Henry I. Yamamura - Publications

Affiliations: 
University of Arizona, Tucson, AZ 

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Year Citation  Score
2011 Yamamoto T, Nair P, Largent-Milnes TM, Jacobsen NE, Davis P, Ma SW, Yamamura HI, Vanderah TW, Porreca F, Lai J, Hruby VJ. Discovery of a potent and efficacious peptide derivative for δ/μ opioid agonist/neurokinin 1 antagonist activity with a 2',6'-dimethyl-L-tyrosine: in vitro, in vivo, and NMR-based structural studies. Journal of Medicinal Chemistry. 54: 2029-38. PMID 21366266 DOI: 10.1021/jm101023r  1
2010 Yamamoto T, Nair P, Jacobsen NE, Kulkarni V, Davis P, Ma SW, Navratilova E, Yamamura HI, Vanderah TW, Porreca F, Lai J, Hruby VJ. Biological and conformational evaluation of bifunctional compounds for opioid receptor agonists and neurokinin 1 receptor antagonists possessing two penicillamines. Journal of Medicinal Chemistry. 53: 5491-501. PMID 20617791 DOI: 10.1021/jm100157m  1
2009 Yamamoto T, Nair P, Jacobsen NE, Vagner J, Kulkarni V, Davis P, Ma SW, Navratilova E, Yamamura HI, Vanderah TW, Porreca F, Lai J, Hruby VJ. Improving metabolic stability by glycosylation: bifunctional peptide derivatives that are opioid receptor agonists and neurokinin 1 receptor antagonists. Journal of Medicinal Chemistry. 52: 5164-75. PMID 20560643 DOI: 10.1021/jm900473p  1
2009 Yamamoto T, Nair P, Ma SW, Davis P, Yamamura HI, Vanderah TW, Porreca F, Lai J, Hruby VJ. The biological activity and metabolic stability of peptidic bifunctional compounds that are opioid receptor agonists and neurokinin-1 receptor antagonists with a cystine moiety. Bioorganic & Medicinal Chemistry. 17: 7337-43. PMID 19762245 DOI: 10.1016/j.bmc.2009.08.035  1
2009 Tumati S, Yamamura HI, Vanderah TW, Roeske WR, Varga EV. Sustained morphine treatment augments capsaicin-evoked calcitonin gene-related peptide release from primary sensory neurons in a protein kinase A- and Raf-1-dependent manner. The Journal of Pharmacology and Experimental Therapeutics. 330: 810-7. PMID 19491327 DOI: 10.1124/jpet.109.151704  1
2009 Nair P, Yamamoto T, Kulkarni V, Moye S, Navratilova E, Davis P, Largent T, Ma SW, Yamamura HI, Vanderah T, Lai J, Porreca F, Hruby VJ. Novel bifunctional peptides as opioid agonists and NK-1 antagonists. Advances in Experimental Medicine and Biology. 611: 537-8. PMID 19400302 DOI: 10.1007/978-0-387-73657-0_235  1
2009 Tumati S, Yamamura HI, St John PA, Vanderah TW, Roeske WR, Varga EV. Sustained cannabinoid agonist treatment augments CGRP release in a PKA-dependent manner. Neuroreport. 20: 815-9. PMID 19387418 DOI: 10.1097/WNR.0b013e32832be50b  1
2008 Varga EV, Georgieva T, Tumati S, Alves I, Salamon Z, Tollin G, Yamamura HI, Roeske WR. Functional selectivity in cannabinoid signaling. Current Molecular Pharmacology. 1: 273-84. PMID 20021440  1
2008 Fioravanti B, De Felice M, Stucky CL, Medler KA, Luo MC, Gardell LR, Ibrahim M, Malan TP, Yamamura HI, Ossipov MH, King T, Lai J, Porreca F, Vanderah TW. Constitutive activity at the cannabinoid CB1 receptor is required for behavioral response to noxious chemical stimulation of TRPV1: antinociceptive actions of CB1 inverse agonists. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 28: 11593-602. PMID 18987195 DOI: 10.1523/JNEUROSCI.3322-08.2008  1
2008 Tumati S, Milnes TL, Yamamura HI, Vanderah TW, Roeske WR, Varga EV. Intrathecal Raf-1-selective siRNA attenuates sustained morphine-mediated thermal hyperalgesia. European Journal of Pharmacology. 601: 207-8. PMID 18976650 DOI: 10.1016/j.ejphar.2008.10.033  1
2008 Yamamoto T, Nair P, Jacobsen NE, Davis P, Ma SW, Navratilova E, Moye S, Lai J, Yamamura HI, Vanderah TW, Porreca F, Hruby VJ. The importance of micelle-bound states for the bioactivities of bifunctional peptide derivatives for delta/mu opioid receptor agonists and neurokinin 1 receptor antagonists. Journal of Medicinal Chemistry. 51: 6334-47. PMID 18821747 DOI: 10.1021/jm800389v  1
2008 Yue X, Tumati S, Navratilova E, Strop D, St John PA, Vanderah TW, Roeske WR, Yamamura HI, Varga EV. Sustained morphine treatment augments basal CGRP release from cultured primary sensory neurons in a Raf-1 dependent manner. European Journal of Pharmacology. 584: 272-7. PMID 18328477 DOI: 10.1016/j.ejphar.2008.02.013  1
2008 Yamamoto T, Nair P, Vagner J, Largent-Milnes T, Davis P, Ma SW, Navratilova E, Moye S, Tumati S, Lai J, Yamamura HI, Vanderah TW, Porreca F, Hruby VJ. A structure-activity relationship study and combinatorial synthetic approach of C-terminal modified bifunctional peptides that are delta/mu opioid receptor agonists and neurokinin 1 receptor antagonists. Journal of Medicinal Chemistry. 51: 1369-76. PMID 18266313 DOI: 10.1021/jm070332f  1
2008 Georgieva T, Devanathan S, Stropova D, Park CK, Salamon Z, Tollin G, Hruby VJ, Roeske WR, Yamamura HI, Varga E. Unique agonist-bound cannabinoid CB1 receptor conformations indicate agonist specificity in signaling. European Journal of Pharmacology. 581: 19-29. PMID 18162180 DOI: 10.1016/j.ejphar.2007.11.053  1
2008 Hruby VJ, Porreca F, Yamamura HI, Tollin G, Agnes RS, Lee YS, Cai M, Alves I, Cowell S, Varga E, Davis P, Salamon Z, Roeske W, Vanderah T, Lai J. New paradigms and tools in drug design for pain and addiction Drug Addiction: From Basic Research to Therapy. 477-494. DOI: 10.1007/978-0-387-76678-2_28  1
2007 Yamamoto T, Nair P, Davis P, Ma SW, Navratilova E, Moye S, Tumati S, Lai J, Vanderah TW, Yamamura HI, Porreca F, Hruby VJ. Design, synthesis, and biological evaluation of novel bifunctional C-terminal-modified peptides for delta/mu opioid receptor agonists and neurokinin-1 receptor antagonists. Journal of Medicinal Chemistry. 50: 2779-86. PMID 17516639 DOI: 10.1021/jm061369n  1
2007 Nissan HP, Lu J, Booth NL, Yamamura HI, Farnsworth NR, Wang ZJ. A red clover (Trifolium pratense) phase II clinical extract possesses opiate activity. Journal of Ethnopharmacology. 112: 207-10. PMID 17350196 DOI: 10.1016/j.jep.2007.02.006  1
2007 Navratilova E, Waite S, Stropova D, Eaton MC, Alves ID, Hruby VJ, Roeske WR, Yamamura HI, Varga EV. Quantitative evaluation of human delta opioid receptor desensitization using the operational model of drug action. Molecular Pharmacology. 71: 1416-26. PMID 17322005 DOI: 10.1124/mol.106.030023  1
2006 Cai M, Varga EV, Stankova M, Mayorov A, Perry JW, Yamamura HI, Trivedi D, Hruby VJ. Cell signaling and trafficking of human melanocortin receptors in real time using two-photon fluorescence and confocal laser microscopy: differentiation of agonists and antagonists. Chemical Biology & Drug Design. 68: 183-93. PMID 17105482 DOI: 10.1111/j.1747-0285.2006.00432.x  1
2006 Hruby VJ, Porreca F, Yamamura HI, Tollin G, Agnes RS, Lee YS, Cai M, Alves I, Cowell S, Varga E, Davis P, Salamon Z, Roeske W, Vanderah T, Lai J. New paradigms and tools in drug design for pain and addiction. The Aaps Journal. 8: E450-60. PMID 17025262 DOI: 10.1208/aapsj080353  1
2006 Yue X, Varga EV, Stropova D, Vanderah TW, Yamamura HI, Roeske WR. Chronic morphine-mediated adenylyl cyclase superactivation is attenuated by the Raf-1 inhibitor, GW5074. European Journal of Pharmacology. 540: 57-9. PMID 16750187 DOI: 10.1016/j.ejphar.2006.04.033  1
2006 Oki T, Maruyama S, Takagi Y, Yamamura HI, Yamada S. Characterization of muscarinic receptor binding and inhibition of salivation after oral administration of tolterodine in mice. European Journal of Pharmacology. 529: 157-63. PMID 16316647 DOI: 10.1016/j.ejphar.2005.11.004  1
2005 Smith EA, Coym JW, Cowell SM, Tokimoto T, Hruby VJ, Yamamura HI, Wirth MJ. Lipid bilayers on polyacrylamide brushes for inclusion of membrane proteins. Langmuir : the Acs Journal of Surfaces and Colloids. 21: 9644-50. PMID 16207048 DOI: 10.1021/la051116h  1
2005 Navratilova E, Eaton MC, Stropova D, Varga EV, Vanderah TW, Roeske WR, Yamamura HI. Morphine promotes phosphorylation of the human delta-opioid receptor at serine 363. European Journal of Pharmacology. 519: 212-4. PMID 16135360 DOI: 10.1016/j.ejphar.2005.07.024  1
2005 Handl HL, Vagner J, Yamamura HI, Hruby VJ, Gillies RJ. Development of a lanthanide-based assay for detection of receptor-ligand interactions at the delta-opioid receptor. Analytical Biochemistry. 343: 299-307. PMID 16004955 DOI: 10.1016/j.ab.2005.05.040  1
2005 Dhanasekaran M, Palian MM, Alves I, Yeomans L, Keyari CM, Davis P, Bilsky EJ, Egleton RD, Yamamura HI, Jacobsen NE, Tollin G, Hruby VJ, Porreca F, Polt R. Glycopeptides related to beta-endorphin adopt helical amphipathic conformations in the presence of lipid bilayers. Journal of the American Chemical Society. 127: 5435-48. PMID 15826181 DOI: 10.1021/ja0432158  1
2005 Varga EV, Hosohata K, Borys D, Navratilova E, Nylen A, Vanderah TW, Porreca F, Roeske WR, Yamamura HI. Antinociception depends on the presence of G protein gamma2-subunits in brain. European Journal of Pharmacology. 508: 93-8. PMID 15680258 DOI: 10.1016/j.ejphar.2004.11.062  1
2005 Gu X, Ying J, Min B, Cain JP, Davis P, Willey P, Navratilova E, Yamamura HI, Porreca F, Hruby VJ. Parallel synthesis and biological evaluation of different sizes of bicyclo[2,3]-Leu-enkephalin analogues. Biopolymers. 80: 151-63. PMID 15660379 DOI: 10.1002/bip.20208  1
