Rob Leurs
Affiliations: | Medicinal Chemistry | Vrije Universiteit Amsterdam, Amsterdam, Netherlands |
Area:
GPCRs, Histamine receptors, Chemokine receptorsWebsite:
http://www.chem.vu.nl/en/research/division-of-medicinal-chemistry/index.aspGoogle:
"Rob Leurs"Mean distance: 13.53 | S | N | B | C | P |
Children
Sign in to add trainee| Martine Joyce Smit | grad student | 1995 | VU Amsterdam |
| Richard M. Van Rijn | grad student | 2002-2006 | VU Amsterdam (Neurotree) |
| Kamonchanok Sansuk | grad student | 2004-2008 | Vrije Universiteit, Amsterdam, Sheffield (Neurotree) |
BETA: Related publications
See more...
Publications
|
You can help our author matching system! If you notice any publications incorrectly attributed to this author, please sign in and mark matches as correct or incorrect. |
| Xia R, Shi S, Xu Z, et al. (2024) Structural basis of ligand recognition and design of antihistamines targeting histamine H receptor. Nature Communications. 15: 2493 |
| Gao M, Dekker ME, Leurs R, et al. (2024) Pharmacological characterization of seven human histamine H receptor isoforms. European Journal of Pharmacology. 968: 176450 |
| Zarca A, Adlere I, Viciano CP, et al. (2024) Pharmacological characterization and radiolabeling of VUF15485, a high-affinity small-molecule agonist for the atypical chemokine receptor ACKR3. Molecular Pharmacology |
| Dekkers S, Comez D, Karsai N, et al. (2023) Small Molecule Fluorescent Ligands for the Atypical Chemokine Receptor 3 (ACKR3). Acs Medicinal Chemistry Letters. 15: 143-148 |
| Rahman SN, Imhaouran F, Leurs R, et al. (2023) Ligand-directed biased agonism at human histamine H receptor isoforms across Gα- and β-arrestin2-mediated pathways. Biochemical Pharmacology. 115988 |
| McNaught-Flores DA, Kooistra AJ, Chen YC, et al. (2023) Pharmacological characterization of the zebrafish () histamine H receptor reveals the involvement of the second extracellular loop in the binding of histamine. Molecular Pharmacology |
| Rahman SN, McNaught-Flores DA, Huppelschoten Y, et al. (2023) Structural and Molecular Determinants for Isoform Bias at Human Histamine H Receptor Isoforms. Acs Chemical Neuroscience |
| Wágner G, Mocking TAM, Ma X, et al. (2022) SAR exploration of the non-imidazole histamine H receptor ligand ZEL-H16 reveals potent inverse agonism. Archiv Der Pharmazie. e2200451 |
| Ma X, Gao M, Vischer HF, et al. (2022) A NanoBRET-Based HR Conformational Biosensor to Study Real-Time H Receptor Pharmacology in Cell Membranes and Living Cells. International Journal of Molecular Sciences. 23 |
| Zheng Y, Wágner G, Hauwert N, et al. (2022) New Chemical Biology Tools for the Histamine Receptor Family. Current Topics in Behavioral Neurosciences |