| Year |
Citation |
Score |
| 2019 |
Borsodi A, Bruchas M, Caló G, Chavkin C, Christie MJ, Civelli O, Connor M, Cox BM, Devi LA, Evans C, Höllt V, Henderson G, Husbands S, Kelly E, Kieffer B, ... ... Simon EJ, et al. Opioid receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database Iuphar/Bps Guide to Pharmacology Cite. 2019. DOI: 10.2218/gtopdb/f50/2019.4 |
0.401 |
|
| 2010 |
Simon EJ, Onoprishvili I. The interaction between the mu opioid receptor and filamin A Neurochemical Research. 35: 1859-1866. PMID 20857334 DOI: 10.1007/S11064-010-0261-9 |
0.457 |
|
| 2009 |
Koob GF, Simon EJ. The Neurobiology of Addiction: Where We Have Been and Where We Are Going. Journal of Drug Issues. 39: 115-132. PMID 20622969 DOI: 10.1177/002204260903900110 |
0.38 |
|
| 2008 |
Onoprishvili I, Ali S, Andria ML, Shpigel A, Simon EJ. Filamin A mutant lacking actin-binding domain restores mu opioid receptor regulation in melanoma cells Neurochemical Research. 33: 2054-2061. PMID 18404377 DOI: 10.1007/S11064-008-9684-Y |
0.385 |
|
| 2007 |
Onoprishvili I, Simon EJ. Chronic morphine treatment up-regulates mu opioid receptor binding in cells lacking filamin A Brain Research. 1177: 9-18. PMID 17897634 DOI: 10.1016/J.Brainres.2007.08.020 |
0.463 |
|
| 2006 |
Ancevska-Taneva N, Onoprishvili I, Andria ML, Hiller JM, Simon EJ. A member of the heat shock protein 40 family, hlj1, binds to the carboxyl tail of the human mu opioid receptor Brain Research. 1081: 28-33. PMID 16542645 DOI: 10.1016/J.Brainres.2006.01.125 |
0.474 |
|
| 2003 |
Onoprishvili I, Andria ML, Kramer HK, Ancevska-Taneva N, Hiller JM, Simon EJ. Interaction Between the μ Opioid Receptor and Filamin A Is Involved in Receptor Regulation and Trafficking Molecular Pharmacology. 64: 1092-1100. PMID 14573758 DOI: 10.1124/Mol.64.5.1092 |
0.512 |
|
| 2002 |
Kramer HK, Onoprishvili I, Andria ML, Hanna K, Sheinkman K, Haddad LB, Simon EJ. Delta opioid activation of the mitogen-activated protein kinase cascade does not require transphosphorylation of receptor tyrosine kinases Bmc Pharmacology [Electronic Resource]. 2: 5. PMID 11897012 DOI: 10.1186/1471-2210-2-5 |
0.423 |
|
| 2002 |
Andria ML, Simon EJ. Erratum to: Identification of a neurorestrictive suppressor element (NRSE) in the human μ-opioid receptor gene Molecular Brain Research. 105: 161. DOI: 10.1016/S0169-328X(02)00165-1 |
0.428 |
|
| 2001 |
Andria ML, Simon EJ. Identification of a neurorestrictive suppressor element (NRSE) in the human μ-opioid receptor gene Molecular Brain Research. 91: 73-80. PMID 11457494 DOI: 10.1016/S0169-328X(01)00124-3 |
0.33 |
|
| 2001 |
Mathieu-Kia AM, Fan LQ, Kreek MJ, Simon EJ, Hiller JM. Mu-, delta- and kappa-opioid receptor populations are differentially altered in distinct areas of postmortem brains of Alzheimer's disease patients. Brain Research. 893: 121-34. PMID 11223000 DOI: 10.1016/S0006-8993(00)03302-3 |
0.504 |
|
| 2000 |
Kramer HK, Andria ML, Esposito DH, Simon EJ. Tyrosine phosphorylation of the δ-opioid receptor: Evidence for its role in mitogen-activated protein kinase activation and receptor internalization Biochemical Pharmacology. 60: 781-792. PMID 10930532 DOI: 10.1016/S0006-2952(00)00400-7 |
0.399 |
|
| 2000 |
Kramer HK, Andria ML, Kushner SA, Esposito DH, Hiller JM, Simon EJ. Mutation of tyrosine 318 (Y318F) in the delta-opioid receptor attenuates tyrosine phosphorylation, agonist-dependent receptor internalization, and mitogen-activated protein kinase activation. Brain Research. Molecular Brain Research. 79: 55-66. PMID 10925143 DOI: 10.1016/S0169-328X(00)00097-8 |
0.432 |
|
| 2000 |
Kramer HK, Simon EJ. μ and δ-opioid receptor agonists induce mitogen-activated protein kinase (MAPK) activation in the absence of receptor internalization Neuropharmacology. 39: 1707-1719. PMID 10884553 DOI: 10.1016/S0028-3908(99)00243-9 |
0.457 |
|
| 1999 |
Onoprishvili I, Andria ML, Vilim FS, Hiller JM, Simon EJ. The bovine mu-opioid receptor: cloning of cDNA and pharmacological characterization of the receptor expressed in mammalian cells. Brain Research. Molecular Brain Research. 73: 129-37. PMID 10581406 DOI: 10.1016/S0169-328X(99)00249-1 |
0.507 |
|
| 1999 |
