| Year |
Citation |
Score |
| 2007 |
Spatola AF, Romanovskis P. Cyclic peptide libraries: Recent developments Combinatorial Peptide and Nonpeptide Libraries: a Handbook. 327-347. DOI: 10.1002/9783527614912.ch11 |
0.424 |
|
| 2005 |
Galande AK, Bramlett KS, Trent JO, Burris TP, Wittliff JL, Spatola AF. Potent inhibitors of LXXLL-based protein-protein interactions. Chembiochem : a European Journal of Chemical Biology. 6: 1991-8. PMID 16222726 DOI: 10.1002/Cbic.200500083 |
0.762 |
|
| 2005 |
Cripps JG, Crespo FA, Romanovskis P, Spatola AF, Fernández-Botrán R. Modulation of acute inflammation by targeting glycosaminoglycan-cytokine interactions. International Immunopharmacology. 5: 1622-32. PMID 16039552 DOI: 10.1016/J.Intimp.2005.04.010 |
0.389 |
|
| 2005 |
Wen JJ, Spatola AF. Synthesis of a cyclic pseudopeptide containing a flexible β-Alaψ[CH2NH]unit Tetrahedron Letters. 46: 2499-2501. DOI: 10.1016/J.Tetlet.2005.01.171 |
0.342 |
|
| 2004 |
Darlak K, Wiegandt Long D, Czerwinski A, Darlak M, Valenzuela F, Spatola AF, Barany G. Facile preparation of disulfide-bridged peptides using the polymer-supported oxidant CLEAR-OX. The Journal of Peptide Research : Official Journal of the American Peptide Society. 63: 303-12. PMID 15049843 DOI: 10.1111/J.1399-3011.2004.00153.X |
0.374 |
|
| 2004 |
Galande AK, Bramlett KS, Burris TP, Wittliff JL, Spatola AF. Thioether side chain cyclization for helical peptide formation: inhibitors of estrogen receptor-coactivator interactions. The Journal of Peptide Research : Official Journal of the American Peptide Society. 63: 297-302. PMID 15049842 DOI: 10.1111/J.1399-3011.2004.00152.X |
0.775 |
|
| 2004 |
Brunel FM, Spatola AF. Synthesis of diketopiperazines with on-resin N-methylation and cyclative release. The Journal of Peptide Research : Official Journal of the American Peptide Society. 63: 213-22. PMID 15049833 DOI: 10.1111/J.1399-3011.2004.00130.X |
0.668 |
|
| 2004 |
Fernandez-Botran R, Romanovskis P, Sun X, Spatola AF. Linear basic peptides for targeting interferon-γ-glycosaminoglycan interactions: Synthesis and inhibitory properties Journal of Peptide Research. 63: 56-62. PMID 15009526 DOI: 10.1111/J.1399-3011.2003.00107.X |
0.414 |
|
| 2003 |
Galande AK, Trent JO, Spatola AF. Understanding base-assisted desulfurization using a variety of disulfide-bridged peptides. Biopolymers. 71: 534-51. PMID 14635094 DOI: 10.1002/Bip.10532 |
0.749 |
|
| 2003 |
Leduc AM, Trent JO, Wittliff JL, Bramlett KS, Briggs SL, Chirgadze NY, Wang Y, Burris TP, Spatola AF. Helix-stabilized cyclic peptides as selective inhibitors of steroid receptor-coactivator interactions. Proceedings of the National Academy of Sciences of the United States of America. 100: 11273-8. PMID 13679575 DOI: 10.1073/Pnas.1934759100 |
0.641 |
|
| 2003 |
Galande AK, Spatola AF. Solid-phase synthesis of disulfide heterodimers of peptides. Organic Letters. 5: 3431-4. PMID 12967292 DOI: 10.1021/Ol0300827 |
0.751 |
|
| 2003 |
Brunel FM, Taylor KG, Spatola AF. Synthesis of permethylated α-D-mannosylacetic acid, a new type of bioconjugate Tetrahedron Letters. 44: 1287-1289. DOI: 10.1016/S0040-4039(02)02770-3 |
0.701 |
|
| 2002 |
Burden JE, Davis P, Porreca F, Spatola AF. Synthesis and biological activities of YkFA analogues: effects of position 4 substitutions and altered ring size on in vitro opioid activity. Bioorganic & Medicinal Chemistry Letters. 12: 213-6. PMID 11755357 DOI: 10.1016/S0960-894X(01)00706-5 |
0.393 |
|
| 2002 |
