Marc O. Anderson, PhD - Publications

Affiliations: 
Chemistry and Biochemistry San Francisco State University, San Francisco, CA, United States 
Area:
Medicinal Chemistry
Website:
http://www.chemistry.sfsu.edu/faculty_anderson/0layout.php

37 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2021 Zhang L, Howland M, Hilgenfeld R, Anderson MO, Eagon S. Identification of Non-Covalent SARS-CoV-2 Main Protease Inhibitors by a Virtual Screen of Commercially Available Drug-Like Compounds. Bioorganic & Medicinal Chemistry Letters. 127990. PMID 33775840 DOI: 10.1016/j.bmcl.2021.127990  0.709
2021 Kahlon G, Lira R, Masvlov N, Pompa E, Brar N, Eagon S, Anderson MO, Andaya A, Chance JP, Fejzic H, Keniston A, Huynh N, Celis N, Vidal B, Trieu N, et al. Corrigendum to "Structure guided development of potent piperazine-derived hydroxamic acid inhibitors targeting falcilysin" [Bioorg. Med. Chem. Lett. 32 (2021) 127683]. Bioorganic & Medicinal Chemistry Letters. 37: 127836. PMID 33588181 DOI: 10.1016/j.bmcl.2021.127836  0.728
2020 Kahlon G, Lira R, Masvlov N, Pompa E, Brar N, Eagon S, Anderson MO, Andaya A, Chance JP, Fejzic H, Keniston A, Vidal B, Trieu N, Rodriguez P, Mallari JP. Structure Guided Development of Potent Piperazine-Derived Hydroxamic Acid Inhibitors Targeting Falcilysin. Bioorganic & Medicinal Chemistry Letters. 127683. PMID 33227414 DOI: 10.1016/j.bmcl.2020.127683  0.742
2020 Eagon S, Hammill JT, Sigal MS, Ahn KJ, Tryhorn JE, Koch G, Belanger B, Chaplan CA, Loop L, Kashtanova AS, Yniguez K, Lazaro H, Wilkinson SP, Rice A, Falade M, ... ... Anderson MO, et al. Synthesis and structure-activity relationship of dual-stage antimalarial pyrazolo[3,4-b]pyridines. Journal of Medicinal Chemistry. PMID 32945666 DOI: 10.1021/Acs.Jmedchem.0C01152  0.727
2019 Bowen LR, Li DJ, Nola DT, Anderson MO, Heying M, Groves AT, Eagon S. Identification of potential Zika virus NS2B-NS3 protease inhibitors via docking, molecular dynamics and consensus scoring-based virtual screening. Journal of Molecular Modeling. 25: 194. PMID 31209577 DOI: 10.1007/S00894-019-4076-6  0.714
2018 Lee S, Cil O, Diez-Cecilia E, Anderson MO, Verkman AS. Nanomolar-potency 1,2,4-triazoloquinoxaline inhibitors of the kidney urea transporter A1 (UT-A1). Journal of Medicinal Chemistry. PMID 29589443 DOI: 10.1021/Acs.Jmedchem.8B00343  0.322
2017 Truong EC, Phuan PW, Reggi AL, Ferrera L, Galietta LJV, Levy SE, Moises AC, Cil O, Diez-Cecilia E, Lee S, Verkman AS, Anderson MO. Substituted 2-acylamino-cycloalkylthiophene-3-carboxylic acid arylamides as inhibitors of the calcium-activated chloride channel transmembrane protein 16A (TMEM16A). Journal of Medicinal Chemistry. PMID 28493701 DOI: 10.1021/Acs.Jmedchem.7B00020  0.415
2017 Tradtrantip L, Jin BJ, Yao X, Anderson MO, Verkman AS. Aquaporin-Targeted Therapeutics: State-of-the-Field. Advances in Experimental Medicine and Biology. 969: 239-250. PMID 28258578 DOI: 10.1007/978-94-024-1057-0_16  0.351
2017 Durham SD, Sierra B, Gomez MJ, Tran JK, Anderson MO, Whittington-Davis NA, Eagon S. Synthesis of β-carbolines via a silver-mediated oxidation of tetrahydro-β-carbolines Tetrahedron Letters. 58: 2747-2750. DOI: 10.1016/J.Tetlet.2017.05.098  0.679
2016 Bayih AG, Folefoc A, Mohon AN, Eagon S, Anderson M, Pillai DR. In vitro and in vivo anti-malarial activity of novel harmine-analog heat shock protein 90 inhibitors: a possible partner for artemisinin. Malaria Journal. 15: 579. PMID 27903279 DOI: 10.1186/S12936-016-1625-7  0.691
