Year |
Citation |
Score |
2016 |
Wagner FF, Weïwer M, Steinbacher S, Schomburg A, Reinemer P, Gale JP, Campbell AJ, Fisher SL, Zhao WN, Reis SA, Hennig KM, Thomas M, Müller P, Jefson MR, Fass DM, et al. Kinetic and structural insights into the binding of histone deacetylase 1 and 2 (HDAC1, 2) inhibitors. Bioorganic & Medicinal Chemistry. PMID 27377864 DOI: 10.1016/J.Bmc.2016.06.040 |
0.333 |
|
2015 |
Wagner FF, Zhang YL, Fass DM, Joseph N, Gale JP, Weïwer M, McCarren P, Fisher SL, Kaya T, Zhao WN, Reis SA, Hennig KM, Thomas M, Lemercier BC, Lewis MC, et al. Kinetically Selective Inhibitors of Histone Deacetylase 2 (HDAC2) as Cognition Enhancers. Chemical Science (Royal Society of Chemistry : 2010). 6: 804-815. PMID 25642316 DOI: 10.1039/C4Sc02130D |
0.311 |
|
2015 |
Benajiba L, Wagner F, Ross L, Galinsky I, DeAngelo DJ, Gale J, Pan J, Zhang Y, Sacher J, Weiwer M, Stone RM, Holson E, Stegmaier K. Identification of a First in Class GSK3-Alpha Selective Inhibitor As a New Differentiation Therapy for AML Blood. 126: 870-870. DOI: 10.1182/Blood.V126.23.870.870 |
0.35 |
|
2013 |
Olson DE, Wagner FF, Kaya T, Gale JP, Aidoud N, Davoine EL, Lazzaro F, Weïwer M, Zhang YL, Holson EB. Discovery of the first histone deacetylase 6/8 dual inhibitors. Journal of Medicinal Chemistry. 56: 4816-20. PMID 23672185 DOI: 10.1021/Jm400390R |
0.354 |
|
2013 |
Wagner FF, Olson DE, Gale JP, Kaya T, Weïwer M, Aidoud N, Thomas M, Davoine EL, Lemercier BC, Zhang YL, Holson EB. Potent and selective inhibition of histone deacetylase 6 (HDAC6) does not require a surface-binding motif. Journal of Medicinal Chemistry. 56: 1772-6. PMID 23368884 DOI: 10.1021/Jm301355J |
0.368 |
|
2012 |
Weïwer M, Spoonamore J, Wei J, Guichard B, Ross NT, Masson K, Silkworth W, Dandapani S, Palmer M, Scherer CA, Stern AM, Schreiber SL, Munoz B. A Potent and Selective Quinoxalinone-Based STK33 Inhibitor Does Not Show Synthetic Lethality in KRAS-Dependent Cells. Acs Medicinal Chemistry Letters. 3: 1034-1038. PMID 23256033 DOI: 10.1021/Ml300246R |
0.335 |
|
2012 |
Dockendorff C, Nagiec MM, Weïwer M, Buhrlage S, Ting A, Nag PP, Germain A, Kim HJ, Youngsaye W, Scherer C, Bennion M, Xue L, Stanton BZ, Lewis TA, Macpherson L, et al. Macrocyclic Hedgehog Pathway Inhibitors: Optimization of Cellular Activity and Mode of Action Studies. Acs Medicinal Chemistry Letters. 3: 808-813. PMID 23074541 DOI: 10.1021/Ml300172P |
0.349 |
|
2012 |
Heidebrecht RW, Mulrooney C, Austin CP, Barker RH, Beaudoin JA, Cheng KC, Comer E, Dandapani S, Dick J, Duvall JR, Ekland EH, Fidock DA, Fitzgerald ME, Foley M, Guha R, et al. Diversity-Oriented Synthesis Yields a Novel Lead for the Treatment of Malaria. Acs Medicinal Chemistry Letters. 3: 112-117. PMID 22328964 DOI: 10.1021/Ml200244K |
0.325 |
|
2012 |
Masuko S, Bera S, Green DE, Weïwer M, Liu J, Deangelis PL, Linhardt RJ. Chemoenzymatic synthesis of uridine diphosphate-GlcNAc and uridine diphosphate-GalNAc analogs for the preparation of unnatural glycosaminoglycans Journal of Organic Chemistry. 77: 1449-1456. PMID 22239739 DOI: 10.1021/Jo202322K |