Brunel FM, Leduc AM, Mashuta MS, Taylor KG, Spatola AF. Synthesis and applications of alkylated C-sugars as peptide bioconjugates Letters in Peptide Science. 9: 111-117. DOI: 10.1007/Bf02576872 |
0.757 |
|
| 2002 |
Galande AK, Spatola AF. A facile method for the direct synthesis of lanthionine containing cyclic peptides Letters in Peptide Science. 8: 247-251. DOI: 10.1007/Bf02446524 |
0.765 |
|
| 2001 |
Leduc AM, Mashuta MS, Spatola AF. Benzyl tert-butoxycarbonyl-α-amino-isobutyrate Acta Crystallographica Section C: Crystal Structure Communications. 57: 487-488. DOI: 10.1107/S010827010100110X |
0.478 |
|
| 2000 |
Spatola AF, Romanovskis P. ChemInform Abstract: Head-to-Tail Cyclic Peptides and Cyclic Peptide Libraries Cheminform. 31: no-no. DOI: 10.1002/chin.200047262 |
0.436 |
|
| 1999 |
Burden JE, Davis P, Porreca F, Spatola AF. Synthesis and biological activities of position one and three transposed analogs of the opioid peptide YKFA. Bioorganic & Medicinal Chemistry Letters. 9: 3441-6. PMID 10617088 DOI: 10.1016/S0960-894X(99)00625-3 |
0.414 |
|
| 1998 |
Romanovskis P, Spatola AF. Preparation of head-to-tail cyclic peptides via side-chain attachment: Implications for library synthesis Journal of Peptide Research. 52: 356-374. PMID 9894841 DOI: 10.1111/J.1399-3011.1998.Tb00660.X |
0.539 |
|
| 1997 |
Crozet Y, Wen JJ, Loo RO, Andrews PC, Spatola AF. Synthesis and characterization of cyclic pseudopeptide libraries containing thiomethylene and thiomethylene-sulfoxide amide bond surrogates Molecular Diversity. 3: 261-276. PMID 9850524 DOI: 10.1023/A:1009665929182 |
0.463 |
|
| 1997 |
Wen JJ, Spatola AF. A systematic approach to the solid-phase synthesis of linear and cyclic pseudopeptide libraries containing Ψ[CH2NH] amide bond surrogates Journal of Peptide Research. 49: 3-14. PMID 9128095 DOI: 10.1111/J.1399-3011.1997.Tb01115.X |
0.522 |
|
| 1997 |
Chen JJ, Spatola AF. Solid phase synthesis of peptide hydroxamic acids Tetrahedron Letters. 38: 1511-1514. DOI: 10.1016/S0040-4039(97)00143-3 |
0.546 |
|
| 1996 |
Spatola AF, Crozet Y, DeWit D, Yanagisawa M. Rediscovering an endothelin antagonist (BQ-123): A self-deconvoluting cyclic pentapeptide library Journal of Medicinal Chemistry. 39: 3842-3846. PMID 8809172 DOI: 10.1021/Jm9604078 |
0.384 |
|
| 1996 |
Hoeg-Jensen T, Spatola AF, Holm A. Amino monothio acids in solid-phase synthesis of peptide thioamides International Journal of Peptide and Protein Research. 47: 190-200. PMID 8740969 DOI: 10.1111/J.1399-3011.1996.Tb01344.X |
0.536 |
|
| 1996 |
Spatola AF, Darlak K, Romanovskis P. An approach to cyclic peptide libraries: Reducing epimerization in medium sized rings during solid phase synthesis Tetrahedron Letters. 37: 591-594. DOI: 10.1016/0040-4039(95)02269-4 |
0.543 |
|
| 1996 |
Chen JJ, Teesch LM, Spatola AF. Using cyclic peptide mixtures as probes for metal ion host-guest interactions Letters in Peptide Science. 3: 17-24. DOI: 10.1007/Bf00131081 |
0.451 |
|
| 1995 |
Ro S, Zhu Q, Lee CW, Goodman M, Darlak K, Spatola AF, Chung NN, Schiller PW, Malmberg AB, Yaksh TL. Highly potent side chain-main chain cyclized dermorphin-deltorphin analogues: an integrated approach including synthesis, bioassays, NMR spectroscopy and molecular modelling. Journal of Peptide Science : An Official Publication of the European Peptide Society. 1: 157-74. PMID 9222993 DOI: 10.1002/Psc.310010303 |
0.417 |
|
| 1993 |
Ma S, Spatola AF. Conformations of ψ[CH2NH] pseudopeptides. Cyclo[Gly-Proψ[CH2NH]Gly-D-Phe-Pro]-TFA and cyclo[Gly-Proψ[CH2NH]Gly-D-Phe-Pro] International Journal of Peptide and Protein Research. 41: 204-206. PMID 8458694 DOI: 10.1111/J.1399-3011.1993.Tb00133.X |
