| Year |
Citation |
Score |
| 2020 |
Beus M, Savijoki K, Patel JZ, Yli-Kauhaluoma J, Fallarero A, Zorc B. Chloroquine fumardiamides as novel quorum sensing inhibitors. Bioorganic & Medicinal Chemistry Letters. 30: 127336. PMID 32631537 DOI: 10.1016/J.Bmcl.2020.127336 |
0.318 |
|
| 2019 |
Jumppanen M, Kinnunen SM, Välimäki MJ, Talman V, Auno S, Bruun T, Boije Af Gennäs G, Xhaard HG, Aumüller IB, Ruskoaho HJ, Yli-Kauhaluoma J. Synthesis, identification and structure-activity relationship analysis of GATA4 and NKX2-5 protein-protein interaction modulators. Journal of Medicinal Chemistry. PMID 31431011 DOI: 10.1021/Acs.Jmedchem.9B01086 |
0.3 |
|
| 2018 |
Bhat C, Ilina P, Tilli I, Voráčová M, Bruun T, Barba V, Hribernik N, Lillsunde KE, Mäki-Lohiluoma E, Rüffer T, Lang H, Yli-Kauhaluoma J, Kiuru P, Tammela P. Synthesis and Antiproliferative Activity of Marine Bromotyrosine Purpurealidin I and Its Derivatives. Marine Drugs. 16. PMID 30513862 DOI: 10.3390/Md16120481 |
0.325 |
|
| 2018 |
Kolsi LE, Leal AS, Yli-Kauhaluoma J, Liby KT, Moreira VM. Dehydroabietic oximes halt pancreatic cancer cell growth in the G1 phase through induction of p27 and downregulation of cyclin D1. Scientific Reports. 8: 15923. PMID 30374056 DOI: 10.1038/S41598-018-34131-1 |
0.307 |
|
| 2018 |
Häkkinen ST, Nygren H, Maiorova N, Haavikko R, Alakurtti S, Yli-Kauhaluoma J, Rischer H, Oksman-Caldentey KM. Biotransformation of Cyclodextrine-Complexed Semisynthetic Betulin Derivatives by Plant Cells. Planta Medica. 84: 743-748. PMID 29518814 DOI: 10.1055/A-0585-6081 |
0.303 |
|
| 2018 |
Zhang Y, Jumppanen M, Maksimainen MM, Auno S, Awol Z, Ghemtio L, Venkannagari H, Lehtiö L, Yli-Kauhaluoma J, Xhaard H, Boije Af Gennäs G. Adenosine analogs bearing phosphate isosteres as human MDO1 ligands. Bioorganic & Medicinal Chemistry. PMID 29501416 DOI: 10.1016/J.Bmc.2018.02.006 |
0.329 |
|
| 2016 |
Chaaban I, El Khawass ES, Abd El Razik HA, El Salamouni NS, Redondo-Horcajo M, Barasoain I, Díaz JF, Yli-Kauhaluoma J, Moreira VM. Synthesis and Anti-Proliferative Activity of Sulfanyltriazolylnaphthalenols and Sulfanyltriazolylnaphthalene-1,4-diones. Archiv Der Pharmazie. PMID 27404773 DOI: 10.1002/Ardp.201600134 |
0.323 |
|
| 2016 |
Pirttimaa M, Nasereddin A, Kopelyanskiy D, Kaiser M, Yli-Kauhaluoma J, Oksman-Caldentey KM, Brun R, Jaffe CL, Moreira VM, Alakurtti S. Abietane-Type Diterpenoid Amides with Highly Potent and Selective Activity against Leishmania donovani and Trypanosoma cruzi. Journal of Natural Products. 79: 362-8. PMID 26849852 DOI: 10.1021/Acs.Jnatprod.5B00990 |
0.32 |
|
| 2016 |
Montalvão S, Leino TO, Kiuru PS, Lillsunde KE, Yli-Kauhaluoma J, Tammela P. Synthesis and Biological Evaluation of 2-Aminobenzothiazole and Benzimidazole Analogs Based on the Clathrodin Structure. Archiv Der Pharmazie. 349: 137-49. PMID 26709468 DOI: 10.1002/Ardp.201500365 |
0.326 |
|
| 2016 |