2005 Egleton RD, Bilsky EJ, Tollin G, Dhanasekaran M, Lowery J, Alves I, Davis P, Porreca F, Yamamura HI, Yeomans L, Keyari CM, Polt R. Biousian glycopeptides penetrate the blood-brain barrier Tetrahedron Asymmetry. 16: 65-75. DOI: 10.1016/j.tetasy.2004.11.038  1
2004 Varga EV, Navratilova E, Stropova D, Jambrosic J, Roeske WR, Yamamura HI. Agonist-specific regulation of the delta-opioid receptor. Life Sciences. 76: 599-612. PMID 15567186 DOI: 10.1016/j.lfs.2004.07.020  1
2004 Gu X, Ying J, Agnes RS, Navratilova E, Davis P, Stahl G, Porreca F, Yamamura HI, Hruby VJ. Novel design of bicyclic beta-turn dipeptides on solid-phase supports and synthesis of [3.3.0]-Bicyclo([2,3])-leu-enkephalin analogues. Organic Letters. 6: 3285-8. PMID 15355033 DOI: 10.1021/ol0488183  1
2004 Alves ID, Ciano KA, Boguslavski V, Varga E, Salamon Z, Yamamura HI, Hruby VJ, Tollin G. Selectivity, cooperativity, and reciprocity in the interactions between the delta-opioid receptor, its ligands, and G-proteins. The Journal of Biological Chemistry. 279: 44673-82. PMID 15317820 DOI: 10.1074/jbc.M404713200  0.56
2004 Handl HL, Vagner J, Yamamura HI, Hruby VJ, Gillies RJ. Lanthanide-based time-resolved fluorescence of in cyto ligand-receptor interactions. Analytical Biochemistry. 330: 242-50. PMID 15203329 DOI: 10.1016/j.ab.2004.04.012  1
2004 Cai M, Stankova M, Pond SJ, Mayorov AV, Perry JW, Yamamura HI, Trivedi D, Hruby VJ. Real time differentiation of G-protein coupled receptor (GPCR) agonist and antagonist by two photon fluorescence laser microscopy. Journal of the American Chemical Society. 126: 7160-1. PMID 15186137 DOI: 10.1021/ja049473m  1
2004 Elmagbari NO, Egleton RD, Palian MM, Lowery JJ, Schmid WR, Davis P, Navratilova E, Dhanasekaran M, Keyari CM, Yamamura HI, Porreca F, Hruby VJ, Polt R, Bilsky EJ. Antinociceptive structure-activity studies with enkephalin-based opioid glycopeptides. The Journal of Pharmacology and Experimental Therapeutics. 311: 290-7. PMID 15166257 DOI: 10.1124/jpet.104.069393  1
2004 Navratilova E, Varga EV, Stropova D, Jambrosic JC, Roeske WR, Yamamura HI. Mutation S363A in the human delta-opioid receptor selectively reduces down-regulation by a peptide agonist. European Journal of Pharmacology. 485: 341-3. PMID 14757159 DOI: 10.1016/j.ejphar.2003.11.067  1
2004 Tóth G, Keresztes A, Tömböly C, Péter A, Fülöp F, Tourwé D, Navratilova E, Varga E, Roeske WR, Yamamura HI, Szucs M, Borsodi A. New endomorphin analogs with μ-agonist and δ-antagonist properties Pure and Applied Chemistry. 76: 951-957.  1
2003 Varga EV, Yamamura HI, Rubenzik MK, Stropova D, Navratilova E, Roeske WR. Molecular mechanisms of excitatory signaling upon chronic opioid agonist treatment. Life Sciences. 74: 299-311. PMID 14607258 DOI: 10.1016/j.lfs.2003.09.017  1
2003 Alves ID, Salamon Z, Varga E, Yamamura HI, Tollin G, Hruby VJ. Direct observation of G-protein binding to the human delta-opioid receptor using plasmon-waveguide resonance spectroscopy. The Journal of Biological Chemistry. 278: 48890-7. PMID 14522991 DOI: 10.1074/jbc.M306866200  1
2003 Varga EV, Rubenzik MK, Stropova D, Sugiyama M, Grife V, Hruby VJ, Rice KC, Roeske WR, Yamamura HI. Converging protein kinase pathways mediate adenylyl cyclase superactivation upon chronic delta-opioid agonist treatment. The Journal of Pharmacology and Experimental Therapeutics. 306: 109-15. PMID 12660310 DOI: 10.1124/jpet.103.049643  1
2003 Hosohata K, Varga EV, Alfaro-Lopez J, Tang X, Vanderah TW, Porreca F, Hruby VJ, Roeske WR, Yamamura HI. (2S,3R) beta-methyl-2',6'-dimethyltyrosine-L-tetrahydroisoquinoline-3-carboxylic acid [(2S,3R)TMT-L-Tic-OH] is a potent, selective delta-opioid receptor antagonist in mouse brain. The Journal of Pharmacology and Experimental Therapeutics. 304: 683-8. PMID 12538822 DOI: 10.1124/jpet.102.042929  1
2003 Okura T, Varga EV, Hosohata Y, Navratilova E, Cowell SM, Rice K, Nagase H, Hruby VJ, Roeske WR, Yamamura HI. Agonist-specific down-regulation of the human delta-opioid receptor. European Journal of Pharmacology. 459: 9-16. PMID 12505529 DOI: 10.1016/S0014-2999(02)02823-6  1
2003 Muramatsu I, Hollenberg MD, Yamamura HI. Life Sciences: Preface Life Sciences. 74: 133-134. DOI: 10.1016/j.lfs.2003.09.001  1
2002 Varga EV, Rubenzik M, Grife V, Sugiyama M, Stropova D, Roeske WR, Yamamura HI. Involvement of Raf-1 in chronic delta-opioid receptor agonist-mediated adenylyl cyclase superactivation. European Journal of Pharmacology. 451: 101-2. PMID 12223234 DOI: 10.1016/S0014-2999(02)02220-3  1
2001 Stamer WD, Golightly SF, Hosohata Y, Ryan EP, Porter AC, Varga E, Noecker RJ, Felder CC, Yamamura HI. Cannabinoid CB(1) receptor expression, activation and detection of endogenous ligand in trabecular meshwork and ciliary process tissues. European Journal of Pharmacology. 431: 277-86. PMID 11730719 DOI: 10.1016/S0014-2999(01)01438-8  1
2001 Rubenzik M, Varga E, Stropova D, Roeske WR, Yamamura HI. Expression of alpha-transducin in Chinese hamster ovary cells stably transfected with the human delta-opioid receptor attenuates chronic opioid agonist-induced adenylyl cyclase superactivation. Molecular Pharmacology. 60: 1076-82. PMID 11641436  1
2001 Witt KA, Huber JD, Egleton RD, Roberts MJ, Bentley MD, Guo L, Wei H, Yamamura HI, Davis TP. Pharmacodynamic and pharmacokinetic characterization of poly(ethylene glycol) conjugation to met-enkephalin analog [D-Pen2, D-Pen5]-enkephalin (DPDPE). The Journal of Pharmacology and Experimental Therapeutics. 298: 848-56. PMID 11454951  1
2001 Hosohata Y, Varga EV, Stropova D, Li X, Knapp RJ, Hruby VJ, Rice KC, Nagase H, Roeske WR, Yamamura HI. Mutation W284L of the human delta opioid receptor reveals agonist specific receptor conformations for G protein activation. Life Sciences. 68: 2233-42. PMID 11358332 DOI: 10.1016/S0024-3205(01)01011-6  1
2001 Liao S, Shenderovich M, Kövér KE, Zhang Z, Hosohata K, Davis P, Porreca F, Yamamura HI, Hurby VJ. Synthesis, biology, NMR and conformation studies of the topographically constrained delta-opioid selective peptide analogs of [beta-iPrPhe(3)]deltorphin I. The Journal of Peptide Research : Official Journal of the American Peptide Society. 57: 257-76. PMID 11328484 DOI: 10.1046/j.1397-002X.2000.00000.x  1
2001 Lipkowski AW, Misicka A, Hosohata K, Davis P, Yamamura HI, Porreca F, Hruby VJ. Biological properties of Phe(o)-opioid peptide analogues. Life Sciences. 68: 969-72. PMID 11213367 DOI: 10.1016/S0024-3205(00)00993-0  1
2000 Salamon Z, Cowell S, Varga E, Yamamura HI, Hruby VJ, Tollin G. Plasmon resonance studies of agonist/antagonist binding to the human delta-opioid receptor: new structural insights into receptor-ligand interactions. Biophysical Journal. 79: 2463-74. PMID 11053123 DOI: 10.1016/S0006-3495(00)76489-7  1
2000 Egleton RD, Mitchell SA, Huber JD, Janders J, Stropova D, Polt R, Yamamura HI, Hruby VJ, Davis TP. Improved bioavailability to the brain of glycosylated Met-enkephalin analogs. Brain Research. 881: 37-46. PMID 11033091 DOI: 10.1016/S0006-8993(00)02794-3  1
2000 Bilsky EJ, Egleton RD, Mitchell SA, Palian MM, Davis P, Huber JD, Jones H, Yamamura HI, Janders J, Davis TP, Porreca F, Hruby VJ, Polt R. Enkephalin glycopeptide analogues produce analgesia with reduced dependence liability. Journal of Medicinal Chemistry. 43: 2586-90. PMID 10891118 DOI: 10.1021/jm000077y  1
2000 Witt KA, Slate CA, Egleton RD, Huber JD, Yamamura HI, Hruby VJ, Davis TP. Assessment of stereoselectivity of trimethylphenylalanine analogues of delta-opioid [D-Pen(2),D-Pen(5)]-enkephalin. Journal of Neurochemistry. 75: 424-35. PMID 10854288 DOI: 10.1046/j.1471-4159.2000.0750424.x  1
2000 Hosohata K, Logan JK, Varga E, Burkey TH, Vanderah TW, Porreca F, Hruby VJ, Roeske WR, Yamamura HI. The role of the G protein gamma(2) subunit in opioid antinociception in mice. European Journal of Pharmacology. 392: R9-R11. PMID 10762674 DOI: 10.1016/S0014-2999(00)00132-1  1
2000 Bonner GG, Davis P, Stropova D, Edsall S, Yamamura HI, Porreca F, Hruby VJ. Opiate aromatic pharmacophore structure-activity relationships in CTAP analogues determined by topographical bias, two-dimensional NMR, and biological activity assays. Journal of Medicinal Chemistry. 43: 569-80. PMID 10691683 DOI: 10.1021/jm9900218  1
2000 Hosohata Y, Vanderah TW, Burkey TH, Ossipov MH, Kovelowski CJ, Sora I, Uhl GR, Zhang X, Rice KC, Roeske WR, Hruby VJ, Yamamura HI, Lai J, Porreca F. delta-Opioid receptor agonists produce antinociception and [35S]GTPgammaS binding in mu receptor knockout mice. European Journal of Pharmacology. 388: 241-8. PMID 10675732 DOI: 10.1016/S0014-2999(99)00897-3  1
2000 Okura T, Cowell SM, Varga E, Burkey TH, Roeske WR, Hruby VJ, Yamamura HI. Differential down-regulation of the human delta-opioid receptor by SNC80 and [D-Pen(2),D-Pen(5)]enkephalin. European Journal of Pharmacology. 387: R11-3. PMID 10650167 DOI: 10.1016/S0014-2999(99)00761-X  1
2000 Varga EV, Stropova D, Kim T, Wang M, Roeske WR, Yamamura HI. Coupling of human delta-opioid receptor to retinal rod transducin in Chinese hamster ovary cells. The Journal of Pharmacology and Experimental Therapeutics. 292: 209-14. PMID 10604950  1
