Year |
Citation |
Score |
2023 |
Nelson S, Harris TJ, Muli CS, Maresh ME, Baker B, Smith C, Neumann C, Trader DJ, Parkinson EI. Discovery and Development of Cyclic Peptide Proteasome Stimulators. Chembiochem : a European Journal of Chemical Biology. e202300671. PMID 38055197 DOI: 10.1002/cbic.202300671 |
0.314 |
|
2022 |
Halder S, Macatangay NJ, Zerfas BL, Salazar-Chaparro AF, Trader DJ. Oleic amide derivatives as small molecule stimulators of the human proteasome's core particle. Rsc Medicinal Chemistry. 13: 1077-1081. PMID 36324496 DOI: 10.1039/d2md00133k |
0.711 |
|
2022 |
Salazar-Chaparro AF, Halder S, Trader DJ. Synthesis and Application of a Clickable Epoxomicin-Based Probe for Proteasome Activity Analysis. Current Protocols. 2: e490. PMID 35849029 DOI: 10.1002/cpz1.490 |
0.71 |
|
2022 |
Salazar-Chaparro AF, Halder S, Maresh ME, Trader DJ. Solid-Phase Synthesis and Application of a Clickable Version of Epoxomicin for Proteasome Activity Analysis. Chembiochem : a European Journal of Chemical Biology. e202100710. PMID 35107861 DOI: 10.1002/cbic.202100710 |
0.715 |
|
2021 |
Tian W, Maresh ME, Trader DJ. Approaches to Evaluate the Impact of a Small-Molecule Binder to a Noncatalytic Site of the Proteasome. Chembiochem : a European Journal of Chemical Biology. PMID 33617657 DOI: 10.1002/cbic.202100023 |
0.329 |
|
2020 |
Maresh ME, Salazar-Chaparro AF, Trader DJ. Methods for the discovery of small molecules to monitor and perturb the activity of the human proteasome. Future Medicinal Chemistry. PMID 33275045 DOI: 10.4155/fmc-2020-0288 |
0.336 |
|
2020 |
Zerfas BL, Coleman RA, Salazar-Chaparro AF, Macatangay NJ, Trader DJ. Fluorescent Probes with Unnatural Amino Acids to Monitor Proteasome Activity in Real-Time. Acs Chemical Biology. PMID 32786259 DOI: 10.1021/Acschembio.0C00634 |
0.452 |
|
2020 |
Borsari C, Trader DJ, Tait A, Costi MP. Designing Chimeric Molecules for Drug Discovery by Leveraging Chemical Biology. Journal of Medicinal Chemistry. PMID 32023055 DOI: 10.1021/Acs.Jmedchem.9B01456 |
0.398 |
|
2020 |
Trader DJ, Zerfas B. Advanced Activity‐Based Probes to Monitor the Proteasome in Live Cells The Faseb Journal. 34: 1-1. DOI: 10.1096/Fasebj.2020.34.S1.09065 |
0.317 |
|
2019 |
Tian W, Trader DJ. Discovery of a Small Molecule Probe to Rpn-6, an Essential Subunit of the 26S Proteasome. Acs Chemical Biology. PMID 31877015 DOI: 10.1021/Acschembio.9B01019 |
0.433 |
|
2019 |
Zerfas BL, Trader DJ. Synthesis and Application of an Activity-Based Peptide-Peptoid Hybrid Probe for the Immunoproteasome. Current Protocols in Chemical Biology. 11: e76. PMID 31860787 DOI: 10.1002/Cpch.76 |
0.465 |
|
2019 |
Zerfas BL, Maresh ME, Trader DJ. The Immunoproteasome: An Emerging Target in Cancer, Autoimmune and Neurological Disorders. Journal of Medicinal Chemistry. PMID 31670954 DOI: 10.1021/Acs.Jmedchem.9B01226 |
0.366 |
|
2019 |
Coleman RA, Trader DJ. Methods to Discover and Evaluate Proteasome Small Molecule Stimulators. Molecules (Basel, Switzerland). 24. PMID 31242677 DOI: 10.3390/Molecules24122341 |
0.41 |
|
2019 |
Zerfas BL, Trader DJ. Monitoring the Immunoproteasome in Live Cells Using an Activity-Based Peptide-Peptoid Hybrid Probe. Journal of the American Chemical Society. PMID 30862160 DOI: 10.1021/Jacs.8B12873 |
0.439 |
|
2019 |
Muli C, Tian W, Trader DJ. Small Molecule Inhibitors of the Proteasome's Regulatory Particle. Chembiochem : a European Journal of Chemical Biology. PMID 30740849 DOI: 10.1002/Cbic.201900017 |