Andria ML, Simon EJ. Localization of promoter elements in the human mu-opioid receptor gene and regulation by DNA methylation. Brain Research. Molecular Brain Research. 70: 54-65. PMID 10381543 DOI: 10.1016/S0169-328X(99)00126-6 |
0.412 |
|
| 1999 |
Gioannini TL, Onoprishvili I, Hiller JM, Simon EJ. Inactivation of the purified bovine mu opioid receptor by sulfhydryl reagents. Neurochemical Research. 24: 37-42. PMID 9973235 DOI: 10.1023/A:1020923928936 |
0.515 |
|
| 1999 |
Kramer HK, Simon EJ. Role of protein kinase C (PKC) in agonist-induced mu-opioid receptor down-regulation: II. Activation and involvement of the alpha, epsilon, and zeta isoforms of PKC. Journal of Neurochemistry. 72: 594-604. PMID 9930731 DOI: 10.1046/J.1471-4159.1999.0720594.X |
0.477 |
|
| 1999 |
Kramer HK, Simon EJ. Role of protein kinase C (PKC) in agonist-induced mu-opioid receptor down-regulation: I. PKC translocation to the membrane of SH-SY5Y neuroblastoma cells is induced by mu-opioid agonists. Journal of Neurochemistry. 72: 585-93. PMID 9930730 DOI: 10.1046/j.1471-4159.1999.0720585.x |
0.418 |
|
| 1998 |
Ehrlich GK, Andria ML, Zheng X, Kieffer B, Gioannini TL, Hiller JM, Rosenkranz JE, Veksler BM, Zukin RS, Simon EJ. Functional significance of cysteine residues in the delta opioid receptor studied by site-directed mutagenesis. Canadian Journal of Physiology and Pharmacology. 76: 269-77. PMID 9673790 DOI: 10.1139/cjpp-76-3-269 |
0.396 |
|
| 1996 |
Wolinsky TD, Carr KD, Hiller JM, Simon EJ. Chronic food restriction alters μ and κ opioid receptor binding in the parabrachial nucleus of the rat: A quantitative autoradiographic study Brain Research. 706: 333-336. PMID 8822378 DOI: 10.1016/0006-8993(95)01337-7 |
0.644 |
|
| 1996 |
Hiller JM, Fan LQ, Simon EJ. Autoradiographic comparison of [3H]DPDPE and [3H]DSLET binding: evidence for distinct delta 1 and delta 2 opioid receptor populations in rat brain. Brain Research. 719: 85-95. PMID 8782867 DOI: 10.1016/0006-8993(96)00090-X |
0.462 |
|
| 1996 |
Galynker I, Schlyer DJ, Dewey SL, Fowler JS, Logan J, Gatley SJ, MacGregor RR, Ferrieri RA, Holland MJ, Brodie J, Simon E, Wolf AP. Opioid receptor imaging and displacement studies with [6-O-[11C] methyl]buprenorphine in baboon brain. Nuclear Medicine and Biology. 23: 325-31. PMID 8782244 DOI: 10.1016/0969-8051(95)02087-X |
0.399 |
|
| 1995 |
Simon EJ. Recent studies on a mu-opioid receptor purified from bovine striatum. Annals of the New York Academy of Sciences. 757: 324-31. PMID 7611689 DOI: 10.1111/J.1749-6632.1995.Tb17490.X |
0.5 |
|
| 1995 |
Fan LQ, Gioannini TL, Wolinsky T, Hiller JM, Simon EJ. Functional reconstitution of a highly purified mu-opioid receptor protein with purified G proteins in liposomes. Journal of Neurochemistry. 65: 2537-42. PMID 7595548 DOI: 10.1046/J.1471-4159.1995.65062537.X |
0.437 |
|
| 1994 |
Hiller JM, Zhang Y, Bing G, Gioannini TL, Stone EA, Simon EJ. Immunohistochemical localization of Mu-opioid receptors in rat brain using antibodies generated against a peptide sequence present in a purified mu-opioid binding protein Neuroscience. 62: 829-841. PMID 7870310 DOI: 10.1016/0306-4522(94)90480-4 |
0.493 |
|
| 1994 |
Wolinsky TD, Carr KD, Hiller JM, Simon EJ. Effects of chronic food restriction on mu and kappa opioid binding in rat forebrain: a quantitative autoradiographic study Brain Research. 656: 274-280. PMID 7820587 DOI: 10.1016/0006-8993(94)91470-2 |
0.648 |
|
| 1994 |
Wolinsky TD, Carr KD, Hiller JM, Simon EJ. The effects of chronic food restriction on mu and kappa opioid receptors in the rat Regulatory Peptides. 54: 325-326. DOI: 10.1016/0167-0115(94)90520-7 |
0.646 |
|
| 1994 |
Andria M, Ehrlich G, Simon E. Molecular characterization of a human mu-opioid receptor gene: Demonstration of promoter activity Regulatory Peptides. 54: 9-10. DOI: 10.1016/0167-0115(94)90363-8 |
0.453 |
|
| 1994 |
Gioannini TL, Fan L-, Hyde L, Ofri D, Hiller JM, Simon EJ. Reconstitution in liposomes of a μ-opioid binding protein purified to homogeneity from bovine striatal membranes Regulatory Peptides. 53. DOI: 10.1016/0167-0115(94)90238-0 |
0.438 |
|
| 1993 |
Simon EJ, Fan LQ, Hiller JM, Seyed-Mozaffari A, Schultz AG, Archer S. Photoaffinity ligands for the mu opioid receptor. Life Sciences. 53: 1173-8. PMID 8396706 DOI: 10.1016/0024-3205(93)90554-G |
