David B. Sattelle - Related publications

University College London, London, United Kingdom 
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50 most relevant papers in past 60 days:
Year Citation  Score
2020 Marcovich I, Moglie MJ, Carpaneto Freixas AE, Trigila AP, Franchini LF, Plazas PV, Lipovsek M, Elgoyhen AB. Distinct Evolutionary Trajectories of Neuronal and Hair Cell Nicotinic Acetylcholine Receptors. Molecular Biology and Evolution. 37: 1070-1089. PMID 31821508 DOI: 10.1093/molbev/msz290   
2020 Rufener L, Kaur K, Sarr A, Aaen SM, Horsberg TE. Nicotinic acetylcholine receptors: Ex-vivo expression of functional, non-hybrid, heteropentameric receptors from a marine arthropod, Lepeophtheirus salmonis. Plos Pathogens. 16: e1008715. PMID 32716968 DOI: 10.1371/journal.ppat.1008715   
2020 Corrie LW, Stokes C, Wilkerson JL, Carroll FI, McMahon LR, Papke RL. Nicotinic Acetylcholine Receptor Accessory Subunits Determine the Activity Profile of Epibatidine Derivatives. Molecular Pharmacology. PMID 32690626 DOI: 10.1124/molpharm.120.000037   
2020 Ghimire M, Cai R, Ling L, Hackett TA, Caspary DM. Nicotinic Receptor Subunit Distribution in Auditory Cortex: Impact of Aging on Receptor Number and Function. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. PMID 32541068 DOI: 10.1523/JNEUROSCI.0093-20.2020   
2020 Oliveira ASF, Ibarra AA, Bermudez I, Casalino L, Gaieb Z, Shoemark DK, Gallagher T, Sessions RB, Amaro RE, Mulholland AJ. Simulations support the interaction of the SARS-CoV-2 spike protein with nicotinic acetylcholine receptors and suggest subtype specificity. Biorxiv : the Preprint Server For Biology. PMID 32743575 DOI: 10.1101/2020.07.16.206680   
2020 Nirthanan S. Snake three-finger α-neurotoxins and nicotinic acetylcholine receptors: molecules, mechanisms and medicine. Biochemical Pharmacology. 114168. PMID 32710970 DOI: 10.1016/j.bcp.2020.114168   
2020 Xu Q, Tae HS, Wang Z, Jiang T, Adams DJ, Yu R. Rational Design of α-Conotoxin RegIIA Analogues Specifically Inhibiting the Human α3β2 Nicotinic Acetylcholine Receptor through Computational Scanning. Acs Chemical Neuroscience. PMID 32649832 DOI: 10.1021/acschemneuro.0c00293   
2020 Johnson K, Yin J, In JG, Kulkarni S, Pasricha P, Tse M, Donowitz M. Cholinergic-induced anion secretion in murine jejunal enteroids involves synergy between muscarinic and nicotinic pathways. American Journal of Physiology. Cell Physiology. PMID 32551856 DOI: 10.1152/ajpcell.00179.2020   
2020 Gelfuso EA, Reis SL, Aguiar DSR, Faggion SA, Gomes FMM, Galan DT, Peigneur S, Pereira AMS, Mortari MR, Cunha AOS, Tytgat J, Beleboni RO. New insights in the mode of action of (+)-erythravine and (+)-11α-hydroxy-erythravine alkaloids. European Journal of Pharmacology. 173390. PMID 32735983 DOI: 10.1016/j.ejphar.2020.173390   
2020 Changeux JP. Golden Anniversary of the Nicotinic Receptor. Neuron. 107: 14-16. PMID 32645305 DOI: 10.1016/j.neuron.2020.05.026   
2020 Falk-Petersen CB, Tsonkov TM, Nielsen MS, Harpsøe K, Bundgaard C, Frølund B, Kristiansen U, Gloriam DE, Wellendorph P. Discovery of a new class of orthosteric antagonists with nanomolar potency at extrasynaptic GABA receptors. Scientific Reports. 10: 10078. PMID 32572053 DOI: 10.1038/s41598-020-66821-0   
