Ashish K Radadiya - Publications

Affiliations: 
Cardiff University, Cardiff, Wales, United Kingdom 
Area:
Medicinal chemistry, organic synthesis, drug-discovery, molecular modelling, chemical biology

18 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2022 Bijani S, Shaikh F, Mirza S, Weng In Siu S, Jain N, Rawal R, Richards NGJ, Shah A, Radadiya A. Novel Dihydropyrimidinone Derivatives as Potential P-Glycoprotein Modulators. Acs Omega. 7: 16278-16287. PMID 35601326 DOI: 10.1021/acsomega.1c05839  0.741
2020 Radadiya A, Zhu W, Coricello A, Alcaro S, Richards NGJ. Improving the Treatment of Acute Lymphoblastic Leukemia. Biochemistry. PMID 32786406 DOI: 10.1021/Acs.Biochem.0C00354  0.428
2020 Gao S, Radadiya A, Li W, Liu H, Zhu W, de Crécy-Lagard V, Richards NGJ, Naismith JH. Uncovering the chemistry of C-C bond formation in C-nucleoside biosynthesis: crystal structure of a C-glycoside synthase/PRPP complex. Chemical Communications (Cambridge, England). PMID 32515440 DOI: 10.1039/D0Cc02834G  0.433
2019 Zhu W, Radadiya A, Bisson C, Wenzel S, Nordin BE, Martínez-Márquez F, Imasaki T, Sedelnikova SE, Coricello A, Baumann P, Berry AH, Nomanbhoy TK, Kozarich JW, Jin Y, Rice DW, et al. Erratum: Author Correction: High-resolution crystal structure of human asparagine synthetase enables analysis of inhibitor binding and selectivity. Communications Biology. 2: 438. PMID 31799439 DOI: 10.1038/s42003-019-0690-1  0.381
2019 Zhu W, Radadiya A, Bisson C, Wenzel S, Nordin BE, Martínez-Márquez F, Imasaki T, Sedelnikova SE, Coricello A, Baumann P, Berry AH, Nomanbhoy TK, Kozarich JW, Jin Y, Rice DW, et al. High-resolution crystal structure of human asparagine synthetase enables analysis of inhibitor binding and selectivity. Communications Biology. 2: 345. PMID 31552298 DOI: 10.1038/s42003-019-0587-z  0.446
2017 Athar M, Yousuf Lone M, M Khedkar V, Radadiya A, Shah A, C Jha P. Structural Investigation of Vinca domain tubulin binders by Pharmacophore, Atom based QSAR, Docking and Molecular Dynamics Simulations. Combinatorial Chemistry & High Throughput Screening. PMID 28486912 DOI: 10.2174/1386207320666170509151253  0.569
2016 Patel S, Shaikh F, Devaraji V, Radadiya A, Shah K, Shah A, Rawal R. Insights Into The Structural Perturbations Of Spliced Variants Of Cd44: A Modelling And Simulation Approach. Journal of Biomolecular Structure & Dynamics. 1-34. PMID 26766750 DOI: 10.1080/07391102.2016.1142476  0.702
2016 Abhinand PA, Shaikh F, Bhakat S, Radadiya A, Bhaskar LV, Shah A, Ragunath PK. Insights on the structural perturbations in human MTHFR Ala222Val mutant by protein modeling and molecular dynamics. Journal of Biomolecular Structure & Dynamics. 34: 892-905. PMID 26273990 DOI: 10.1080/07391102.2015.1057866  0.71
2015 Radadiya A, Shah A. Bioactive benzofuran derivatives: An insight on lead developments, radioligands and advances of the last decade. European Journal of Medicinal Chemistry. 97: 356-376. PMID 25703339 DOI: 10.1016/J.Ejmech.2015.01.021  0.554