1999 LeVan TD, Babin EA, Yamamura HI, Bloom JW. Pharmacological characterization of glucocorticoid receptors in primary human bronchial epithelial cells. Biochemical Pharmacology. 57: 1003-9. PMID 10796070 DOI: 10.1016/S0006-2952(99)00008-8  1
1999 Alfaro-Lopez J, Okayama T, Hosohata K, Davis P, Porreca F, Yamamura HI, Hruby VJ. Exploring the structure-activity relationships of [1-(4-tert-butyl-3'-hydroxy)benzhydryl-4-benzylpiperazine] (SL-3111), a high-affinity and selective delta-opioid receptor nonpeptide agonist ligand. Journal of Medicinal Chemistry. 42: 5359-68. PMID 10639279 DOI: 10.1021/jm990337f  1
1999 Hosohata K, Burkey TH, Alfaro-Lopez J, Hruby VJ, Roeske WR, Yamamura HI. (2S,3R)TMT-L-Tic-OH is a potent inverse agonist at the human delta-opioid receptor. European Journal of Pharmacology. 380: R9-10. PMID 10513562 DOI: 10.1016/S0014-2999(99)00516-6  1
1999 Lipkowski AW, Misicka A, Davis P, Stropova D, Janders J, Lachwa M, Porreca F, Yamamura HI, Hruby VJ. Biological activity of fragments and analogues of the potent dimeric opioid peptide, biphalin. Bioorganic & Medicinal Chemistry Letters. 9: 2763-6. PMID 10509931 DOI: 10.1016/S0960-894X(99)00464-3  1
1999 Quock RM, Burkey TH, Varga E, Hosohata Y, Hosohata K, Cowell SM, Slate CA, Ehlert FJ, Roeske WR, Yamamura HI. The delta-opioid receptor: molecular pharmacology, signal transduction, and the determination of drug efficacy. Pharmacological Reviews. 51: 503-32. PMID 10471416  1
1999 Bartosz-Bechowski H, Davis P, Slaninova J, Malatynska E, Stropova D, Porreca F, Yamamura HI, Hruby VJ. Cyclic enkephalin analogs that are hybrids of DPDPE-related peptides and metenkephalin-Arg-Gly-Leu: prohormone analogs that retain good potency and selectivity for delta opioid receptors. The Journal of Peptide Research : Official Journal of the American Peptide Society. 53: 329-36. PMID 10231722 DOI: 10.1034/j.1399-3011.1999.00033.x  1
1999 Varga EV, Stropova D, Rubenzik M, Waite S, Roeske WR, Yamamura HI. Phosphorylation of adenylyl cyclase VI upon chronic delta-opioid receptor stimulation. European Journal of Pharmacology. 364: R1-3. PMID 9932732 DOI: 10.1016/S0014-2999(98)00847-4  1
1999 Hau VS, Campos C, Hoshata K, Lipokowski A, Yamamura HI, Hruby VJ, Davis TP. Guanidino cationization effects on the blood-brain barrier permeability, in vitro stability and receptor binding of endomorphins Journal of Investigative Medicine. 47: 34A.  1
1998 Li G, Haq W, Xiang L, Lou BS, Hughes R, De Leon IA, Davis P, Gillespie TJ, Romanowski M, Zhu X, Misicka A, Lipkowski AW, Porreca F, Davis TP, Yamamura HI, et al. Modifications of the 4,4'-residues and SAR studies of Biphalin, a highly potent opioid receptor active peptide. Bioorganic & Medicinal Chemistry Letters. 8: 555-60. PMID 9871617 DOI: 10.1016/S0960-894X(98)00065-1  1
1998 Malatynska E, Waite S, Wei HB, Knapp RJ, Yamamura HI, Roeske WR. Structural correlates for down-regulation of m1 and m2 muscarinic receptor subtypes. Brain Research Bulletin. 47: 285-90. PMID 9865862 DOI: 10.1016/S0361-9230(98)00110-5  1
1998 Liao S, Alfaro-Lopez J, Shenderovich MD, Hosohata K, Lin J, Li X, Stropova D, Davis P, Jernigan KA, Porreca F, Yamamura HI, Hruby VJ. De novo design, synthesis, and biological activities of high-affinity and selective non-peptide agonists of the delta-opioid receptor. Journal of Medicinal Chemistry. 41: 4767-76. PMID 9822547 DOI: 10.1021/jm980374r  1
1998 Varga EV, Stropova D, Rubenzik M, Wang M, Landsman RS, Roeske WR, Yamamura HI. Identification of adenylyl cyclase isoenzymes in CHO and B82 cells. European Journal of Pharmacology. 348: R1-2. PMID 9652350 DOI: 10.1016/S0014-2999(98)00258-1  1
1998 Hosohata K, Burkey TH, Alfaro-Lopez J, Varga E, Hruby VJ, Roeske WR, Yamamura HI. Endomorphin-1 and endomorphin-2 are partial agonists at the human mu-opioid receptor. European Journal of Pharmacology. 346: 111-4. PMID 9617760 DOI: 10.1016/S0014-2999(98)00117-4  1
1998 Burkey TH, Ehlert FJ, Hosohata Y, Quock RM, Cowell S, Hosohata K, Varga E, Stropova D, Li X, Slate C, Nagase H, Porreca F, Hruby VJ, Roeske WR, Yamamura HI. The efficacy of delta-opioid receptor-selective drugs. Life Sciences. 62: 1531-6. PMID 9585131 DOI: 10.1016/S0024-3205(98)00102-7  1
1998 Slaninova J, Appleyard SM, Misicka A, Lipkowski AW, Knapp RJ, Weber SJ, Davis TP, Yamamura HI, Hruby VJ. [125I-Tyr1]biphalin binding to opioid receptors of rat brain and NG108-15 cell membranes. Life Sciences. 62: PL199-204. PMID 9570343  1
1998 Landsman RS, Makriyannis A, Deng H, Consroe P, Roeske WR, Yamamura HI. AM630 is an inverse agonist at the human cannabinoid CB1 receptor. Life Sciences. 62: PL109-13. PMID 9496703 DOI: 10.1016/S0024-3205(97)01187-9  1
1998 Kovacs I, Yamamura HI, Waite SL, Varga EV, Roeske WR. Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line. The Journal of Pharmacology and Experimental Therapeutics. 284: 500-7. PMID 9454790  1
1998 Olczak J, Kaczmarek K, Maszczyńska I, Lisowski M, Stropova D, Hruby VJ, Yamamura HI, Lipkowski AW, Zabrocki J. Consequences of cis-amide bond simulation in opioid peptides International Journal of Peptide Research and Therapeutics. 5: 437-440.  1
1997 Hruby VJ, Bartosz-Bechowski H, Davis P, Slaninova J, Zalewska T, Stropova D, Porreca F, Yamamura HI. Cyclic enkephalin analogues with exceptional potency and selectivity for delta-opioid receptors. Journal of Medicinal Chemistry. 40: 3957-62. PMID 9397176 DOI: 10.1021/jm9704762  1
1997 Burkey TH, Quock RM, Consroe P, Ehlert FJ, Hosohata Y, Roeske WR, Yamamura HI. Relative efficacies of cannabinoid CB1 receptor agonists in the mouse brain. European Journal of Pharmacology. 336: 295-8. PMID 9384246 DOI: 10.1016/S0014-2999(97)01255-7  1
1997 Landsman RS, Burkey TH, Consroe P, Roeske WR, Yamamura HI. SR141716A is an inverse agonist at the human cannabinoid CB1 receptor. European Journal of Pharmacology. 334: R1-2. PMID 9346339 DOI: 10.1016/S0014-2999(97)01160-6  1
1997 Haaseth RC, Zalewska T, Davis P, Yamamura HI, Porreca F, Hruby VJ. Para-substituted phenylalanine-4 analogues of [L-Ala3]DPDPE: highly selective delta opioid receptor ligands. The Journal of Peptide Research : Official Journal of the American Peptide Society. 50: 171-7. PMID 9309580 DOI: 10.1111/J.1399-3011.1997.TB01182.X  1
1997 Katsura Y, Zhang X, Homma K, Rice KC, Calderon SN, Rothman RB, Yamamura HI, Davis P, Flippen-Anderson JL, Xu H, Becketts K, Foltz EJ, Porreca F. Probes for narcotic receptor-mediated phenomena. 25. Synthesis and evaluation of N-alkyl-substituted (alpha-piperazinylbenzyl)benzamides as novel, highly selective delta opioid receptor agonists. Journal of Medicinal Chemistry. 40: 2936-47. PMID 9288176 DOI: 10.1021/jm970106d  1
1997 Hosohata K, Quock RM, Hosohata Y, Burkey TH, Makriyannis A, Consroe P, Roeske WR, Yamamura HI. AM630 is a competitive cannabinoid receptor antagonist in the guinea pig brain. Life Sciences. 61: PL115-8. PMID 9284087 DOI: 10.1016/S0024-3205(97)00596-1  1
1997 Misicka A, Cavagnero S, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Synthesis and biological properties of beta-MePhe3 analogues of deltorphin I and dermenkephalin: influence of biased chi 1 Phe3 residues on peptide recognition for delta-opioid receptors. The Journal of Peptide Research : Official Journal of the American Peptide Society. 50: 48-54. PMID 9273887 DOI: 10.1111/J.1399-3011.1997.TB00619.X  1
1997 Quock RM, Hosohata Y, Knapp RJ, Burkey TH, Hosohata K, Zhang X, Rice KC, Nagase H, Hruby VJ, Porreca F, Roeske WR, Yamamura HI. Relative efficacies of delta-opioid receptor agonists at the cloned human delta-opioid receptor. European Journal of Pharmacology. 326: 101-4. PMID 9178661 DOI: 10.1016/S0014-2999(97)83488-7  1
1997 Patel D, McKinley BD, Davis TP, Porreca F, Yamamura HI, Hruby VJ. Peptide targeting and delivery across the blood-brain barrier utilizing synthetic triglyceride esters: design, synthesis, and bioactivity. Bioconjugate Chemistry. 8: 434-41. PMID 9177851 DOI: 10.1021/bc970027g  1
1997 Burkey TH, Quock RM, Consroe P, Roeske WR, Yamamura HI. delta 9-Tetrahydrocannabinol is a partial agonist of cannabinoid receptors in mouse brain. European Journal of Pharmacology. 323: R3-4. PMID 9128853 DOI: 10.1016/S0014-2999(97)00146-5  1
1997 Bonner GG, Davis P, Stropova D, Ferguson R, Yamamura HI, Porreca F, Hruby VJ. Opioid peptides: simultaneous delta agonism and mu antagonism in somatostatin analogues. Peptides. 18: 93-100. PMID 9114458 DOI: 10.1016/S0196-9781(96)00242-2  1
1997 Misicka A, Lipkowski AW, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Structure-activity relationship of biphalin. The synthesis and biological activities of new analogues with modifications in positions 3 and 4. Life Sciences. 60: 1263-9. PMID 9096243 DOI: 10.1016/S0024-3205(97)00069-6  1
1997 Hosohata Y, Quock RM, Hosohata K, Makriyannis A, Consroe P, Roeske WR, Yamamura HI. AM630 antagonism of cannabinoid-stimulated [35S]GTP gamma S binding in the mouse brain. European Journal of Pharmacology. 321: R1-3. PMID 9083796 DOI: 10.1016/S0014-2999(97)00047-2  1