2016 Esteva-Font C, Jin BJ, Lee S, Phuan PW, Anderson MO, Verkman AS. Experimental evaluation of proposed small-molecule inhibitors of water channel aquaporin-1. Molecular Pharmacology. PMID 26993802 DOI: 10.1124/Mol.116.103929  0.306
2016 Piechowicz KA, Truong EC, Javed KM, Chaney RR, Wu JY, Phuan PW, Verkman AS, Anderson MO. Synthesis and evaluation of 5,6-disubstituted thiopyrimidine aryl aminothiazoles as inhibitors of the calcium-activated chloride channel TMEM16A/Ano1. Journal of Enzyme Inhibition and Medicinal Chemistry. 1-7. PMID 26796863 DOI: 10.3109/14756366.2015.1135912  0.41
2015 Lee S, Esteva-Font C, Phuan PW, Anderson MO, Verkman AS. Discovery, synthesis and structure-activity analysis of symmetrical 2,7-disubstituted fluorenones as urea transporter inhibitors. Medchemcomm. 6: 1278-1284. PMID 26191399 DOI: 10.1039/C5Md00198F  0.384
2015 Esteva-Font C, Phuan PW, Lee S, Su T, Anderson MO, Verkman AS. Structure-activity analysis of thiourea analogs as inhibitors of UT-A and UT-B urea transporters. Biochimica Et Biophysica Acta. 1848: 1075-80. PMID 25613743 DOI: 10.1016/J.Bbamem.2015.01.004  0.348
2015 Esteva-Font C, Anderson MO, Verkman AS. Urea transporter proteins as targets for small-molecule diuretics. Nature Reviews. Nephrology. 11: 113-23. PMID 25488859 DOI: 10.1038/Nrneph.2014.219  0.344
2014 Verkman AS, Esteva-Font C, Cil O, Anderson MO, Li F, Li M, Lei T, Ren H, Yang B. Small-molecule inhibitors of urea transporters. Sub-Cellular Biochemistry. 73: 165-77. PMID 25298345 DOI: 10.1007/978-94-017-9343-8_11  0.354
2014 Esteva-Font C, Cil O, Phuan PW, Su T, Lee S, Anderson MO, Verkman AS. Diuresis and reduced urinary osmolality in rats produced by small-molecule UT-A-selective urea transport inhibitors. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 28: 3878-90. PMID 24843071 DOI: 10.1096/Fj.14-253872  0.402
2014 Eagon S, Anderson MO. Microwave-assisted synthesis of tetrahydro-β-carbolines and β-carbolines European Journal of Organic Chemistry. 2014: 1653-1665. DOI: 10.1002/Ejoc.201301580  0.674
2013 Esteva-Font C, Phuan PW, Anderson MO, Verkman AS. A small molecule screen identifies selective inhibitors of urea transporter UT-A. Chemistry & Biology. 20: 1235-44. PMID 24055006 DOI: 10.1016/J.Chembiol.2013.08.005  0.339
2013 Choy CJ, Fulton MD, Davis AL, Hopkins M, Choi JK, Anderson MO, Berkman CE. Rationally designed sulfamides as glutamate carboxypeptidase II inhibitors. Chemical Biology & Drug Design. 82: 612-9. PMID 23773397 DOI: 10.1111/Cbdd.12174  0.368
2013 Liu Y, Esteva-Font C, Yao C, Phuan PW, Verkman AS, Anderson MO. 1,1-Difluoroethyl-substituted triazolothienopyrimidines as inhibitors of a human urea transport protein (UT-B): new analogs and binding model. Bioorganic & Medicinal Chemistry Letters. 23: 3338-41. PMID 23597791 DOI: 10.1016/J.Bmcl.2013.03.089  0.391
2012 O'Donoghue AJ, Eroy-Reveles AA, Knudsen GM, Ingram J, Zhou M, Statnekov JB, Greninger AL, Hostetter DR, Qu G, Maltby DA, Anderson MO, Derisi JL, McKerrow JH, Burlingame AL, Craik CS. Global identification of peptidase specificity by multiplex substrate profiling. Nature Methods. 9: 1095-100. PMID 23023596 DOI: 10.1038/Nmeth.2182  0.333
2012 Phuan PW, Anderson MO, Tradtrantip L, Zhang H, Tan J, Lam C, Bennett JL, Verkman AS. A small-molecule screen yields idiotype-specific blockers of neuromyelitis optica immunoglobulin G binding to aquaporin-4. The Journal of Biological Chemistry. 287: 36837-44. PMID 22989877 DOI: 10.1074/Jbc.M112.408716  0.326
2012 Anderson MO, Zhang J, Liu Y, Yao C, Phuan PW, Verkman AS. Nanomolar potency and metabolically stable inhibitors of kidney urea transporter UT-B. Journal of Medicinal Chemistry. 55: 5942-50. PMID 22694147 DOI: 10.1021/Jm300491Y  0.369
