Year |
Citation |
Score |
2021 |
Estrada CD, Ang HT, Vetter KM, Ponich AA, Hall DG. Enantioselective Desymmetrization of 2-Aryl-1,3-propanediols by Direct -Alkylation with a Rationally Designed Chiral Hemiboronic Acid Catalyst That Mitigates Substrate Conformational Poisoning. Journal of the American Chemical Society. PMID 33719442 DOI: 10.1021/jacs.1c00759 |
0.318 |
|
2020 |
Hackney HE, Paladino M, Fu H, Hall DG. Diazaboryl-Naphthyl-Ketone: a New Scaffold with Bright Fluorescence, Aggregation-Induced Emission, and Application in the Quantitation of Trace Boronic Acids in Pharma Intemediates. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 32681577 DOI: 10.1002/Chem.202003248 |
0.361 |
|
2020 |
Bhangu J, Whittal RM, Hall DG. Design, synthesis and structure of a frustrated benzoxaborole and its applications in the complexation of amines, amino acids, and protein modification. Organic & Biomolecular Chemistry. PMID 32338262 DOI: 10.1039/D0Ob00572J |
0.447 |
|
2020 |
Li X, Hall DG. Stereodivergent Asymmetric Synthesis of α,β-Disubstituted β Aminoalkylboronic Acid Derivatives via Group-Selective Protodeboronation Enabling Access to the Elusive anti Isomer. Journal of the American Chemical Society. PMID 32320234 DOI: 10.1021/Jacs.0C03207 |
0.367 |
|
2020 |
Li X, Hall DG. Synthesis and Applications of β Aminoalkylboronic Acid Derivatives Advanced Synthesis & Catalysis. DOI: 10.1002/Adsc.202000690 |
0.379 |
|
2020 |
Clement HA, Hall DG. Recent Advances in the Stereoselective Additions of Allylic Boronates to Carbonyl Compounds Patai's Chemistry of Functional Groups. 1-86. DOI: 10.1002/9780470682531.Pat0968 |
0.326 |
|
2019 |
Clement HA, Boghi M, McDonald RM, Bernier L, Coe JW, Farrell W, Helal CJ, Reese MR, Sach NW, Lee JC, Hall DG. High-Throughput Ligand Screening Enables the Enantioselective Conjugate Borylation of Cyclobutenones to Access Synthetically Versatile Tertiary Cyclobutylboronates. Angewandte Chemie (International Ed. in English). PMID 31591755 DOI: 10.1002/Anie.201909308 |
0.607 |
|
2019 |
Ang HT, Rygus JPG, Hall DG. Two-component boronic acid catalysis for increased reactivity in challenging Friedel-Crafts alkylations with deactivated benzylic alcohols. Organic & Biomolecular Chemistry. PMID 31166346 DOI: 10.1039/C9Ob01043B |
0.385 |
|
2019 |
Hall DG. Boronic acid catalysis. Chemical Society Reviews. PMID 31089632 DOI: 10.1039/C9Cs00191C |
0.454 |
|
2019 |
Tailor J, Hall DG. Tandem Aza Organic Letters. 2: 3715-8. PMID 11073683 DOI: 10.1021/Ol006626B |
0.421 |
|
2019 |
Wu D, Wang W, Diaz-Dussan D, Peng Y, Chen Y, Narain R, Hall DG. In Situ Forming, Dual-Crosslink Network, Self-Healing Hydrogel Enabled by a Bioorthogonal Nopoldiol–Benzoxaborolate Click Reaction with a Wide pH Range Chemistry of Materials. 31: 4092-4102. DOI: 10.1021/Acs.Chemmater.9B00769 |
0.338 |
|
2018 |
Li X, Hall DG. Diastereocontrolled Monoprotodeboronation of β-Sulfinimido gem-Bis(boronates): A General and Stereoselective Access to α,β-Disubstituted β-Aminoalkylboronates. Angewandte Chemie (International Ed. in English). PMID 29932490 DOI: 10.1002/Anie.201804277 |
0.37 |
|
2018 |
Hall DG, Akgun B. Boronic Acids as Bioorthogonal Probes in Site-Selective Labeling of Proteins. Angewandte Chemie (International Ed. in English). PMID 29723444 DOI: 10.1002/Anie.201712611 |
0.41 |
|
2018 |
Mo X, Morgan TDR, Ang HT, Hall DG. Scope and Mechanism of a True Organocatalytic Beckmann Rear-rangement with a Boronic Acid / Perfluoropinacol System under Ambient Conditions. Journal of the American Chemical Society. PMID 29565116 DOI: 10.1021/Jacs.8B01618 |
0.472 |
|
2018 |
Clement HA, Hall DG. Synthesis of α-hydroxyalkyl dehydroazepanes via catalytic enantioselective borylative migration of an enol nonaflate Tetrahedron Letters. 59: 4334-4339. DOI: 10.1016/J.Tetlet.2018.10.053 |
0.454 |
|
2017 |
Akgun B, Li C, Hao Y, Lambkin G, Derda R, Hall DG. Synergic 'Click' Boronate/Thiosemicarbazone System for Fast and Irreversible Bioorthogonal Conjugation in Live Cells. Journal of the American Chemical Society. PMID 28891646 DOI: 10.1021/Jacs.7B08693 |
0.406 |
|
2017 |
Verdelet T, Ward RM, Hall DG. Direct Sulfonamidation of Primary and Secondary Benzylic Alcohols Catalyzed by a Boronic Acid/Oxalic Acid System European Journal of Organic Chemistry. 2017: 5729-5738. DOI: 10.1002/Ejoc.201700621 |
0.42 |
|
2016 |
Vshyvenko S, Clapson ML, Suzuki I, Hall DG. Characterization of the Dynamic Equilibrium between Closed and Open Forms of the Benzoxaborole Pharmacophore. Acs Medicinal Chemistry Letters. 7: 1097-1101. PMID 27994745 DOI: 10.1021/Acsmedchemlett.6B00300 |
0.33 |
|
2016 |
Hall DG, Rybak T, Verdelet T. Multicomponent Hetero-[4 + 2] Cycloaddition/Allylboration Reaction: From Natural Product Synthesis to Drug Discovery. Accounts of Chemical Research. PMID 27753496 DOI: 10.1021/Acs.Accounts.6B00403 |