1997 Liao S, Lin J, Shenderovich MD, Han Y, Hasohata K, Davis P, Qiu W, Porreca F, Yamamura HI, Hruby VJ. The stereochemical requirements of the novel δ-opioid selective dipeptide antagonist TMT-Tic Bioorganic and Medicinal Chemistry Letters. 7: 3049-3052.  1
1997 Hruby VJ, Davis TP, O'Brien DF, Porreca F, Yamamura HI. Design of peptides and peptidomimetics that are selective, stable and can cross membrane barriers Protein Engineering. 10: 76.  1
1996 Millard SL, Bloom JW, Yamamura HI. Heterogeneity of tachykinin receptors in the rabbit lung. Neurochemical Research. 21: 277-83. PMID 9182253 DOI: 10.1007/BF02529145  1
1996 Varga EV, Li X, Stropova D, Zalewska T, Landsman RS, Knapp RJ, Malatynska E, Kawai K, Mizusura A, Nagase H, Calderon SN, Rice K, Hruby VJ, Roeske WR, Yamamura HI. The third extracellular loop of the human delta-opioid receptor determines the selectivity of delta-opioid agonists. Molecular Pharmacology. 50: 1619-24. PMID 8967985  1
1996 Qian X, Liao S, Stropova D, Yamamura HI, Hruby VJ. Novel scaffolds for non-peptide mimetics of delta opioid receptor agonists based on peptide leads. Regulatory Peptides. 65: 79-82. PMID 8876039 DOI: 10.1016/0167-0115(96)00075-4  1
1996 Boteju LW, Nikiforovich GV, Haskell-Luevano C, Fang SN, Zalewska T, Stropova D, Yamamura HI, Hruby VJ. The use of topographical constraints in receptor mapping: investigation of the topographical requirements of the tryptophan 30 residue for receptor binding of Asp-Tyr-D-Phe-Gly-Trp-(N-Me)Nle-Asp-Phe-NH2 (SNF 9007), a cholecystokinin (26-33) analogue that binds to both CCK-B and delta-opioid receptors. Journal of Medicinal Chemistry. 39: 4120-4. PMID 8831778 DOI: 10.1021/jm960078j  1
1996 Malatynska E, Wang Y, Knapp RJ, Waite S, Calderon S, Rice K, Hruby VJ, Yamamura HI, Roeske WR. Human delta opioid receptor: functional studies on stably transfected Chinese hamster ovary cells after acute and chronic treatment with the selective nonpeptidic agonist SNC-80. The Journal of Pharmacology and Experimental Therapeutics. 278: 1083-9. PMID 8819489  1
1996 Misicka A, Maszczynska I, Lipkowski AW, Stropova D, Yamamura HI, Hruby VJ. Synthesis and biological properties of gamma-glutamyl-dermorphin, a prodrug. Life Sciences. 58: 905-11. PMID 8786696 DOI: 10.1016/0024-3205(96)00033-1  1
1996 Vanderah TW, Bernstein RN, Yamamura HI, Hruby VJ, Porreca F. Enhancement of morphine antinociception by a CCKB antagonist in mice is mediated via opioid delta receptors. The Journal of Pharmacology and Experimental Therapeutics. 278: 212-9. PMID 8764354  1
1996 Li X, Varga EV, Stropova D, Zalewska T, Malatynska E, Knapp RJ, Roeske WR, Yamamura HI. delta-Opioid receptor: the third extracellular loop determines naltrindole selectivity. European Journal of Pharmacology. 300: R1-2. PMID 8741185  1
1996 Edsall SA, Knapp RJ, Vanderah TW, Roeske WR, Consroe P, Yamamura HI. Antisense oligodeoxynucleotide treatment to the brain cannabinoid receptor inhibits antinociception. Neuroreport. 7: 593-6. PMID 8730837  1
1996 Lung FD, Meyer JP, Lou BS, Xiang L, Li G, Davis P, DeLeon IA, Yamamura HI, Porreca F, Hruby VJ. Effects of modifications of residues in position 3 of dynorphin A(1-11)-NH2 on kappa receptor selectivity and potency. Journal of Medicinal Chemistry. 39: 2456-60. PMID 8691442 DOI: 10.1021/jm950655o  1
1996 Lung FD, Collins N, Stropova D, Davis P, Yamamura HI, Porreca F, Hruby VJ. Design, synthesis, and biological activities of cyclic lactam peptide analogues of dynorphine A(1-11)-NH2. Journal of Medicinal Chemistry. 39: 1136-41. PMID 8676350 DOI: 10.1021/jm950369c  1
1996 Knapp RJ, Santoro G, De Leon IA, Lee KB, Edsall SA, Waite S, Malatynska E, Varga E, Calderon SN, Rice KC, Rothman RB, Porreca F, Roeske WR, Yamamura HI. Structure-activity relationships for SNC80 and related compounds at cloned human delta and mu opioid receptors. The Journal of Pharmacology and Experimental Therapeutics. 277: 1284-91. PMID 8667189  1
1996 Qian X, Shenderovich MD, Kover KE, Davis P, Horvath R, Zalewska T, Yamamura HI, Porreca F, Hruby VJ. Probing the stereochemical requirements for receptor recognition of δ opioid agonists through topographic modifications in position 1 Journal of the American Chemical Society. 118: 7280-7290. DOI: 10.1021/ja954241w  1
1995 Knapp RJ, Landsman R, Waite S, Malatynska E, Varga E, Haq W, Hruby VJ, Roeske WR, Nagase H, Yamamura HI. Properties of TAN-67, a nonpeptidic delta-opioid receptor agonist, at cloned human delta- and mu-opioid receptors. European Journal of Pharmacology. 291: 129-34. PMID 8566162 DOI: 10.1016/0922-4106(95)90134-5  1
1995 Lung FD, Meyer JP, Li G, Lou BS, Stropova D, Davis P, Yamamura HI, Porreca F, Hruby VJ. Highly kappa receptor-selective dynorphin A analogues with modifications in position 3 of dynorphin A(1-11)-NH2. Journal of Medicinal Chemistry. 38: 585-6. PMID 7861405 DOI: 10.1021/JM00004A002  1
1995 Slaninova J, Knapp RJ, Weber SJ, Davis TP, Fang SN, Hruby VJ, Yamamura HI. [125I]SNF 8702: a selective radioligand for CCKB receptors. Peptides. 16: 221-4. PMID 7784252 DOI: 10.1016/0196-9781(94)00168-5  1
1995 Knapp RJ, Malatynska E, Collins N, Fang L, Wang JY, Hruby VJ, Roeske WR, Yamamura HI. Molecular biology and pharmacology of cloned opioid receptors. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 9: 516-25. PMID 7737460  1
1995 Witt-Enderby PA, Yamamura HI, Halonen M, Lai J, Palmer JD, Bloom JW. Regulation of airway muscarinic cholinergic receptor subtypes by chronic anticholinergic treatment. Molecular Pharmacology. 47: 485-90. PMID 7700247  1
1995 Malatynska E, Knapp RJ, Stropova D, Varga E, Yamamura HI. The role of the Val353 residue in antagonist binding to rat CCK-B receptors. Neuroreport. 6: 1325-9. PMID 7669996  1
1995 Meyer JP, Davis P, Lee KB, Porreca F, Yamamura HI, Hruby VJ. Synthesis using a Fmoc-based strategy and biological activities of some reduced peptide bond pseudopeptide analogues of dynorphin A1. Journal of Medicinal Chemistry. 38: 3462-8. PMID 7658433 DOI: 10.1021/JM00018A006  1
1995 Hruby VJ, Yamamura HI, Porreca F. Molecular organization of receptors. Efficacy, agonists, and antagonists. Annals of the New York Academy of Sciences. 757: 7-22. PMID 7611710 DOI: 10.1111/j.1749-6632.1995.tb17461.x  1
1995 Malatynska E, De Leon I, Allen D, Yamamura HI. Effects of amitriptyline on GABA-stimulated 36CI- uptake in relation to a behavioral model of depression. Brain Research Bulletin. 37: 53-9. PMID 7606479 DOI: 10.1016/0361-9230(94)00257-6  1
1995 Malatynska E, Wang Y, Knapp RJ, Santoro G, Li X, Waite S, Roeske WR, Yamamura HI. Human delta opioid receptor: a stable cell line for functional studies of opioids. Neuroreport. 6: 613-6. PMID 7605911  1
1995 Knapp RJ, Waite S, Landsman R, Santoro G, De Leon IA, Malatynska E, Varga E, Nagase H, Calderon SN, Rice K. Efficacy of peptide and nonpeptidic agonists at the cloned human delta opioid receptor. Proceedings of the Western Pharmacology Society. 38: 141-3. PMID 7480008  1
1995 Misicka A, Lipkowski AW, Slaninova J, Davis P, Yamamura HI, Porreca F, Hruby VJ. The synthesis and opioid receptor binding affinities of analogues of dermorphin and its N-terminal tetrapeptide fragment with dibasic acids in position 2. Life Sciences. 57: 1633-40. PMID 7475903 DOI: 10.1016/0024-3205(95)02142-6  1
1995 Misicka A, Lipkowski AW, Stropova D, Davis P, Porreca F, Yamamura HI, Hruby VJ. Amino acids with amphiphilic side chains: Deltorphin analogues with Phe3 replaced by all β-hydroxyphenylalanine diastereoisomers Letters in Peptide Science. 2: 203-205. DOI: 10.1007/BF00119153  1
1995 Lipkowski AW, Misicka A, Porreca F, Davis P, Yamamura HI, Stropova D, Hruby VJ. Benzomorphan alkaloids: Natural peptidomimetics of opioid peptide pharmacophores Letters in Peptide Science. 2: 177-181. DOI: 10.1007/BF00119147  1
1994 Bartosz-Bechowski H, Davis P, Zalewska T, Slaninova J, Porreca F, Yamamura HI, Hruby VJ. Cyclic enkephalin analogs with exceptional potency at peripheral delta opioid receptors. Journal of Medicinal Chemistry. 37: 146-50. PMID 8289188 DOI: 10.1021/JM00027A018  1
1994 Misicka A, Lipkowski AW, Horvath R, Davis P, Yamamura HI, Porreca F, Hruby VJ. Design of cyclic deltorphins and dermenkephalins with a disulfide bridge leads to analogues with high selectivity for delta-opioid receptors. Journal of Medicinal Chemistry. 37: 141-5. PMID 8289187 DOI: 10.1021/JM00027A017  1
1994 Knapp RJ, Malatynska E, Fang L, Li X, Babin E, Nguyen M, Santoro G, Varga EV, Hruby VJ, Roeske WR. Identification of a human delta opioid receptor: cloning and expression. Life Sciences. 54: PL463-9. PMID 8201839 DOI: 10.1016/0024-3205(94)90138-4  1
1994 Haaseth RC, Horan PJ, Bilsky EJ, Davis P, Zalewska T, Slaninova J, Yamamura HI, Weber SJ, Davis TP, Porreca F. [L-Ala3]DPDPE: a new enkephalin analog with a unique opioid receptor activity profile. Further evidence of delta-opioid receptor multiplicity. Journal of Medicinal Chemistry. 37: 1572-7. PMID 8201592 DOI: 10.1021/JM00037A007  1
1994 Knapp RJ, Malatynska E, Hashimoto S, Fang S, Hunt M, Wamsley JK, Peterson P, Zalewska T, Hruby VJ, Yamamura HI. [3H]SNF8702 autoradiography of CCK-B receptors in guinea pig brain and studies with a cloned rat CCK-B receptor. Annals of the New York Academy of Sciences. 713: 380-3. PMID 8185194 DOI: 10.1111/j.1749-6632.1994.tb44099.x  1