0.41 |
|
2019 |
Maresh ME, Trader DJ. Development of a Method to Prioritize Protein-Ligand Pairs on Beads Using Protein Conjugated to a Near-IR Dye. Acs Combinatorial Science. PMID 30677288 DOI: 10.1021/Acscombsci.8B00165 |
0.366 |
|
2018 |
Coleman RA, Muli CS, Zhao Y, Bhardwaj A, Newhouse TR, Trader DJ. Analysis of chain length, substitution patterns, and unsaturation of AM-404 derivatives as 20S proteasome stimulators. Bioorganic & Medicinal Chemistry Letters. PMID 30587447 DOI: 10.1016/J.Bmcl.2018.12.030 |
0.415 |
|
2018 |
Coleman RA, Trader DJ. A Sensitive High-Throughput Screening Method for Identifying Small Molecule Stimulators of the Core Particle of the Proteasome. Current Protocols in Chemical Biology. e52. PMID 30285317 DOI: 10.1002/Cpch.52 |
0.427 |
|
2018 |
Coleman R, Trader DJ. Development and Application of a Sensitive Peptide Reporter to Discover 20S Proteasome Stimulators. Acs Combinatorial Science. PMID 29553711 DOI: 10.1021/Acscombsci.7B00193 |
0.385 |
|
2017 |
Trader DJ, Simanski S, Dickson P, Kodadek T. Establishment of a suite of assays that support the discovery of proteasome stimulators. Biochimica Et Biophysica Acta. 1861: 892-899. PMID 28065760 DOI: 10.1016/J.Bbagen.2017.01.003 |
0.568 |
|
2015 |
Trader DJ, Carlson EE. Chemoselective enrichment as a tool to increase access to bioactive natural products: Case study borrelidin. Bioorganic & Medicinal Chemistry Letters. 25: 4767-9. PMID 26255540 DOI: 10.1016/J.Bmcl.2015.07.062 |
0.638 |
|
2015 |
Trader DJ, Simanski S, Kodadek T. A reversible and highly selective inhibitor of the proteasomal ubiquitin receptor rpn13 is toxic to multiple myeloma cells. Journal of the American Chemical Society. 137: 6312-9. PMID 25914958 DOI: 10.1021/Jacs.5B02069 |
0.556 |
|
2015 |
Trader DJ, Carlson EE. Chemoselective enrichment as a tool to increase access to bioactive natural products: Case study borrelidin Bioorganic and Medicinal Chemistry Letters. DOI: 10.1016/j.bmcl.2015.07.062 |
0.539 |
|
2014 |
Trader DJ, Carlson EE. Toward the development of solid-supported reagents for separation of alcohol-containing compounds by steric environment Tetrahedron. 70: 4191-4196. DOI: 10.1016/J.Tet.2014.03.040 |
0.617 |
|
2013 |
Trader DJ, Carlson EE. Taming of a superbase for selective phenol desilylation and natural product isolation. The Journal of Organic Chemistry. 78: 7349-55. PMID 23815363 DOI: 10.1021/Jo4010298 |
0.623 |
|
2013 |
Sidebottom AM, Johnson AR, Karty JA, Trader DJ, Carlson EE. Integrated metabolomics approach facilitates discovery of an unpredicted natural product suite from Streptomyces coelicolor M145. Acs Chemical Biology. 8: 2009-16. PMID 23777274 DOI: 10.1021/Cb4002798 |
0.718 |
|
2012 |
Trader DJ, Carlson EE. Chemoselective hydroxyl group transformation: an elusive target. Molecular Biosystems. 8: 2484-93. PMID 22695722 DOI: 10.1039/C2Mb25122A |
0.618 |
|
2011 |
Odendaal AY, Trader DJ, Carlson EE. Chemoselective enrichment for natural products discovery. Chemical Science. 2: 760-764. PMID 24926410 DOI: 10.1039/C0Sc00620C |
0.679 |
|
2011 |
Trader DJ, Carlson EE. Siloxyl ether functionalized resins for chemoselective enrichment of carboxylic acids. Organic Letters. 13: 5652-5. PMID 21957886 DOI: 10.1021/Ol202376M |
0.647 |
|
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