Vahermo M, Krogerus S, Nasereddin A, Kaiser M, Brun R, Jaffe CL, Yli-Kauhaluoma J, Moreira VM. Antiprotozoal activity of dehydroabietic acid derivatives against Leishmania donovani and Trypanosoma cruzi Medchemcomm. 7: 457-463. DOI: 10.1039/C5Md00498E |
0.322 |
|
| 2015 |
Leino TO, Baumann M, Yli-Kauhaluoma J, Baxendale IR, Wallén EA. Synthesis of 1,3,6-Trisubstituted Azulenes. The Journal of Organic Chemistry. 80: 11513-20. PMID 26528547 DOI: 10.1021/Acs.Joc.5B02271 |
0.312 |
|
| 2015 |
Keurulainen L, Siiskonen A, Nasereddin A, Kopelyanskiy D, Sacerdoti-Sierra N, Leino TO, Tammela P, Yli-Kauhaluoma J, Jaffe CL, Kiuru P. Synthesis and biological evaluation of 2-arylbenzimidazoles targeting Leishmania donovani. Bioorganic & Medicinal Chemistry Letters. 25: 1933-7. PMID 25827525 DOI: 10.1016/J.Bmcl.2015.03.027 |
0.306 |
|
| 2015 |
Keurulainen L, Heiskari M, Nenonen S, Nasereddin A, Kopelyanskiy D, Leino TO, Yli-Kauhaluoma J, Jaffe CL, Kiuru P. Synthesis of carboxyimidamide-substituted benzo[c][1,2,5]oxadiazoles and their analogs, and evaluation of biological activity against Leishmania donovani Medchemcomm. 6: 1673-1678. DOI: 10.1039/C5Md00119F |
0.335 |
|
| 2015 |
Rossi D, Talman V, Gennäs GBA, Marra A, Picconi P, Nasti R, Serra M, Ann J, Amadio M, Pascale A, Tuominen RK, Yli-Kauhaluoma J, Lee J, Collina S. Beyond the affinity for protein kinase C: exploring 2-phenyl-3-hydroxypropyl pivalate analogues as C1 domain-targeting ligands Medchemcomm. 6: 547-554. DOI: 10.1039/C4Md00564C |
0.305 |
|
| 2014 |
Chaaban I, El Khawass el SM, Abd El Razik HA, El Salamouni NS, Redondo-Horcajo M, Barasoain I, Díaz JF, Yli-Kauhaluoma J, Moreira VM. Synthesis and biological evaluation of new oxadiazoline-substituted naphthalenyl acetates as anticancer agents. European Journal of Medicinal Chemistry. 87: 805-13. PMID 25440882 DOI: 10.1016/J.Ejmech.2014.10.015 |
0.339 |
|
| 2014 |
Talman V, Provenzani R, Boije af Gennäs G, Tuominen RK, Yli-Kauhaluoma J. C1 domain-targeted isophthalates as protein kinase C modulators: structure-based design, structure-activity relationships and biological activities. Biochemical Society Transactions. 42: 1543-9. PMID 25399568 DOI: 10.1042/Bst20140181 |
0.333 |
|
| 2014 |
Alcazar W, López AS, Alakurtti S, Tuononen ML, Yli-Kauhaluoma J, Ponte-Sucre A. Betulin derivatives impair Leishmania braziliensis viability and host-parasite interaction. Bioorganic & Medicinal Chemistry. 22: 6220-6. PMID 25240731 DOI: 10.1016/J.Bmc.2014.08.023 |
0.313 |
|
| 2014 |
Kiuru P, D?Auria MV, Muller CD, Tammela P, Vuorela H, Yli-Kauhaluoma J. Exploring marine resources for bioactive compounds. Planta Medica. 80: 1234-46. PMID 25203732 DOI: 10.1055/S-0034-1383001 |
0.303 |
|
| 2014 |
Haque S, Nawrot DA, Alakurtti S, Ghemtio L, Yli-Kauhaluoma J, Tammela P. Screening and characterisation of antimicrobial properties of semisynthetic betulin derivatives. Plos One. 9: e102696. PMID 25032708 DOI: 10.1371/Journal.Pone.0102696 |
0.327 |
|
| 2014 |