1994 Fang L, Knapp RJ, Horvath R, Matsunaga TO, Haaseth RC, Hruby VJ, Porreca F, Yamamura HI. Characterization of [3H]naltrindole binding to delta opioid receptors in mouse brain and mouse vas deferens: evidence for delta opioid receptor heterogeneity. The Journal of Pharmacology and Experimental Therapeutics. 268: 836-46. PMID 8113996  1
1994 Rao RK, Levenson S, Fang SN, Hruby VJ, Yamamura HI, Porreca F. Characterization of SNF 9007, a novel cholecystokinin/opoid ligand in mouse ileum in vitro: evidence for involvement of cholecystokininA and cholecystokininB receptors in regulation of ion transport. The Journal of Pharmacology and Experimental Therapeutics. 268: 1003-9. PMID 8113956  1
1994 Polt R, Porreca F, Szabò LZ, Bilsky EJ, Davis P, Abbruscato TJ, Davis TP, Harvath R, Yamamura HI, Hruby VJ. Glycopeptide enkephalin analogues produce analgesia in mice: evidence for penetration of the blood-brain barrier. Proceedings of the National Academy of Sciences of the United States of America. 91: 7114-8. PMID 8041755 DOI: 10.1073/pnas.91.15.7114  1
1994 Qian X, Kövér KE, Shenderovich MD, Lou BS, Misicka A, Zalewska T, Horváth R, Davis P, Bilsky EJ, Porreca F, Yamamura HI, Hruby VJ. Newly discovered stereochemical requirements in the side-chain conformation of δ opioid agonists for recognizing opioid δ receptors Journal of Medicinal Chemistry. 37: 1746-1757. PMID 8021915 DOI: 10.1021/JM00038A004  1
1994 Ehlert FJ, Roeske WR, Yamamura HI. Muscarinic receptors and novel strategies for the treatment of age-related brain disorders. Life Sciences. 55: 2135-45. PMID 7997072 DOI: 10.1016/0024-3205(94)00394-7  1
1994 Wild KD, Porreca F, Yamamura HI, Raffa RB. Differentiation of receptor subtypes by thermodynamic analysis: application to opioid delta receptors. Proceedings of the National Academy of Sciences of the United States of America. 91: 12018-21. PMID 7991576 DOI: 10.1073/pnas.91.25.12018  1
1994 Meyer JP, Collins N, Lung FD, Davis P, Zalewska T, Porreca F, Yamamura HI, Hruby VJ. Design, synthesis, and biological properties of highly potent cyclic dynorphin A analogues. Analogues cyclized between positions 5 and 11. Journal of Medicinal Chemistry. 37: 3910-7. PMID 7966152 DOI: 10.1021/JM00049A010  1
1994 Sora I, Richman J, Santoro G, Wei HB, Wang Y, Vanderah T, Horvath R, Nguyen M, Waite S, Roeske WR, Yamamura HI. The Cloning and Expression of a Human Creatine Transporter Biochemical and Biophysical Research Communications. 204: 419-427. PMID 7945388 DOI: 10.1006/bbrc.1994.2475  1
1994 Knapp RJ, Malatynska E, Peterson P, Zalewska T, Fang S, Hruby VJ, Smith TL, Yamamura HI. [N-methylnorleucine-(28,31)]cholecystokinin-(26-33) (SNF 8702) activity at a cloned rat CCKB receptor. European Journal of Pharmacology. 269: 133-8. PMID 7851490 DOI: 10.1016/0922-4106(94)90079-5  1
1994 Wei HB, Yamamura HI, Roeske WR. Down-regulation and desensitization of the muscarinic M1 and M2 receptors in transfected fibroblast B82 cells. European Journal of Pharmacology. 268: 381-91. PMID 7805762 DOI: 10.1016/0922-4106(94)90063-9  1
1994 Misicka A, Lipkowski AW, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Delta opioid receptor selective ligands; DPLPE-deltorphin chimeric peptide analogues. International Journal of Peptide and Protein Research. 44: 80-4. PMID 7718035 DOI: 10.1111/J.1399-3011.1994.TB00407.X  1
1994 Misicka A, Lipkowski AW, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Delta opioid receptor selective ligands; DPLPE-deltorphin chimeric peptide analogues. International Journal of Peptide and Protein Research. 44: 607. PMID 7705984  1
1994 Vanderah TW, Lai J, Yamamura HI, Porreca F. Antisense oligodeoxynucleotide to the CCKB receptor produces naltrindole- and [Leu5]enkephalin antiserum-sensitive enhancement of morphine antinociception. Neuroreport. 5: 2601-5. PMID 7696612  1
1994 Mania-Farnell BL, Merrill BJ, Yamamura HI, Davis TP. Second messenger activators regulate CCK mRNA in the human neuroepithelioma cell line SK-N-MCIXC. Annals of the New York Academy of Sciences. 713: 446-8. PMID 7514375 DOI: 10.1111/j.1749-6632.1994.tb44122.x  1
1994 Rao RK, Levenson S, Fang SN, Hruby VJ, Yamamura HI, Porreca F. Role of substance P in the regulation of ion transport by CCKA and CCKB receptors in mouse ileum. Annals of the New York Academy of Sciences. 713: 420-1. PMID 7514373 DOI: 10.1111/j.1749-6632.1994.tb44113.x  1
1994 Hruby VJ, Collins N, Lung FD, Meyer JP, Davis TP, Yamamura HI, Porreca F. Design of peptides and peptidomimetics for delta and kappa opioid receptor subtypes Regulatory Peptides. 54: 123-124. DOI: 10.1016/0167-0115(94)90420-0  1
1994 Misicka A, Lipkowski AW, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Structure-activity relationships of analogues of higly potent opioid peptide, biphalin Regulatory Peptides. 53: S131-S132. DOI: 10.1016/0167-0115(94)90276-3  1
1994 Misicka A, Lipkowski AW, Horvath R, Davis P, Porreca F, Yamamura HI, Hruby VJ. Topographic model of delta opioid selective ligands; DPLPE-deltorphin hybrid analogues Regulatory Peptides. 53: S129-S130. DOI: 10.1016/0167-0115(94)90275-5  1
1994 Hruby VJ, Misicka A, Lipkowski AW, Haaseth R, Bartosz H, Qian X, Collins N, Meyer JP, Szabo L, Polt R, Porreca F, Davis T, Yamamura HI. New opioid compounds in analgesia Regulatory Peptides. 53: S71-S72. DOI: 10.1016/0167-0115(94)90246-1  1
1993 Wild KD, Horan PJ, Misicka A, Lipkowski A, Haaseth RC, Matsunaga TO, Hruby VJ, Toth G, Borsodi A, Yamamura HI. Pseudoirreversible binding characteristics of [D-Ala2,Glu4]deltorphin and its Cys4 substituted derivative to delta-opioid receptors. European Journal of Pharmacology. 246: 25-31. PMID 8394818 DOI: 10.1016/0922-4106(93)90005-T  1
1993 Horan PJ, Mattia A, Bilsky EJ, Weber S, Davis TP, Yamamura HI, Malatynska E, Appleyard SM, Slaninova J, Misicka A. Antinociceptive profile of biphalin, a dimeric enkephalin analog. The Journal of Pharmacology and Experimental Therapeutics. 265: 1446-54. PMID 8389867  1
1993 Horan PJ, Wild KD, Misicka A, Lipkowski A, Haaseth RC, Hruby VJ, Weber SJ, Davis TP, Yamamura HI, Porreca F. Agonist and antagonist profiles of [D-Ala2,Glu4]deltorphin and its [Cys4]- and [Ser4]-substituted derivatives: further evidence of opioid delta receptor multiplicity. The Journal of Pharmacology and Experimental Therapeutics. 265: 896-902. PMID 8388462  1
1993 Henderson AK, Roeske WR, Smith TL, Yamamura HI. Desensitization of neurokinin A receptors expressed by B82 fibroblasts. European Journal of Pharmacology. 245: 75-8. PMID 8386670 DOI: 10.1016/0922-4106(93)90172-6  1
1993 Horan PJ, Wild KD, Kazmierski WM, Ferguson R, Hruby VJ, Weber SJ, Davis TP, Fang L, Knapp RJ, Yamamura HI. Unexpected antinociceptive potency of cyclic [D-Tca1]CTAP: potential for a novel mechanism of action. European Journal of Pharmacology. 233: 53-62. PMID 8386089 DOI: 10.1016/0014-2999(93)90348-L  1
1993 Parola AL, Yamamura HI, Laird HE. Peripheral-type benzodiazepine receptors. Life Sciences. 52: 1329-42. PMID 8385255 DOI: 10.1016/0024-3205(93)90168-3  1
1993 Wild KD, Fang L, McNutt RW, Chang KJ, Toth G, Borsodi A, Yamamura HI, Porreca F. Binding of BW 373U86, a non-peptidic delta opioid receptor agonist, is not regulated by guanine nucleotides and sodium. European Journal of Pharmacology. 246: 289-92. PMID 8223952 DOI: 10.1016/0922-4106(93)90044-A  1
1993 Kawasaki AM, Knapp RJ, Kramer TH, Walton A, Wire WS, Hashimoto S, Yamamura HI, Porreca F, Burks TF, Hruby VJ. Design and synthesis of highly potent and selective cyclic dynorphin A analogs. 2. New analogs. Journal of Medicinal Chemistry. 36: 750-7. PMID 8096246 DOI: 10.1021/JM00058A012  1
1993 Fujiwara Y, Tomita H, Hikiji M, Kashihara K, Otsuki S, Ohnuki T, Hamagishi Y, Oki T, Sora I, Roeske WR, Yamamura HI. Characterization of a cloned rat serotonin 5-HT1A receptor expressed in the HeLa cell line Life Sciences. 52: 949-958. PMID 8095315 DOI: 10.1016/0024-3205(93)90530-G  1
1993 Kawasaki AM, Knapp RJ, Walton A, Wire WS, Zalewska T, Yamamura HI, Porreca F, Burks TF, Hruby VJ. Syntheses, opioid binding affinities, and potencies of dynorphin A analogues substituted in positions, 1, 6, 7, 8 and 10. International Journal of Peptide and Protein Research. 42: 411-9. PMID 7906258 DOI: 10.1111/J.1399-3011.1993.TB00148.X  1
1993 Witt-Enderby PA, Yamamura HI, Halonen M, Palmer JD, Bloom JW. Chronic exposure to a beta 2-adrenoceptor agonist increases the airway response to methacholine. European Journal of Pharmacology. 241: 121-3. PMID 7901034 DOI: 10.1016/0014-2999(93)90942-B  1
1993 Boteju LW, Zalewska T, Yamamura HI, Hruby VJ. Tryptophan-norleucine 1,5-disubstituted tetrazoles as cis peptide bond mimics: Investigation of the bioactive conformation of a potent and selective peptide for the cholecystokinin-B receptor Bioorganic and Medicinal Chemistry Letters. 3: 2011-2016. DOI: 10.1016/S0960-894X(01)81005-2  1
1993 Hristova-Kazmierski MK, Horan P, Davis P, Yamamura HI, Kramer T, Horvath R, Kazmierski WM, Porreca F, Hruby VJ. A new approach to enhance bioavailability of biologically active peptides: conjugation of a δ opioid agonist to β-cyclodextrin Bioorganic and Medicinal Chemistry Letters. 3: 831-834. DOI: 10.1016/S0960-894X(00)80675-7  1