0.368 |
|
| 1993 |
Ma S, Richardson JF, Spatola AF. Crystal structures of two cyclic pseudopentapeptides containing psi[CH2S] and psi[CH2SO] backbone surrogates. Biopolymers. 33: 1101-10. PMID 8343587 DOI: 10.1002/Bip.360330712 |
0.445 |
|
| 1992 |
Spatola AF, Anwer MK, Rao MN. Phase transfer catalysis in solid phase peptide synthesis. Preparation of cyclo[Xxx-Pro-Gly-Yyy-Pro-Gly] model peptides and their conformational analysis International Journal of Peptide and Protein Research. 40: 322-332. PMID 1478790 DOI: 10.1111/J.1399-3011.1992.Tb00308.X |
0.537 |
|
| 1992 |
Lankiewicz L, Bowers CY, Reynolds GA, Labroo V, Cohen LA, Vonhof S, Sirén AL, Spatola AF. Biological activities of thionated thyrotropin-releasing hormone analogs Biochemical and Biophysical Research Communications. 184: 359-366. PMID 1314591 DOI: 10.1016/0006-291X(92)91201-Z |
0.367 |
|
| 1992 |
Anwer MK, Spatola AF. Cleavage of peptides bound to merrifield resins by potassium carbonate in the presence of a phase transfer reagent Tetrahedron Letters. 33: 3121-3124. DOI: 10.1016/S0040-4039(00)79829-7 |
0.482 |
|
| 1990 |
Anwer MK, Sherman DB, Spatola AF. Backbone modifications in cyclic peptides. Conformational analysis of a cyclic pseudopentapeptide containing a thiomethylene ether amide bond replacement International Journal of Peptide and Protein Research. 36: 392-399. PMID 2079394 DOI: 10.1111/J.1399-3011.1990.Tb01299.X |
0.434 |
|
| 1990 |
Sherman DB, Spatola AF. Compatibility of thioamides with reverse turn features: Synthesis and conformational analysis of two model cyclic pseudopeptides containing thioamides as backbone modifications Journal of the American Chemical Society. 112: 433-441. DOI: 10.1021/Ja00157A064 |
0.431 |
|
| 1990 |
Deterding LJ, Tomer KB, Spatola AF. Tandem mass spectrometry for the structural determination of backbone-modified peptides Journal of the American Society For Mass Spectrometry. 1: 174-182. DOI: 10.1016/1044-0305(90)85054-P |
0.485 |
|
| 1989 |
Sherman DB, Spatola AF, Wire WS, Burks TF, Nguyen TMD, Schiller PW. Biological activities of cyclic enkephalin pseudopeptides containing thioamides as amide bond replacements Biochemical and Biophysical Research Communications. 162: 1126-1132. PMID 2764921 DOI: 10.1016/0006-291X(89)90790-0 |
0.351 |
|
| 1989 |
Anwer MK, Sherman DB, Roney JG, Spatola AF. Applications of ammonium formate catalytic transfer hydrogenation. 6. Analysis of catalyst, donor quantity, and solvent effects upon the efficacy of dechlorination Journal of Organic Chemistry. 54: 1284-1289. DOI: 10.1021/Jo00267A012 |
0.305 |
|
| 1988 |
Darlak K, Benovitz DE, Spatola AF, Grzonka Z. Dermorphin analogs: Resistance to in vitro enzymatic degradation is not always increased by additional D-amino acid substitutions Biochemical and Biophysical Research Communications. 156: 125-130. PMID 2902857 DOI: 10.1016/S0006-291X(88)80813-1 |
0.351 |
|
| 1988 |
Darlak K, Franklin G, Woost P, Sonnenfeld E, Twardzik D, Spatola A, Schultz G. Assessment of biological activity of synthetic fragments of transforming growth factor-alpha. Journal of Cellular Biochemistry. 36: 341-52. PMID 2897968 DOI: 10.1002/Jcb.240360404 |
0.304 |
|
| 1988 |
Spatola AF, Darlak K. Amide bond surrogates: pseudopeptides and macrocycles Tetrahedron. 44: 821-833. DOI: 10.1016/S0040-4020(01)86119-6 |
0.43 |
|
| 1987 |