2020 Fujii N, McGarr GW, Ghassa R, Schmidt MD, McCormick JJ, Nishiyasu T, Kenny GP. Sex-differences in cholinergic, nicotinic, and β-adrenergic cutaneous vasodilation: Roles of nitric oxide synthase, cyclooxygenase, and K channels. Microvascular Research. 131: 104030. PMID 32531353 DOI: 10.1016/j.mvr.2020.104030   
2020 Tsetlin VI, Kasheverov IE, Utkin YN. Three-finger proteins from snakes and humans acting on nicotinic receptors: old and new. Journal of Neurochemistry. PMID 32648941 DOI: 10.1111/jnc.15123   
2020 Gillet C, Kurth S, Kuenzel T. Muscarinic modulation of M and h currents in gerbil spherical bushy cells. Plos One. 15: e0226954. PMID 31940388 DOI: 10.1371/journal.pone.0226954   
2020 Ihara M, Furutani S, Shigetou S, Shimada S, Niki K, Komori Y, Kamiya M, Koizumi W, Magara L, Hikida M, Noguchi A, Okuhara D, Yoshinari Y, Kondo S, Tanimoto H, et al. Cofactor-enabled functional expression of fruit fly, honeybee, and bumblebee nicotinic receptors reveals picomolar neonicotinoid actions. Proceedings of the National Academy of Sciences of the United States of America. PMID 32611810 DOI: 10.1073/pnas.2003667117   
2020 Tsetlin VI. Acetylcholine and Acetylcholine Receptors: Textbook Knowledge and New Data. Biomolecules. 10. PMID 32503306 DOI: 10.3390/biom10060852   
2020 Homem RA, Buttery B, Richardson EE, Tan Y, Field LM, Williamson MS, Davies TGE. Evolutionary trade-offs of insecticide resistance - the fitness costs associated with target-site mutations in the nAChR of Drosophila melanogaster. Molecular Ecology. PMID 32510730 DOI: 10.1111/mec.15503   
2020 Salazar H, Mischke S, Plested AJR. Measurements of the Timescale and Conformational Space of AMPA Receptor Desensitization. Biophysical Journal. PMID 32559412 DOI: 10.1016/j.bpj.2020.05.029   
2020 Park J, Fu Z, Frangaj A, Liu J, Mosyak L, Shen T, Slavkovich VN, Ray KM, Taura J, Cao B, Geng Y, Zuo H, Kou Y, Grassucci R, Chen S, et al. Structure of human GABA receptor in an inactive state. Nature. PMID 32581365 DOI: 10.1038/s41586-020-2452-0   
2020 Huynh PN, Harvey PJ, Gajewiak J, Craik DJ, Michael McIntosh J. Critical residue properties for potency and selectivity of α-Conotoxin RgIA towards α9α10 nicotinic acetylcholine receptors. Biochemical Pharmacology. 114124. PMID 32593612 DOI: 10.1016/j.bcp.2020.114124   
2020 Germann AL, Reichert DE, Burbridge AB, Pierce SR, Evers AS, Steinbach JH, Akk G. Analysis of modulation of the ρ1 GABAA receptor by combinations of inhibitory and potentiating neurosteroids reveals shared and distinct binding sites. Molecular Pharmacology. PMID 32675382 DOI: 10.1124/mol.120.119842   
2020 Dalby NO, Falk-Petersen CB, Leurs U, Scholze P, Krall J, Frølund B, Wellendorph P. Silencing of spontaneous activity at α4β1/3δ GABA receptors in hippocampal granule cells reveals different ligand pharmacology. British Journal of Pharmacology. PMID 32484592 DOI: 10.1111/bph.15146   
2020 Liu JYH, Du P, Rudd JA. Acetylcholine Exerts Inhibitory and Excitatory Actions on Mouse Ileal Pacemaker Activity: The Role of Muscarinic versus Nicotinic Receptors. American Journal of Physiology. Gastrointestinal and Liver Physiology. PMID 32475128 DOI: 10.1152/ajpgi.00003.2020   
2020 Mitra S, Khatri SN, Maulik M, Bult-Ito A, Schulte M. Allosterism of Nicotinic Acetylcholine Receptors: Therapeutic Potential for Neuroinflammation Underlying Brain Trauma and Degenerative Disorders. International Journal of Molecular Sciences. 21. PMID 32664647 DOI: 10.3390/ijms21144918   