0.432 |
|
| 1993 |
Hiller JM, Fan LQ, Simon EJ. Alterations in delta opioid receptor levels in discrete areas of the neocortex and in the globus pallidus of the aging guinea pig: a quantitative autoradiographic study. Brain Research. 614: 86-98. PMID 8394190 DOI: 10.1016/0006-8993(93)91021-J |
0.43 |
|
| 1993 |
Gioannini TL, Fan LQ, Hyde L, Ofri D, Yao YH, Hiller JM, Simon EJ. Reconstitution of a purified mu-opioid binding protein in liposomes: selective, high affinity, GTP gamma S-sensitive mu-opioid agonist binding is restored. Biochemical and Biophysical Research Communications. 194: 901-8. PMID 8393673 DOI: 10.1006/Bbrc.1993.1906 |
0.488 |
|
| 1992 |
Stein EA, Hiller JM, Simon EJ. Effects of stress on opioid receptor binding in the rat central nervous system. Neuroscience. 51: 683-90. PMID 1336824 DOI: 10.1016/0306-4522(92)90307-N |
0.505 |
|
| 1992 |
Hiller JM, Fan LQ, Simon EJ. Age-related changes in kappa opioid receptors in the guinea-pig brain: a quantitative autoradiographic study. Neuroscience. 50: 663-73. PMID 1331867 DOI: 10.1016/0306-4522(92)90455-B |
0.413 |
|
| 1992 |
Ofri D, Fan LQ, Simon EJ, Hiller JM. Lesioning of the nucleus basalis of Meynert has differential effects on mu, delta and kappa opioid receptor binding in rat brain: a quantitative autoradiographic study. Brain Research. 581: 252-60. PMID 1327399 DOI: 10.1016/0006-8993(92)90715-L |
0.495 |
|
| 1992 |
Simon EJ, Gioannini TL, Yao YH, Hiller JM. Opioid receptors and their biochemistry. Clinical Neuropharmacology. 15: 48A-49A. PMID 1323402 DOI: 10.1097/00002826-199201001-00027 |
0.394 |
|
| 1992 |
Gioannini TL, Weiss ER, Johnson GL, Hiller JM, Simon EJ. Immunoblots with rhodopsin antisera suggest that a purified mu opioid binding protein has structural characteristics of a G-protein-coupled receptor. Proceedings of the National Academy of Sciences of the United States of America. 89: 52-5. PMID 1309617 DOI: 10.1073/Pnas.89.1.52 |
0.455 |
|
| 1992 |
Ofri D, Ritter AM, Liu YF, Gioannini TL, Hiller JM, Simon EJ. Characterization of solubilized opioid receptors: reconstitution and uncoupling of guanine nucleotide-sensitive agonist binding. Journal of Neurochemistry. 58: 628-35. PMID 1309566 DOI: 10.1111/J.1471-4159.1992.Tb09764.X |
0.495 |
|
| 1992 |
Wang BC, Hiller JM, Simon EJ, Li D, Rosenberg C, Turndorf H. Analgesia following Subarachnoid Sodium Ibuprofen in rats Anesthesiology. 77. DOI: 10.1097/00000542-199209001-00862 |
0.305 |
|
| 1991 |
Simon EJ. Opioid receptors and endogenous opioid peptides Medicinal Research Reviews. 11: 357-374. PMID 1652044 DOI: 10.1002/Med.2610110402 |
0.404 |
|
| 1991 |
Carr KD, Aleman DO, Bak TH, Simon EJ. Effects of parabrachial opioid antagonism on stimulation-induced feeding Brain Research. 545: 283-286. PMID 1650277 DOI: 10.1016/0006-8993(91)91298-F |
0.667 |
|
| 1990 |
Hiller JM, Fan LQ, Simon EJ. Differential effects of cyanogen bromide on ligand binding by mu, delta and kappa opioid receptors. Life Sciences. 47: 2225-30. PMID 2176264 DOI: 10.1016/0024-3205(90)90153-I |
0.52 |
|
| 1990 |
Klein P, Nelson WL, Yao YH, Simon EJ. Electrophilic α-methylene-γ-lactone and isothiocyanate opioid ligands related to etorphine Journal of Medicinal Chemistry. 33: 2286-2296. PMID 2165166 DOI: 10.1021/Jm00170A038 |
0.353 |
|
| 1990 |
Olsen LD, Klein P, Nelson WL, Yao YH, Simon EJ. Conjugate addition ligands of opioid antagonists. Methacrylate esters and ethers of 6α- and 6β-naltrexol Journal of Medicinal Chemistry. 33: 737-741. PMID 2153826 DOI: 10.1021/Jm00164A043 |
0.419 |
|
| 1990 |
Stein EA, Carr KD, Simon EJ. Brain stimulation-induced feeding alters regional opioid receptor binding in the rat: an in vivo autoradiographic study Brain Research. 533: 213-222. PMID 1963108 DOI: 10.1016/0006-8993(90)91342-E |
0.666 |
|
| 1990 |
Wang BC, Hiller JM, Simon EJ, Li D, Rosenberg C, Turndorf H. A806 Low Dose Epidural Clonidine Enhances Morphine Analgesia Without Causing Hypotension in Rabbits Anesthesiology. 73. DOI: 10.1097/00000542-199009001-00804 |
0.34 |
|
| 1990 |