Anwer MK, Porter RA, Spatola AF. Applications of ammonium formate-catalytic transfer hydrogenation. Part V (1). Transfer hydrogenolysis of peptides containing p-chlorophenylalanine as a convenient method for preparation of deuterium labeled peptides International Journal of Peptide and Protein Research. 30: 489-497. PMID 2962959 DOI: 10.1111/J.1399-3011.1987.Tb03357.X |
0.405 |
|
| 1986 |
Spatola AF, Saneii H, Edwards JV, Bettag AL, Anwer MK, Rowell P, Browne B, Lahti R, Von Voigtlander P. Structure-activity relationships of enkephalins containing serially replaced thiomethylene amide bond surrogates Life Sciences. 38: 1243-1249. PMID 3959753 DOI: 10.1016/0024-3205(86)90416-9 |
0.354 |
|
| 1986 |
Gray RD, Miller RB, Spatola AF. Inhibition of mammalian collagenases by thiol-containing peptides Journal of Cellular Biochemistry. 32: 71-77. PMID 3021790 DOI: 10.1002/Jcb.240320108 |
0.366 |
|
| 1986 |
Edwards JV, Spatola AF, Lemieux C, Schiller PW. In vitro activity profiles of cyclic and linear enkephalin pseudopeptide analogs Biochemical and Biophysical Research Communications. 136: 730-736. PMID 3010995 DOI: 10.1016/0006-291X(86)90500-0 |
0.494 |
|
| 1986 |
Spatola AF, Anwer MK, Rockwell AL, Gierasch LM. Compatibility of .beta.- and .gamma.-turn features with a peptide backbone modification: synthesis and conformational analysis of a model cyclic pseudopentapeptide Journal of the American Chemical Society. 108: 825-831. DOI: 10.1021/Ja00264A041 |
0.489 |
|
| 1986 |
Spatola AF, Anwer MK, Rockwell AL, Gierasch LM. Compatibility of β- and γ-turn features with a peptide backbone modification: Synthesis and conformational analysis of a model cyclic pseudopentapeptide Journal of the American Chemical Society. 108: 825-831. |
0.377 |
|
| 1985 |
Benovitz DE, Spatola AF. Enkephalin pseudopeptides: Resistance to in vitro proteolytic degradation afforded by amide bond replacements extends to remote sites Peptides. 6: 257-261. PMID 4034413 DOI: 10.1016/0196-9781(85)90049-X |
0.465 |
|
| 1985 |
Spatola AF, Benovitz DE. Improved detection limits in the analysis of tyrosine-containing polypeptide hormones by using electrochemical detection Journal of Chromatography A. 327: 165-171. DOI: 10.1016/S0021-9673(01)81645-9 |
0.423 |
|
| 1985 |
Anwer MK, Clausen K, Spatola AF. Synthetic peptide analogs which elicit or inhibit growth hormone release Federation Proceedings. 44. |
0.338 |
|
| 1985 |
Gray RD, Edwards JV, Harrod JW, Spatola AF. Inhibition of tumor collagenase by peptide analogues of the collagen cleavage site Federation Proceedings. 44: No. 5970. |
0.324 |
|
| 1984 |
Clausen K, Spatola AF, Lemieux C, Schiller PW, Lawesson SO. Evidence of a peptide backbone contribution toward selective receptor recognition for leucine enkephalin thioamide analogs Biochemical and Biophysical Research Communications. 120: 305-310. PMID 6324793 DOI: 10.1016/0006-291X(84)91449-9 |
0.491 |
|
| 1984 |
Clausen K, Thorsen M, Lawesson SO, Spatola AF. Studies on amino acids and peptides. Part 6. Methods for introducing thioamide bonds into the peptide backbone: Synthesis of the four monothio analogues of leucine enkephalin Journal of the Chemical Society, Perkin Transactions 1. 785-798. DOI: 10.1039/P19840000785 |
0.521 |
|
| 1983 |
Anwer MK, Spatola AF, Bossinger CD, Flanigan E, Liu RC, Olsen DB, Stevenson D. Quantitative removal of a pentadecapeptide ACTH fragment analogue from a Merrifield resin using ammonium formate catalytic transfer hydrogenation: Synthesis of [Asp25,Ala26,Gly27,Gln 30]-ACTH-(25-39)-OH Journal of Organic Chemistry. 48: 3503-3507. DOI: 10.1002/Chin.198412323 |
0.356 |
|
| 1983 |