2020 Pandey T, Smita SS, Mishra A, Sammi SR, Pandey R. Swertiamarin, a secoiridoid glycoside modulates nAChR and AChE activity. Experimental Gerontology. 111010. PMID 32590127 DOI: 10.1016/j.exger.2020.111010   
2020 Eom S, Kim C, Yeom HD, Lee J, Lee S, Baek YB, Na J, Park SI, Kim GY, Lee CM, Lee JH. Molecular Regulation of α3β4 Nicotinic Acetylcholine Receptors by Lupeol in Cardiovascular System. International Journal of Molecular Sciences. 21. PMID 32570692 DOI: 10.3390/ijms21124329   
2020 Chou TH, Tajima N, Romero-Hernandez A, Furukawa H. Structural Basis of Functional Transitions in Mammalian NMDA Receptors. Cell. PMID 32610085 DOI: 10.1016/j.cell.2020.05.052   
2020 Evenseth LSM, Ocello R, Gabrielsen M, Masetti M, Recanatini M, Sylte I, Cavalli A. Exploring Conformational Dynamics of the Extracellular Domain of the GABA Receptor: A Path-Metadynamics Study. Journal of Chemical Information and Modeling. 60: 2294-2303. PMID 32233432 DOI: 10.1021/acs.jcim.0c00163   
2020 Markus F, Angelini C, Trimouille A, Rudolf G, Lesca G, Goizet C, Lasseaux E, Arveiler B, van Slegtenhorst M, Brooks AS, Abou Jamra R, Korenke GC, Neidhardt J, Owczarek-Lipska M. Rare variants in the GABA receptor subunit ε identified in patients with a wide spectrum of epileptic phenotypes. Molecular Genetics & Genomic Medicine. e1388. PMID 32588540 DOI: 10.1002/mgg3.1388   
2020 Yu Liao VW, Kusay AS, Balle T, Ahring PK. Heterologous expression of concatenated nicotine acetylcholine receptors: pros and cons of subunit concatenation and recommendations for construct designs. British Journal of Pharmacology. PMID 32627170 DOI: 10.1111/bph.15188   
2020 Friedman S, Tauber M, Ben-Chaim Y. Sodium ions allosterically modulate the M2 muscarinic receptor. Scientific Reports. 10: 11177. PMID 32636499 DOI: 10.1038/s41598-020-68133-9   
2020 Papasergi-Scott MM, Robertson MJ, Seven AB, Panova O, Mathiesen JM, Skiniotis G. Structures of metabotropic GABA receptor. Nature. PMID 32580208 DOI: 10.1038/s41586-020-2469-4   
2020 Akk G, Germann AL, Sugasawa Y, Pierce SR, Evers AS, Steinbach JH. Enhancement of muscimol binding and gating by allosteric modulators of the GABA receptor: relating occupancy to state functions. Molecular Pharmacology. PMID 32723768 DOI: 10.1124/molpharm.120.000066   
2020 Islam MT, Molla S, Zihad SMNK, Umer M, Rahman MS, Zaman F, Das AK, Afzal MI, Salehi B, Akter MS, Mubarak MS, Martins N, Imran M, Chaudhary N, Iqbal Z, et al. Ascorbic acid antagonizes the sedative effect of diazepam possibly through inhibition of GABA(Aρ₁) and GABA(B1) receptors. Cellular and Molecular Biology (Noisy-Le-Grand, France). 66: 15-19. PMID 32583769   
2020 Sun HS, Yang QR, Bai YY, Hu NW, Liu DX, Qin CY. Gene testing for osteonecrosis of the femoral head in systemic lupus erythematosus using targeted next-generation sequencing: A pilot study. World Journal of Clinical Cases. 8: 2530-2541. PMID 32607330 DOI: 10.12998/wjcc.v8.i12.2530   
2020 Zheng N, Christensen S, Blakely A, Dowell C, Purushottam L, McIntosh JM, Chou DH. Development of Conformationally Constrained α-RgIA Analogues as Stable Peptide Antagonists of Human α9α10 Nicotinic Acetylcholine Receptors. Journal of Medicinal Chemistry. PMID 32597184 DOI: 10.1021/acs.jmedchem.0c00613   
2020 Motawe ZY, Abdelmaboud SS, Cuevas J, Breslin JW. PRE-084 as a tool to uncover potential therapeutic applications for selective sigma-1 receptor activation. The International Journal of Biochemistry & Cell Biology. 126: 105803. PMID 32668330 DOI: 10.1016/j.biocel.2020.105803   