Parkkari T, Haavikko R, Laitinen T, Navia-Paldanius D, Rytilahti R, Vaara M, Lehtonen M, Alakurtti S, Yli-Kauhaluoma J, Nevalainen T, Savinainen JR, Laitinen JT. Discovery of triterpenoids as reversible inhibitors of α/β-hydrolase domain containing 12 (ABHD12). Plos One. 9: e98286. PMID 24879289 DOI: 10.1371/Journal.Pone.0098286 |
0.317 |
|
| 2014 |
Haavikko R, Nasereddin A, Sacerdoti-Sierra N, Kopelyanskiy D, Alakurtti SA, Tikka M, Jaffe CL, Yli-Kauhaluoma J. Heterocycle-fused lupane triterpenoids inhibit Leishmania donovani amastigotes Medchemcomm. 5: 445-451. DOI: 10.1039/C3Md00282A |
0.334 |
|
| 2013 |
Fallarero A, Skogman M, Kujala J, Rajaratnam M, Moreira VM, Yli-Kauhaluoma J, Vuorela P. (+)-Dehydroabietic Acid, an Abietane-Type Diterpene, Inhibits Staphylococcus aureus Biofilms in Vitro. International Journal of Molecular Sciences. 14: 12054-72. PMID 23739682 DOI: 10.3390/Ijms140612054 |
0.307 |
|
| 2013 |
Manevski N, Troberg J, Svaluto-Moreolo P, Dziedzic K, Yli-Kauhaluoma J, Finel M. Albumin stimulates the activity of the human UDP-glucuronosyltransferases 1A7, 1A8, 1A10, 2A1 and 2B15, but the effects are enzyme and substrate dependent. Plos One. 8: e54767. PMID 23372764 DOI: 10.1371/Journal.Pone.0054767 |
0.322 |
|
| 2013 |
Leikoski T, Wrigstedt P, Matikainen J, Sipilä J, Yli-Kauhaluoma J. Erratum: Solid-phase synthesis of N-(buta-2,3,-dien-1-yl)amides by the Crabbé reaction Canadian Journal of Chemistry. 91: 38-42. DOI: 10.1139/Cjc-2012-0255 |
0.323 |
|
| 2013 |
Leikoski T, Wrigstedt P, Helminen J, Matikainen J, Sipilä J, Yli-Kauhaluoma J. The Heck reaction of polymer-supported allylamine with aryl iodides Tetrahedron. 69: 839-843. DOI: 10.1016/J.Tet.2012.10.092 |
0.351 |
|
| 2012 |
Manevski N, Yli-Kauhaluoma J, Finel M. UDP-glucuronic acid binds first and the aglycone substrate binds second to form a ternary complex in UGT1A9-catalyzed reactions, in both the presence and absence of bovine serum albumin. Drug Metabolism and Disposition: the Biological Fate of Chemicals. 40: 2192-203. PMID 22912433 DOI: 10.1124/Dmd.112.047746 |
0.315 |
|
| 2012 |
Siiskonen A, Keurulainen L, Salin O, Kiuru P, Pohjala L, Vuorela P, Yli-Kauhaluoma J. Conformation study of 2-arylbenzimidazoles as inhibitors of Chlamydia pneumoniae growth. Bioorganic & Medicinal Chemistry Letters. 22: 4882-6. PMID 22695128 DOI: 10.1016/J.Bmcl.2012.05.023 |
0.311 |
|
| 2011 |
Talman V, Tuominen RK, Boije af Gennäs G, Gennäs GB, Yli-Kauhaluoma J, Ekokoski E. C1 Domain-targeted isophthalate derivatives induce cell elongation and cell cycle arrest in HeLa cells. Plos One. 6: e20053. PMID 21629792 DOI: 10.1371/Journal.Pone.0020053 |
0.307 |
|
| 2011 |
Wert L, Alakurtti S, Corral MJ, Sánchez-Fortún S, Yli-Kauhaluoma J, Alunda JM. Toxicity of betulin derivatives and in vitro effect on promastigotes and amastigotes of Leishmania infantum and L. donovani. The Journal of Antibiotics. 64: 475-81. PMID 21522160 DOI: 10.1038/Ja.2011.34 |
0.322 |
|
| 2011 |