2014 Radadiya A, Khedkar V, Bavishi A, Vala H, Thakrar S, Bhavsar D, Shah A, Coutinho E. Synthesis and 3D-QSAR study of 1,4-dihydropyridine derivatives as MDR cancer reverters. European Journal of Medicinal Chemistry. 74: 375-87. PMID 24486418 DOI: 10.1016/J.Ejmech.2014.01.011  0.745
2014 Shaikh F, Bhakat S, Thakur A, Radadiya A, Soliman MES, Shah A. Identification of Novel GSK1070916 Analogs as Potential Aurora B Inhibitors: Insights from Molecular Dynamics and MM/GBSA Based Rescoring Letters in Drug Design & Discovery. 12: 2-13. DOI: 10.2174/1570180811666140725184953  0.544
2014 Thakrar S, Bavishi A, Radadiya A, Vala H, Parekh S, Bhavsar D, Chaniyara R, Shah A. An efficient microwave-assisted synthesis and antimicrobial activity of novel 2-amino 3-cyano pyridine derivatives using two reusable solid acids as catalysts Journal of Heterocyclic Chemistry. 51: 555-561. DOI: 10.1002/Jhet.1641  0.653
2013 Thakrar S, Bavishi A, Radadiya A, Parekh S, Bhavsar D, Vala H, Pandya N, Shah A. Microwave-Assisted Rapid Synthesis of Novel 1,5-Benzodiazepine Derivatives as Potent Antimicrobial Agent Journal of Heterocyclic Chemistry. 50: E73-E79. DOI: 10.1002/Jhet.1065  0.68
2012 Thakrar S, Bavishi A, Bhavsar D, Parekh S, Vala H, Radadiya A, Parmar M, Savant M, Shah A. Efficient and rapid synthesis of highly functionalized novel symmetric 1,4-dihydropyridines using glacial acetic acid as solvent Synthetic Communications. 42: 3269-3278. DOI: 10.1080/00397911.2011.576448  0.635
2011 Manvar A, Bavishi A, Radadiya A, Patel J, Vora V, Dodia N, Rawal K, Shah A. Diversity oriented design of various hydrazides and their in vitro evaluation against Mycobacterium tuberculosis H37Rv strains. Bioorganic & Medicinal Chemistry Letters. 21: 4728-31. PMID 21752642 DOI: 10.1016/J.Bmcl.2011.06.074  0.655
2011 Bhavsar D, Trivedi J, Parekh S, Savant M, Thakrar S, Bavishi A, Radadiya A, Vala H, Lunagariya J, Parmar M, Paresh L, Loddo R, Shah A. Synthesis and in vitro anti-HIV activity of N-1,3-benzo[d]thiazol-2-yl-2-(2-oxo-2H-chromen-4-yl)acetamide derivatives using MTT method. Bioorganic & Medicinal Chemistry Letters. 21: 3443-6. PMID 21515046 DOI: 10.1016/J.Bmcl.2011.03.105  0.701
2011 Upadhyay K, Bavishi A, Thakrar S, Radadiya A, Vala H, Parekh S, Bhavsar D, Savant M, Parmar M, Adlakha P, Shah A. Synthesis and biological evaluation of 4-styrylcoumarin derivatives as inhibitors of TNF-α and IL-6 with anti-tubercular activity. Bioorganic & Medicinal Chemistry Letters. 21: 2547-9. PMID 21396814 DOI: 10.1016/J.Bmcl.2011.02.016  0.69
2011 Parekh S, Bhavsar D, Savant M, Thakrar S, Bavishi A, Parmar M, Vala H, Radadiya A, Pandya N, Serly J, Molnár J, Shah A. Synthesis of some novel benzofuran-2-yl(4,5-dihyro-3,5-substituted diphenylpyrazol-1-yl) methanones and studies on the antiproliferative effects and reversal of multidrug resistance of human MDR1-gene transfected mouse lymphoma cells in vitro. European Journal of Medicinal Chemistry. 46: 1942-8. PMID 21396744 DOI: 10.1016/J.Ejmech.2011.02.045  0.773
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