2020 Thomas P, Pang Y. Anti-apoptotic Actions of Allopregnanolone and Ganaxolone Mediated Through Membrane Progesterone Receptors (PAQRs) in Neuronal Cells. Frontiers in Endocrinology. 11: 417. PMID 32670200 DOI: 10.3389/fendo.2020.00417   
2020 Al Noman MA, Kyzer J, Chung SSW, Wolgemuth DJ, Georg GI. Retinoic acid receptor antagonists for male contraception: Current status. Biology of Reproduction. PMID 32671394 DOI: 10.1093/biolre/ioaa122   
2020 Magno AL, Leatherbarrow KM, Brown SJ, Wilson SG, Walsh JP, Ward BK. Functional Analysis of Calcium-Sensing Receptor Variants Identified in Families Provisionally Diagnosed with Familial Hypocalciuric Hypercalcaemia. Calcified Tissue International. PMID 32638038 DOI: 10.1007/s00223-020-00715-1   
2020 Bolchi C, Bavo F, Appiani R, Roda G, Pallavicini M. 1,4-Benzodioxane, an evergreen, versatile scaffold in medicinal chemistry: A review of its recent applications in drug design. European Journal of Medicinal Chemistry. 200: 112419. PMID 32502862 DOI: 10.1016/j.ejmech.2020.112419   
2020 Fischer JP, Els-Heindl S, Beck-Sickinger AG. Adrenomedullin - Current Perspective on a Peptide Hormone with Significant Therapeutic Potential. Peptides. 170347. PMID 32569606 DOI: 10.1016/j.peptides.2020.170347   
2020 Lillo A, Martínez-Pinilla E, Reyes-Resina I, Navarro G, Franco R. Adenosine A and A Receptors Are Able to Interact with Each Other. A Further Piece in the Puzzle of Adenosine Receptor-Mediated Signaling. International Journal of Molecular Sciences. 21. PMID 32709103 DOI: 10.3390/ijms21145070   
2020 Kim SH, Kim W. GABA-B Receptor Encephalitis Triggered by Enterovirus Encephalitis in a Patient With Small Cell Lung Cancer: A Case Report. The Neurologist. 25: 106-108. PMID 32618841 DOI: 10.1097/NRL.0000000000000283   
2020 Rumpret M, Drylewicz J, Ackermans LJE, Borghans JAM, Medzhitov R, Meyaard L. Functional categories of immune inhibitory receptors. Nature Reviews. Immunology. PMID 32612208 DOI: 10.1038/s41577-020-0352-z   
2020 Abbott JA, Popescu GK. Hydroxynorketamine Blocks NMDA Receptor Currents by Binding to Closed Receptors. Molecular Pharmacology. PMID 32606205 DOI: 10.1124/mol.120.119784   
2020 Zhang X, Meng R, Wang H, Xing J. Differential Effects of Components in Artemisia annua Extract on the Induction of Drug-Metabolizing Enzyme Expression Mediated by Nuclear Receptors. Planta Medica. PMID 32557519 DOI: 10.1055/a-1178-0852   
2020 Richendrfer HA, Levy MM, Elsaid KA, Schmidt TA, Zhang L, Cabezas R, Jay GD. Recombinant Human Proteoglycan-4 Mediates Interleukin-6 Response in Both Human and Mouse Endothelial Cells Induced Into a Sepsis Phenotype. Critical Care Explorations. 2: e0126. PMID 32695993 DOI: 10.1097/CCE.0000000000000126   
2020 Pflüger P, Regner GG, Luft JG, Gonçalves DA, Krebs C, Fontenla JA, Pereira P. Gamma-decanolactone attenuates acute and chronic seizures in mice: a possible role of adenosine A1 receptors. Behavioural Pharmacology. PMID 32701527 DOI: 10.1097/FBP.0000000000000554   
2020 Gallagher CI, Sheipouri D, Shimmon S, Rawling T, Vandenberg RJ. Identification of N-acyl amino acids that are positive allosteric modulators of glycine receptors. Biochemical Pharmacology. 114117. PMID 32579961 DOI: 10.1016/j.bcp.2020.114117