Warm BC, Haler JM, Simon EJ, Rosenberg C, Li D, Tumdorf H. A preliminary evaluation of analgesic latency of epidural analgesics in rabbits Pain. 41. DOI: 10.1016/0304-3959(90)92390-C |
0.317 |
|
| 1989 |
Wang BC, Hiller JM, Simon EJ, Hillman DE, Rosenberg C, Turndorf H. Distribution of 3H-morphine following lumbar subarachnoid injection in unanesthetized rabbits. Anesthesiology. 70: 817-24. PMID 2719317 DOI: 10.1097/00000542-198905000-00019 |
0.354 |
|
| 1989 |
Gioannini TL, Liu YF, Park YH, Hiller JM, Simon EJ. Evidence for the presence of disulfide bridges in opioid receptors essential for ligand binding. Possible role in receptor activation. Journal of Molecular Recognition : Jmr. 2: 44-8. PMID 2561526 DOI: 10.1002/jmr.300020107 |
0.41 |
|
| 1989 |
Carr KD, Bak TH, Simon EJ, Portoghese PS. Effects of the selective kappa opioid antagonist, nor-binaltorphimine, on electrically-elicited feeding in the rat Life Sciences. 45: 1787-1792. PMID 2556617 DOI: 10.1016/0024-3205(89)90518-3 |
0.677 |
|
| 1989 |
Schoffelmeer AN, Yao YH, Simon EJ. Cross-linking of human 125I-beta-endorphin to a mu-delta opioid receptor complex in rat striatum. European Journal of Pharmacology. 166: 357-8. PMID 2551701 DOI: 10.1016/0014-2999(89)90085-X |
0.438 |
|
| 1989 |
Archer S, Seyed-Mozaffari A, Simon EJ, Gioannini TL. Opioid ligands related to tifluadom European Journal of Medicinal Chemistry. 24: 569-572. DOI: 10.1016/0223-5234(89)90022-6 |
0.467 |
|
| 1988 |
Wang BC, Hiller JM, Simon EJ, Hillman DE, Turndorf H. Intravenous cystogram for study of urinary retention following intrathecal morphine in unanesthetized rabbits. Anesthesiology. 68: 962-4. PMID 3377245 DOI: 10.1097/00000542-198806000-00031 |
0.404 |
|
| 1988 |
Keren O, Gioannini TL, Hiller JM, Simon EJ. Affinity crosslinking of 125I-labeled human beta-endorphin to cell lines possessing either mu- or delta-type opioid binding sites. Brain Research. 440: 280-4. PMID 2833993 DOI: 10.1016/0006-8993(88)90996-1 |
0.49 |
|
| 1987 |
Simon EJ. Subunit structure and purification of opioid receptors. Journal of Receptor Research. 7: 105-32. PMID 3040975 DOI: 10.3109/10799898709054982 |
0.411 |
|
| 1987 |
Hiller JM, Itzhak Y, Simon EJ. Selective changes in μ, δ and κ{script} opioid receptor binding in certain limbic regions of the brain in Alzheimer's disease patients Brain Research. 406: 17-23. PMID 3032356 DOI: 10.1016/0006-8993(87)90764-5 |
0.403 |
|
| 1987 |
Valette A, Rouge P, Coulais E, Potonnier G, Cros J, Simon EJ. Interaction with lectin of kappa opioid binding sites solubilized from human placenta. Life Sciences. 40: 535-40. PMID 3027488 DOI: 10.1016/0024-3205(87)90366-3 |
0.461 |
|
| 1987 |
Carr KD, Bak TH, Gioannini TL, Simon EJ. Antibodies to dynorphin A(1-13) but not β-endorphin inhibit electrically elicited feeding in the rat Brain Research. 422: 384-388. PMID 2890420 DOI: 10.1016/0006-8993(87)90950-4 |
0.565 |
|
| 1987 |
Adams JU, Andrews JS, Hiller JM, Simon EJ, Holtzman SG. Effects of stress and beta-funal trexamine pretreatment on morphine analgesia and opioid binding in rats. Life Sciences. 41: 2835-44. PMID 2826950 DOI: 10.1016/0024-3205(87)90430-9 |
0.48 |
|
| 1987 |
Wang BC, Hiller JM, Holland MJ, Simon EJ, Hillman DE, Turndorf H. Distribution Of 3H Morphine Following Lumbar Subarachnoid Administration In Rabbits Anesthesia & Analgesia. 66. DOI: 10.1213/00000539-198702001-00185 |
0.362 |
|
| 1987 |
Wang BC, Hiller JM, Holland MJ, Simon EJ, Hillman DE, Turndorf H. Distribution Of 3H-Morphine Following Lumbar Epidural Administration In Rabbits Anesthesiology. 67. DOI: 10.1097/00000542-198709001-00253 |
0.363 |
|
| 1986 |
Simon EJ. Recent studies on opioid receptors: heterogeneity and purification. Annals of the New York Academy of Sciences. 463: 31-45. PMID 3013065 DOI: 10.1111/J.1749-6632.1986.Tb21501.X |
0.49 |
|
| 1986 |
Appelmans N, Carroll JA, Rance MJ, Simon EJ, Traynor JR. Sodium ions increase the binding of the antagonist peptide ICI 174864 to the delta-opiate receptor. Neuropeptides. 7: 139-43. PMID 3010168 DOI: 10.1016/0143-4179(86)90089-2 |
0.412 |
|
| 1986 |
Tempel A, Crain SM, Peterson ER, Simon EJ, Zukin RS. Antagonist-induced opiate receptor upregulation in cultures of fetal mouse spinal cord-ganglion explants. Brain Research. 390: 287-91. PMID 3006869 DOI: 10.1016/0165-3806(86)90218-X |
