| Year |
Citation |
Score |
| 2017 |
Detroja DP, Chen TL, Lin YW, Yen TY, Wu MH, Tsai TH, Maheriya K, Kakadiya R, Lee TC, Shah A, Su TL. Novel N-mustard-benzimidazoles/benzothiazoles hybrids, synthesis and anticancer evaluation. Anti-Cancer Agents in Medicinal Chemistry. PMID 28530540 DOI: 10.2174/1871520617666170522120200 |
0.655 |
|
| 2016 |
Viradiya D, Mirza S, Shaikh F, Kakadiya R, Rathod A, Jain N, Rawal R, Shah A. Design and synthesis of 1,4-dihydropyridine derivatives as anti-cancer agent. Anti-Cancer Agents in Medicinal Chemistry. PMID 27924733 DOI: 10.2174/1871520616666161206143251 |
0.568 |
|
| 2014 |
Marvania B, Kakadiya R, Christian W, Chen TL, Wu MH, Suman S, Tala K, Lee TC, Shah A, Su TL. The synthesis and biological evaluation of new DNA-directed alkylating agents, phenyl N-mustard-4-anilinoquinoline conjugates containing a urea linker. European Journal of Medicinal Chemistry. 83: 695-708. PMID 25014640 DOI: 10.1016/J.Ejmech.2014.06.066 |
0.7 |
|
| 2014 |
Sanjiv K, Chen CW, Kakadiya R, Tala S, Suman S, Wu MH, Chen YH, Su TL, Lee TC. PI3K Inhibition Augments the Therapeutic Efficacy of a 3a-aza-Cyclopenta[α]indene Derivative in Lung Cancer Cells. Translational Oncology. 7: 256-266.e5. PMID 24913674 DOI: 10.1016/j.tranon.2014.02.012 |
0.352 |
|
| 2014 |
Tala SD, Ou TH, Lin YW, Tala KS, Chao SH, Wu MH, Tsai TH, Kakadiya R, Suman S, Chen CH, Lee TC, Su TL. Design and synthesis of potent antitumor water-soluble phenyl N-mustard-benzenealkylamide conjugates via a bioisostere approach. European Journal of Medicinal Chemistry. 76: 155-69. PMID 24583355 DOI: 10.1016/j.ejmech.2014.02.018 |
0.486 |
|
| 2013 |
Su TL, Lee TC, Kakadiya R. The development of bis(hydroxymethyl)pyrrole analogs as bifunctional DNA cross-linking agents and their chemotherapeutic potential. European Journal of Medicinal Chemistry. 69: 609-21. PMID 24095754 DOI: 10.1016/j.ejmech.2013.09.016 |
0.383 |
|
| 2013 |
Chaniyara R, Tala S, Chen CW, Zang X, Kakadiya R, Lin LF, Chen CH, Chien SI, Chou TC, Tsai TH, Lee TC, Shah A, Su TL. Novel antitumor indolizino[6,7-b]indoles with multiple modes of action: DNA cross-linking and topoisomerase I and II inhibition. Journal of Medicinal Chemistry. 56: 1544-63. PMID 23360284 DOI: 10.1021/Jm301788A |
0.681 |
|
| 2012 |
Chaniyara R, Tala S, Chen CW, Lee PC, Kakadiya R, Dong H, Marvania B, Chen CH, Chou TC, Lee TC, Shah A, Su TL. Synthesis and antitumor evaluation of novel benzo[d]pyrrolo[2,1-b]thiazole derivatives. European Journal of Medicinal Chemistry. 53: 28-40. PMID 22507893 DOI: 10.1016/J.Ejmech.2012.03.030 |
0.686 |
|
| 2012 |
Sanjiv K, Su TL, Suman S, Kakadiya R, Lai TC, Wang HY, Hsiao M, Lee TC. The novel DNA alkylating agent BO-1090 suppresses the growth of human oral cavity cancer in xenografted and orthotopic mouse models. International Journal of Cancer. 130: 1440-50. PMID 21500194 DOI: 10.1002/ijc.26142 |
0.408 |
|
| 2011 |