0.488 |
|
2016 |
Mo X, Hall DG. Dual Catalysis Using Boronic Acid and Chiral Amine: Acyclic Quaternary Carbons via Enantioselective Alkylation of Branched Aldehydes with Allylic Alcohols. Journal of the American Chemical Society. PMID 27518200 DOI: 10.1021/Jacs.6B06101 |
0.414 |
|
2016 |
Kim YR, Hall DG. Optimization and multigram scalability of a catalytic enantioselective borylative migration for the synthesis of functionalized chiral piperidines. Organic & Biomolecular Chemistry. PMID 27143333 DOI: 10.1039/C6Ob00685J |
0.429 |
|
2016 |
Akgun B, Hall DG. Fast and Tight Boronate Formation for Click Bioorthogonal Conjugation. Angewandte Chemie (International Ed. in English). PMID 26913832 DOI: 10.1002/Anie.201510321 |
0.358 |
|
2015 |
Rybak T, Hall DG. Stereoselective and Regiodivergent Allylic Suzuki-Miyaura Cross-Coupling of 2-Ethoxydihydropyranyl Boronates: Synthesis and Confirmation of Absolute Stereochemistry of Diospongin B. Organic Letters. 17: 4156-9. PMID 26291472 DOI: 10.1021/Acs.Orglett.5B01906 |
0.402 |
|
2015 |
Mo X, Yakiwchuk J, Dansereau J, McCubbin JA, Hall DG. Unsymmetrical Diarylmethanes by Ferroceniumboronic Acid Catalyzed Direct Friedel-Crafts Reactions with Deactivated Benzylic Alcohols: Enhanced Reactivity due to Ion-Pairing Effects. Journal of the American Chemical Society. 137: 9694-703. PMID 26158198 DOI: 10.1021/Jacs.5B05076 |
0.436 |
|
2015 |
Lee JC, Sun HY, Hall DG. Optimization of Reaction and Substrate Activation in the Stereoselective Cross Coupling of Chiral 3,3-Diboronyl Amides. The Journal of Organic Chemistry. PMID 26090783 DOI: 10.1021/Acs.Joc.5B00991 |
0.573 |
|
2015 |
Sun HY, Kubota K, Hall DG. Reaction Optimization, Scalability, and Mechanistic Insight on the Catalytic Enantioselective Desymmetrization of 1,1-Diborylalkanes via Suzuki-Miyaura Cross-Coupling. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 25829225 DOI: 10.1002/Chem.201406680 |
0.416 |
|
2015 |
Ricardo CL, Mo X, McCubbin JA, Hall DG. A surprising substituent effect provides a superior boronic acid catalyst for mild and metal-free direct Friedel-Crafts alkylations and prenylations of neutral arenes. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 4218-23. PMID 25678266 DOI: 10.1002/Chem.201500020 |
0.404 |
|
2015 |
Fatemi S, Gernigon N, Hall DG. A multigram-scale lower E-factor procedure for MIBA-catalyzed direct amidation and its application to the coupling of alpha and beta aminoacids Green Chemistry. 17: 4016-4028. DOI: 10.1039/C5Gc00659G |
0.424 |
|
2014 |
Ding J, Rybak T, Hall DG. Synthesis of chiral heterocycles by ligand-controlled regiodivergent and enantiospecific Suzuki Miyaura cross-coupling. Nature Communications. 5: 5474. PMID 25403650 DOI: 10.1038/Ncomms6474 |
0.402 |
|
2014 |
Al-Zoubi RM, Hall DG. Catalytic enantioselective diversity-oriented synthesis of a small library of polyhydroxylated pyrans inspired from thiomarinol antibiotics. Molecular Diversity. 18: 701-19. PMID 25151273 DOI: 10.1007/S11030-014-9542-6 |
0.72 |
|
2014 |
Bhakta U, Sullivan E, Hall DG. Catalytic enantioselective allylboration of propargylic aldehydes Tetrahedron. 70: 678-683. DOI: 10.1016/J.Tet.2013.11.095 |
0.441 |
|
2014 |
Elford TG, Hall DG. Total synthesis of chinensiolide B: An exercise in functional group selectivity with the help of a fortuitous side product and a good nose Strategies and Tactics in Organic Synthesis. 10: 79-112. DOI: 10.1016/B978-0-12-417185-5.00004-1 |
0.441 |
|
2013 |
Gao D, Sand R, Fu H, Sharmin N, Gallin WJ, Hall DG. Synthesis of the non-peptidic snail toxin 6-bromo-2-mercaptotryptamine dimer (BrMT)(2), its lower and higher thio homologs and their ability to modulate potassium ion channels. Bioorganic & Medicinal Chemistry Letters. 23: 5503-6. PMID 24021461 DOI: 10.1016/J.Bmcl.2013.08.070 |
0.319 |
|
2013 |
Ding J, Hall DG. Concise synthesis and antimalarial activity of all four mefloquine stereoisomers using a highly enantioselective catalytic borylative alkene isomerization. Angewandte Chemie (International Ed. in English). 52: 8069-73. PMID 23818420 DOI: 10.1002/Anie.201303931 |
0.415 |
|
2013 |
Gernigon N, Zheng H, Hall DG. Solid-supported ortho-iodoarylboronic acid catalyst for direct amidation of carboxylic acids Tetrahedron Letters. 54: 4475-4478. DOI: 10.1016/J.Tetlet.2013.06.043 |
0.595 |
|
2013 |
Zheng H, Lejkowski M, Hall DG. Mild boronic acid catalyzed Nazarov cyclization of divinyl alcohols in tandem with Diels-Alder cycloaddition Tetrahedron Letters. 54: 91-94. DOI: 10.1016/J.Tetlet.2012.10.100 |
0.591 |
|
2012 |
Tomsho JW, Pal A, Hall DG, Benkovic SJ. Ring Structure and Aromatic Substituent Effects on the pK a of the Benzoxaborole Pharmacophore. Acs Medicinal Chemistry Letters. 3: 48-52. PMID 24900370 DOI: 10.1021/Ml200215J |