0.462 |
|
| 1986 |
Howard AD, Sarne Y, Gioannini TL, Hiller JM, Simon EJ. Identification of distinct binding site subunits of μ and δ opioid receptors Biochemistry. 25: 357-360. PMID 3006757 DOI: 10.1021/Bi00350A012 |
0.427 |
|
| 1986 |
Klopman G, Macina OT, Simon EJ, Hiller JM. Computer automated structure evaluation of opiate alkaloids Journal of Molecular Structure: Theochem. 134: 299-308. DOI: 10.1016/0166-1280(86)80002-1 |
0.354 |
|
| 1986 |
Hwang D, Feliu AL, Wolf AP, Macgregor RR, Fowler JS, Amett CD, Holland HJ, Carr K, Simon EJ. Synthesis and evaluation of fluorinated derivatives of fentanyl as candidates for opiate receptor studies using positron emission tomograpry Journal of Labelled Compounds and Radiopharmaceuticals. 23: 277-293. DOI: 10.1002/Jlcr.2580230306 |
0.639 |
|
| 1986 |
Archer S, Michael J, Osei-Gyimah P, Seyed-Mozaffari A, Zukin RS, Maneckjee R, Simon EJ, Gioannini TL. Hybromet: A Ligand for Purifying Opioid Receptors. Cheminform. 17. DOI: 10.1002/Chin.198614360 |
0.475 |
|
| 1985 |
Archer S, Michael J, Osei-Gyimah P, Seyed-Mozaffari A, Zukin RS, Maneckjee R, Simon EJ, Gioannini TL. Hybromet: a ligand for purifying opioid receptors. Journal of Medicinal Chemistry. 28: 1950-3. PMID 2999408 DOI: 10.1021/Jm00150A032 |
0.428 |
|
| 1985 |
Hui KS, Gioannini T, Hui M, Simon EJ, Lajtha A. An opiate receptor-associated aminopeptidase that degrades enkephalins. Neurochemical Research. 10: 1047-58. PMID 2997642 DOI: 10.1007/Bf00965880 |
0.383 |
|
| 1985 |
Bianchetti A, Dragonetti M, Giudice A, Tarantino A, Ferrarese N, Manara L, Appelmans N, Simon EJ. Relative affinities of the quaternary narcotic antagonist, N-methyl levallorphan (SR 58002), for different types of opioid receptors. Neuropeptides. 5: 379-82. PMID 2987738 DOI: 10.1016/0143-4179(85)90033-2 |
0.5 |
|
| 1985 |
Carr KD, Hiller JM, Simon EJ. Diphenhydramine potentiates narcotic but not endogenous opioid analgesia Neuropeptides. 5: 411-414. PMID 2860599 DOI: 10.1016/0143-4179(85)90041-1 |
0.643 |
|
| 1985 |
Archer S, Michael J, Michael M, Simon EJ, Abdelhamid EME, Nelson WL, Koolpe GA. Chloroacryloyl amides and alpha-methylenelactones from naltrexone, oxymorphone and fentanyl Neuropeptides. 5: 395-398. PMID 2582304 DOI: 10.1016/0143-4179(85)90037-X |
0.342 |
|
| 1985 |
Koolpe GA, Nelson WL, Gioannini TL, Angel L, Appelmans N, Simon EJ. Opioid agonists and antagonists. 6-Desoxy-6-substituted lactone, epoxide, and glycidate ester derivatives of naltrexone and oxymorphone. Journal of Medicinal Chemistry. 28: 949-57. PMID 2409280 DOI: 10.1021/Jm00145A018 |
0.31 |
|
| 1985 |
Gioannini TL, Howard AD, Hiller JM, Simon EJ. Purification of an active opioid-binding protein from bovine striatum. Journal of Biological Chemistry. 260: 15117-15121. DOI: 10.1016/s0021-9258(18)95710-8 |
0.342 |
|
| 1985 |
KOOLPE GA, NELSON WL, GIOANNINI TL, ANGEL L, APPELMANS N, SIMON EJ. ChemInform Abstract: OPIOID AGONISTS AND ANTAGONISTS. 6-DESOXY-6-SUBSTITUTED LACTONE, EPOXIDE, AND GLYCIDATE ESTER DERIVATIVES OF NALTREXONE AND OXYMORPHONE Chemischer Informationsdienst. 16. DOI: 10.1002/Chin.198544212 |
0.465 |
|
| 1985 |
KOOLPE GA, NELSON WL, GIOANNINI TL, ANGEL L, SIMON EJ. ChemInform Abstract: DIASTEREOMERIC 6-DESOXY-6-SPIRO-α-METHYLENE-Γ-BUTYROLACTONE DERIVATIVES OF NALTREXONE AND OXYMORPHONE. SELECTIVE IRREVERSIBLE INHIBITION OF NALTREXONE BINDING IN AN OPIOID RECEPTOR PREPARATION BY A CONFORMATIONALLY RESTRICTED MICHAEL Chemischer Informationsdienst. 16. DOI: 10.1002/Chin.198523209 |
0.481 |
|
| 1984 |
Holland MJ, Simon EJ. Etorphine pharmacokinetics in the rat: experimental data and mathematical model. Neuropeptides. 5: 65-8. PMID 6531076 DOI: 10.1016/0143-4179(84)90028-3 |
0.336 |
|
| 1984 |
Carr KD, Aleman DO, Holland MJ, Simon EJ. Analgesic effects of ethylketocyclazocine and morphine in rat and toad Life Sciences. 35: 997-1003. PMID 6433131 DOI: 10.1016/0024-3205(84)90666-0 |
0.631 |
|
| 1984 |
Itzhak Y, Hiller JM, Simon EJ. Solubilization and characterization of μ, δ, and κ opioid binding sites from guinea pig brain: Physical separation of κ receptors Proceedings of the National Academy of Sciences of the United States of America. 81: 4217-4221. PMID 6330751 DOI: 10.1073/Pnas.81.13.4217 |
