Year |
Citation |
Score |
2023 |
Jia X, Schols D, Meier C. Lipophilic Nucleoside Triphosphate Prodrugs of Anti-HIV Active Nucleoside Analogs as Potential Antiviral Compounds. Advanced Science (Weinheim, Baden-Wurttemberg, Germany). e2306021. PMID 37884485 DOI: 10.1002/advs.202306021 |
0.312 |
|
2020 |
Jia X, Weber S, Schols D, Meier C. Membrane Permeable, Bioreversibly Modified Prodrugs of Nucleoside Diphosphate-γ-Phosphonates. Journal of Medicinal Chemistry. 63: 11990-12007. PMID 32991174 DOI: 10.1021/acs.jmedchem.0c01294 |
0.33 |
|
2020 |
Jia X, Schols D, Meier C. Lipophilic Triphosphate Prodrugs of various Nucleoside Analogues. Journal of Medicinal Chemistry. PMID 32515595 DOI: 10.1021/Acs.Jmedchem.0C00358 |
0.383 |
|
2020 |
Jia X, Schols D, Meier C. Anti-HIV-Active Nucleoside Triphosphate Prodrugs. Journal of Medicinal Chemistry. 63: 6003-6027. PMID 32421343 DOI: 10.1021/Acs.Jmedchem.0C00271 |
0.354 |
|
2020 |
Fehling H, Choy SL, Ting F, Landschulze D, Bernin H, Lender SC, Mühlenpfordt M, Bifeld E, Eick J, Marggraff C, Kottmayr N, Groneberg M, Hoenow S, Sellau J, Clos J, ... Meier C, et al. Anti-leishmanial effects of synthetic PIb analogs derived from the lipopeptidephosphoglycan. Antimicrobial Agents and Chemotherapy. PMID 32393489 DOI: 10.1128/Aac.00161-20 |
0.312 |
|
2020 |
Meier C, Zhao C, Weber S, Schols D, Balzarini J. Prodrugs of γ-Alkyl-modified Nucleoside Triphosphates - improved Inhibition of HIV Reverse Transcriptase. Angewandte Chemie (International Ed. in English). PMID 32379948 DOI: 10.1002/Anie.202003073 |
0.388 |
|
2018 |
Weising S, Sterrenberg V, Schols D, Meier C. Synthesis and Antiviral Evaluation of TriPPPro-AbacavirTP, TriPPPro-CarbovirTP, and Their 1',2'-cis-Disubstituted Analogues Chemmedchem. 13: 1771-1778. PMID 29943432 DOI: 10.1002/Cmdc.201800361 |
0.402 |
|
2018 |
Weising S, Dekiert P, Schols D, Neyts J, Meier C. Synthesis of Enantiomerically Pure 1′,2′-cis-dideoxy, -dideoxydidehydro, -ribo and -deoxy Carbocyclic Nucleoside Analogues Synthesis. 50: 2266-2280. DOI: 10.1055/S-0037-1609493 |
0.385 |
|
2017 |
Meier C. Nucleoside diphosphate and triphosphate prodrugs – An unsolvable task?: Antiviral Chemistry & Chemotherapy. 25: 69-82. PMID 29096525 DOI: 10.1177/2040206617738656 |
0.364 |
|
2017 |
Pahnke K, Meier C. Synthesis of a Bioreversibly Masked Lipophilic Adenosine Diphosphate Ribose Derivative Chembiochem. 18: 1616-1626. PMID 28589630 DOI: 10.1002/Cbic.201700232 |
0.377 |
|
2017 |
Ehrit J, Keys TG, Sutherland M, Meier C, Wolf S, Falconer R, Gerardy-Schahn R. Exploring and Exploiting Acceptor Preferences of the Human Polysialyltransferases as a Basis for an Inhibitor Screen. Chembiochem : a European Journal of Chemical Biology. PMID 28472541 DOI: 10.1002/Cbic.201700157 |
0.327 |
|
2017 |
Ordonez P, Kunzelmann S, Groom HC, Yap MW, Weising S, Meier C, Bishop KN, Taylor IA, Stoye JP. SAMHD1 enhances nucleoside-analogue efficacy against HIV-1 in myeloid cells. Scientific Reports. 7: 42824. PMID 28220857 DOI: 10.1038/Srep42824 |
0.331 |
|
2017 |
Weising S, Torquati I, Meier C. Stereoselective Synthesis of 1′,2′-cis-Disubstituted Carbocyclic ribo-Nucleoside Analogues Synthesis. 50: 1264-1274. DOI: 10.1055/S-0036-1591732 |
0.378 |
|
2017 |
Huchting J, Winkler M, Nasser H, Meier C. Cover Picture: Synthesis of T‐705‐Ribonucleoside and T‐705‐Ribonucleotide and Studies of Chemical Stability (ChemMedChem 9/2017) Chemmedchem. 12: 621-621. DOI: 10.1002/Cmdc.201700255 |
0.32 |
|
2016 |
Sarac I, Meier C. Solid-Phase Synthesis of DNA and RNA 5'-O-Triphosphates Using cycloSal Chemistry. Current Protocols in Human Genetics. 64. PMID 31820581 DOI: 10.1002/0471142700.Nc0467S64 |
0.351 |
|
2016 |
Gollnest T, Dinis de Oliveira T, Rath A, Hauber I, Schols D, Balzarini J, Meier C. Membrane-permeable Triphosphate Prodrugs of Nucleoside Analogues. Angewandte Chemie (International Ed. in English). 55: 5255-8. PMID 27008042 DOI: 10.1002/anie.201511808 |
0.309 |
|
2016 |
Schröder M, Kolodzik A, Windshügel B, Krepstakies M, Priyadarshini P, Hartjen P, van Lunzen J, Rarey M, Hauber J, Meier C. Linker-Region Modified Derivatives of the Deoxyhypusine Synthase Inhibitor CNI-1493 Suppress HIV-1 Replication. Archiv Der Pharmazie. 349: 91-103. PMID 26725082 DOI: 10.1002/Ardp.201500323 |
0.369 |
|
2016 |
Gollnest T, De Oliveira TD, Rath A, Hauber I, Schols D, Balzarini J, Meier C. Membrane-permeable Triphosphate Prodrugs of Nucleoside Analogues Angewandte Chemie - International Edition. 55: 5255-5258. DOI: 10.1002/Anie.201511808 |
0.421 |
|
2015 |
Meier C, Jessen HJ, Schulz T, Weinschenk L, Pertenbreiter F, Balzarini J. Rational Development of Nucleoside Diphosphate Prodrugs: DiPPro-Compounds. Current Medicinal Chemistry. 22: 3933-50. PMID 26303175 DOI: 10.2174/0929867322666150825163119 |
0.374 |
|
2015 |
Höfler K, Sarac I, Meier C. Synthesis of C8-N-Arylamine-Modified 2'-Deoxyguanosine-5'-Triphosphates and Their Effects on Primer Extension by DNA Polymerases. Chembiochem : a European Journal of Chemical Biology. 16: 2046-53. PMID 26222706 DOI: 10.1002/Cbic.201500293 |
0.329 |
|
2015 |
