Year |
Citation |
Score |
2022 |
Quirke JCK, Sati GC, Sonousi A, Gysin M, Haldimann K, Bottger EC, Vasella A, Hobbie SN, Crich D. Structure-Activity Relationships for 5''-Modifications of 4,5-Aminoglycoside Antibiotics. Chemmedchem. PMID 35385605 DOI: 10.1002/cmdc.202200120 |
0.631 |
|
2021 |
Lubriks D, Zogota R, Sarpe VA, Matsushita T, Sati GC, Haldimann K, Gysin M, Böttger EC, Vasella A, Suna E, Hobbie SN, Crich D. Synthesis and Antibacterial Activity of Propylamycin Derivatives Functionalized at the 5''- and Other Positions with a View to Overcoming Resistance Due to Aminoglycoside Modifying Enzymes. Acs Infectious Diseases. PMID 34114793 DOI: 10.1021/acsinfecdis.1c00158 |
0.61 |
|
2019 |
Waduge P, Sati GC, Crich D, Chow CS. Use of a fluorescence assay to determine relative affinities of semisynthetic aminoglycosides to small RNAs representing bacterial and mitochondrial A sites. Bioorganic & Medicinal Chemistry. 115121. PMID 31610941 DOI: 10.1016/J.Bmc.2019.115121 |
0.422 |
|
2019 |
Sati GC, Sarpe VA, Furukawa T, Mondal S, Mantovani M, Hobbie SN, Vasella A, Böttger EC, Crich D. Modification at the 2'-Position of the 4,5-Series of 2-Deoxystreptamine Aminoglycoside Antibiotics to Resist Aminoglycoside Modifying Enzymes and Increase Ribosomal Target Selectivity. Acs Infectious Diseases. PMID 31436080 DOI: 10.1021/Acsinfecdis.9B00128 |
0.61 |
|
2019 |
Matsushita T, Sati G, Kondasinghe N, Pirrone M, Kato T, Waduge P, Kumar H, Sanchon A, Dobosz-Bartoszek M, Shcherbakov D, Juhas M, Hobbie SN, Schrepfer T, Chow CS, Polikanov Y, et al. Design, Multigram Synthesis, and in Vitro and in Vivo Evaluation of Propylamycin: A Semisynthetic 4,5-Deoxystreptamine Class Aminoglycoside for the Treatment of Drug-Resistant Enterobacteriaceae and Other Gram-Negative Pathogens. Journal of the American Chemical Society. PMID 30793894 DOI: 10.1021/jacs.9b01693 |
0.615 |
|
2018 |
Anneken JH, Angoa-Perez M, Sati GC, Crich D, Kuhn DM. Dissociation between hypothermia and neurotoxicity caused by mephedrone and methcathinone in TPH2 knockout mice. Psychopharmacology. PMID 30074064 DOI: 10.1007/S00213-018-4991-8 |
0.339 |
|
2017 |
Anneken JH, Angoa-Perez M, Sati GC, Crich D, Kuhn DM. Assessing the role of dopamine in the differential neurotoxicity patterns of methamphetamine, mephedrone, methcathinone and 4-methylmethamphetamine. Neuropharmacology. PMID 28851615 DOI: 10.1016/J.Neuropharm.2017.08.033 |
0.384 |
|
2017 |
Sati GC, Scherbakov D, Hobbie SN, Vasella A, Böttger EC, Crich D. N6', N6''' and O4' Modifications to Neomycin Affect Ribosomal Selectivity Without Compromising Antibacterial Activity. Acs Infectious Diseases. PMID 28343384 DOI: 10.1021/Acsinfecdis.6B00214 |
0.548 |
|
2016 |
Anneken JH, Angoa-Perez M, Sati GC, Crich D, Kuhn DM. Dissecting the influence of two structural substituents on the differential neurotoxic effects of methamphetamine and mephedrone on dopamine nerve endings with the use of 4-methylmethamphetamine and methcathinone. The Journal of Pharmacology and Experimental Therapeutics. PMID 28039330 DOI: 10.1124/Jpet.116.237768 |
0.424 |
|
2015 |
Sati GC, Crich D. Facile Synthesis of 3-N-Alkyl Pyrimidin-2,4-diones from N-Sulfonyloxy Maleimides and Amines. Organic Letters. 17: 4122-4. PMID 26267613 DOI: 10.1021/acs.orglett.5b02079 |
0.371 |
|
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