Nicholas Griggs
Affiliations: | University of Michigan, Ann Arbor, Ann Arbor, MI |
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| Montgomery D, Anand JP, Griggs N, et al. (2019) Novel Dimethyltyrosine-Tetrahydroisoquinoline Peptidomimetics with Aromatic Tetrahydroisoquinoline Substitutions Show In Vitro Kappa and Mu Opioid Receptor Agonism. Acs Chemical Neuroscience |
| Henry S, Fernandez TM, Anand JP, et al. (2019) Structural Simplification of a Tetrahydroquinoline Core Peptidomimetic µ-Opioid-Receptor (MOR) Agonist/ δ-Opioid Receptor (DOR) Antagonist Produces Improved Metabolic Stability . Journal of Medicinal Chemistry |
| Nastase AF, Anand JP, Bender AM, et al. (2019) Dual Pharmacophores Explored via Structure-Activity Relationship (SAR) Matrix: Insights into Potent, Bifunctional Opioid Ligand Design. Journal of Medicinal Chemistry |
| Nastase AF, Griggs NW, Anand JP, et al. (2018) Synthesis and pharmacological evaluation of novel C-8 substituted tetrahydroquinolines as balanced-affinity mu/delta opioid ligands for the treatment of pain. Acs Chemical Neuroscience |
| Anand JP, Kochan KE, Nastase AF, et al. (2018) In Vivo Effects of μ Opioid Receptor Agonist/δ Opioid Receptor Antagonist Peptidomimetics Following Acute and Repeated Administration. British Journal of Pharmacology |
| Harland AA, Pogozheva ID, Griggs NW, et al. (2017) Placement of hydroxy moiety on pendant of peptidomimetic scaffold modulates mu and kappa opioid receptor efficacy. Acs Chemical Neuroscience |
| Healy JR, Bezawada P, Griggs NW, et al. (2016) Benzylideneoxymorphone: A new lead for development of bifunctional mu/delta opioid receptor ligands. Bioorganic & Medicinal Chemistry Letters |
| Harland AA, Bender AM, Griggs NW, et al. (2016) Effects of N-Substitutions on the Tetrahydroquinoline (THQ) core of Mixed-Efficacy μ-Opioid Receptor (MOR)/ δ-Opioid Receptor (DOR) Ligands. Journal of Medicinal Chemistry |
| Bender AM, Griggs NW, Gao C, et al. (2015) Rapid Synthesis of Boc-2',6'-dimethyl-l-tyrosine and Derivatives and Incorporation into Opioid Peptidomimetics. Acs Medicinal Chemistry Letters. 6: 1199-203 |
| Yao XQ, Malik R, Griggs NW, et al. (2015) Dynamic coupling and allosteric networks in the alpha subunit of heterotrimeric G proteins. The Journal of Biological Chemistry |