Weinschenk L, Schols D, Balzarini J, Meier C. Nucleoside Diphosphate Prodrugs: Nonsymmetric DiPPro-Nucleotides Journal of Medicinal Chemistry. 58: 6114-6130. PMID 26125628 DOI: 10.1021/Acs.Jmedchem.5B00737 |
0.381 |
|
2015 |
Weinschenk L, Gollnest T, Schols D, Balzarini J, Meier C. Bis(benzoyloxybenzyl)-DiPPro nucleoside diphosphates of anti-HIV active nucleoside analogues Chemmedchem. 10: 891-900. PMID 25847660 DOI: 10.1002/Cmdc.201500063 |
0.434 |
|
2015 |
Pertenbreiter F, Balzarini J, Meier C. Nucleoside mono- and diphosphate prodrugs of 2′,3′-dideoxyuridine and 2′,3′-dideoxy-2′,3′-didehydrouridine Chemmedchem. 10: 94-106. PMID 25209965 DOI: 10.1002/Cmdc.201402295 |
0.376 |
|
2015 |
Gollnest T, De Oliveira TD, Schols D, Balzarini J, Meier C. Lipophilic prodrugs of nucleoside triphosphates as biochemical probes and potential antivirals Nature Communications. 6. DOI: 10.1038/Ncomms9716 |
0.376 |
|
2015 |
Höfler K, Zimmermann T, Peña Fuentes D, Vogel C, Meier C. Synthesis of Homo-C-Nucleoside Phosphoramidites and Their Site-Specific Incorporation into Oligonucleotides European Journal of Organic Chemistry. 2015: 6841-6849. DOI: 10.1002/Ejoc.201500996 |
0.303 |
|
2015 |
Sarac I, Meier C. Efficient Automated Solid-Phase Synthesis of DNA and RNA 5′-Triphosphates Chemistry - a European Journal. 21: 16421-16426. DOI: 10.1002/Chem.201502844 |
0.362 |
|
2014 |
Seelhorst K, Piernitzki T, Lunau N, Meier C, Hahn U. Synthesis and analysis of potential α1,3-fucosyltransferase inhibitors Bioorganic and Medicinal Chemistry. 22: 6430-6437. PMID 25438767 DOI: 10.1016/J.Bmc.2014.09.038 |
0.323 |
|
2014 |
Schulz T, Balzarini J, Meier C. The DiPPro approach: synthesis, hydrolysis, and antiviral activity of lipophilic d4T diphosphate prodrugs. Chemmedchem. 9: 762-775. PMID 24616176 DOI: 10.1002/Cmdc.201300500 |
0.418 |
|
2014 |
Schroeder M, Kolodzik A, Pfaff K, Priyadarshini P, Krepstakies M, Hauber J, Rarey M, Meier C. In silico design, synthesis, and screening of novel deoxyhypusine synthase inhibitors targeting HIV-1 replication. Chemmedchem. 9: 940-52. PMID 24616161 DOI: 10.1002/Cmdc.201300481 |
0.371 |
|
2014 |
Huchting J, Meier C. Synthesis of Pyranonucleoside-6′-triphosphates through the cycloSal-Method European Journal of Organic Chemistry. 2014: 3423-3429. DOI: 10.1002/Ejoc.201402047 |
0.399 |
|
2014 |
Schulz T, Balzarini J, Meier C. Back Cover: The DiPPro Approach: Synthesis, Hydrolysis, and Antiviral Activity of Lipophilic d4T Diphosphate Prodrugs (ChemMedChem 4/2014) Chemmedchem. 9: 860-860. DOI: 10.1002/Cmdc.201490014 |
0.373 |
|
2013 |
Lunau N, Seelhorst K, Kahl S, Tscherch K, Stacke C, Rohn S, Thiem J, Hahn U, Meier C. Fluorescently labeled substrates for monitoring α1,3-fucosyltransferase IX activity. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 17379-90. PMID 24258785 DOI: 10.1002/Chem.201302601 |
0.306 |
|
2013 |
Huchting J, Ruthenbeck A, Meier C. Synthesis of cycloSal-(Glycopyranosyl-6)-phosphates as Activated Sugar Phosphates European Journal of Organic Chemistry. 2013: 6907-6916. DOI: 10.1002/Ejoc.201300852 |
0.342 |
|
2012 |
Wolf S, Warnecke S, Ehrit J, Freiberger F, Gerardy‐Schahn R, Meier C. Chemical synthesis and enzymatic testing of CMP-sialic acid derivatives. Chembiochem. 13: 2605-2615. PMID 23129454 DOI: 10.1002/Cbic.201200471 |
0.362 |
|
2012 |
Mahler M, Reichardt B, Hartjen P, van Lunzen J, Meier C. Stereoselective synthesis of D- and L-carbocyclic nucleosides by enzymatically catalyzed kinetic resolution. Chemistry (Weinheim An Der Bergstrasse, Germany). 18: 11046-62. PMID 22829408 DOI: 10.1002/Chem.201200733 |
0.344 |
|
2012 |
Morales EHR, Balzarini J, Meier C. Stereoselective Synthesis and Antiviral Activity of Methyl-Substituted cycloSal-Pronucleotides Journal of Medicinal Chemistry. 55: 7245-7252. PMID 22827702 DOI: 10.1021/Jm3008085 |
0.37 |
|
2012 |
Lunau N, Meier C. Synthesis of L‐Altrose and Some Derivatives European Journal of Organic Chemistry. 2012: 6260-6270. DOI: 10.1002/Ejoc.201200938 |
0.338 |
|
2011 |
Tonn VC, Meier C. Solid‐Phase Synthesis of (Poly)phosphorylated Nucleosides and Conjugates Chemistry: a European Journal. 17: 9832-9842. PMID 21766366 DOI: 10.1002/Chem.201101291 |
0.367 |
|
2011 |
Morales EHR, Balzarini J, Meier C. Diastereoselective synthesis of cyclosaligenyl-nucleosyl-phosphotriesters. Chemistry: a European Journal. 17: 1649-1659. PMID 21268168 DOI: 10.1002/Chem.201002657 |
0.404 |
|
2011 |
Meier C, Morales EHR, Román CA, Balzarini J. Stereoselective synthesis of 3-methyl- cyclo Sal-nucleotides Collection of Czechoslovak Chemical Communications. 12: 33-41. DOI: 10.1135/Css201112033 |
0.33 |
|
2011 |
Meier C, Hander RME, Cristina AR, Nadine L, Jan B. Stereoselective synthesis of different types of nucleotide prodrugs Antiviral Research. 90. DOI: 10.1016/J.Antiviral.2011.03.156 |
0.332 |
|
2011 |
Wolf S, Berrio RM, Meier C. Synthesis of Nonnatural Nucleoside Diphosphate Sugars European Journal of Organic Chemistry. 2011: 6304-6313. DOI: 10.1002/Ejoc.201100906 |
0.374 |
|
2011 |