Šilhár P, Alakurtti S, ?apková K, Xiaochuan F, Shoemaker CB, Yli-Kauhaluoma J, Janda KD. Synthesis and evaluation of library of betulin derivatives against the botulinum neurotoxin A protease. Bioorganic & Medicinal Chemistry Letters. 21: 2229-31. PMID 21421315 DOI: 10.1016/J.Bmcl.2011.02.115 |
0.468 |
|
| 2011 |
Kiriazis A, Aumüller IB, Yli-Kauhaluoma J. Synthesis of 4-aminoguaiazulene and its δ-lactam derivatives Tetrahedron Letters. 52: 1151-1153. DOI: 10.1016/J.Tetlet.2011.01.016 |
0.342 |
|
| 2010 |
Salin O, Alakurtti S, Pohjala L, Siiskonen A, Maass V, Maass M, Yli-Kauhaluoma J, Vuorela P. Inhibitory effect of the natural product betulin and its derivatives against the intracellular bacterium Chlamydia pneumoniae. Biochemical Pharmacology. 80: 1141-51. PMID 20615390 DOI: 10.1016/J.Bcp.2010.06.051 |
0.337 |
|
| 2010 |
Alakurtti S, Bergström P, Sacerdoti-Sierra N, Jaffe CL, Yli-Kauhaluoma J. Anti-leishmanial activity of betulin derivatives. The Journal of Antibiotics. 63: 123-6. PMID 20139867 DOI: 10.1016/J.Ejps.2008.02.105 |
0.35 |
|
| 2010 |
Alakurtti S, Heiska T, Kiriazis A, Sacerdoti-Sierra N, Jaffe CL, Yli-Kauhaluoma J. Synthesis and anti-leishmanial activity of heterocyclic betulin derivatives. Bioorganic & Medicinal Chemistry. 18: 1573-82. PMID 20116263 DOI: 10.1016/J.Bmc.2010.01.003 |
0.326 |
|
| 2010 |
Taylor MJ, Yli-Kauhaluoma JT, Ashley JA, Wirsching P, Lerner RA, Janda KD. ChemInform Abstract: The α-Ketoamide Group: A New Motif for the Elicitation of Catalytic Antibodies for Acyl-Transfer Reactions. Cheminform. 30: no-no. DOI: 10.1002/CHIN.199938222 |
0.393 |
|
| 2010 |
Taylor MJ, Hoffman TZ, Yli-Kauhaluoma JT, Lerner RA, Janda KD. ChemInform Abstract: A Light-Activated Antibody Catalyst. Cheminform. 30: no-no. DOI: 10.1002/CHIN.199917044 |
0.34 |
|
| 2010 |
YLI-KAUHALUOMA JT, HARWIG CW, WENTWORTH PJ, JANDA KD. ChemInform Abstract: Unexpected 1,3-Oxazolidine Formation in the Attempted Oxidation of N-Aryl-N-methyl Substituted β-Amino Alcohols Using Pyridinium Dichromate. Cheminform. 29: no-no. DOI: 10.1002/CHIN.199829101 |
0.352 |
|
| 2010 |
YLI-KAUHALUOMA JT, JANDA KD. ChemInform Abstract: An Expedient Synthesis of Isopropyl Anisoles and Veratroles. Cheminform. 25: no-no. DOI: 10.1002/CHIN.199446109 |
0.358 |
|
| 2009 |
Aumüller IB, Yli-Kauhaluoma J. Benzo[cd]azulene skeleton: azulene, heptafulvene, and tropone derivatives. Organic Letters. 11: 5363-5. PMID 19904921 DOI: 10.1021/Ol902283Q |
0.323 |
|
| 2009 |
Pohjala L, Alakurtti S, Ahola T, Yli-Kauhaluoma J, Tammela P. Betulin-derived compounds as inhibitors of alphavirus replication. Journal of Natural Products. 72: 1917-26. PMID 19839605 DOI: 10.1021/Np9003245 |
0.311 |
|
| 2009 |
Alonen A, Gartman M, Aitio O, Finel M, Yli-Kauhaluoma J, Kostiainen R. Synthesis, structure characterization, and enzyme screening of clenbuterol glucuronides. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. 37: 581-7. PMID 19447177 DOI: 10.1016/J.Ejps.2009.05.003 |
0.301 |
|
| 2009 |