2011 Blank BR, Alayoglu P, Engen W, Choi JK, Berkman CE, Anderson MO. N-substituted glutamyl sulfonamides as inhibitors of glutamate carboxypeptidase II (GCP2). Chemical Biology & Drug Design. 77: 241-7. PMID 21219587 DOI: 10.1111/J.1747-0285.2011.01085.X  0.378
2010 Zhang Y, Anderson M, Weisman JL, Lu M, Choy CJ, Boyd VA, Price J, Sigal M, Clark J, Connelly M, Zhu F, Guiguemde WA, Jeffries C, Yang L, Lemoff A, et al. Evaluation of Diarylureas for Activity Against Plasmodium falciparum. Acs Medicinal Chemistry Letters. 1: 460-465. PMID 21243104 DOI: 10.1021/Ml100083C  0.587
2010 Engen W, O'Brien TE, Kelly B, Do J, Rillera L, Stapleton LK, Youngren JF, Anderson MO. Synthesis of aryl-heteroaryl ureas (AHUs) based on 4-aminoquinoline and their evaluation against the insulin-like growth factor receptor (IGF-1R). Bioorganic & Medicinal Chemistry. 18: 5995-6005. PMID 20643554 DOI: 10.1016/J.Bmc.2010.06.071  0.384
2008 Wu LY, Do JC, Kazak M, Page H, Toriyabe Y, Anderson MO, Berkman CE. Phosphoramidate derivatives of hydroxysteroids as inhibitors of prostate-specific membrane antigen. Bioorganic & Medicinal Chemistry Letters. 18: 281-4. PMID 18023582 DOI: 10.1016/J.Bmcl.2007.10.096  0.314
2007 Wu LY, Anderson MO, Toriyabe Y, Maung J, Campbell TY, Tajon C, Kazak M, Moser J, Berkman CE. The molecular pruning of a phosphoramidate peptidomimetic inhibitor of prostate-specific membrane antigen. Bioorganic & Medicinal Chemistry. 15: 7434-43. PMID 17869524 DOI: 10.1016/J.Bmc.2007.07.028  0.368
2007 Blecha JE, Anderson MO, Chow JM, Guevarra CC, Pender C, Penaranda C, Zavodovskaya M, Youngren JF, Berkman CE. Inhibition of IGF-1R and lipoxygenase by nordihydroguaiaretic acid (NDGA) analogs. Bioorganic & Medicinal Chemistry Letters. 17: 4026-9. PMID 17502145 DOI: 10.1016/J.Bmcl.2007.04.092  0.324
2006 Anderson MO, Yu H, Penaranda C, Maddux BA, Goldfine ID, Youngren JF, Guy RK. Parallel synthesis of diarylureas and their evaluation as inhibitors of insulin-like growth factor receptor. Journal of Combinatorial Chemistry. 8: 784-90. PMID 16961415 DOI: 10.1021/cc050136z  0.509
2006 May BC, Witkop J, Sherrill J, Anderson MO, Madrid PB, Zorn JA, Prusiner SB, Cohen FE, Guy RK. Structure-activity relationship study of 9-aminoacridine compounds in scrapie-infected neuroblastoma cells. Bioorganic & Medicinal Chemistry Letters. 16: 4913-6. PMID 16860557 DOI: 10.1016/J.Bmcl.2006.06.050  0.73
2006 Anderson MO, Sherrill J, Madrid PB, Liou AP, Weisman JL, DeRisi JL, Guy RK. Parallel synthesis of 9-aminoacridines and their evaluation against chloroquine-resistant Plasmodium falciparum. Bioorganic & Medicinal Chemistry. 14: 334-43. PMID 16216519 DOI: 10.1016/J.Bmc.2005.08.017  0.73
2005 Anderson MO, Shelat AA, Guy RK. A solid-phase approach to the phallotoxins: total synthesis of [Ala7]-phalloidin. The Journal of Organic Chemistry. 70: 4578-84. PMID 15932292 DOI: 10.1021/jo0503153  0.611
2004 Anderson MO, Moser J, Sherrill J, Guy RK. A convenient procedure for parallel ester hydrolysis Synlett. 2391-2393. DOI: 10.1055/s-2004-832828  0.387
2002 Braslau R, Anderson MO, Rivera F, Jimenez A, Haddad T, Axon JR. Acyl hydrazines as precursors to acyl radicals Tetrahedron. 58: 5513-5523. DOI: 10.1016/S0040-4020(02)00490-8  0.705
1998 Braslau R, Anderson MO. Abstraction of deuterium from dideuteroglycine by aryl radical: A model for 1,4-benzene diradical reactions with proteins Tetrahedron Letters. 39: 4227-4230. DOI: 10.1016/S0040-4039(98)00791-6  0.606
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