Román CA, Wasserthal P, Balzarini J, Meier C. Diastereoselective Synthesis of (Aryloxy)phosphoramidate Prodrugs European Journal of Organic Chemistry. 2011: 4899-4909. DOI: 10.1002/Ejoc.201100614 |
0.448 |
|
2011 |
Morales EHR, Román CA, Thomann JO, Meier C. Linear Synthesis of Chiral cycloSal‐Pronucleotides European Journal of Organic Chemistry. 2011: 4397-4408. DOI: 10.1002/Ejoc.201100334 |
0.422 |
|
2010 |
Roman CA, Balzarini J, Meier C. Diastereoselective synthesis of aryloxy phosphoramidate prodrugs of 3'-deoxy-2',3'-didehydrothymidine monophosphate. Journal of Medicinal Chemistry. 53: 7675-81. PMID 20945915 DOI: 10.1021/Jm100817F |
0.41 |
|
2010 |
Wolf S, Zismann T, Lunau N, Warnecke S, Wendicke S, Meier C. A convenient synthesis of nucleoside diphosphate glycopyranoses and other polyphosphorylated bioconjugates. European Journal of Cell Biology. 89: 63-75. PMID 20045214 DOI: 10.1016/J.Ejcb.2009.10.013 |
0.362 |
|
2010 |
Schulz T, Balzarini J, Meier C. Lipophilic nucleoside diphosphate prodrugs – synthesis and properties Antiviral Research. 86. DOI: 10.1016/J.Antiviral.2010.02.470 |
0.36 |
|
2010 |
Schroeder M, Kolodzik A, Windshuegel B, Krepstakies M, Priyadarshini P, Rarey M, Hauber J, Meier C. Rational Drug Design—Screening and Synthesis of Potential Deoxyhypusine Synthase Inhibitors Targeting HIV-1 Replication Antiviral Research. 86. DOI: 10.1016/J.Antiviral.2010.02.469 |
0.311 |
|
2010 |
Morales ER, Roman CA, Balzarini J, Meier C. First diastereoselective synthesis of pronucleotides Antiviral Research. 86. DOI: 10.1016/J.Antiviral.2010.02.465 |
0.359 |
|
2010 |
Pertenbreiter F, Meier C. 151Nucleoside Diphosphate Prodrugs of Antivirally Active Nucleosides Antiviral Research. 86. DOI: 10.1016/J.Antiviral.2010.02.461 |
0.334 |
|
2010 |
Mahler M, Reichardt B, Balzarini J, Meier C. A chemoenzymatic synthesis of carbocyclic nucleosides and nucleotides Antiviral Research. 86. DOI: 10.1016/J.Antiviral.2010.02.454 |
0.373 |
|
2009 |
Boyer PL, Vu BC, Ambrose Z, Julias JG, Warnecke S, Liao C, Meier C, Marquez VE, Hughes SH. The nucleoside analogue D-carba T blocks HIV-1 reverse transcription. Journal of Medicinal Chemistry. 52: 5356-64. PMID 19678643 DOI: 10.1021/Jm801176E |
0.31 |
|
2009 |
Gisch N, Balzarini J, Meier C. Doubly Loaded cycloSaligenyl-Pronucleotides – 5,5′-Bis-(cycloSaligenyl-2′,3′-dideoxy-2′,3′-didehydrothymidine Monophosphates) Journal of Medicinal Chemistry. 52: 3464-3473. PMID 19438207 DOI: 10.1021/Jm900164G |
0.397 |
|
2009 |
Warnecke S, Meier C. Synthesis of Nucleoside Di- and Triphosphates and Dinucleoside Polyphosphates with cycloSal-Nucleotides Journal of Organic Chemistry. 74: 3024-3030. PMID 19320463 DOI: 10.1021/Jo802348H |
0.383 |
|
2009 |
Böge N, Jacobsen MI, Szombati Z, Baerns S, Di Pasquale F, Marx A, Meier C. Synthesis of DNA strands site-specifically damaged by c8-arylamine purine adducts and effects on various DNA polymerases. Chemistry (Weinheim An Der Bergstrasse, Germany). 14: 11194-208. PMID 18988239 DOI: 10.1002/Chem.200800979 |
0.315 |
|
2009 |
Elshehry MF, Balzarini J, Meier C. Synthesis of New Cyclic and Acyclic 5-Halouridine Derivatives as Potential Antiviral Agents Synthesis. 2009: 841-847. DOI: 10.1055/S-0028-1083369 |
0.422 |
|
2009 |
Pertenbreiter F, Meier C. Synthesis and Properties of CycloSal-phosphatetriesters of Fluorescent Bicyclic Nucleoside Analogues (BCNAS) Antiviral Research. 82. DOI: 10.1016/J.Antiviral.2009.02.149 |
0.312 |
|
2008 |
Gisch N, Pertenbreiter F, Balzarini J, Meier C. 5-(1-Acetoxyvinyl)-cycloSaligenyl-2',3'-dideoxy-2',3'- didehydrothymidine monophosphates, a second type of new, enzymatically activated cycloSaligenyl pronucleotides. Journal of Medicinal Chemistry. 51: 8115-8123. PMID 19053827 DOI: 10.1021/Jm801197F |
0.399 |
|
2008 |
Gisch N, Balzarini J, Meier C. Studies on enzyme-cleavable dialkoxymethyl-cyclosaligenyl-2',3'-dideoxy-2',3'-didehydrothymidine monophosphates. Journal of Medicinal Chemistry. 51: 6752-6760. PMID 18834186 DOI: 10.1021/Jm800853P |
0.361 |
|
2008 |
Jessen HJ, Balzarini J, Meier C. Intracellular trapping of cycloSal-pronucleotides: modification of prodrugs with amino acid esters. Journal of Medicinal Chemistry. 51: 6592-8. PMID 18826203 DOI: 10.1021/Jm800815B |
0.357 |
|
2008 |
Randhawa P, Zemlicka J, Sauerbrei A, Meier C, Hostetler KY, Beadle JR, Farasati NA, Huang Y, Bradley M. Anti-BK virus activity of nucleoside analogs. Antimicrobial Agents and Chemotherapy. 52: 1519-21. PMID 18285481 DOI: 10.1128/Aac.01241-07 |
0.302 |
|
2008 |
Wendicke S, Warnecke S, Meier C. Efficient synthesis of nucleoside diphosphate glycopyranoses. Angewandte Chemie. 47: 1500-1502. PMID 18033710 DOI: 10.1002/Anie.200703237 |
0.345 |
|
2008 |
Böge N, Krüger S, Meier C. Synthesis of N 2 - and C8- N -Ac-DNA-adducts of aromatic amines Collection of Czechoslovak Chemical Communications. 10: 137-141. DOI: 10.1135/Css200810137 |
0.316 |
|
2008 |
Boge N, Schröder M, Meier C. First Route to Phosphoramidites of N2-Hydrazinoaryl- and N2-Azoaryl-dG Adducts and Their Site-Selective Incorporation into DNA Oligonucleotides Synlett. 2008: 1066-1070. DOI: 10.1055/S-2008-1072659 |