0.342 |
|
2012 |
Gernigon N, Al-Zoubi RM, Hall DG. Direct amidation of carboxylic acids catalyzed by ortho-iodo arylboronic acids: catalyst optimization, scope, and preliminary mechanistic study supporting a peculiar halogen acceleration effect. The Journal of Organic Chemistry. 77: 8386-400. PMID 23013456 DOI: 10.1021/Jo3013258 |
0.705 |
|
2012 |
Ding J, Lee JC, Hall DG. Stereoselective preparation of β-aryl-β-boronyl enoates and their copper-catalyzed enantioselective conjugate reduction. Organic Letters. 14: 4462-5. PMID 22894652 DOI: 10.1021/Ol301958X |
0.59 |
|
2012 |
Zheng H, Ghanbari S, Nakamura S, Hall DG. Boronic acid catalysis as a mild and versatile strategy for direct carbo- and heterocyclizations of free allylic alcohols. Angewandte Chemie (International Ed. in English). 51: 6187-90. PMID 22589004 DOI: 10.1002/Anie.201201620 |
0.543 |
|
2012 |
Hall DG, Lee JCH, Ding J. Catalytic enantioselective transformations of borylated substrates: Preparation and synthetic applications of chiral alkylboronates Pure and Applied Chemistry. 84: 2263-2277. DOI: 10.1351/Pac-Con-12-02-04 |
0.472 |
|
2012 |
Knochel P, Barl NM, Lee JCH, McDonald R, Hall DG. Enantioselective Preparation and Chemo-selective Coupling of 1,1-Diboronyls Synfacts. 8: 89-89. DOI: 10.1055/S-0031-1289469 |
0.329 |
|
2012 |
Ding J, Hall DG. Preparation of chiral secondary boronic esters via copper-catalyzed enantioselective conjugate reduction of β-boronyl-β-alkyl α,β-unsaturated esters Tetrahedron. 68: 3428-3434. DOI: 10.1016/J.Tet.2011.07.088 |
0.368 |
|
2012 |
Zilke L, Hall DG. Synthetic studies towards the core tricyclic ring system of pradimicin A European Journal of Organic Chemistry. 4153-4163. DOI: 10.1002/Ejoc.201200294 |
0.415 |
|
2011 |
Lee JC, McDonald R, Hall DG. Enantioselective preparation and chemoselective cross-coupling of 1,1-diboron compounds. Nature Chemistry. 3: 894-9. PMID 22024887 DOI: 10.1038/Nchem.1150 |
0.572 |
|
2011 |
Zheng H, Lejkowski M, Hall DG. Mild and selective boronic acid catalyzed 1,3-transposition of allylic alcohols and Meyer-Schuster rearrangement of propargylic alcohols Chemical Science. 2: 1305-1310. DOI: 10.1039/C1Sc00140J |
0.555 |
|
2011 |
Lee JCH, Hall DG. Gold-catalyzed cycloisomerization reactions of boronated enynes Tetrahedron Letters. 52: 321-324. DOI: 10.1016/J.Tetlet.2010.11.051 |
0.403 |
|
2010 |
Al-Zoubi RM, Hall DG. Mild silver(I)-mediated regioselective iodination and bromination of arylboronic acids. Organic Letters. 12: 2480-3. PMID 20450213 DOI: 10.1021/Ol100537X |
0.721 |
|
2010 |
Zheng H, McDonald R, Hall DG. Boronic acid catalysis for mild and selective [3+2] dipolar cycloadditions to unsaturated carboxylic acids. Chemistry (Weinheim An Der Bergstrasse, Germany). 16: 5454-60. PMID 20373314 DOI: 10.1002/Chem.200903484 |
0.61 |
|
2010 |
Lee JC, Hall DG. Chiral boronate derivatives via catalytic enantioselective conjugate addition of Grignard reagents on 3-boronyl unsaturated esters and thioesters. Journal of the American Chemical Society. 132: 5544-5. PMID 20355729 DOI: 10.1021/Ja9104057 |
0.631 |
|
2010 |
Lu JY, Hall DG. Fragmentation enables complexity in the first total synthesis of vinigrol. Angewandte Chemie (International Ed. in English). 49: 2286-8. PMID 20187053 DOI: 10.1002/Anie.200906826 |
0.335 |
|
2010 |
Mothana S, Grassot JM, Hall DG. Multistep phase-switch synthesis by using liquid-liquid partitioning of boronic acids: productive tags with an expanded repertoire of compatible reactions. Angewandte Chemie (International Ed. in English). 49: 2883-7. PMID 20146294 DOI: 10.1002/Anie.200906710 |
0.394 |
|
2010 |
Elford TG, Hall DG. Total synthesis of (+)-chinensiolide B via tandem allylboration/lactonization. Journal of the American Chemical Society. 132: 1488-9. PMID 20067261 DOI: 10.1021/Ja9104478 |
0.397 |
|
2010 |
Sivasubramaniam U, Hall DG. Stereoselective preparation of oxygenated heterocycles using stereocontrolled tandem double-allylation of carbonyl compounds with a boron-silicon reagent Heterocycles. 80: 1449-1456. DOI: 10.3987/Com-09-S(S)50 |
0.404 |
|
2010 |
Penner M, Rauniyar V, Kaspar LT, Hall DG. Asymmetric Synthesis of Palmerolide A Synfacts. 2010: 381-381. DOI: 10.1055/S-0029-1219448 |
0.409 |
|
2010 |
Elford TG, Hall DG. Advances in 2-(alkoxycarbonyl)allylboration of carbonyl compounds and other direct methods for the preparation of α-exo-alkylidene γ-lactones Synthesis. 893-907. DOI: 10.1055/S-0029-1218664 |
0.392 |
|
2010 |
Zheng H, Hall DG. Zirconium-catalyzed Nagata reaction for the synthesis of 2-aryl-1,3,2-aryldioxaborins via a mild three-component condensation of phenols, aldehydes, and boronic acid Tetrahedron Letters. 51: 4256-4259. DOI: 10.1016/J.Tetlet.2010.06.035 |
0.634 |