Kakadiya R, Wu YC, Dong H, Kuo HH, Yih LH, Chou TC, Su TL. Novel 2-substituted quinolin-4-yl-benzenesulfonate derivatives: synthesis, antiproliferative activity, and inhibition of cellular tubulin polymerization. Chemmedchem. 6: 1119-29. PMID 21542133 DOI: 10.1002/cmdc.201100121 |
0.423 |
|
| 2011 |
Marvania B, Lee PC, Chaniyara R, Dong H, Suman S, Kakadiya R, Chou TC, Lee TC, Shah A, Su TL. Design, synthesis and antitumor evaluation of phenyl N-mustard-quinazoline conjugates. Bioorganic & Medicinal Chemistry. 19: 1987-98. PMID 21356592 DOI: 10.1016/J.Bmc.2011.01.055 |
0.722 |
|
| 2011 |
Chaniyara R, Kapuriya N, Dong H, Lee PC, Suman S, Marvania B, Chou TC, Lee TC, Kakadiya R, Shah A, Su TL. Novel bifunctional alkylating agents, 5,10-dihydropyrrolo[1,2-b]isoquinoline derivatives, synthesis and biological activity. Bioorganic & Medicinal Chemistry. 19: 275-86. PMID 21144756 DOI: 10.1016/J.Bmc.2010.11.030 |
0.68 |
|
| 2011 |
Kapuriya N, Kakadiya R, Dong H, Kumar A, Lee PC, Zhang X, Chou TC, Lee TC, Chen CH, Lam K, Marvania B, Shah A, Su TL. Design, synthesis, and biological evaluation of novel water-soluble N-mustards as potential anticancer agents. Bioorganic & Medicinal Chemistry. 19: 471-85. PMID 21106377 DOI: 10.1016/J.Bmc.2010.11.005 |
0.702 |
|
| 2010 |
Lee PC, Kakadiya R, Su TL, Lee TC. Combination of bifunctional alkylating agent and arsenic trioxide synergistically suppresses the growth of drug-resistant tumor cells. Neoplasia (New York, N.Y.). 12: 376-87. PMID 20454509 |
0.407 |
|
| 2010 |
Kakadiya R, Dong H, Kumar A, Narsinh D, Zhang X, Chou TC, Lee TC, Shah A, Su TL. Potent DNA-directed alkylating agents: Synthesis and biological activity of phenyl N-mustard-quinoline conjugates having a urea or hydrazinecarboxamide linker. Bioorganic & Medicinal Chemistry. 18: 2285-99. PMID 20181487 DOI: 10.1016/J.Bmc.2010.01.061 |
0.748 |
|
| 2009 |
Kakadiya R, Dong H, Lee PC, Kapuriya N, Zhang X, Chou TC, Lee TC, Kapuriya K, Shah A, Su TL. Potent antitumor bifunctional DNA alkylating agents, synthesis and biological activities of 3a-aza-cyclopenta[a]indenes. Bioorganic & Medicinal Chemistry. 17: 5614-26. PMID 19576785 DOI: 10.1016/J.Bmc.2009.06.018 |
0.677 |
|
| 2008 |
Chen CH, Lin YW, Zhang X, Chou TC, Tsai TJ, Kapuriya N, Kakadiya R, Su TL. Synthesis and in vitro cytotoxicity of 9-anilinoacridines bearing N-mustard residue on both anilino and acridine rings. European Journal of Medicinal Chemistry. 44: 3056-9. PMID 18752869 DOI: 10.1016/j.ejmech.2008.07.016 |
0.369 |
|
| 2008 |
Kapuriya N, Kapuriya K, Zhang X, Chou TC, Kakadiya R, Wu YT, Tsai TH, Chen YT, Lee TC, Shah A, Naliapara Y, Su TL. Synthesis and biological activity of stable and potent antitumor agents, aniline nitrogen mustards linked to 9-anilinoacridines via a urea linkage. Bioorganic & Medicinal Chemistry. 16: 5413-23. PMID 18450456 DOI: 10.1016/J.Bmc.2008.04.024 |
0.758 |
|
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