0.301 |
|
2008 |
Schulz T, Balzarini J, Meier C. Synthesis and Properties of Glycosyl-functionalised CycloSal–Pronucleotides Antiviral Research. 78. DOI: 10.1016/J.Antiviral.2008.01.137 |
0.338 |
|
2008 |
Wendicke S, Warnecke S, Meier C. Effiziente Synthese von Nucleosiddiphosphat‐Glycopyranosen Angewandte Chemie. 120: 1523-1525. DOI: 10.1002/Ange.200703237 |
0.359 |
|
2007 |
Gisch N, Balzarini J, Meier C. 5-Diacetoxymethyl-cycloSal-d4TMP—A prototype of enzymatically activated cycloSal-pronucleotides Nucleosides, Nucleotides & Nucleic Acids. 26: 861-864. PMID 18066914 DOI: 10.1080/15257770701504025 |
0.371 |
|
2007 |
Görbig U, Balzarini J, Meier C. New cycloAmb-nucleoside phosphonate prodrugs. Nucleosides, Nucleotides & Nucleic Acids. 26: 831-834. PMID 18066909 DOI: 10.1080/15257770701503894 |
0.384 |
|
2007 |
Jessen HJ, Tonn V, Meier C. Intracellular Trapping of CycloSal-Pronucleotides by Enzymatic Cleavage Nucleosides, Nucleotides & Nucleic Acids. 26: 827-830. PMID 18066908 DOI: 10.1080/15257770701503886 |
0.325 |
|
2007 |
Böge N, Szombati Z, Meier C. Synthesis of DNA-Oligonucleotides Damaged by Arylamine-Modified 2′-Deoxyguanosine Nucleosides, Nucleotides & Nucleic Acids. 26: 705-708. PMID 18066884 DOI: 10.1080/15257770701490738 |
0.377 |
|
2007 |
Vukadinović-Tenter D, Balzarini J, Meier C. New developments of the "lock-in" modified cycloSal-d4TMPs. Nucleosides, Nucleotides & Nucleic Acids. 26: 1325-1328. PMID 18066777 DOI: 10.1080/15257770701530707 |
0.344 |
|
2007 |
Jacobsen MI, Meier C. Synthesis of C8-modified 2''-deoxyadenosine with carcinogenic arylamines. Nucleosides, Nucleotides & Nucleic Acids. 26: 1217-1220. PMID 18066755 DOI: 10.1080/15257770701527976 |
0.341 |
|
2007 |
Jessel S, Hense E, Meier C. Cyclopentane-Nucleobase Coupling in the Synthesis of Carbocyclic L-Nucleosides: is A S N 2-Reaction an Alternative to the Mitsunobu-Reaction? Nucleosides, Nucleotides & Nucleic Acids. 26: 1181-1184. PMID 18058561 DOI: 10.1080/15257770701527745 |
0.323 |
|
2007 |
Reichardt B, Meier C. A New and Short Convergent Synthetic Strategy to Carbocyclic Nucleosides Nucleosides, Nucleotides & Nucleic Acids. 26: 935-937. PMID 18058512 DOI: 10.1080/15257770701507937 |
0.394 |
|
2007 |
Gisch N, Balzarini J, Meier C. Enzymatically activated cycloSal-d4T-monophosphates: The third generation of cycloSal-pronucleotides. Journal of Medicinal Chemistry. 50: 1658-1667. PMID 17335187 DOI: 10.1021/Jm0613267 |
0.395 |
|
2007 |
Ducho C, Görbig U, Jessel S, Gisch N, Balzarini J, Meier C. Bis-cycloSal-d4T-monophosphates: Drugs That Deliver Two Molecules of Bioactive Nucleotides Journal of Medicinal Chemistry. 50: 1335-1346. PMID 17328534 DOI: 10.1021/Jm0611713 |
0.38 |
|
2007 |
Böge N, Krüger S, Schröder M, Meier C. A New Short and Efficient Synthetic Route to C8-N-Acetylarylamine 2'-Deoxyguanosine Phosphoramidites Synthesis. 2007: 3907-3914. DOI: 10.1055/S-2007-990913 |
0.361 |
|
2006 |
Böge N, Gräsl S, Meier C. Synthesis and properties of oligonucleotides containing C8-deoxyguanosine arylamine adducts of borderline carcinogens. Journal of Organic Chemistry. 71: 9728-9738. PMID 17168591 DOI: 10.1021/Jo061803T |
0.334 |
|
2006 |
Meier C, Balzarini J. Application of the cycloSal-prodrug approach for improving the biological potential of phosphorylated biomolecules Antiviral Research. 71: 282-292. PMID 16735066 DOI: 10.1016/J.Antiviral.2006.04.011 |
0.316 |
|
2006 |
Meerbach A, Meier C, Sauerbrei A, Meckel H, Wutzler P. Antiviral activity of cyclosaligenyl prodrugs of the nucleoside analogue bromovinyldeoxyuridine against herpes viruses International Journal of Antimicrobial Agents. 27: 423-430. PMID 16621459 DOI: 10.1016/J.Ijantimicag.2005.11.021 |
0.358 |
|
2006 |
Sauerbrei A, Meier C, Meerbach A, Wutzler P. Inhibitory Efficacy of CycloSal-Nucleoside Monophosphates of Aciclovir and Brivudin on DNA Synthesis of Orthopoxviruses Antiviral Chemistry & Chemotherapy. 17: 25-31. PMID 16542003 DOI: 10.1177/095632020601700104 |
0.326 |
|
2006 |
Reichardt B, Ludek OR, Meier C. New and Efficient Synthesis of Racemic Cyclopent-3-en-1-yl Nucleoside Analogues and Their Derivatives Collection of Czechoslovak Chemical Communications. 71: 1011-1028. DOI: 10.1135/Cccc20061011 |
0.398 |
|
2006 |
Jacobsen MI, Meier C. First synthesis of C8-arylamine adducts of 2'-deoxyadenosine and incorporation of the phosphoramidite into an oligonucleotide Synlett. 2006: 2411-2414. DOI: 10.1055/S-2006-950411 |
0.302 |
|
2006 |
Ludek OR, Meier C. Regioselective O- and N-Alkylation of Pyrimidine Nucleosides via the Mitsunobu Reaction Synfacts. 2006: 775-775. DOI: 10.1055/S-2006-941975 |
0.311 |
|
2006 |
Ludek OR, Krämer T, Balzarini J, Meier C. Divergent synthesis and biological evaluation of carbocyclic α-, iso- and 3′-epi-nucleosides and their lipophilic nucleotide prodrugs Synthesis. 2006: 1313-1324. DOI: 10.1055/S-2006-926411 |
0.404 |
|
2006 |
Ludek OR, Meier C. Influence of the N3‐Protection Group on N1‐ vs. O2‐Alkylation in the Mitsunobu Reaction European Journal of Organic Chemistry. 2006: 941-946. DOI: 10.1002/Ejoc.200500801 |
0.362 |