1992 Lai J, Nunan L, Waite SL, Ma SW, Bloom JW, Roeske WR, Yamamura HI. Chimeric M1/M2 muscarinic receptors: correlation of ligand selectivity and functional coupling with structural modifications. The Journal of Pharmacology and Experimental Therapeutics. 262: 173-80. PMID 1625198  1
1992 Mahesh VK, Nunan LM, Halonen M, Yamamura HI, Palmer JD, Bloom JW. A minority of muscarinic receptors mediate rabbit tracheal smooth muscle contraction. American Journal of Respiratory Cell and Molecular Biology. 6: 279-86. PMID 1540392 DOI: 10.1165/ajrcmb/6.3.279  1
1992 Weber SJ, Greene DL, Hruby VJ, Yamamura HI, Porreca F, Davis TP. Whole body and brain distribution of [3H]cyclic [D-Pen2,D-Pen5] enkephalin after intraperitoneal, intravenous, oral and subcutaneous administration. The Journal of Pharmacology and Experimental Therapeutics. 263: 1308-16. PMID 1469637  1
1992 Kazmierski WM, Ferguson RD, Knapp RJ, Lui GK, Yamamura HI, Hruby VJ. Reduced peptide bond cyclic somatostatin based opioid octapeptides. Synthesis, conformational properties and pharmacological characterization. International Journal of Peptide and Protein Research. 39: 401-14. PMID 1358847  1
1992 Knapp RJ, Yamamura HI. Delta opioid receptor radioligands. Biochemical Pharmacology. 44: 1687-95. PMID 1333204 DOI: 10.1016/0006-2952(92)90060-V  1
1992 Fang L, Knapp RJ, Matsunaga T, Weber SJ, Davis T, Hruby VJ, Yamamura HI. Synthesis of [D-Ala2,4'-125I-Phe3,Glu4]deltorphin and characterization of its delta opioid receptor binding properties. Life Sciences. 51: PL189-93. PMID 1331636 DOI: 10.1016/0024-3205(92)90628-3  1
1992 Misicka A, Lipkowski AW, Horvath R, Davis P, Kramer TH, Yamamura HI, Hruby VJ. Topographical requirements for delta opioid ligands: common structural features of dermenkephalin and deltorphin. Life Sciences. 51: 1025-32. PMID 1326067 DOI: 10.1016/0024-3205(92)90501-F  1
1992 Kashihara K, Varga EV, Waite SL, Roeske WR, Yamamura HI. Cloning of the rat M3, M4 and M5 muscarinic acetylcholine receptor genes by the polymerase chain reaction (PCR) and the pharmacological characterization of the expressed genes. Life Sciences. 51: 955-71. PMID 1325587 DOI: 10.1016/0024-3205(92)90403-C  1
1992 Tourwé D, Couder J, Ceusters M, Meert D, Burks TF, Kramer TH, Davis P, Knapp R, Yamamura HI, Leysen JE. Synthesis and biological activities of linear and cyclic enkephalin analogues containing a psi (E,CH = CH) or psi (CH2CH2) isosteric replacement. International Journal of Peptide and Protein Research. 39: 131-6. PMID 1325415  1
1992 Toth G, Russell KC, Landis G, Kramer TH, Fang L, Knapp R, Davis P, Burks TF, Yamamura HI, Hruby VJ. Ring substituted and other conformationally constrained tyrosine analogues of [D-Pen2,D-Pen5]enkephalin with delta opioid receptor selectivity. Journal of Medicinal Chemistry. 35: 2384-91. PMID 1320122  1
1992 Yamamura MS, Horvath R, Toth G, Otvos F, Malatynska E, Knapp RJ, Porreca F, Hruby VJ, Yamamura HI. Characterization of [3H]naltrindole binding to delta opioid receptors in rat brain. Life Sciences. 50: PL119-24. PMID 1313133 DOI: 10.1016/0024-3205(92)90464-Z  1
1992 Henderson AK, Yamamura HI, Maggi CA, Buck SH, Van Giersbergen PL, Roeske WR. Demonstration of a neurokinin A receptor subtype in transfected fibroblasts. European Journal of Pharmacology. 225: 175-8. PMID 1312943 DOI: 10.1016/0922-4106(92)90099-H  1
1992 Horan P, Taylor J, Yamamura HI, Porreca F. Extremely long-lasting antagonistic actions of nor-binaltorphimine (nor-BNI) in the mouse tail-flick test. The Journal of Pharmacology and Experimental Therapeutics. 260: 1237-43. PMID 1312164  1
1992 Wei HB, Roeske WR, Lai J, Wanibuchi F, Hidaka K, Usuda S, Yamamura HI. Pharmacological characterization of a novel muscarinic partial agonist, YM796, in transfected cells expressing the m1 or m2 muscarinic receptor gene. Life Sciences. 50: 355-63. PMID 1310135 DOI: 10.1016/0024-3205(92)90437-T  1
1992 Sora I, Fujiwara Y, Tomita H, Ishizu H, Akiyama K, Otsuki S, Yamamura HI. Lack of effect of haloperidol or methamphetamine treatment on the mRNA levels of two dopamine D2 receptor isoforms in rat brain. The Japanese Journal of Psychiatry and Neurology. 46: 967-73. PMID 1304623  0.56
1992 Misicka A, Nikiforovich G, Lipkowski AW, Horvath R, Davis P, Kramer TH, Yamamura HI, Hruby VJ. Topographical requirements for delta opioid ligands: The synthesis and biological properties of a cyclic analogue of deltorphin I Bioorganic and Medicinal Chemistry Letters. 2: 547-552. DOI: 10.1016/S0960-894X(01)81195-1  1
1992 Lai J, Roeske W, Yamamura HI. Structure-function correlation of muscarinic acetylfholine receptors European Neuropsychopharmacology. 2: 227-228. DOI: 10.1016/0924-977X(92)90078-M  1
1991 Malatynska E, Dilsaver SC, Knapp RJ, Giroux ML, Ikeda M, Yamamura HI. The interaction of a benzodiazepine receptor antagonist (Ro15-1788) with GABA and GABA receptor antagonists at the GABA(A) receptor chloride-ionophore complex. Neurochemistry International. 18: 405-10. PMID 20504718  0.68
1991 Davis TP, Gillespie TJ, Shook J, Kramer TH, Hoyer G, Hawkins K, Davis P, Yamamura HI, Burks TF. Changes in opioid receptor selectivity following processing of peptide E: effect on gut motility. Gastroenterology. 100: 1603-15. PMID 1850373  1
1991 van Giersbergen PL, Shatzer SA, Henderson AK, Lai J, Nakanishi S, Yamamura HI, Buck SH. Characterization of a tachykinin peptide NK2 receptor transfected into murine fibroblast B82 cells. Proceedings of the National Academy of Sciences of the United States of America. 88: 1661-5. PMID 1848006  1
1991 Fujiwara Y, Sora I, Tomita H, Akiyama K, Otsuki S, Yamamura HI. Localization of the mRNAs for two dopamine D2 receptor isoforms in the rat brain. The Japanese Journal of Psychiatry and Neurology. 45: 897-902. PMID 1813683  0.56
1991 Weber SJ, Greene DL, Sharma SD, Yamamura HI, Kramer TH, Burks TF, Hruby VJ, Hersh LB, Davis TP. Distribution and analgesia of [3H][D-Pen2, D-Pen5]enkephalin and two halogenated analogs after intravenous administration. The Journal of Pharmacology and Experimental Therapeutics. 259: 1109-17. PMID 1762065  1
1991 Lai J, Smith TL, Mei L, Ikeda M, Fujiwara Y, Gomez J, Halonen M, Roeske WR, Yamamura HI. The molecular properties of the M1 muscarinic receptor and its regulation of cytosolic calcium in a eukaryotic gene expression system. Advances in Experimental Medicine and Biology. 287: 313-30. PMID 1759615  1
1991 Mei L, Lai J, Yamamura HI, Roeske WR. Pharmacologic comparison of selected agonists for the M1 muscarinic receptor in transfected murine fibroblast cells (B82). The Journal of Pharmacology and Experimental Therapeutics. 256: 689-94. PMID 1704434  1
1991 Slaninova J, Knapp RJ, Wu JJ, Fang SN, Kramer T, Burks TF, Hruby VJ, Yamamura HI. Opioid receptor binding properties of analgesic analogues of cholecystokinin octapeptide. European Journal of Pharmacology. 200: 195-8. PMID 1663041 DOI: 10.1016/0014-2999(91)90688-M  1
1991 Misicka A, Lipkowski AW, Fang L, Knapp RJ, Davis P, Kramer T, Burks TF, Yamamura HI, Carr DB, Hruby VJ. Topographical requirements for delta opioid ligands: presence of a carboxyl group in position 4 is not critical for deltorphin high delta receptor affinity and analgesic activity. Biochemical and Biophysical Research Communications. 180: 1290-7. PMID 1659410 DOI: 10.1016/S0006-291X(05)81335-X  1
1991 Lai J, Waite SL, Bloom JW, Yamamura HI, Roeske WR. The m2 muscarinic acetylcholine receptors are coupled to multiple signaling pathways via pertussis toxin-sensitive guanine nucleotide regulatory proteins. The Journal of Pharmacology and Experimental Therapeutics. 258: 938-44. PMID 1653846  1
1991 Knapp RJ, Sharma SD, Toth G, Duong MT, Fang L, Bogert CL, Weber SJ, Hunt M, Davis TP, Wamsley JK. [D-Pen2,4'-125I-Phe4,D-Pen5]enkephalin: a selective high affinity radioligand for delta opioid receptors with exceptional specific activity. The Journal of Pharmacology and Experimental Therapeutics. 258: 1077-83. PMID 1653834  1
1991 Cavagnero S, Misicka A, Knapp RJ, Davis P, Fang L, Burks TF, Yamamura HI, Hruby VJ. Delta opioid receptor-selective ligands: [D-Pen2,D-Pen5]enkephalin-dermenkephalin chimeric peptides. Life Sciences. 49: 495-503. PMID 1650414 DOI: 10.1016/0024-3205(91)90066-K  1
1991 Henderson AK, Yamamura HI, Maggi CA, Roeske WR, Smith TL. Neurokinin A receptors are coupled to calcium mobilization in transfected fibroblasts. European Journal of Pharmacology. 206: 251-3. PMID 1649764 DOI: 10.1016/S0922-4106(05)80026-4  1
1991 Hruby VJ, Toth G, Gehrig CA, Kao LF, Knapp R, Lui GK, Yamamura HI, Kramer TH, Davis P, Burks TF. Topographically designed analogues of [D-Pen,D-Pen5]enkephalin. Journal of Medicinal Chemistry. 34: 1823-30. PMID 1648137  1
1991 Parola AL, Yamamura HI. Pharmacological and molecular basis for reclassifying peripheral-type benzodiazepine receptors as τ (tau) receptors European Neuropsychopharmacology. 1: 289-294. DOI: 10.1016/0924-977X(91)90533-Z  1