|
2010 |
Zheng H, Hall DG. Mild and efficient boronic acid catalysis of Diels-Alder cycloadditions to 2-alkynoic acids Tetrahedron Letters. 51: 3561-3564. DOI: 10.1016/J.Tetlet.2010.04.132 |
0.575 |
|
2010 |
DORY YL, HALL DG, DESLONGCHAMPS P. ChemInform Abstract: Mechanism of the Diels-Alder Reaction of Enal Dienophiles. Competitive Reactivity and ab initio Calculations Using a Transannular Probe. Cheminform. 30: no-no. DOI: 10.1002/chin.199903037 |
0.462 |
|
2010 |
DROUIN M, HALL DG, CAILLE A, DESLONGCHAMPS P. ChemInform Abstract: Unique trans-syn-cis [6.6.7] Tricycle Derivative from Transannular Diels-Alder Contraction of a Model 15-Membered trans-cis-cis Macrocyclic Triene. Cheminform. 29: no-no. DOI: 10.1002/chin.199807027 |
0.421 |
|
2010 |
HALL DG, SCHULTZ PG. ChemInform Abstract: Synthesis of Diverse Ethoxyformacetal Oligomers. Toward Libraries of Metal-Coordinating Unnatural Biopolymers. Cheminform. 29: no-no. DOI: 10.1002/chin.199806117 |
0.4 |
|
2010 |
HALL DG, MUELLER R, DESLONGCHAMPS P. ChemInform Abstract: Studies on the Transannular Diels-Alder Reaction of 15-Membered Macrocyclic Trienes Containing a trans-trans Diene. Part 2. Evidence for Unsymmetrical Transition States in the Formation of A.B.C.(6.6.7) Tricyclic Products. Cheminform. 27: no-no. DOI: 10.1002/chin.199618103 |
0.498 |
|
2010 |
HALL DG, MUELLER R, DESLONGCHAMPS P. ChemInform Abstract: Studies on the Transannular Diels-Alder Reaction of 15-Membered Macrocyclic Trienes Containing a trans-trans Diene. Part 1. Synthesis and Isomerization of Various Model Cyclopentadecatrienes. Cheminform. 27: no-no. DOI: 10.1002/chin.199618088 |
0.549 |
|
2010 |
HALL DG, CAILLE A, DROUIN M, LAMOTHE S, MUELLER R, DESLONGCHAMPS P. ChemInform Abstract: A Stereospecific Transannular Diels-Alder Approach to the (6.6.7) Tricyclic Skeleton Related to Aphidicolin and Scopadulan Natural Products. Cheminform. 27: no-no. DOI: 10.1002/chin.199602225 |
0.464 |
|
2010 |
HALL DG, CHAPDELAINE D, PREVILLE P, DESLONGCHAMPS P. ChemInform Abstract: Stereocontrolled Synthesis of Acyclic Tri- and Tetra-C-Substituted . alpha.-Alkoxymethyl α,β-Unsaturated Esters. Cheminform. 25: no-no. DOI: 10.1002/chin.199451111 |
0.773 |
|
2010 |
HALL DG, MUELLER R, DESLONGCHAMPS P. ChemInform Abstract: Transannular Diels-Alder Reaction of Trans-Trans-Trans 15-Membered Macrocyclic Trienes (I), (IV). Cheminform. 24: no-no. DOI: 10.1002/chin.199303081 |
0.504 |
|
2009 |
Penner M, Rauniyar V, Kaspar LT, Hall DG. Catalytic asymmetric synthesis of palmerolide A via organoboron methodology. Journal of the American Chemical Society. 131: 14216-7. PMID 19764721 DOI: 10.1021/Ja906429C |
0.777 |
|
2009 |
Lessard S, Peng F, Hall DG. Alpha-hydroxyalkyl heterocycles via chiral allylic boronates: Pd-catalyzed borylation leading to a formal enantioselective isomerization of allylic ether and amine. Journal of the American Chemical Society. 131: 9612-3. PMID 19552416 DOI: 10.1021/Ja903946F |
0.442 |
|
2009 |
Touré BB, Hall DG. Natural product synthesis using multicomponent reaction strategies. Chemical Reviews. 109: 4439-86. PMID 19480390 DOI: 10.1021/Cr800296P |
0.402 |
|
2009 |
Rauniyar V, Hall DG. Rationally improved chiral Brønsted acid for catalytic enantioselective allylboration of aldehydes with an expanded reagent scope. The Journal of Organic Chemistry. 74: 4236-41. PMID 19422213 DOI: 10.1021/Jo900553F |
0.466 |
|
2009 |
Elford TG, Ulaczyk-Lesanko A, De Pascale G, Wright GD, Hall DG. Diversity-oriented synthesis and preliminary biological screening of highly substituted five-membered lactones and lactams originating from an allyboration of aldehydes and imines. Journal of Combinatorial Chemistry. 11: 155-68. PMID 19072614 DOI: 10.1021/Cc8001487 |
0.351 |
|
2009 |
Marion O, Gao X, Marcus S, Hall DG. Synthesis and preliminary antibacterial evaluation of simplified thiomarinol analogs. Bioorganic & Medicinal Chemistry. 17: 1006-17. PMID 18234501 DOI: 10.1016/J.Bmc.2008.01.001 |
0.361 |
|
2009 |
Lachance H, Hall DG. Allylboration of Carbonyl Compounds Organic Reactions. DOI: 10.1002/0471264180.Or073.01 |
0.469 |
|
2008 |
Bérubé M, Dowlut M, Hall DG. Benzoboroxoles as efficient glycopyranoside-binding agents in physiological conditions: structure and selectivity of complex formation. The Journal of Organic Chemistry. 73: 6471-9. PMID 18549270 DOI: 10.1021/Jo800788S |
0.317 |
|
2008 |
Rauniyar V, Zhai H, Hall DG. Catalytic enantioselective allyl- and crotylboration of aldehydes using chiral diol x SnCl4 complexes. optimization, substrate scope and mechanistic investigations. Journal of the American Chemical Society. 130: 8481-90. PMID 18540580 DOI: 10.1021/Ja8016076 |
0.429 |
|
2008 |