0.663 |
|
2012 |
Kemp MM, Weïwer M, Koehler AN. Unbiased binding assays for discovering small-molecule probes and drugs. Bioorganic & Medicinal Chemistry. 20: 1979-89. PMID 22230199 DOI: 10.1016/J.Bmc.2011.11.071 |
0.6 |
|
2010 |
Liu R, Xu Y, Chen M, Weïwer M, Zhou X, Bridges AS, DeAngelis PL, Zhang Q, Linhardt RJ, Liu J. Chemoenzymatic design of heparan sulfate oligosaccharides. The Journal of Biological Chemistry. 285: 34240-9. PMID 20729556 DOI: 10.1074/Jbc.M110.159152 |
0.513 |
|
2009 |
Weïwer M, Chen CC, Kemp MM, Linhardt RJ. Synthesis and Biological Evaluation of Non-Hydrolizable 1,2,3-Triazole Linked Sialic Acid Derivatives as Neuraminidase Inhibitors. European Journal of Organic Chemistry. 2009. PMID 24223493 DOI: 10.1002/Ejoc.200900117 |
0.68 |
|
2009 |
Mora-Pale M, Weïwer M, Yu J, Linhardt RJ, Dordick JS. Inhibition of human vascular NADPH oxidase by apocynin derived oligophenols. Bioorganic & Medicinal Chemistry. 17: 5146-52. PMID 19523836 DOI: 10.1016/J.Bmc.2009.05.061 |
0.55 |
|
2009 |
Weïwer M, Chen C, Kemp MM, Linhardt RJ. Synthesis and Biological Evaluation of Non-Hydrolyzable 1,2,3-Triazole-Linked Sialic Acid Derivatives as Neuraminidase Inhibitors (Eur. J. Org. Chem. 16/2009) European Journal of Organic Chemistry. 2009: 2587-2587. DOI: 10.1002/Ejoc.200990041 |
0.668 |
|
2009 |
Weiwer M, Huang F, Chen C, Yuan X, Tokuzaki K, Tomiyama H, Linhardt RJ. ChemInform Abstract: Synthesis and Evaluation of Anticancer Vaccine Candidates: C-Glycoside Analogues of STn and PSA Cheminform. 40. DOI: 10.1002/chin.200934253 |
0.301 |
|
2009 |
Weiwer M, Sherwood T, Linhardt RJ. ChemInform Abstract: Synthesis of Floridoside. Cheminform. 40. DOI: 10.1002/chin.200920180 |
0.344 |
|
2008 |
Weïwer M, Sherwood T, Green DE, Chen M, DeAngelis PL, Liu J, Linhardt RJ. Synthesis of uridine 5'-diphosphoiduronic acid: a potential substrate for the chemoenzymatic synthesis of heparin. The Journal of Organic Chemistry. 73: 7631-7. PMID 18759479 DOI: 10.1021/Jo801409C |
0.576 |
|
2008 |
Zhang Z, Weïwer M, Li B, Kemp MM, Daman TH, Linhardt RJ. Oversulfated chondroitin sulfate: impact of a heparin impurity, associated with adverse clinical events, on low-molecular-weight heparin preparation. Journal of Medicinal Chemistry. 51: 5498-501. PMID 18754653 DOI: 10.1021/Jm800785T |
0.642 |
|
2008 |
Yu J, Weïwer M, Linhardt RJ, Dordick JS. The role of the methoxyphenol apocynin, a vascular NADPH oxidase inhibitor, as a chemopreventative agent in the potential treatment of cardiovascular diseases. Current Vascular Pharmacology. 6: 204-17. PMID 18673160 DOI: 10.2174/157016108784911984 |
0.559 |
|
2008 |
Weïwer M, Sherwood T, Linhardt RJ. Synthesis of Floridoside Journal of Carbohydrate Chemistry. 27: 420-427. DOI: 10.1080/07328300802408843 |
0.404 |
|
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