|
2006 |
Ludek OR, Balzarini J, Meier C. Synthesis and Antiviral Evaluation of Carbocyclic 3′‐Azidothymidine (AZT) Analogues and Their cycloSal‐Phosphate Triesters European Journal of Organic Chemistry. 2006: 932-940. DOI: 10.1002/Ejoc.200500719 |
0.397 |
|
2006 |
Meier C. cycloSal phosphates as chemical trojan horses for intracellular nucleotide and glycosylmonophosphate delivery - Chemistry meets biology European Journal of Organic Chemistry. 1081-1102. DOI: 10.1002/Ejoc.200500671 |
0.354 |
|
2006 |
Jessen HJ, Fendrich W, Meier C. Synthesis and Properties of Fluorescent cycloSal Nucleotides Based on the Pyrimidine Nucleoside m5K and Its 2′,3′-Dideoxy Analog dm5K European Journal of Organic Chemistry. 2006: 924-931. DOI: 10.1002/Ejoc.200500532 |
0.371 |
|
2006 |
Meier C, Ducho C, Jessen H, Vukadinović-Tenter D, Balzarini J. Second-Generation cycloSal-d4TMP Pronucleotides Bearing Esterase-Cleavable Sites — The “Trapping” Concept European Journal of Organic Chemistry. 2006: 197-206. DOI: 10.1002/Ejoc.200500490 |
0.396 |
|
2005 |
Meier C, Görbig U, Müller C, Balzarini J. cycloSal-PMEA and cycloAmb-PMEA: potentially new phosphonate prodrugs based on the cycloSal-pronucleotide approach. Journal of Medicinal Chemistry. 48: 8079-8086. PMID 16335932 DOI: 10.1021/Jm050641A |
0.366 |
|
2005 |
Meier C, Gräsl S, Detmer I, Marx A. Synthesis of oligonucleotides bearing an arylamine modification in the C8-position of 2'-deoxyguanosine. Nucleosides, Nucleotides & Nucleic Acids. 24: 691-4. PMID 16248016 DOI: 10.1081/Ncn-200060267 |
0.343 |
|
2005 |
Ludek OR, Meier C. Synthesis of carbocyclic nucleotides as potential substrates for thymidylate kinase. Nucleosides, Nucleotides & Nucleic Acids. 24: 683-686. PMID 16248014 DOI: 10.1081/Ncn-200060251 |
0.337 |
|
2005 |
Ducho C, Jessel S, Gisch N, Balzarini J, Meier C. Novel cyclosal nucleotides with reduced inhibitory potency toward human butyrylcholinesterase. Nucleosides, Nucleotides & Nucleic Acids. 24: 519-522. PMID 16247982 DOI: 10.1081/Ncn-200061791 |
0.332 |
|
2005 |
Sauerbrei A, Meier C, Meerbach A, Schiel M, Helbig B, Wutzler P. In vitro activity of cycloSal-nucleoside monophosphates and polyhydroxycarboxylates against orthopoxviruses. Antiviral Research. 67: 147-154. PMID 16076502 DOI: 10.1016/J.Antiviral.2005.06.001 |
0.341 |
|
2005 |
Ludek OR, Meier C. Synthesis of carbocyclic pyrimidine nucleosides using the mitsunobu reaction - Part II: Influence of the solvent on N1- versus O2-alkylation Synlett. 2005: 3145-3147. DOI: 10.1055/S-2005-922746 |
0.329 |
|
2004 |
Meier C, Ducho C, Görbig U, Esnouf R, Balzarini J. Interaction of cycloSal-pronucleotides with cholinesterases from different origins. A structure-activity relationship. Journal of Medicinal Chemistry. 47: 2839-2852. PMID 15139762 DOI: 10.1021/Jm031032A |
0.301 |
|
2004 |
Meier C, Ruppel MFH, Vukadinovic D, Balzarini J. Lock-in"-cycloSal-pronucleotides - a new generation of chemical Trojan Horses? Mini-Reviews in Medicinal Chemistry. 4: 383-394. PMID 15134541 DOI: 10.2174/1389557043403972 |
0.306 |
|
2004 |
Meier C, Ruppel MFH, Vukadinović D, Balzarini J. Second Generation of cycloSal‐Pronucleotides with Esterase‐Cleavable Sites: The ”Lock‐In”‐Concept Nucleosides, Nucleotides & Nucleic Acids. 23: 89-115. PMID 15043139 DOI: 10.1081/Ncn-120027820 |
0.387 |
|
2004 |
Meier C, Meerbach A, Balzarini J. Cyclosal-pronucleotides--development of first and second generation chemical trojan horses for antiviral chemotherapy. Frontiers in Bioscience. 9: 873-890. PMID 14766416 DOI: 10.2741/1283 |
0.355 |
|
2004 |
Muus U, Kranz C, Marquardt T, Meier C. cycloSaligenyl-mannose-1-monophosphates as a new strategy in CDG-Ia therapy: Hydrolysis, mechanistic insights and biological activity European Journal of Organic Chemistry. 1228-1235. DOI: 10.1002/Ejoc.200300681 |
0.335 |
|
2003 |
Fendrich W, Meier C. Determination of the absolute P-configuration of a phthalidyl-phosphonate thymidine-thymidine dimer. Nucleosides, Nucleotides & Nucleic Acids. 22: 1127-1129. PMID 14565361 DOI: 10.1081/Ncn-120022817 |
0.303 |
|
2003 |
Hohlfeld A, Meier C. α-Hydroxybenzylphosphonate modified oligonucleotides: Synthesis, properties, and a novel route via monomer building blocks Nucleosides, Nucleotides & Nucleic Acids. 22: 1123-1125. PMID 14565360 DOI: 10.1081/Ncn-120022816 |
0.351 |
|
2003 |
Gräsl S, Meier C. Synthesis of oligonucleotide building blocks of 2'-deoxyguanosine bearing a C8-arylamine modification. Nucleosides, Nucleotides & Nucleic Acids. 22: 1119-1121. PMID 14565359 DOI: 10.1081/Ncn-120022751 |
0.369 |
|
2003 |
Meier C, Renze JT, Balzarini J, De Clercq E. d4TMP delivery from 7-substituted cycloSal-d4TMPs Nucleosides, Nucleotides and Nucleic Acids. 22: 825-827. PMID 14565288 DOI: 10.1081/Ncn-120022663 |
0.323 |
|
2003 |
Müller HC, Meier C, Balzarini J, Reinstein J. Novel nucleotide analogues as potential substrates for TMPK, a key enzyme in the metabolism of AZT. Nucleosides, Nucleotides & Nucleic Acids. 22: 821-3. PMID 14565287 DOI: 10.1081/Ncn-120022662 |
0.324 |
|
2003 |