Al-Zoubi RM, Marion O, Hall DG. Direct and waste-free amidations and cycloadditions by organocatalytic activation of carboxylic acids at room temperature. Angewandte Chemie (International Ed. in English). 47: 2876-9. PMID 18324651 DOI: 10.1002/Anie.200705468 |
0.66 |
|
2008 |
Hall DG. New preparative methods for allylic boronates and their application in stereoselective catalytic allylborations Pure and Applied Chemistry. 80: 913-927. DOI: 10.1351/Pac200880050913 |
0.49 |
|
2008 |
Rauniyar V, Zhai H, Hall DG. Convenient preparation of cycloalkenyl boronic acid pinacol esters Synthetic Communications. 38: 3984-3995. DOI: 10.1080/00397910802245762 |
0.458 |
|
2008 |
Elford TG, Hall DG. Imine allylation using 2-alkoxycarbonyl allylboronates as an expedient three-component reaction to polysubstituted α-exo-methylene-γ-lactams Tetrahedron Letters. 49: 6995-6998. DOI: 10.1016/J.Tetlet.2008.09.112 |
0.41 |
|
2008 |
Lachance H, Marion O, Hall DG. Synthetic studies toward the pyran core and the amide side chain of psymberin Tetrahedron Letters. 49: 6061-6064. DOI: 10.1016/J.Tetlet.2008.07.170 |
0.463 |
|
2007 |
Carosi L, Hall DG. Catalytic enantioselective preparation of alpha-substituted allylboronates: one-pot addition to functionalized aldehydes and a route to chiral allylic trifluoroborate reagents. Angewandte Chemie (International Ed. in English). 46: 5913-5. PMID 17579908 DOI: 10.1002/Anie.200700975 |
0.398 |
|
2007 |
Ulaczyk-Lesanko A, Pelletier E, Lee M, Prinz H, Waldmann H, Hall DG. Optimization of three- and four-component reactions for polysubstituted piperidines: application to the synthesis and preliminary biological screening of a prototype library. Journal of Combinatorial Chemistry. 9: 695-703. PMID 17521171 DOI: 10.1021/Cc0700344 |
0.398 |
|
2007 |
Mothana S, Chahal N, Vanneste S, Hall DG. Phase-switch synthesis with boronic acids as productive tags. Journal of Combinatorial Chemistry. 9: 193-6. PMID 17348725 DOI: 10.1021/Cc060149S |
0.379 |
|
2007 |
Peng F, Hall DG. Simple, stable, and versatile double-allylation reagents for the stereoselective preparation of skeletally diverse compounds. Journal of the American Chemical Society. 129: 3070-1. PMID 17315879 DOI: 10.1021/Ja068985T |
0.434 |
|
2007 |
Elford TG, Arimura Y, Yu SH, Hall DG. Triflic acid-catalyzed additions of 2-alkoxycarbonyl allylboronates to aldehydes. Study of scope and mechanistic investigation of the reaction stereochemistry. The Journal of Organic Chemistry. 72: 1276-84. PMID 17288375 DOI: 10.1021/Jo062151B |
0.432 |
|
2007 |
Manku S, Hall DG. Synthesis, decoding, and preliminary screening of a bead-supported split-pool library of triboronic acid receptors for complex oligosaccharides Australian Journal of Chemistry. 60: 824-828. DOI: 10.1071/Ch07263 |
0.766 |
|
2007 |
Rauniyar V, Hall DG. Preparation of a C2-symmetric binol-derived diol and its application in the catalytic enantioselective and catalyst-controlled diastereoselective allylboration of aldehydes Synthesis. 3421-3426. DOI: 10.1055/S-2007-983832 |
0.444 |
|
2007 |
Hall DG. Lewis and Brønsted acid catalyzed allylboration of carbonyl compounds: From discovery to mechanism and applications Synlett. 1644-1655. DOI: 10.1055/S-2007-980384 |
0.476 |
|
2007 |
Peng F, Hall DG. Preparation of α-substituted allylboronates by chemoselective iridium-catalyzed asymmetric allylic alkylation of 1-propenylboronates Tetrahedron Letters. 48: 3305-3309. DOI: 10.1016/J.Tetlet.2007.02.124 |
0.453 |
|
2006 |
Manku S, Hall DG. Screening of a combinatorial library of synthetic polyamines displaying selectivity in multiple ion-pairing interactions with model polyanionic compounds in aqueous organic solutions. Journal of Combinatorial Chemistry. 8: 551-61. PMID 16827568 DOI: 10.1021/Cc0501559 |
0.741 |
|
2006 |
Dowlut M, Hall DG. An improved class of sugar-binding boronic acids, soluble and capable of complexing glycosides in neutral water. Journal of the American Chemical Society. 128: 4226-7. PMID 16568987 DOI: 10.1021/Ja057798C |
0.356 |
|
2006 |
Rauniyar V, Hall DG. Catalytic enantioselective and catalyst-controlled diastereofacial-selective additions of allyl- and crotylboronates to aldehydes using chiral Brønsted acids. Angewandte Chemie (International Ed. in English). 45: 2426-8. PMID 16526087 DOI: 10.1002/Anie.200504432 |
0.384 |
|
2006 |
Gao X, Hall DG, Deligny M, Favre A, Carreaux F, Carboni B. Catalytic enantioselective three-component hetero-[4+2] cycloaddition/allylboration approach to alpha-hydroxyalkyl pyrans: scope, limitations, and mechanistic proposal. Chemistry (Weinheim An Der Bergstrasse, Germany). 12: 3132-42. PMID 16440389 DOI: 10.1002/Chem.200501197 |
0.422 |
|
2006 |
Hall D, Rauniyar V. Asymmetric Additions of Allyl- and Crotylboronates to Aldehydes Synfacts. 2006: 0697-0697. DOI: 10.1055/s-2006-941923 |
0.326 |
|
2006 |