Spatola AF, Gierasch LM, Rockwell AL. Conformational comparison of cyclic peptide and pseudopeptide structures with intramolecular hydrogen bonding Biopolymers. 22: 147-151. DOI: 10.1002/Bip.360220123 |
0.412 |
|
| 1982 |
Saneii H, Spatola AF. Amino acids surrogates: an indirect method for the synthesis of peptides containing the thioasparaginyl residue Tetrahedron Letters. 23: 149-152. DOI: 10.1016/S0040-4039(00)86771-4 |
0.411 |
|
| 1981 |
Gray RD, Saneii HH, Spatola AF. Metal binding peptide inhibitors of vertebrate collagenase Biochemical and Biophysical Research Communications. 101: 1251-1258. PMID 6272777 DOI: 10.1016/0006-291X(81)91582-5 |
0.48 |
|
| 1981 |
Spatola AF, Bettag AL. Pseudodipeptides: A novel route to serine-containing diastereomeric analogues Journal of Organic Chemistry. 46: 2393-2394. DOI: 10.1021/Jo00324A038 |
0.318 |
|
| 1981 |
Spatola AF. Chapter 19. Peptides of the Hypothalamus Annual Reports in Medicinal Chemistry. 16: 199-211. DOI: 10.1016/S0065-7743(08)61286-5 |
0.538 |
|
| 1981 |
Anwer MK, Spatola AF. A rapid non-acidolytic method for deprotection and removal of peptides from solid phase resins - applications of ammonium formate catalytic transfer hydrogenation Tetrahedron Letters. 22: 4369-4372. DOI: 10.1016/S0040-4039(01)82959-2 |
0.461 |
|
| 1980 |
Spatola AF, Agarwal NS. A highly potent antiovulatory LH-RH analogue with no 1-position side chain Biochemical and Biophysical Research Communications. 97: 1571-1574. PMID 7011319 DOI: 10.1016/S0006-291X(80)80045-3 |
0.31 |
|
| 1980 |
Spatola AF, Agarwal NS, Bettag AL, Yankeelov JA, Bowers CY, Vale WW. Synthesis and biological activities of pseudopeptide analogues of LH-RH: Agonists and antagonists Biochemical and Biophysical Research Communications. 97: 1014-1023. PMID 6258597 DOI: 10.1016/0006-291X(80)91477-1 |
0.374 |
|
| 1979 |
Hruby VJ, Deb KK, Spatola AF, Upson DA, Yamamoto D. Carbon-13 NMR studies of the Peptide hormones oxytocin, arginine vasopressin, isotocin, mesotocin, glumitocin, aspartocin, related analogs, and diastereoisomers. Use of specifically deuterated hormone derivatives for assignments and effects of structural changes on carbon-13 NMR chemical shifts in peptides Journal of the American Chemical Society. 101: 202-212. DOI: 10.1021/Ja00495A033 |
0.514 |
|
| 1979 |
HRUBY VJ, DEB KK, SPATOLA AF, UPSON DA, YAMAMOTO D. ChemInform Abstract: CARBON-13 NMR STUDIES OF THE HORMONES OXYTOC Chemischer Informationsdienst. 10. DOI: 10.1002/Chin.197915050 |
0.31 |
|
| 1979 |
Hruby VJ, Deb KK, Spatola AF, Upson DA, Yamamoto D. 13C nuclear magnetic resonance studies of the peptide hormones oxytocin, arginine vasopressin, isotocin, mesotocin, glumitocin, aspartocin, related analogues, and diastereoisomers. Use of specifically deuterated hormone derivatives for assignments and effects of structural changes on 13C NMR chemical shifts in peptides Journal of the American Chemical Society. 101: 202-212. |
0.407 |
|
| 1975 |
Hruby VJ, Spatola AF, Glasel JA, McKelvy JF. Equilibrium dialysis studies of hormone-neurophysin binding. Annals of the New York Academy of Sciences. 248: 451-7. PMID 235234 DOI: 10.1111/J.1749-6632.1975.Tb34205.X |
0.301 |
|
| 1974 |
Spatola AF, Cornelius DA, Hruby VJ, Blomquist AT. Synthesis of oxytocin and related diastereomers deuterated in the half-cystine positions. Comparison of solid-phase and solution methods. The Journal of Organic Chemistry. 39: 2207-12. PMID 4859518 DOI: 10.1002/Chin.197446430 |
0.592 |
|
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