Year |
Citation |
Score |
2012 |
Sarkis M, Tran DN, Kolb S, Miteva MA, Villoutreix BO, Garbay C, Braud E. Design and synthesis of novel bis-thiazolone derivatives as micromolar CDC25 phosphatase inhibitors: Effect of dimerisation on phosphatase inhibition Bioorganic and Medicinal Chemistry Letters. 22: 7345-7350. PMID 23141909 DOI: 10.1016/J.Bmcl.2012.10.072 |
0.691 |
|
2012 |
Amombo GM, Kramer T, Lo Monte F, Göring S, Fach M, Smith S, Kolb S, Schubenel R, Baumann K, Schmidt B. Modification of a promiscuous inhibitor shifts the inhibition from γ-secretase to FLT-3. Bioorganic & Medicinal Chemistry Letters. 22: 7634-40. PMID 23107479 DOI: 10.1016/j.bmcl.2012.10.016 |
0.59 |
|
2011 |
Besset T, Braud E, Jarray R, Garbay C, Kolb S, Leo P, Morin C. Preparation and evaluation of a set of bis(methoxycarbonylmethylthio) heteroquinones as CDC25B phosphatase inhibitors European Journal of Chemistry. 2: 433-440. DOI: 10.5155/Eurjchem.2.4.433-440.400 |
0.752 |
|
2010 |
Kolb S, Goddard ML, Loukaci A, Mondésert O, Ducommun B, Braud E, Garbay C. 5-Substituted [1]pyrindine derivatives with antiproliferative activity. European Journal of Medicinal Chemistry. 45: 896-901. PMID 19969400 DOI: 10.1016/J.Ejmech.2009.11.028 |
0.658 |
|
2009 |
Duval R, Kolb S, Braud E, Genest D, Garbay C. Rapid discovery of triazolobenzylidene-thiazolopyrimidines (TBTP) as CDC25 phosphatase inhibitors by parallel click chemistry and in situ screening. Journal of Combinatorial Chemistry. 11: 947-50. PMID 19835352 DOI: 10.1021/Cc900140F |
0.56 |
|
2009 |
Kolb S, Mondésert O, Goddard ML, Jullien D, Villoutreix BO, Ducommun B, Garbay C, Braud E. Development of novel thiazolopyrimidines as CDC25B phosphatase inhibitors. Chemmedchem. 4: 633-48. PMID 19212959 DOI: 10.1002/Cmdc.200800415 |
0.78 |
|
2009 |
Kolb S, Mondésert O, Goddard M, Jullien D, Villoutreix BO, Ducommun B, Garbay C, Braud E. Inside Cover: Development of Novel Thiazolopyrimidines as CDC25B Phosphatase Inhibitors (ChemMedChem 4/2009) Chemmedchem. 4: 482-482. DOI: 10.1002/Cmdc.200990016 |
0.679 |
|
2008 |
Braud E, Goddard ML, Kolb S, Brun MP, Mondésert O, Quaranta M, Gresh N, Ducommun B, Garbay C. Novel naphthoquinone and quinolinedione inhibitors of CDC25 phosphatase activity with antiproliferative properties. Bioorganic & Medicinal Chemistry. 16: 9040-9. PMID 18789703 DOI: 10.1016/J.Bmc.2008.08.009 |
0.72 |
|
2008 |
Montes M, Braud E, Miteva MA, Goddard ML, Mondésert O, Kolb S, Brun MP, Ducommun B, Garbay C, Villoutreix BO. Receptor-based virtual ligand screening for the identification of novel CDC25 phosphatase inhibitors. Journal of Chemical Information and Modeling. 48: 157-65. PMID 18154280 DOI: 10.1021/Ci700313E |
0.698 |
|
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