1991 Malatynska E, Dilsaver SC, Knapp RJ, Giroux ML, Ikeda M, Yamamura HI. The interaction of a benzodiazepine receptor antagonist (Ro15-1788) with GABA and GABA receptor antagonists at the GABAA receptor chloride-ionophore complex Neurochemistry International. 18: 405-410. DOI: 10.1016/0197-0186(91)90173-B  1
1991 Kazmierski WM, Yamamura HI, Hruby VJ. Topographic Design of Peptide Neurotransmitters and Hormones on Stable Backbone Templates: Relation of Conformation and Dynamics to Bioactivity Journal of the American Chemical Society. 113: 2275-2283.  1
1990 Hruby VJ, Fang SA, Knapp R, Kazmierski W, Lui GK, Yamamura HI. Cholecystokinin analogues with high affinity and selectivity for brain membrane receptors. International Journal of Peptide and Protein Research. 35: 566-73. PMID 2401597  1
1990 Mei L, Roeske WR, Izutsu KT, Yamamura HI. Characterization of muscarinic acetylcholine receptors in human labial salivary glands. European Journal of Pharmacology. 176: 367-70. PMID 2328757 DOI: 10.1016/0014-2999(90)90032-2  1
1990 Fujiwara Y, Nelson DL, Kashihara K, Varga E, Roeske WR, Yamamura HI. The cloning and sequence analysis of the rat serotonin-1A receptor gene. Life Sciences. 47: PL127-32. PMID 2273937  0.8
1990 Knapp RJ, Vaughn LK, Fang SN, Bogert CL, Yamamura MS, Hruby VJ, Yamamura HI. A new, highly selective CCK-B receptor radioligand ([3H][N-methyl-Nle28,31]CCK26-33): evidence for CCK-B receptor heterogeneity. The Journal of Pharmacology and Experimental Therapeutics. 255: 1278-86. PMID 2262906  1
1990 Lai J, Bloom JW, Yamamura HI, Roeske WR. Amplification of the rat M2 muscarinic receptor gene by the polymerase chain reaction: functional expression of the M2 muscarinic receptor. Life Sciences. 47: 1001-13. PMID 2172674 DOI: 10.1016/0024-3205(90)90472-4  1
1990 Gomez J, Bloom JW, Yamamura HI, Halonen M. Characterization of receptors for platelet-activating factor in guinea pig lung membranes. American Journal of Respiratory Cell and Molecular Biology. 3: 259-64. PMID 2167700 DOI: 10.1165/ajrcmb/3.3.259  1
1990 Knapp RJ, Yamamura HI. [3H][D-Pen2, D-Pen5]enkephalin binding to delta opioid receptors on intact neuroblastoma-glioma (NG 108-15) hybrid cells. Life Sciences. 46: 1457-63. PMID 2161068 DOI: 10.1016/0024-3205(90)90462-Z  1
1990 Vaughn LK, Wire WS, Davis P, Shimohigashi Y, Toth G, Knapp RJ, Hruby VJ, Burks TF, Yamamura HI. Differentiation between rat brain and mouse vas deferens delta opioid receptors. European Journal of Pharmacology. 177: 99-101. PMID 2160370 DOI: 10.1016/0014-2999(90)90556-L  1
1990 Knapp RJ, Malatynska E, Yamamura HI. From binding studies to the molecular biology of GABA receptors. Neurochemical Research. 15: 105-12. PMID 2159117 DOI: 10.1007/BF00972199  1
1990 Toth G, Kramer TH, Knapp R, Lui G, Davis P, Burks TF, Yamamura HI, Hruby VJ. [D-Pen2,D-Pen5]enkephalin analogues with increased affinity and selectivity for delta opioid receptors. Journal of Medicinal Chemistry. 33: 249-53. PMID 2153205  1
1990 Kawasaki AM, Knapp RJ, Kramer TH, Wire WS, Vasquez OS, Yamamura HI, Burks TF, Hruby VJ. Design and synthesis of highly potent and selective cyclic dynorphin A analogues. Journal of Medicinal Chemistry. 33: 1874-9. PMID 1972964  1
1990 Henderson AK, Lai J, Buck SH, Fujiwara Y, Singh G, Yamamura MS, Nakanishi S, Roeske WR, Yamamura HI. Accelerated communication a cloned NK2 receptor mediates phosphatidylinositol hydrolysis in a transfected murine fibrolast Life Sciences. 47: PL7-PL12. DOI: 10.1016/0024-3205(90)90329-P  1
1990 Roeske WR, Lai J, Mei L, Bloom JW, Yamamura HI. Pharmacologic comparison of the cloned M1 and M2 muscarinic receptors of the rat expressed in murine fibroblast cells European Journal of Pharmacology. 183: 1618. DOI: 10.1016/0014-2999(90)91905-Q  1
1990 Hruby VJ, Kazmierski W, Pelton JT, Yamamura HI, Burks TF. Conversion of somatostatin to an opioid peptide: design using a conformational template and topographical constraints European Journal of Pharmacology. 183: 54. DOI: 10.1016/0014-2999(90)91304-T  1
1989 Mei L, Lai J, Yamamura HI, Roeske WR. The relationship between agonist states of the M1 muscarinic receptor and the hydrolysis of inositol lipids in transfected murine fibroblast cells (B82) expressing different receptor densities. The Journal of Pharmacology and Experimental Therapeutics. 251: 90-7. PMID 2795474  1
1989 Palfreyman MG, Dudley MW, Cheng HC, Mir AK, Yamada S, Roeske WR, Obata T, Yamamura HI. Lactamimides: a novel chemical class of calcium antagonists with diltiazem-like properties. Biochemical Pharmacology. 38: 2459-65. PMID 2757648  0.8
1989 Wang JX, Roeske WR, Hawkins KN, Gehlert DR, Yamamura HI. Quantitative autoradiography of M2 muscarinic receptors in the rat brain identified by using a selective radioligand [3H]AF-DX 116. Brain Research. 477: 322-6. PMID 2702492  0.8
1989 Ikeda M, Weber KH, Bechtel WD, Malatynska E, Yamamura HI. Relative efficacies of 1,4-diazepines on GABA-stimulated chloride influx in rat brain vesicles. Life Sciences. 45: 349-58. PMID 2569655 DOI: 10.1016/0024-3205(89)90145-8  1
1989 Hawkins KN, Knapp RJ, Lui GK, Gulya K, Kazmierski W, Wan YP, Pelton JT, Hruby VJ, Yamamura HI. [3H]-[H-D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Pen-Thr-NH2] ([3H]CTOP), a potent and highly selective peptide for mu opioid receptors in rat brain. The Journal of Pharmacology and Experimental Therapeutics. 248: 73-80. PMID 2563293  0.64
1989 Speth RC, Mei L, Yamamura HI. Angiotensin II receptor binding and actions in NG108-15 cells. Peptide Research. 2: 232-9. PMID 2562484  0.44
1989 Ikeda M, Knapp RJ, Malatynska E, Yamamura HI. Amoxapine inhibition of GABA-stimulated chloride conductance: investigations of potential sites of activity. Life Sciences. 45: 1903-10. PMID 2557507 DOI: 10.1016/0024-3205(89)90544-4  1
1989 Mei L, Roeske WR, Yamamura HI. The coupling of muscarinic receptors to hydrolysis of inositol lipids in human neuroblastoma SH-SY5Y cells. Brain Research. 504: 7-14. PMID 2557126 DOI: 10.1016/0006-8993(89)91591-6  1
1989 Vaughn LK, Knapp RJ, Toth G, Wan YP, Hruby VJ, Yamamura HI. A high affinity, highly selective ligand for the delta opioid receptor: [3H]-[D-Pen2, pCl-Phe4, d-Pen5]enkephalin. Life Sciences. 45: 1001-8. PMID 2552241  0.8
1989 Fujiwara Y, Bloom JW, Mantione CR, Yamamura HI. Identification of B2 bradykinin binding sites in the guinea pig nasal turbinate. Peptides. 10: 701-3. PMID 2550915 DOI: 10.1016/0196-9781(89)90163-0  1
1989 Malatynska E, Knapp R, Ikeda M, Yamamura HI. Beta-carboline interactions at the BZ-GABA receptor chloride-ionophore complex in the rat cerebral cortex. Brain Research Bulletin. 22: 845-8. PMID 2548678 DOI: 10.1016/0361-9230(89)90028-2  1
1989 Fujiwara Y, Mantione CR, Vavrek RJ, Stewart JM, Yamamura HI. Characterization of [3H]bradykinin binding sites in guinea-pig central nervous system: possible existence of B2 subtypes. Life Sciences. 44: 1645-53. PMID 2543876  0.56
1989 Knapp RJ, Kazmierski W, Hruby VJ, Yamamura HI. Structural characteristics of two highly selective opioid peptides. Bioessays : News and Reviews in Molecular, Cellular and Developmental Biology. 10: 58-61. PMID 2541696 DOI: 10.1002/bies.950100206  0.8
1989 Landis G, Lui G, Shook JE, Yamamura HI, Burks TF, Hruby VJ. Synthesis of highly mu and delta opioid receptor selective peptides containing a photoaffinity group. Journal of Medicinal Chemistry. 32: 638-43. PMID 2537426  1
1989 Mei L, Lai J, Roeske WR, Fraser CM, Venter JC, Yamamura HI. Pharmacological characterization of the M1 muscarinic receptors expressed in murine fibroblast B82 cells. The Journal of Pharmacology and Experimental Therapeutics. 248: 661-70. PMID 2537406  1
1989 Mei L, Roeske WR, Yamamura HI. Molecular pharmacology of muscarinic receptor heterogeneity. Life Sciences. 45: 1831-51. PMID 2513460 DOI: 10.1016/0024-3205(89)90537-7  1
1988 Mei L, Yamamura HI, Roeske WR. Muscarinic receptor-mediated hydrolysis of phosphatidylinositols in human neuroblastoma (SH-SY5Y) cells is sensitive to pertussis toxin. Brain Research. 447: 360-3. PMID 3390705 DOI: 10.1016/0006-8993(88)91140-7  1
1988 Lai J, Mei L, Roeske WR, Chung FZ, Yamamura HI, Venter JC. The cloned murine M1 muscarinic receptor is associated with the hydrolysis of phosphatidylinositols in transfected murine B82 cells. Life Sciences. 42: 2489-502. PMID 3374268  1
1988 Wang JX, Roeske WR, Wang W, Yamamura HI. Himbacine recognizes a high affinity subtype of M2 muscarinic cholinergic receptors in the rat cerebral cortex. Brain Research. 446: 155-8. PMID 3370478 DOI: 10.1016/0006-8993(88)91306-6  1
1988 Serra M, Mei L, Roeske WR, Lui GK, Watson M, Yamamura HI. The intact human neuroblastoma cell (SH-SY5Y) exhibits high-affinity [3H]pirenzepine binding associated with hydrolysis of phosphatidylinositols. Journal of Neurochemistry. 50: 1513-21. PMID 3361307  0.8
1988 Malatynska E, Serra M, Ikeda M, Biggio G, Yamamura HI. Modulation of GABA-stimulated chloride influx by beta-carbolines in rat brain membrane vesicles. Brain Research. 443: 395-7. PMID 3359279  0.68
1988 Bloom JW, Halonen M, Yamamura HI. Characterization of muscarinic cholinergic receptor subtypes in human peripheral lung. The Journal of Pharmacology and Experimental Therapeutics. 244: 625-32. PMID 3346839  1