0.406 |
|
| 1984 |
Carr KD, Simon EJ. Potentiation of reward by hunger is opioid mediated Brain Research. 297: 369-373. PMID 6326944 DOI: 10.1016/0006-8993(84)90578-X |
0.605 |
|
| 1984 |
Gioannini TL, Howard A, Hiller JM, Simon EJ. Affinity chromatography of solubilized opioid binding sites using CH-Sepharose modified with a new naltrexone derivative. Biochemical and Biophysical Research Communications. 119: 624-629. PMID 6324770 DOI: 10.1016/S0006-291X(84)80295-8 |
0.449 |
|
| 1984 |
Yossefit, Hiller JM, Gioannini TL, Simon EJ. Effect of digitonin on the binding of opiate agonists and antagonists to membrane-bound and soluble opioid binding sites Brain Research. 291: 309-315. PMID 6320961 DOI: 10.1016/0006-8993(84)91263-0 |
0.462 |
|
| 1984 |
Koolpe GA, Nelson WL, Gioannini TL, Angel L, Simon EJ. Diastereomeric 6-desoxy-6-spiro-α-methylene-γ-butyrolactone derivatives of naltrexone and oxymorphone. Selective irreversible inhibition of naltrexone binding in an opioid receptor preparation by a conformationally restricted Michael acceptor ligand Journal of Medicinal Chemistry. 27: 1718-1723. PMID 6209395 DOI: 10.1021/Jm00378A032 |
0.331 |
|
| 1984 |
Itzhak Y, Hiller JM, Simon EJ. Solubilization and characterization of kappa opioid binding sites from guinea pig cerebellum Neuropeptides. 5: 201-204. PMID 6099497 DOI: 10.1016/0143-4179(84)90062-3 |
0.435 |
|
| 1984 |
Aucélio JG, Hiller JM, Gioannini T, Simon EJ. Differential sensitivity of major types of opioid binding sites to U.V. irradiation. Neuropeptides. 5: 141-144. PMID 6099483 DOI: 10.1016/0143-4179(84)90047-7 |
0.406 |
|
| 1984 |
Simon EJ, Hiller JM, Itzhak Y, Gioannini TL. SOLUBILIZATION AND CHARACTERIZATION OF ACTIVE OPIOID RECEPTORS BINDING SITES Clinical Neuropharmacology. 7: S24. DOI: 10.1097/00002826-198406001-00023 |
0.498 |
|
| 1983 |
Carr KD, Simon EJ. Effects of naloxone and its quarternary analogue on stimulation-induced feeding Neuropharmacology. 22: 127-130. PMID 6843782 DOI: 10.1016/0028-3908(83)90272-1 |
0.621 |
|
| 1983 |
Carr KD, Simon EJ. The role of opioids in feeding and reward elicited by lateral hypothalamic electrical stimulation Life Sciences. 33: 563-566. PMID 6664237 DOI: 10.1016/0024-3205(83)90565-9 |
0.634 |
|
| 1983 |
Inturrisi CE, Schultz M, Shin S, Umans JG, Angel L, Simon EJ. Evidence from opiate binding studies that heroin acts through its metabolites Life Sciences. 33: 773-776. PMID 6319928 DOI: 10.1016/0024-3205(83)90616-1 |
0.458 |
|
| 1983 |
Bianchetti A, Nisato D, Sacilotto R, Dragonetti M, Picerno N, Tarantino A, Manara L, Angel LM, Simon EJ. Quaternary derivatives of narcotic antagonists: Stereochemical requirements at the chiral nitrogen for in vitro and in vivo activity Life Sciences. 33: 415-418. PMID 6319895 DOI: 10.1016/0024-3205(83)90530-1 |
0.369 |
|
| 1983 |
Itzhak Y, Hiller JM, Gioannini TL, Simon EJ. Evidence for the solubilization of multiple opioid binding sites from mammalian brain Life Sciences. 33: 191-194. PMID 6319858 DOI: 10.1016/0024-3205(83)90475-7 |
0.48 |
|
| 1983 |
Maryanoff BE, Simon EJ, Gioannini T, Gorissen H. Potential Affinity Labels For The Opiate Receptor Based On Fentanyl And Related Compounds Cheminform. 14. DOI: 10.1002/Chin.198302188 |
0.386 |
|
| 1982 |
Carr KD, Bonnet KA, Simon EJ. Medial thalamic lesions reduce the aversion-gating action of lateral hypothalamic stimulation Brain Research. 246: 342-346. PMID 7127104 DOI: 10.1016/0006-8993(82)91189-1 |
0.516 |
|
| 1982 |
Simon EJ. Opiate receptors and opioid peptides: An overview Annals of the New York Academy of Sciences. 327-339. PMID 6297357 DOI: 10.1111/J.1749-6632.1982.Tb39504.X |
0.44 |
|
| 1982 |
Simon EJ, Hiller JM, Groth J, Itzhak Y, Holland MJ, Beck SG. The nature of opiate receptors in toad brain Life Sciences. 31: 1367-1370. PMID 6292631 DOI: 10.1016/0024-3205(82)90383-6 |
0.398 |
|
| 1982 |
Itzhak Y, Bonnet KA, Groth J, Hiller JM, Simon EJ. Multiple opiate binding sites in human brain regions: Evidence for κ and σ sites Life Sciences. 31: 1363-1366. PMID 6292630 DOI: 10.1016/0024-3205(82)90382-4 |
0.365 |
|
| 1982 |