Harju K, Vesterinen J, Yli-Kauhaluoma J. Solid-phase synthesis of amino acid derived N-unsubstituted pyrazoles via sydnones. Organic Letters. 11: 2219-21. PMID 19419217 DOI: 10.1021/Ol900704B |
0.307 |
|
| 2007 |
Bichlmaier I, Finel M, Sippl W, Yli-Kauhaluoma J. Stereochemical and steric control of the UDP-glucuronosyltransferase-catalyzed conjugation reaction: a rational approach for the design of inhibitors for the human UGT2B7. Chemmedchem. 2: 1730-40. PMID 17943712 DOI: 10.1002/Cmdc.200700122 |
0.354 |
|
| 2007 |
Bichlmaier I, Kurkela M, Siiskonen A, Finel M, Yli-Kauhaluoma J. Eudismic analysis of tricyclic sesquiterpenoid alcohols: lead structures for the design of potent inhibitors of the human UDP-glucuronosyltransferase 2B7. Bioorganic Chemistry. 35: 386-400. PMID 17706742 DOI: 10.1016/J.Bioorg.2007.07.002 |
0.308 |
|
| 2007 |
Bichlmaier I, Kurkela M, Joshi T, Siiskonen A, Rüffer T, Lang H, Finel M, Yli-Kauhaluoma J. Potent inhibitors of the human UDP-glucuronosyltransferase 2B7 derived from the sesquiterpenoid alcohol longifolol. Chemmedchem. 2: 881-9. PMID 17479992 DOI: 10.1002/Cmdc.200600246 |
0.303 |
|
| 2007 |
Bichlmaier I, Kurkela M, Joshi T, Siiskonen A, Rüffer T, Lang H, Suchanova B, Vahermo M, Finel M, Yli-Kauhaluoma J. Isoform-selective inhibition of the human UDP-glucuronosyltransferase 2B7 by isolongifolol derivatives. Journal of Medicinal Chemistry. 50: 2655-64. PMID 17474732 DOI: 10.1021/Jm061204E |
0.329 |
|
| 2007 |
Kiriazis A, Rüffer T, Jäntti S, Lang H, Yli-Kauhaluoma J. Stereoselective aza Diels-Alder reaction on solid phase: a facile synthesis of hexahydrocinnoline derivatives. Journal of Combinatorial Chemistry. 9: 263-6. PMID 17348732 DOI: 10.1021/Cc060125L |
0.348 |
|
| 2007 |
Mutikainen I, Kiriazis A, Leikoski T, Yli-Kauhaluoma J. 2-Ethyl-1,3-dioxo-2,3,3a,4,7,7a-hexahydro-1H-isoindole-4-carboxylic acid Acta Crystallographica Section E-Structure Reports Online. 63. DOI: 10.1107/S1600536807027900 |
0.367 |
|
| 2006 |
Alakurtti S, Mäkelä T, Koskimies S, Yli-Kauhaluoma J. Pharmacological properties of the ubiquitous natural product betulin. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. 29: 1-13. PMID 16716572 DOI: 10.1016/J.Ejps.2006.04.006 |
0.309 |
|
| 2006 |
Harju K, Kylänlahti I, Paananen T, Polamo M, Nielsen J, Yli-Kauhaluoma J. Solid-phase synthesis of pyrazolopyridines from polymer-bound alkyne and azomethine imines. Journal of Combinatorial Chemistry. 8: 344-9. PMID 16677003 DOI: 10.1021/cc050138j |
0.468 |
|
| 2006 |
Bichlmaier I, Siiskonen A, Kurkela M, Finel M, Yli-Kauhaluoma J. Chiral distinction between the enantiomers of bicyclic alcohols by UDP-glucuronosyltransferases 2B7 and 2B17. Biological Chemistry. 387: 407-16. PMID 16606339 DOI: 10.1515/Bc.2006.055 |
0.309 |
|
| 2006 |
Bichlmaier I, Siiskonen A, Finel M, Yli-Kauhaluoma J. Stereochemical sensitivity of the human UDP-glucuronosyltransferases 2B7 and 2B17. Journal of Medicinal Chemistry. 49: 1818-27. PMID 16509597 DOI: 10.1021/Jm051142C |
0.302 |
|
| 2005 |