Muus U, Clercq ED, Balzarini J, Naesens L, Meier C. Study of different substituted cyclic and acyclic benzylpronucleotides of d4T relative to their hydrolytic stability and antiviral activity. Nucleosides, Nucleotides & Nucleic Acids. 22: 791-795. PMID 14565280 DOI: 10.1081/Ncn-120022636 |
0.375 |
|
2003 |
Ludek OR, Meier C. Synthesis of carbocyclic analogues of thymidine. Nucleosides, Nucleotides & Nucleic Acids. 22: 683-685. PMID 14565253 DOI: 10.1081/Ncn-120022700 |
0.38 |
|
2003 |
Mazzon C, Rampazzo C, Scaini MC, Gallinaro L, Karlsson A, Meier C, Balzarini J, Reichard P, Bianchi V. Cytosolic and mitochondrial deoxyribonucleotidases: activity with substrate analogs, inhibitors and implications for therapy. Biochemical Pharmacology. 66: 471-479. PMID 12907246 DOI: 10.1016/S0006-2952(03)00290-9 |
0.321 |
|
2003 |
Ostermann N, Segura-Peña D, Meier C, Veit T, Monnerjahn C, Konrad M, Lavie A. Structures of human thymidylate kinase in complex with prodrugs: implications for the structure-based design of novel compounds. Biochemistry. 42: 2568-77. PMID 12614151 DOI: 10.1021/Bi027302T |
0.323 |
|
2003 |
Ludek OR, Meier C. New Convergent Synthesis of Carbocyclic Nucleoside Analogues Synthesis. 2003: 2101-2109. DOI: 10.1055/S-2003-41455 |
0.387 |
|
2003 |
Ducho C, Wendicke S, Görbig U, Balzarini J, Meier C. 3,5-Di-(tert-Butyl)-6-fluoro-cycloSal-d4TMP − A Pronucleotide with a Considerably Improved Masking Group European Journal of Organic Chemistry. 2003: 4786-4791. DOI: 10.1002/Ejoc.200300537 |
0.359 |
|
2002 |
Meier C, Lomp A, Meerbach aA, Wutzler P. CycloSal-BVDUMP pronucleotides: how to convert an antiviral-inactive nucleoside analogue into a bioactive compound against EBV. Journal of Medicinal Chemistry. 45: 5157-5172. PMID 12408726 DOI: 10.1021/Jm0209275 |
0.39 |
|
2002 |
Meier C. cycloSal-pronucleotides design of chemical trojan horses Mini Reviews in Medicinal Chemistry. 2: 219-234. PMID 12370064 DOI: 10.2174/1389557023406205 |
0.33 |
|
2002 |
Ducho C, Balzarini J, Naesens L, Clercq ED, Meier C. Aryl-Substituted and Benzo-Annulated CycloSal-Derivatives of 2′,3′-Dideoxy-2′,3′-Didehydrothymidine Monophosphate — Correlation of Structure, Hydrolysis Properties and Anti-HIV Activity Antiviral Chemistry & Chemotherapy. 13: 129-141. PMID 12238530 DOI: 10.1177/095632020201300206 |
0.426 |
|
2002 |
Meier C, Muus U, Renze J, Naesens L, De Clercq E, Balzarini J. Comparative study of bis(benzyl)phosphate triesters of 2′,3′-dideoxy-2′,3′-didehydrothymidine (d4t) and cycloSal-d4TMP - Hydrolysis, mechanistic insights and anti-HIV activity Antiviral Chemistry and Chemotherapy. 13: 101-114. PMID 12238528 DOI: 10.1177/095632020201300204 |
0.448 |
|
2002 |
Meier C, Renze J, Ducho C, Balzarini J. cycloSal-d4TMP Pronucleotides-Structural Variations, Mechanistic Insights and Antiviral Activity Current Topics in Medicinal Chemistry. 2: 1111-1121. PMID 12173970 DOI: 10.2174/1568026023393183 |
0.351 |
|
2002 |
Nifantiev EE, Khrebtova SB, Kulikova YV, Predvoditelv DA, Kukhareva TS, Petrovskii PV, Rose M, Meier C. Formation of Benzooxaphosphole Oxide Heterocyclic System by the Ring-Contractive Arbuzov-Michaelis Isomerization of Alkoxy-Substituted Benzodioxaphosphorins Phosphorus Sulfur and Silicon and the Related Elements. 177: 251-259. DOI: 10.1080/10426500210234 |
0.308 |
|
2002 |
Meier C, Gräsl S. Highly efficient synthesis of a phosphoramidite building block of C8-deoxyguanosine adducts of aromatic amines Synlett. 2002: 802-804. DOI: 10.1055/S-2002-25354 |
0.381 |
|
2001 |
Balzarini J, Haller-Meier F, Clercq ED, Meier C. Antiviral Activity of Cyclosaligenyl Prodrugs of Acyclovir, Carbovir and Abacavir Antiviral Chemistry & Chemotherapy. 12: 301-306. PMID 11900349 DOI: 10.1177/095632020101200505 |
0.357 |
|
2001 |
Meier C, Lomp A, Meerbach A, Wutzler P. Synthesis, hydrolysis and anti-EBV activity of a series of 3'-modified cycloSal-BVDUMP pronucleotides. Nucleosides, Nucleotides & Nucleic Acids. 20: 307-314. PMID 11563042 DOI: 10.1081/Ncn-100002301 |
0.415 |
|
2000 |
Balzarini J, Aquaro S, Knispel T, Rampazzo C, Bianchi V, Perno CF, Clercq ED, Meier C. Cyclosaligenyl-2',3'-didehydro-2',3'-dideoxythymidine monophosphate: efficient intracellular delivery of d4TMP. Molecular Pharmacology. 58: 928-935. PMID 11040039 DOI: 10.1124/Mol.58.5.928 |
0.319 |
|
2000 |
Meerbach A, Klöcking R, Meier C, Lomp A, Helbig B, Wutzler P. Inhibitory effect of cycloSaligenyl-nucleoside monophosphates (cycloSal-NMP) of acyclic nucleoside analogues on HSV-1 and EBV. Antiviral Research. 45: 69-77. PMID 10774591 DOI: 10.1016/S0166-3542(99)00076-5 |
0.33 |
|
1999 |
Balzarini J, Naesens L, Aquaro S, Knispel T, Perno C-, Clercq ED, Meier C. Intracellular Metabolism Of Cyclosaligenyl 3'-Azido-2', 3'-Dideoxythymidine Monophosphate, A Prodrug Of 3'-Azido-2', 3'-Dideoxythymidine (Zidovudine) Molecular Pharmacology. 56: 1354-1361. PMID 10570065 DOI: 10.1124/Mol.56.6.1354 |
0.327 |
|
1999 |
Lorey M, Meier C. A new cyclic phosphoramidate D4T prodrug approach cycloAmb-D4T-phosphoramidates. Nucleosides, Nucleotides & Nucleic Acids. 18: 947-948. PMID 10432716 DOI: 10.1080/15257779908041608 |