Carosi L, Lachance H, Hall DG. Additions of Functionalized α-Substituted Allylboronates to Aldehydes under the Novel Lewis and Broensted Acid Catalyzed Manifolds. Cheminform. 37. DOI: 10.1002/chin.200615052 |
0.308 |
|
2005 |
Yu SH, Ferguson MJ, McDonald R, Hall DG. Brønsted acid-catalyzed allylboration: short and stereodivergent synthesis of all four eupomatilone diastereomers with crystallographic assignments. Journal of the American Chemical Society. 127: 12808-9. PMID 16159268 DOI: 10.1021/Ja054171L |
0.461 |
|
2005 |
Ulaczyk-Lesanko A, Hall DG. Wanted: new multicomponent reactions for generating libraries of polycyclic natural products. Current Opinion in Chemical Biology. 9: 266-76. PMID 15939328 DOI: 10.1016/J.Cbpa.2005.04.003 |
0.391 |
|
2005 |
Lachance H, St-Onge M, Hall DG. Practical and efficient multigram preparation of a camphor-derived diol for the enantioselective Lewis acid catalyzed allylboration of aldehydes. The Journal of Organic Chemistry. 70: 4180-3. PMID 15876115 DOI: 10.1021/Jo050207G |
0.471 |
|
2005 |
Gao X, Hall DG. Catalytic asymmetric synthesis of a potent thiomarinol antibiotic. Journal of the American Chemical Society. 127: 1628-9. PMID 15700983 DOI: 10.1021/Ja042827P |
0.42 |
|
2005 |
Gravel M, Toure BB, Hall DG. Practical Procedure for the Preparation of Functionalized (E)-1-Alkenylboronic Acids Including the Unprecedented 1-Alkoxycarbonyl Derivatives. Cheminform. 36. DOI: 10.1080/00304940409355974 |
0.735 |
|
2005 |
Hall D, Yu S, Ferguson M, McDonald R. Synthesis of Eupomatilone-6 Synfacts. 2006: 0010-0010. DOI: 10.1055/S-2005-921661 |
0.387 |
|
2005 |
Carosi L, Lachance H, Hall DG. Additions of functionalized α-substituted allylboronates to aldehydes under the novel Lewis and Brønsted acid catalyzed manifolds Tetrahedron Letters. 46: 8981-8985. DOI: 10.1016/J.Tetlet.2005.10.115 |
0.436 |
|
2005 |
Li D, Hall DG. Design and solid-phase synthesis of chiral acyclic and cyclic diamine ligands Tetrahedron: Asymmetry. 16: 1733-1736. DOI: 10.1016/J.Tetasy.2005.03.029 |
0.36 |
|
2005 |
Touré BB, Hall DG. Multicomponent Reactions in the Total Synthesis of Natural Products Multicomponent Reactions. 342-397. DOI: 10.1002/3527605118.ch12 |
0.679 |
|
2004 |
Touré BB, Hall DG. Design of a nonreductive method for chemoselective cleavage of hydrazines in the presence of unsaturations: application to a stereoconvergent three-component synthesis of (-)-methyl palustramate. The Journal of Organic Chemistry. 69: 8429-36. PMID 15549817 DOI: 10.1021/Jo048581O |
0.429 |
|
2004 |
Kennedy JW, Hall DG. Lewis acid catalyzed allylboration: discovery, optimization, and application to the formation of stereogenic quaternary carbon centers. The Journal of Organic Chemistry. 69: 4412-28. PMID 15202896 DOI: 10.1021/Jo049773M |
0.62 |
|
2004 |
Rauniyar V, Hall DG. Lewis acids catalyze the addition of allylboronates to aldehydes by electrophilic activation of the dioxaborolane in a closed transition structure. Journal of the American Chemical Society. 126: 4518-9. PMID 15070360 DOI: 10.1021/Ja049446W |
0.374 |
|
2004 |
Touré BB, Hall DG. Three-component sequential aza[4+2] cycloaddition/allylboration/retro-sulfinyl-ene reaction: a new stereocontrolled entry to palustrine alkaloids and other 2,6-disubstituted piperidines. Angewandte Chemie (International Ed. in English). 43: 2001-4. PMID 15065285 DOI: 10.1002/Anie.200353152 |
0.69 |
|
2004 |
Stones D, Manku S, Lu X, Hall DG. Modular solid-phase synthetic approach to optimize structural and electronic properties of oligoboronic acid receptors and sensors for the aqueous recognition of oligosaccharides. Chemistry (Weinheim An Der Bergstrasse, Germany). 10: 92-100. PMID 14695554 DOI: 10.1002/Chem.200305400 |
0.755 |
|
2004 |
Gravel M, Touré BB, Hall DG. PRACTICAL PROCEDURE FOR THE PREPARATION OF FUNCTIONALIZED (E)-1-ALKENYLBORONIC ACIDS INCLUDING THE UNPRECEDENTED 1-ALKOXYCARBONYL DERIVATIVES Organic Preparations and Procedures International. 36: 573-579. DOI: 10.1080/00304940409355974 |
0.646 |
|
2004 |
Hall DG, Gravel M, Lachance H, Lu X. Scope and Limitations of the Scandium-Catalyzed Enantioselective Addition of Chiral Allylboronates to Aldehydes Synthesis. 2004: 1290-1302. DOI: 10.1055/S-2004-822359 |
0.633 |
|
2004 |
Gravel M, Hall DG. DEAM-PS: Solid-Phase Chemistry for Boronic Acids Cheminform. 35. DOI: 10.1002/chin.200434284 |
0.532 |
|
2003 |
Kennedy JW, Hall DG. Recent advances in the activation of boron and silicon reagents for stereocontrolled allylation reactions. Angewandte Chemie (International Ed. in English). 42: 4732-9. PMID 14562340 DOI: 10.1002/Anie.200301632 |
0.61 |
|
2003 |
Lachance H, Lu X, Gravel M, Hall DG. Scandium-catalyzed allylboration of aldehydes as a practical method for highly diastereo- and enantioselective construction of homoallylic alcohols. Journal of the American Chemical Society. 125: 10160-1. PMID 12926924 DOI: 10.1021/Ja036807J |
