell JB, Tobin AB, Sexton PM, et al. Crystal structure of the M muscarinic acetylcholine receptor. Proceedings of the National Academy of Sciences of the United States of America. PMID 31772027 DOI: 10.2210/Pdb6Ol9/Pdb  0.567
2017 Swarbrick J, Dennis M, Lee M, Harjani J, Ahmed M, Debono A, Pitcher N, Wang ZC, Chhabra S, Barlow N, Rahmani R, Cleary B, Dolezal O, Hattarki M, Aurelio L, et al. 8-Mercaptoguanine derivatives as inhibitors of dihydropteroate synthase. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 29171692 DOI: 10.1002/Chem.201704730  0.602
2016 Johnson S, Rahmani R, Drew DR, Williams MJ, Wilkinson M, Tan YH, Huang JX, Tonkin CJ, Beeson JG, Baum J, Smith BJ, Baell JB. Truncated Latrunculins as Actin Inhibitors Targeting Plasmodium falciparum Motility and Host Cell Invasion. Journal of Medicinal Chemistry. 59: 10994-11005. PMID 28002959 DOI: 10.1021/Acs.Jmedchem.6B01109  0.6
2016 Russell S, Rahmani R, Jones AJ, Newson H, Neilde K, Cotillo I, Rahmani Khajouei M, Ferrins L, Qureishi S, Nguyen N, Martínez-Martínez MS, Weaver DF, Kaiser M, Riley J, Thomas J, et al. Hit-to-Lead Optimisation of a Novel Class of Potent, Broad-Spectrum Trypanosomacides. Journal of Medicinal Chemistry. PMID 27548560 DOI: 10.1021/Acs.Jmedchem.6B00442  0.772
2016 Dennis ML, Pitcher NP, Lee MD, Debono AJ, Wang ZC, Harjani JR, Rahmani R, Cleary B, Peat TS, Baell JB, Swarbrick JD. Structural Basis for the Selective Binding of Inhibitors to 6-Hydroxymethyl-7,8-dihydropterin Pyrophosphokinase from Staphylococcus aureus and Escherichia coli. Journal of Medicinal Chemistry. PMID 27094768 DOI: 10.1021/Acs.Jmedchem.6B00002  0.606
2016 Stoessel D, Nowell CJ, Jones AJ, Ferrins L, Ellis KM, Riley J, Rahmani R, Read KD, McConville MJ, Avery VM, Baell JB, Creek DJ. Metabolomics and lipidomics reveal perturbation of sphingolipid metabolism by a novel anti-trypanosomal 3-(oxazolo[4,5-b]pyridine-2-yl)anilide Metabolomics. 12. DOI: 10.1007/S11306-016-1062-1  0.75
2015 Rahmani R, Ban K, Jones AJ, Ferrins L, Ganame D, Sykes ML, Avery VM, White KL, Ryan E, Kaiser M, Charman SA, Baell JB. 6-Arylpyrazine-2-carboxamides: A New Core for Trypanosoma brucei Inhibitors. Journal of Medicinal Chemistry. 58: 6753-65. PMID 26247439 DOI: 10.1021/Acs.Jmedchem.5B00438  0.773
2014 Dennis ML, Chhabra S, Wang ZC, Debono A, Dolezal O, Newman J, Pitcher NP, Rahmani R, Cleary B, Barlow N, Hattarki M, Graham B, Peat TS, Baell JB, Swarbrick JD. Structure-based design and development of functionalized Mercaptoguanine derivatives as inhibitors of the folate biosynthesis pathway enzyme 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase from Staphylococcus aureus. Journal of Medicinal Chemistry. 57: 9612-26. PMID 25357262 DOI: 10.1021/jm501417f  0.593
2014 Ferrins L, Gazdik M, Rahmani R, Varghese S, Sykes ML, Jones AJ, Avery VM, White KL, Ryan E, Charman SA, Kaiser M, Bergström CA, Baell JB. Pyridyl benzamides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei. Journal of Medicinal Chemistry. 57: 6393-402. PMID 24978605 DOI: 10.1021/Jm500191U  0.759