0.321 |
|
1999 |
Mugnier F, Meier C. Phosphoramidite Chemistry for the Synthesis of cycloSal-Pro-Nucleotides Nucleosides, Nucleotides & Nucleic Acids. 18: 941-942. PMID 10432714 DOI: 10.1080/15257779908041605 |
0.389 |
|
1999 |
Meier C, Knispel T, Marquez VE, Clercq ED, Balzarini J. CycloSal-2'-ara(ribo)-fluoro-2',3'-dideoxyadenosine monophosphates--an effort to solve the structure-activity relationship of 2'-fluoro-ddA. Nucleosides, Nucleotides & Nucleic Acids. 18: 907-912. PMID 10432708 DOI: 10.1080/15257779908041598 |
0.37 |
|
1999 |
Meier C, Knispel T, Marquez VE, Siddiqui MA, Clercq ED, Balzarini J. cycloSal-Pronucleotides of 2'-fluoro-ara- and 2'-fluoro-ribo-2',3'- dideoxyadenosine as a strategy to bypass a metabolic blockade. Journal of Medicinal Chemistry. 42: 1615-1624. PMID 10229630 DOI: 10.1021/Jm981097R |
0.329 |
|
1999 |
Meier C, Knispel T, Clercq ED, Balzarini J. cycloSal-Pronucleotides of 2',3'-dideoxyadenosine and 2', 3'-dideoxy-2',3'-didehydroadenosine: synthesis and antiviral evaluation of a highly efficient nucleotide delivery system. Journal of Medicinal Chemistry. 42: 1604-1614. PMID 10229629 DOI: 10.1021/Jm981096Z |
0.389 |
|
1999 |
Knispel T, Meier C. N,O-Selectivity in the Synthesis of 3-Me-CycloSal-ddAMP Nucleosides, Nucleotides & Nucleic Acids. 18: 945-946. DOI: 10.1080/15257779908041607 |
0.302 |
|
1998 |
Meier C, Habel L, Haller-Meier F, Lomp A, Herderich M, Klöcking R, Meerbach A, Wutzler P. Chemistry and anti-herpes simplex virus type 1 evaluation of cycloSal-nucleotides of acyclic nucleoside analogues Antiviral Chemistry & Chemotherapy. 9: 389-402. PMID 9875392 DOI: 10.1177/095632029800900503 |
0.379 |
|
1998 |
Meier C, Aubertin AM, de Monte M, Faraj A, Sommadossi JP, Périgaud C, Imbach JL, Gosselin G. Synthesis and antiviral evaluation of SATE-foscarnet prodrugs and new foscarnet-AZT conjugates. Antiviral Chemistry & Chemotherapy. 9: 41-52. PMID 9875376 DOI: 10.1177/095632029800900105 |
0.436 |
|
1998 |
Meier C, Lorey M, De Clercq E, Balzarini J. cycloSal-2',3'-dideoxy-2',3'-didehydrothymidine monophosphate (cycloSal-d4TMP): synthesis and antiviral evaluation of a new d4TMP delivery system. Journal of Medicinal Chemistry. 41: 1417-27. PMID 9554875 DOI: 10.1021/JM970664S |
0.311 |
|
1998 |
Meier C, Clercq ED, Balzarini J. Nucleotide Delivery from cycloSaligenyl‐3′‐azido‐3′‐deoxythymidine Monophosphates (cycloSal‐AZTMP) European Journal of Organic Chemistry. 1998: 837-846. DOI: 10.1002/(Sici)1099-0690(199805)1998:5<837::Aid-Ejoc837>3.0.Co;2-7 |
0.368 |
|
1997 |
Habel LW, Meier C. Di-ddU-α-Hydroxyphosphonate and α-Hydroxy- α- METHYLPHOSPHONATES as Potential Prodrugs of Antiviral Nucleoside Analogues Nucleosides, Nucleotides & Nucleic Acids. 16: 1311-1314. DOI: 10.1080/07328319708006178 |
0.336 |
|
1997 |
Lorey M, Meier C, Clercq ED, Balzarini J. Cyclo-saligenyl-5-fluoro-2′-deoxyuridinemonophosphate (cycloSal-FdUMP) — A New Prodrug Approach for FdUMP Nucleosides, Nucleotides & Nucleic Acids. 16: 1307-1310. DOI: 10.1080/07328319708006177 |
0.368 |
|
1997 |
Meier C, Lorey M, Clercq ED, Balzarini J. Cyclo-saligenyl-2′,3′-dideoxy-2′,3′-didehydroythymidinemonophosphate (cycloSal-d4TMP) — A New Pro-Nucleotide Approach Nucleosides, Nucleotides & Nucleic Acids. 16: 1303-1306. DOI: 10.1080/07328319708006176 |
0.388 |
|
1997 |
Mauritz RP, Meier C, Uhlmann E. Synthesis of 3′,5′-Dithymidylyl-α-hydroxyphosphonate Dimer Building Blocks for Oligonucleotide Synthesis—A New Pro-oliguncleotide Nucleosides, Nucleotides & Nucleic Acids. 16: 1209-1212. DOI: 10.1080/07328319708006159 |
0.372 |
|
1997 |
Mauritz RP, Meier C. Fpmp-Protected α-Hydroxyphosphonate Diesters for The Synthesis of Pro-Oligonucleotides Nucleosides, Nucleotides & Nucleic Acids. 16: 675-678. DOI: 10.1080/07328319708002933 |
0.374 |
|
1997 |
Meier C, Knispel T, Clercq ED, Balzarini J. ADA-Bypass by lipophilic cycloSal-ddAMP pro-nucleotides A second example of the efficiency of the cycloSal-Concept Bioorganic & Medicinal Chemistry Letters. 7: 1577-1582. DOI: 10.1016/S0960-894X(97)00265-5 |
0.354 |
|
1997 |
Meier C, Lorey M, Clercq ED, Balzarini J. Cyclic saligenyl phosphotriesters of 2′,3′-dideoxy-2′,3′-didehydrothymidine (d4T) — a new pro-nucleotide approach Bioorganic & Medicinal Chemistry Letters. 7: 99-104. DOI: 10.1016/S0960-894X(96)00597-5 |
0.394 |
|
1996 |
Meier C, Laux WHG. Asymmetric synthesis of chiral, Nonracemic dialkyl-α-hydroxyalkylphosphonates via a (−)-Chlorodiiso-pinocampheylborane (Ipc2B-Cl) reduction Tetrahedron-Asymmetry. 7: 89-94. DOI: 10.1016/0957-4166(95)00424-6 |
0.363 |
|
1996 |
Meier C, Laux WHG. Enantioselective synthesis of diisopropyl α-, β-, and γ-hydroxyarylalkylphosphonates from ketophosphonates: A study on the effect of the phosphonyl group Tetrahedron. 52: 589-598. DOI: 10.1016/0040-4020(95)00855-1 |
0.314 |
|
1996 |
Meier C. 2‐Nucleos‐5′‐O‐yl‐4H‐1,3,2‐benzodioxaphos‐phinin‐2‐oxides—A New Concept for Lipophilic, Potential Prodrugs of Biologically Active Nucleoside Monophosphates Angewandte Chemie. 35: 70-72. DOI: 10.1002/Anie.199600701 |
0.316 |
|
1996 |