0.601 |
|
2003 |
Gao X, Hall DG. 3-Boronoacrolein as an exceptional heterodiene in the highly enantio- and diastereoselective Cr(III)-catalyzed three-component [4+2]/allylboration. Journal of the American Chemical Society. 125: 9308-9. PMID 12889956 DOI: 10.1021/Ja036368O |
0.416 |
|
2003 |
Zhu N, Hall DG. Effect of additives on the stereochemical integrity and reactivity of alpha-alkoxycarbonyl alkenylcopper intermediates. Optimal conditions for the synthesis of isomerically pure tetrasubstituted alkenes. The Journal of Organic Chemistry. 68: 6066-9. PMID 12868953 DOI: 10.1021/Jo034465U |
0.408 |
|
2003 |
Manku S, Wang F, Hall DG. Synthesis and high performance liquid chromatography/electrospray mass spectrometry single-bead decoding of split-pool structural libraries of polyamines supported on polystyrene and polystyrene/ethylene glycol resins. Journal of Combinatorial Chemistry. 5: 379-91. PMID 12857106 DOI: 10.1021/Cc0201142 |
0.778 |
|
2003 |
Touré BB, Hoveyda HR, Tailor J, Ulaczyk-Lesanko A, Hall DG. A three-component reaction for diversity-oriented synthesis of polysubstituted piperidines: solution and solid-phase optimization of the first tandem aza[4+2]/allylboration. Chemistry (Weinheim An Der Bergstrasse, Germany). 9: 466-74. PMID 12532296 DOI: 10.1002/Chem.200390049 |
0.735 |
|
2003 |
Gao X, Hall DG. New Electronically Enriched Boronobutadienes for the Synthesis of Hydroxylated Cyclohexenes via Tandem [4 + 2]/Allylboration. Cheminform. 34. DOI: 10.1016/S0040-4039(03)00164-3 |
0.421 |
|
2003 |
Kennedy JW, Hall DG. Design of chiral boronate-substituted acrylanilides. Journal of Organometallic Chemistry. 680: 263-270. DOI: 10.1016/S0022-328X(03)00400-5 |
0.621 |
|
2002 |
Kennedy JW, Hall DG. Dramatic rate enhancement with preservation of stereospecificity in the first metal-catalyzed additions of allylboronates. Journal of the American Chemical Society. 124: 11586-7. PMID 12296710 DOI: 10.1021/Ja027453J |
0.62 |
|
2002 |
Kopac DS, Hall DG. General solid-phase approach to the synthesis of chiral triazacycloalkane ligands with stereogenic backbone substituents. Journal of Combinatorial Chemistry. 4: 251-4. PMID 12099840 DOI: 10.1021/Cc020015O |
0.372 |
|
2002 |
Kennedy JW, Hall DG. Novel isomerically pure tetrasubstituted allylboronates: stereocontrolled synthesis of alpha-exomethylene gamma-lactones as aldol-like adducts with a stereogenic quaternary carbon center. Journal of the American Chemical Society. 124: 898-9. PMID 11829585 DOI: 10.1021/Ja016391E |
0.582 |
|
2002 |
Gravel M, Thompson KA, Zak M, Bérubé C, Hall DG. Universal solid-phase approach for the immobilization, derivatization, and resin-to-resin transfer reactions of boronic acids. The Journal of Organic Chemistry. 67: 3-15. PMID 11777432 DOI: 10.1021/Jo0106501 |
0.651 |
|
2002 |
Manku S, Hall DG. Combinatorial approach to selective multivalent ion pairing in mixed aqueous-organic media using bead-supported libraries of unnatural polyamines. Organic Letters. 4: 31-4. PMID 11772083 DOI: 10.1021/Ol016827V |
0.732 |
|
2002 |
Kennedy JWJ, Hall DG. Self-Activation and 1,8-Stereoinduction in a Boronate-substituted Dienophile Synlett. 2002: 0477-0479. DOI: 10.1055/S-2002-20470 |
0.375 |
|
2001 |
Hoveyda HR, Hall DG. Solid-phase synthesis of cleavable N-arylmaleimides: applications in 1,3-dipolar cycloaddition and in thiol scavenging. Organic Letters. 3: 3491-4. PMID 11678690 DOI: 10.1021/Ol016533+ |
0.428 |
|
2001 |
Manku S, Laplante C, Kopac D, Chan T, Hall DG. A mild and general solid-phase method for the synthesis of chiral polyamines. Solution studies on the cleavage of borane-amine intermediates from the reduction of secondary amides. The Journal of Organic Chemistry. 66: 874-85. PMID 11430107 DOI: 10.1021/Jo005647G |
0.798 |
|
2001 |
Laplante C, Hall DG. Direct mono-N-methylation of solid-supported amino acids: a useful application of the Matteson rearrangement of alpha-aminoalkylboronic esters. Organic Letters. 3: 1487-90. PMID 11388848 DOI: 10.1021/Ol015803L |
0.409 |
|
2001 |
Hall DG, Manku S, Wang F. Solution- and solid-phase strategies for the design, synthesis, and screening of libraries based on natural product templates: a comprehensive survey. Journal of Combinatorial Chemistry. 3: 125-50. PMID 11300852 DOI: 10.1021/Cc0001001 |
0.752 |
|
2001 |
Hall DG. Organic Synthesis on Solid Phase. Supports, Linkers, Reactions By Florencio Zaragoza Dörwald (Novo Nordisk A/S MedChem Research, Malov, Denmark). Wiley-VCH: Weinheim. 2000. xx + 474 pp. DM 268 (approximately $125.00). ISBN 3-527-29950-5. Journal of the American Chemical Society. 123: 6463-6464. DOI: 10.1021/Ja004860R |
0.359 |
|
2001 |