2014 Drujon J, Rahmani R, Héran V, Blanc R, Carissan Y, Tuccio B, Commeiras L, Parrain JL. trans-1,2-Disiloxybenzocyclobutene, an adequate partner for the auto-oxidation: EPR/spin trapping and theoretical studies. Physical Chemistry Chemical Physics : Pccp. 16: 7513-20. PMID 24626812 DOI: 10.1039/C3Cp55077J  0.475
2014 Dror RO, Green HF, Valant C, Borhani DW, Valcourt JR, Pan AC, Arlow DH, Canals M, Lane JR, Rahmani R, Baell JB, Sexton PM, Christopoulos A, Shaw DE. Structural Basis for Modulation of a GPCR by Allosteric Drugs Biophysical Journal. 106: 100a. DOI: 10.1016/J.Bpj.2013.11.626  0.56
2013 Ferrins L, Rahmani R, Baell JB. Drug discovery and human African trypanosomiasis: a disease less neglected? Future Medicinal Chemistry. 5: 1801-41. PMID 24144414 DOI: 10.4155/Fmc.13.162  0.735
2013 Dror RO, Green HF, Valant C, Borhani DW, Valcourt JR, Pan AC, Arlow DH, Canals M, Lane JR, Rahmani R, Baell JB, Sexton PM, Christopoulos A, Shaw DE. Structural basis for modulation of a G-protein-coupled receptor by allosteric drugs. Nature. 503: 295-9. PMID 24121438 DOI: 10.1038/Nature12595  0.556
2013 Ferrins L, Rahmani R, Sykes ML, Jones AJ, Avery VM, Teston E, Almohaywi B, Yin J, Smith J, Hyland C, White KL, Ryan E, Campbell M, Charman SA, Kaiser M, et al. 3-(Oxazolo[4,5-b]pyridin-2-yl)anilides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei, the causative agent for human African trypanosomiasis. European Journal of Medicinal Chemistry. 66: 450-65. PMID 23831695 DOI: 10.1016/J.Ejmech.2013.05.007  0.767
2012 Dubois S, Rodier F, Blanc R, Rahmani R, Héran V, Thibonnet J, Commeiras L, Parrain JL. Dramatic influence of the substitution of alkylidene-5H-furan-2-ones in Diels-Alder cycloadditions with o-quinonedimethide as diene partner: en route to the CDEF polycyclic ring system of lactonamycin. Organic & Biomolecular Chemistry. 10: 4712-9. PMID 22580446 DOI: 10.1039/C2Ob25299F  0.537
2012 Rahmani R, Matsumoto M, Yamashita Y, Kobayashi S. Direct-type aldol reactions of fluorenylidene-protected/activated glycine esters with aldehydes for the synthesis of β-hydroxy-α-amino acid derivatives. Chemistry, An Asian Journal. 7: 1191-4. PMID 22461460 DOI: 10.1002/Asia.201200081  0.385
2010 Blanc R, Héran V, Rahmani R, Commeiras L, Parrain JL. Diels-Alder cycloaddition of o-quinonedimethides and alkylidene-5H-furan-2-ones: new and rapid access to lambertellol cores and arthrinone derivatives. Organic & Biomolecular Chemistry. 8: 5490-4. PMID 20936215 DOI: 10.1039/C0Ob00448K  0.548
2009 Inack-Ngi S, Rahmani R, Commeiras L, Chouraqui G, Thibonnet J, Duchene A, Abarbri M, Parrain J. ChemInform Abstract: Copper-Catalyzed Preparation of γ-Alkylidenebutenolides and Isocoumarins under Mild Palladium-Free Conditions. Cheminform. 40. DOI: 10.1002/chin.200930036  0.442
2009 Inack-Ngi S, Rahmani R, Commeiras L, Chouraqui G, Thibonnet J, Duchêne A, Abarbri M, Parrain JL. Copper-catalyzed preparation of γ-alkylidenebutenolides and isocoumarins under mild palladium-free conditions Advanced Synthesis and Catalysis. 351: 779-788. DOI: 10.1002/Adsc.200800757  0.462
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