Meier C. 2‐Nucleos‐5′‐O‐yl‐4H‐1,3,2‐benzodioxaphosphinin‐2‐oxide—ein neues Konzept für lipophile, potentielle Prodrugs biologisch' aktiver Nucleosidmonophosphate Angewandte Chemie. 108: 77-79. DOI: 10.1002/Ange.19961080112 |
0.317 |
|
1995 |
Meier C, Mauritz R. Synthesis Of Protected 3',5'-Dl-2'-deoxythymidine-(α-hydroxy-2-nitrobenzyl)-phosphonatediesters as dimer building blocks for oligonucleotides Nucleosides and Nucleotides. 14: 803-804. DOI: 10.1080/15257779508012475 |
0.34 |
|
1995 |
Meier C, Habel L, Laux W, Clercq ED, Balzarini J. Homo Dinucleoside-α-hydroxyphosphonate Diesters as Prodrugs of the Antiviral Nucleoside Analogues 2′,3′-Dideoxythymidine and 3′-Azido-2′,3′-dideoxythymidine Nucleosides, Nucleotides & Nucleic Acids. 14: 759-762. DOI: 10.1080/15257779508012466 |
0.419 |
|
1995 |
Meier C, Laux WHG. Asymmetric synthesis of chiral, nonracemic dialkyl-α-, β-, and γ-hydroxyalkylphosphonates via a catalyzed enantioselective catecholborane reduction Tetrahedron-Asymmetry. 6: 1089-1092. DOI: 10.1016/0957-4166(95)00132-9 |
0.332 |
|
1995 |
Meier C, Habel LW, Balzarini J, Clercq ED. 5′,5′‐di‐O‐nucleosyl‐O′‐benzylphosphotriesters as potential prodrugs of 3′‐azido‐2′,3′‐dideoxythymidine‐5′‐monophosphate Liebigs Annalen. 1995: 2203-2208. DOI: 10.1002/Jlac.1995199512306 |
0.428 |
|
1995 |
Meier C, Habel LW, Balzarini J, Clercq ED. Lipophilic α‐hydroxybenzylphosphonates as prodrugs of 3′‐azido‐2′,3′‐dideoxythymidine (AZT) Liebigs Annalen. 1995: 2195-2202. DOI: 10.1002/Jlac.1995199512305 |
0.414 |
|
1995 |
Meier C, Laux WHG, Bats JW. Asymmetric synthesis of chiral, nonracemic dialkyl α‐hydroxyarylmethyl‐and α‐, β‐ and γ‐hydroxyalkylphosphonates from keto phosphonates Liebigs Annalen. 1995: 1963-1979. DOI: 10.1002/Jlac.1995199511276 |
0.386 |
|
1993 |
Meier C. Lipophilic 5′,5′‐O‐Dinucleoside‐α‐hydroxybenzylphosphonic Acid Esters as Potential Prodrugs of 2′,3′‐Dideoxythymidine (ddT) Angewandte Chemie. 32: 1704-1706. DOI: 10.1002/Anie.199317041 |
0.325 |
|
1992 |
Meier C, Neumann JM, Andre F, Henin Y, Tam HD. O-Alkyl-5',5'-dinucleoside phosphates as prodrugs of 3'-azidothymidine and cordycepin Journal of Organic Chemistry. 57: 7300-7308. DOI: 10.1021/Jo00052A053 |
0.309 |
|
1991 |
Meier C, Boche G. The modification of guanine nucleosides and nucleotides by the borderline arylamine carcinogens 4-methyl- and 4-methoxyaniline: Chemishy and structural characterization Carcinogenesis. 12: 1633-1640. PMID 1893521 DOI: 10.1093/Carcin/12.9.1633 |
0.513 |
|
1991 |
Meier C, Huynh-Dinh T. O-alkyl-5′-,5′-dinucleoside-phosphates as combined prodrugs of antiviral and antibiotic compounds Bioorganic & Medicinal Chemistry Letters. 1: 527-530. DOI: 10.1016/S0960-894X(01)80459-5 |
0.4 |
|
1990 |
Meier C, Boche G. N-acetoxy-4-methoxyaniline, a model compound for the ultimate carcinogen of the phenacetin belated 4-ethoxyaniline Tetrahedron Letters. 31: 1693-1696. DOI: 10.1016/S0040-4039(00)88856-5 |
0.505 |
|
1990 |
Meier C, Boche G. N- (α-aminoacyloxy)-N-arylamines: Activation of aromatic amines to ultimate carcinogens by amino acids Tetrahedron Letters. 31: 1685-1688. DOI: 10.1016/S0040-4039(00)88854-1 |
0.519 |
|
1990 |
MEIER C, BOCHE G. ChemInform Abstract: 1H and 13C NMR Conformational Analysis and Minimal-Potential-Energy Calculations with Deoxyguanosine, Guanosine and 5′-Guanosinemonophosphate Adducts of the Borderline Carcinogen 4-Methylaniline. Cheminform. 21. DOI: 10.1002/CHIN.199045313 |
0.427 |
|
1990 |
MEIER C, BOCHE G. ChemInform Abstract: N-Aryl-O-(α-aminoacyl)hydroxylamines: Model Reactions with Deoxyguanosine, Guanosine and 5′-Guanosinemonophosphate for the Activation of Monocyclic Aromatic Amines (e.g. Phenacetin) into Ultimate Carcinogens. Cheminform. 21. DOI: 10.1002/CHIN.199044275 |
0.49 |
|
1990 |
MEIER C, BOCHE G. ChemInform Abstract: N-Aryl-O-(α-aminoacyl)hydroxylamines: Model Reactions for the Activation of Monocyclic Aromatic Amines into Ultimate Carcinogens with α-Amino Acids. Cheminform. 21. DOI: 10.1002/CHIN.199044274 |
0.489 |
|
1990 |
Meier C, Boche G. 1H- und 13C-NMR-Konformationsanalysen und Minimal-Potential-Energie-Rechnungen an Desoxyguanosin-, Guanosin- und 5′-Guanosinmonophosphat-Addukten des Grenzcarcinogens 4-Methylanilin Chemische Berichte. 123: 1707-1713. DOI: 10.1002/Cber.19901230821 |
0.517 |
|
1990 |
Meier C, Boche G. N‐Aryl‐O‐(α‐aminoacyl)hydroxylamine: Modellreaktionen mit Desoxyguanosin, Guanosin und 5′‐Guanosinmonophosphat zur Aktivierung monocyclischer aromatischer Amine (z. B. Phenacetin) zu ultimaten Carcinogenen Chemische Berichte. 123: 1699-1705. DOI: 10.1002/Cber.19901230820 |
0.563 |
|
1990 |
Meier C, Boche G. N‐Aryl‐O‐(α‐aminoacyl)hydroxylamine: Modellreaktionen zur Aktivierung von monocyclischen aromatischen Aminen zu ultimaten Carcinogenen durch α‐Aminosäuren Chemische Berichte. 123: 1691-1698. DOI: 10.1002/Cber.19901230819 |
0.543 |
|
1988 |
Boche G, Meier C, Kleemiβ W. Hydrazines and azo compounds from O-diphenylphosphinoyl arylhydroxylamines Tetrahedron Letters. 29: 1777-1779. DOI: 10.1016/S0040-4039(00)82041-9 |
0.534 |
|
Show low-probability matches. |