Gioannini TL, Howells RD, Miller JM, Simon EJ. Solubilization in good yield of active opiate binding sites from mammalian brain. Life Sciences. 31: 1315-1318. PMID 6292621 DOI: 10.1016/0024-3205(82)90370-8 |
0.427 |
|
| 1982 |
Carr KD, Bonnet KA, Simon EJ. Mu and kappa opioid agonists elevate brain stimulation threshold for escape by inhibiting aversion Brain Research. 245: 389-393. PMID 6289969 DOI: 10.1016/0006-8993(82)90824-1 |
0.645 |
|
| 1982 |
Crain SM, Crain B, Peterson ER, Hiller JM, Simon EJ. Exposure to 4-aminopyridine prevents depressant effects of opiates on sensory-evoked dorsal-horn network responses in spinal cord cultures. Life Sciences. 31: 235-40. PMID 6289031 DOI: 10.1016/0024-3205(82)90583-5 |
0.375 |
|
| 1982 |
Maryanoff BE, Simon EJ, Gioannini T, Gorissen H. Potential affinity labels for the opiate receptor based on fentanyl and related compounds. Journal of Medicinal Chemistry. 25: 913-919. PMID 6288945 DOI: 10.1021/Jm00350A006 |
0.432 |
|
| 1982 |
Gioannini T, Foucaud B, Hiller JM, Hatten ME, Simon EJ. Lectin binding of solubilized opiate receptors: evidence for their glycoprotein nature. Biochemical and Biophysical Research Communications. 105: 1128-34. PMID 6284164 DOI: 10.1016/0006-291X(82)91087-7 |
0.445 |
|
| 1982 |
Rüegg UT, Cuénoud S, Fulpius BW, Simon EJ. Inactivation and solubilization of opiate receptors by phospholipases A2. Biochimica Et Biophysica Acta. 685: 241-248. PMID 6279149 DOI: 10.1016/0005-2736(82)90063-3 |
0.383 |
|
| 1982 |
Monferini E, Adler MW, Simon EJ. Binding characteristics of mu and kappa agonists in rat brain subcellular fractions. Life Sciences. 31: 1295-8. PMID 6128655 DOI: 10.1016/0024-3205(82)90365-4 |
0.369 |
|
| 1982 |
Simon EJ. Opiate Receptors and Endorphins Advances in Alcohol and Substance Abuse. 1: 13-31. DOI: 10.1300/J251V01N01_03 |
0.464 |
|
| 1981 |
Hiller J, Angel L, Simon E. Multiple opiate receptors: alcohol selectively inhibits binding to delta receptors. Science. 214: 468-469. PMID 6270788 DOI: 10.1126/Science.6270788 |
0.388 |
|
| 1981 |
Ruegg UT, Cuenod S, Hiller JM, Gioannini T, Howells RD, Simon EJ. Characterization and partial purification of solubilized active opiate receptors from toad brain. Proceedings of the National Academy of Sciences of the United States of America. 78: 4635-4638. PMID 6270689 DOI: 10.1073/Pnas.78.7.4635 |
0.419 |
|
| 1981 |
Bonnet KA, Groth J, Gioannini T, Cortes M, Simon EJ. Opiate receptor heterogeneity in human brain regions. Brain Research. 221: 437-440. PMID 6269694 DOI: 10.1016/0006-8993(81)90797-6 |
0.424 |
|
| 1981 |
Simon LD, Simon FR, Mohasci E, Berger L, Simon EJ. Effect of the position of the phenolic group in morphinans on their affinity for oplate receptor binding Life Sciences. 28: 2769-2772. PMID 6267396 DOI: 10.1016/0024-3205(81)90179-X |
0.346 |
|
| 1981 |
Simon EJ. Opiate receptors: some recent developments Trends in Pharmacological Sciences. 2: 155-158. DOI: 10.1016/0165-6147(81)90296-0 |
0.437 |
|
| 1980 |
Howells RD, Simon EJ. Benzodiazepine binding in chicken retina and its interaction with γ-aminobutyric acid European Journal of Pharmacology. 67: 133-137. PMID 7418728 DOI: 10.1016/0014-2999(80)90021-7 |
0.316 |
|
| 1980 |
Pearson J, Brandeis L, Simon E, Hiller J. Radioautography of binding of tritiated diprenorphine to opiate receptors in the rat. Life Sciences. 26: 1047-1052. PMID 6248701 DOI: 10.1016/0024-3205(80)90250-7 |
0.425 |
|
| 1980 |
Rüegg UT, Hiller JM, Simon EJ. Solubilization of an active opiate receptor from Bufo marinus. European Journal of Pharmacology. 64: 367-368. PMID 6248353 DOI: 10.1016/0014-2999(80)90247-2 |
0.375 |
|
| 1980 |
Smith JR, Simon EJ. Selective protection of stereospecific enkephalin and opiate binding against inactivation by N-ethylmaleimide: evidence for two classes of opiate receptors. Proceedings of the National Academy of Sciences of the United States of America. 77: 281-284. PMID 6244551 DOI: 10.1073/Pnas.77.1.281 |
0.412 |
|
| 1979 |
Howells RD, Hiller JM, Simon EJ. Benzodiazepine binding sites are present in retina. Life Sciences. 25: 2131-2136. PMID 537471 DOI: 10.1016/0024-3205(79)90207-8 |
0.379 |
|
| 1979 |