Tailor J, Hall DG. ChemInform Abstract: Tandem Aza[4 + 2]/Allylboration: A Novel Multicomponent Reaction for the Stereocontrolled Synthesis of α-Hydroxyalkyl Piperidine Derivatives. Cheminform. 32: no-no. DOI: 10.1002/chin.200114159 |
0.324 |
|
2000 |
Wang F, Manku S, Hall DG. Solid phase syntheses of polyamine toxins HO-416b and PhTX-433. Use of an efficient polyamide reduction strategy that facilitates access to branched analogues. Organic Letters. 2: 1581-3. PMID 10841484 DOI: 10.1021/Ol005817B |
0.775 |
|
2000 |
Gravel M, Berube CD, Hall DG. Resin-to-resin suzuki coupling of solid supported arylboronic acids Journal of Combinatorial Chemistry. 2: 228-31. PMID 10827927 DOI: 10.1021/Cc990082R |
0.584 |
|
2000 |
Thompson KA, Hall DG. Resin-to-resin Petasis borono-Mannich reaction between dialkylamino resins and supported boronic acids Chemical Communications. 2379-2380. DOI: 10.1039/B006279K |
0.393 |
|
1999 |
Hall DG, Laplante C, Manku S, Nagendran J. Mild Oxidative Cleavage of Borane-Amine Adducts from Amide Reductions: Efficient Solution- and Solid-Phase Synthesis of N-Alkylamino Acids and Chiral Oligoamines. The Journal of Organic Chemistry. 64: 698-699. PMID 11674134 DOI: 10.1021/Jo982290W |
0.776 |
|
1999 |
Hall DG, Tailor J, Gravel M. N,N-Diethanolaminomethyl Polystyrene: An Efficient Solid Support to Immobilize Boronic Acids. Angewandte Chemie (International Ed. in English). 38: 3064-3067. PMID 10540423 DOI: 10.1002/(Sici)1521-3773(19991018)38:20<3064::Aid-Anie3064>3.0.Co;2-T |
0.609 |
|
1999 |
Conn MM, Kappock J, Drueckhammer D, Cammack R, Hall D, Cass T, Stewart JD, Cousins GR, Sanders JK, Flitsch S, Lowden PA, Newman R. Chemical biology Current Opinion in Chemical Biology. 3: 631-638. DOI: 10.1016/S1367-5931(99)00038-1 |
0.719 |
|
1999 |
Hall DG, Tailor J, Gravel M. N,N-Diethanolaminomethylpolystyrol: ein effizienter fester Träger für die Immobilisierung von Boronsäuren Angewandte Chemie. 111: 3250-3253. DOI: 10.1002/(Sici)1521-3757(19991018)111:20<3250::Aid-Ange3250>3.0.Co;2-V |
0.499 |
|
1998 |
Dory YL, Hall DG, Deslongchamps P. On the mechanism of the Diels-Alder reaction of enal dienophiles. Competitive reactivity and ab initio calculations using a transannular probe Tetrahedron. 54: 12279-12288. DOI: 10.1016/S0040-4020(98)00764-9 |
0.561 |
|
1997 |
Drouin M, Hall DG, Caillé A, Deslongchamps P. Uniquetrans-syn-cis[6.6.7] Tricycle Derivative from Transannular Diels–Alder Contraction of a Model 15-Memberedtrans-cis-cisMacrocyclic Triene Acta Crystallographica Section C Crystal Structure Communications. 53: 1490-1493. DOI: 10.1107/S0108270197005635 |
0.505 |
|
1997 |
Hall DG, Schultz PG. Synthesis of diverse ethoxyformacetal oligomers. Toward libraries of metal-coordinating unnatural biopolymers Tetrahedron Letters. 38: 7825-7828. DOI: 10.1016/S0040-4039(97)10094-6 |
0.505 |
|
1996 |
Hall DG, Deslongchamps P. Transannular Diels-Alder/Intramolecular Aldol Tandem Reaction as a Stereocontrolled Route to (+)-Aphidicolin and its Isosteric C8-Epimer. The Journal of Organic Chemistry. 61: 2914. PMID 11667138 DOI: 10.1021/Jo9640027 |
0.559 |
|
1995 |
Hall DG, Müller R, Deslongchamps P. Studies on the transannular Diels–Alder reaction of 15-membered macrocyclic trienes containing a trans-trans diene. Part II: Evidence for unsymmetrical transition states in the formation of A.B.C.[6.6.7] tricyclic products Canadian Journal of Chemistry. 73: 1695-1710. DOI: 10.1139/V95-208 |
0.597 |
|
1995 |
Hall DG, Müller R, Deslongchamps P. Studies on the transannular Diels–Alder reaction of 15-membered macrocyclic trienes containing a trans-trans diene. Part I: Synthesis and isomerization of various model cyclopentadecatrienes Canadian Journal of Chemistry. 73: 1675-1694. DOI: 10.1139/V95-207 |
0.597 |
|
1995 |
Hall DG, Caillé A, Drouin M, Lamothe S, Müller R, Deslongchamps P. A Stereospecific Transannular Diels-Alder Approach to the [6.6.7] Tricyclic Skeleton Related to Aphidicolin and Scopadulan Natural Products Synthesis. 1995: 1081-1088. DOI: 10.1055/S-1995-4077 |
0.511 |
|
1994 |
Hall DG, Chapdelaine D, Préville P, Deslongchamps P. Stereocontrolled Synthesis of Acyclic Tri- and Tetra-C-Substituted α-Alkoxymethyl α,β-Unsaturated Esters Synlett. 1994: 660-662. DOI: 10.1055/S-1994-22966 |
0.766 |
|
1992 |
Hall DG, Müller R, Deslongchamps P. Transannular diels-alder reaction of trans-trans-cis 15-membered macrocyclic trienes. Evidence for asynchronous transition state. Tetrahedron Letters. 33: 5221-5224. DOI: 10.1016/S0040-4039(00)79137-4 |
0.549 |
|
1992 |
Hall DG, Müller R, Deslongchamps P. Transannular diels-alder reaction of trans-trans-trans 15-membered macrocyclic trienes Tetrahedron Letters. 33: 5217-5220. DOI: 10.1016/S0040-4039(00)79136-2 |
0.57 |
|
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