Toker JD, Tremblay MR, Yli-Kauhaluoma J, Wentworth AD, Zhou B, Wentworth P, Janda KD. Exploring the scope of the 29G12 antibody catalyzed 1,3-dipolar cycloaddition reaction. The Journal of Organic Chemistry. 70: 7810-5. PMID 16277300 DOI: 10.1021/Jo050410B |
0.689 |
|
| 2005 |
Samanta SK, Kylänlahti I, Yli-Kauhaluoma J. Microwave-assisted synthesis of imidazoles: reaction of p-toluenesulfonylmethyl isocyanide and polymer-bound imines. Bioorganic & Medicinal Chemistry Letters. 15: 3717-9. PMID 15993061 DOI: 10.1016/J.Bmcl.2005.05.066 |
0.338 |
|
| 2005 |
Harju K, Yli-Kauhaluoma J. Recent advances in 1,3-dipolar cycloaddition reactions on solid supports. Molecular Diversity. 9: 187-207. PMID 15789565 DOI: 10.1007/S11030-005-1339-1 |
0.326 |
|
| 2005 |
Samanta SK, Yli-Kauhaluoma J. Polymer-supported 1,3-oxazolium-5-olates: synthesis of 1,2,4-triazoles. Journal of Combinatorial Chemistry. 7: 142-6. PMID 15638494 DOI: 10.1021/Cc049905P |
0.31 |
|
| 1999 |
Taylor MJ, Yli-Kauhaluoma JT, Ashley JA, Wirsching P, Lerner RA, Janda KD. The α-ketoamide group: A new motif for the elicitation of catalytic antibodies for acyl-transfer reactions Journal of the Chemical Society - Perkin Transactions 1. 1133-1134. DOI: 10.1039/A902475A |
0.394 |
|
| 1998 |
Heine A, Stura EA, Yli-Kauhaluoma JT, Gao C, Deng Q, Beno BR, Houk KN, Janda KD, Wilson IA. An antibody exo Diels-Alderase inhibitor complex at 1.95 angstrom resolution. Science (New York, N.Y.). 279: 1934-40. PMID 9506943 DOI: 10.1126/Science.279.5358.1934 |
0.58 |
|
| 1998 |
Taylor MJ, Hoffman TZ, Yli-Kauhaluoma JT, Lerner RA, Janda KD. A light-activated antibody catalyst Journal of the American Chemical Society. 120: 12783-12790. DOI: 10.1021/Ja982711R |
0.411 |
|
| 1998 |
Yli-Kauhaluoma JT, Harwig CW, Wentworth P, Janda KD. Unexpected 1,3-oxazolidine formation in the attempted oxidation of N-aryl-N-methyl substituted β-amino alcohols using pyridinium dichromate Tetrahedron Letters. 39: 2269-2272. DOI: 10.1016/S0040-4039(98)00289-5 |
0.369 |
|
| 1996 |
Yli-Kauhaluoma JT, Ashley JA, Lo CL, Coakley J, Wirsching P, Janda KD. Catalytic Antibodies with Peptidyl−Prolyl Cis−Trans Isomerase Activity Journal of the American Chemical Society. 118: 5496-5497. DOI: 10.1021/Ja954206P |
0.363 |
|
| 1995 |
Yli-Kauhaluoma JT, Ashley JA, Lo C, Tucker L, Wolfe MM, Janda KD. Anti-Metallocene Antibodies: A New Approach to Enantioselective Catalysis of the Diels-Alder Reaction Journal of the American Chemical Society. 117: 7041-7047. DOI: 10.1021/Ja00132A001 |
0.392 |
|
| 1994 |
Yli-Kauhaluoma J, Janda KD. Twisted α-keto amides as transition-state analogues for acyl-transfer reactions: Synthesis of the immunoconjugates Bioorganic and Medicinal Chemistry. 2: 521-528. PMID 7528089 DOI: 10.1016/0968-0896(94)80022-7 |
0.475 |
|
| 1994 |
Yli-Kauhaluoma JT, Janda KD. An expedient synthesis of isopropyl anisoles and veratroles Tetrahedron Letters. 35: 4509-4510. DOI: 10.1016/S0040-4039(00)60713-X |
0.416 |
|
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