Crain SM, Crain B, Finnigan T, Simon EJ. Development of tolerance to opiates and opioid peptides in organotypic cultures of mouse spinal cord Life Sciences. 25: 1797-1802. PMID 529987 DOI: 10.1016/0024-3205(79)90426-0 |
0.376 |
|
| 1979 |
Hiller JM, Simon EJ. 3H-ethylketocyclazocine binding: Lack of evidence for a separate κ receptor in rats CNS European Journal of Pharmacology. 60: 389-390. PMID 230985 DOI: 10.1016/0014-2999(79)90249-8 |
0.402 |
|
| 1979 |
Simon EJ, Bonnet KA, Hiller JM, Rieman MW, Merrifield RB. Opioid activity of synthetic and naturally occurring enkephalin peptides. Biochemical Pharmacology. 28: 3333-7. PMID 230849 DOI: 10.1016/0006-2952(79)90129-1 |
0.319 |
|
| 1978 |
Persky-Brosh S, Young JR, Holland MJ, Simon EJ. Effect of morphine analogues on chemotaxis in Escherichia coli. Journal of General Microbiology. 107: 53-8. PMID 366075 DOI: 10.1099/00221287-107-1-53 |
0.387 |
|
| 1978 |
Crain SM, Crain B, Peterson ER, Simon EJ. Selective depression by opioid peptides of sensory-evoked dorsal-horn network responses in organized spinal cord cultures. Brain Research. 157: 196-201. PMID 212165 DOI: 10.1016/0006-8993(78)91014-4 |
0.309 |
|
| 1978 |
Simon EJ, Hiller JM. The opiate receptors. Annual Review of Pharmacology and Toxicology. 18: 371-394. PMID 206194 DOI: 10.1146/Annurev.Pa.18.040178.002103 |
0.423 |
|
| 1978 |
Lin H, Simon EJ. Phospholipase A inhibition of opiate receptor binding can be reversed by albumin Nature. 271: 383-384. PMID 202879 DOI: 10.1038/271383A0 |
0.428 |
|
| 1977 |
Stahl KD, Bever WV, Janssen P, Simon EJ. Receptor affinity and pharmacological potency of a series of narcotic analgesic, anti-diarrheal and neuroleptic drugs. European Journal of Pharmacology. 46: 199-205. PMID 22440 DOI: 10.1016/0014-2999(77)90334-X |
0.446 |
|
| 1976 |
Simon EJ. The opiate receptors. Neurochemical Research. 1: 3-28. PMID 24271240 DOI: 10.1007/Bf00965627 |
0.39 |
|
| 1976 |
Clendeninn NJ, Petraitis M, Simon EJ. Ontological development of opiate receptors in rodent brain. Brain Research. 118: 157-160. PMID 186159 DOI: 10.1016/0006-8993(76)90852-0 |
0.378 |
|
| 1975 |
Simon EJ, Hiller JM, Edelman I. Solubilization of a stereospecific opiate-macromolecular complex from rat brain Science. 190: 389-390. PMID 1182043 DOI: 10.1126/Science.1182043 |
0.365 |
|
| 1975 |
Simon EJ, Hiller JM, Edelman I, Groth J, Stahl KD. Opiate receptors and their interactions with agonists and antagonists Life Sciences. 16: 1795-1800. PMID 1152605 DOI: 10.1016/0024-3205(75)90277-5 |
0.449 |
|
| 1975 |
Simon EJ, Groth J. Kinetics of opiate receptor inactivation by sulfhydryl reagents: evidence for conformational change in presence of sodium ions Proceedings of the National Academy of Sciences of the United States of America. 72: 2404-2407. PMID 1056036 DOI: 10.1073/Pnas.72.6.2404 |
0.411 |
|
| 1973 |
Simon EJ. In search of the opiate receptor American Journal of the Medical Sciences. 266: 160-168. PMID 4583407 DOI: 10.1097/00000441-197309000-00001 |
0.446 |
|
| 1973 |
Simon EJ, Hiller JM, Edelman I. Stereospecific binding of the potent narcotic analgesic (3H) Etorphine to rat-brain homogenate. Proceedings of the National Academy of Sciences of the United States of America. 70: 1947-1949. PMID 4516196 DOI: 10.1073/Pnas.70.7.1947 |
0.429 |
|
| 1972 |
Simon EJ, Dole WP, Hiller JM. Coupling of a New, Active Morphine Derivative to Sepharose for Affinity Chromatography Proceedings of the National Academy of Sciences of the United States of America. 69: 1835-1837. PMID 4505662 DOI: 10.1073/Pnas.69.7.1835 |
0.449 |
|
| 1971 |
Wurster N, Elsbach P, Simon EJ, Pettis P, Lebow S. The effects of the morphine analogue levorphanol on leukocytes: Metabolic effects at rest and during phagocytosis Journal of Clinical Investigation. 50: 1091-1099. PMID 4928264 DOI: 10.1172/Jci106580 |
0.329 |
|
| 1966 |
Praag DV, Simon EJ. Studies on the intracellular distribution and tissue binding of dihydromorphine-7,8-H3 in the rat. Experimental Biology and Medicine. 122: 6-11. PMID 5944896 DOI: 10.3181/00379727-122-31036 |
0.385 |
|
| 1964 |
Simon EJ. Inhibition Of Bacterial Growth By Drugs Of The Morphine Series. Science. 144: 543-544. PMID 14194101 DOI: 10.1126/Science.144.3618.543 |
0.314 |
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