1988 Watson M, Roeske WR, Yamamura HI. Decreased muscarinic receptor density in the aged rat brain. Proceedings of the Western Pharmacology Society. 31: 61-5. PMID 3211923  1
1988 Bloom JW, Baumgartener-Folkerts C, Palmer JD, Yamamura HI, Halonen M. A muscarinic receptor subtype modulates vagally stimulated bronchial contraction. Journal of Applied Physiology (Bethesda, Md. : 1985). 65: 2144-50. PMID 3209557 DOI: 10.1152/jappl.1988.65.5.2144  0.56
1988 Wang JX, Yamamura HI, Wang W, Roeske WR. Irreversible inhibition by tyrosine-directed alkylating reagents of muscarinic cholinergic receptors in membranes from rat forebrain and heart. Biochemical Pharmacology. 37: 3787-90. PMID 3178894  0.8
1988 Berzetei IP, Fong A, Yamamura HI, Duckles SP. Characterization of kappa opioid receptors in the rabbit ear artery. European Journal of Pharmacology. 151: 449-55. PMID 2905660 DOI: 10.1016/0014-2999(88)90542-0  1
1988 Kazmierski W, Wire WS, Lui GK, Knapp RJ, Shook JE, Burks TF, Yamamura HI, Hruby VJ. Design and synthesis of somatostatin analogues with topographical properties that lead to highly potent and specific mu opioid receptor antagonists with greatly reduced binding at somatostatin receptors. Journal of Medicinal Chemistry. 31: 2170-7. PMID 2903246  1
1988 Obata T, Morelli M, Concas A, Serra M, Yamamura HI. Modulation of GABA-stimulated chloride influx into membrane vesicles from rat cerebral cortex by benzodiazepines and nonbenzodiazepines. Advances in Biochemical Psychopharmacology. 45: 175-87. PMID 2902742  0.44
1988 Hawkins KN, Knapp RJ, Gehlert DR, Lui GK, Yamamura MS, Roeske LC, Hruby VJ, Yamamura HI. Quantitative autoradiography of [3H]CTOP binding to mu opioid receptors in rat brain. Life Sciences. 42: 2541-51. PMID 2898716  0.8
1988 Fujiwara Y, Mantione CR, Yamamura HI. Identification of B2 bradykinin binding sites in guinea-pig brain. European Journal of Pharmacology. 147: 487-8. PMID 2897921 DOI: 10.1016/0014-2999(88)90187-2  1
1988 Obata T, Yamamura HI. Modulation of GABA-stimulated chloride influx into membrane vesicles from rat cerebral cortex by triazolobenzodiazepines. Life Sciences. 42: 659-65. PMID 2893237 DOI: 10.1016/0024-3205(88)90457-2  1
1988 Obata T, Yamamura HI, Malatynska E, Ikeda M, Laird H, Palmer CJ, Casida JE. Modulation of gamma-aminobutyric acid-stimulated chloride influx by bicycloorthocarboxylates, bicyclophosphorus esters, polychlorocycloalkanes and other cage convulsants. The Journal of Pharmacology and Experimental Therapeutics. 244: 802-6. PMID 2855243  1
1988 Sugg EE, Serra M, Shook JE, Yamamura HI, Burks TF, Korc M, Hruby VJ. Cholecystokinic activity of N alpha-hydroxysulfonyl-[Nle28,31]CCK26-33 analogues modified at the C-terminal residue. International Journal of Peptide and Protein Research. 31: 514-9. PMID 2457563  1
1988 Malatynska E, Knapp RJ, Ikeda M, Yamamura HI. Antidepressants and seizure-interactions at the GABA-receptor chloride-ionophore complex. Life Sciences. 43: 303-7. PMID 2456440 DOI: 10.1016/0024-3205(88)90107-5  1
1987 Bloom JW, Halonen M, Lawrence LJ, Rould E, Seaver NA, Yamamura HI. Characterization of high affinity [3H]pirenzepine and (-)-[3H] quinuclidinyl benzilate binding to muscarinic cholinergic receptors in rabbit peripheral lung. The Journal of Pharmacology and Experimental Therapeutics. 240: 51-8. PMID 3806397  0.56
1987 Yamada S, Gehlert DR, Hawkins KN, Nakayama K, Roeske WR, Yamamura HI. Autoradiographic localization of nicotinic receptor binding in rat brain using [3H]methylcarbamylcholine, a novel radioligand. Life Sciences. 41: 2851-61. PMID 3695812  0.8
1987 Smith TL, Yamamura HI. Competitive inhibition of phosphoinositide hydrolysis by the muscarinic receptor antagonist AF-DX 116 is of low affinity in mouse cerebral cortex. Brain Research. 420: 362-4. PMID 3676767 DOI: 10.1016/0006-8993(87)91257-1  1
1987 Wang JX, Yamamura HI, Wang W, Roeske WR. Differential regulation of M2 muscarinic receptors by guanine nucleotides in rat cerebral cortical and cardiac membranes. European Journal of Pharmacology. 139: 357-8. PMID 3666011  0.8
1987 Wang JX, Roeske WR, Gulya K, Wang W, Yamamura HI. [3H]AF-DX 116 labels subsets of muscarinic cholinergic receptors in rat brain and heart. Life Sciences. 41: 1751-60. PMID 3657382 DOI: 10.1016/0024-3205(87)90604-7  1
1987 Mei L, Wang JX, Roeske WR, Yamamura HI. Thermodynamic analyses of pirenzepine binding to membrane-bound and solubilized muscarinic receptors from rat forebrain and heart. The Journal of Pharmacology and Experimental Therapeutics. 242: 991-1000. PMID 3656121  1
1987 Lemcke PK, Sugg E, Malarchik M, Lui G, Serra M, Yamamura HI, Hruby VJ, Shook JE, Burks TF. N-terminal cyclization of a nonsulfated CCK analogue exhibits opioid antagonist activity in vitro. Proceedings of the Western Pharmacology Society. 30: 223-6. PMID 3628282  1
1987 Obata T, Yamamura HI. Inhibition of GABA-stimulated chloride influx by the convulsant benzodiazepines Ro 5-3663 and Ro 5-4864 into membrane vesicles from rat cerebral cortex. European Journal of Pharmacology. 136: 447-8. PMID 3609129 DOI: 10.1016/0014-2999(87)90324-4  1
1987 Bloom JW, Halonen M, Seaver NA, Yamamura HI. Heterogeneity of the M1 muscarinic receptor subtype between peripheral lung and cerebral cortex demonstrated by the selective antagonist AF-DX 116. Life Sciences. 41: 491-6. PMID 3600190 DOI: 10.1016/0024-3205(87)90226-8  0.56
1987 Duckles SP, Yamamura HI, Lee V. AF-DX 116 discriminates between muscarinic M2 receptors of the heart and vasculature. Life Sciences. 40: 1507-11. PMID 3561162 DOI: 10.1016/0024-3205(87)90383-3  1
1987 Bloom JW, Yamamura HI, Baumgartener C, Halonen M. A muscarinic receptor with high affinity for pirenzepine mediates vagally induced bronchoconstriction. European Journal of Pharmacology. 133: 21-7. PMID 3556389 DOI: 10.1016/0014-2999(87)90201-9  1
1987 Wang JX, Mei L, Yamamura HI, Roeske WR. Solubilization with digitonin alters the kinetics of pirenzepine binding to muscarinic receptors from rat forebrain and heart. The Journal of Pharmacology and Experimental Therapeutics. 242: 981-90. PMID 3116203  0.8
1987 Earle ME, Concas A, Wamsley JK, Yamamura HI. Temperature dependence and GABA modulation of [3H]triazolam binding in the rat brain. Life Sciences. 41: 397-403. PMID 3037225 DOI: 10.1016/0024-3205(87)90214-1  1
1987 Hawkins KN, Morelli M, Gulya K, Chang KJ, Yamamura HI. Autoradiographic localization of [3H] [MePhe3,D-Pro4]morphiceptin ([3H]PL017) to mu opioid receptors in rat brain. European Journal of Pharmacology. 133: 351-2. PMID 3030778 DOI: 10.1016/0014-2999(87)90033-1  1
1987 Nelson DL, Monroe PJ, Lambert G, Yamamura HI. [3H]spiroxatrine labels a serotonin1A-like site in the rat hippocampus. Life Sciences. 41: 1567-76. PMID 2957559 DOI: 10.1016/0024-3205(87)90723-5  1
1987 Berzetei IP, Yamamura HI, Duckles SP. Characterization of rabbit ear artery opioid receptors using a delta-selective agonist and antagonist. European Journal of Pharmacology. 139: 61-6. PMID 2820755 DOI: 10.1016/0014-2999(87)90497-3  1
1987 Fox DA, Ayres EA, Wire WS, Lui G, Yamamura HI, Burks TF. Kentsin: tetrapeptide from hamster embryos produces naloxone-sensitive effects without binding to opioid receptors. Peptides. 8: 613-8. PMID 2819832 DOI: 10.1016/0196-9781(87)90034-9  1
1986 Brinton RE, Gehlert DR, Wamsley JK, Wan YP, Yamamura HI. Vasopressin metabolite, AVP4-9, binding sites in brain: distribution distinct from that of parent peptide. Life Sciences. 38: 443-52. PMID 3945171  0.6
1986 Hynes MR, Banner W, Yamamura HI, Duckles SP. Characterization of muscarinic receptors of the rabbit ear artery smooth muscle and endothelium. The Journal of Pharmacology and Experimental Therapeutics. 238: 100-5. PMID 3755169  1
1986 Watson M, Roeske WR, Yamamura HI. [3H]pirenzepine and (-)-[3H]quinuclidinyl benzilate binding to rat cerebral cortical and cardiac muscarinic cholinergic sites. II. Characterization and regulation of antagonist binding to putative muscarinic subtypes. The Journal of Pharmacology and Experimental Therapeutics. 237: 419-27. PMID 3754581  1
1986 Watson M, Yamamura HI, Roeske WR. [3H]pirenzepine and (-)-[3H]quinuclidinyl benzilate binding to rat cerebral cortical and cardiac muscarinic cholinergic sites. I. Characterization and regulation of agonist binding to putative muscarinic subtypes. The Journal of Pharmacology and Experimental Therapeutics. 237: 411-8. PMID 3754580  1
1986 Brinton RE, Gruener R, Deshmukh P, Yamamura HI. In vitro inhibition of vasopressin release in brain by behaviorally relevant ethanol concentrations. Neuroscience Letters. 67: 213-7. PMID 3725210 DOI: 10.1016/0304-3940(86)90400-3  1
1986 Clark JA, Itzhak Y, Hruby VJ, Yamamura HI, Pasternak GW. [D-Pen2,D-Pen5]enkephalin (DPDPE): a delta-selective enkephalin with low affinity for mu 1 opiate binding sites. European Journal of Pharmacology. 128: 303-4. PMID 3025000 DOI: 10.1016/0014-2999(86)90784-3  1
1986 Serra M, Smith TL, Yamamura HI. Phorbol esters alter muscarinic receptor binding and inhibit polyphosphoinositide breakdown in human neuroblastoma (SH-SY5Y) cells. Biochemical and Biophysical Research Communications. 140: 160-6. PMID 3022714 DOI: 10.1016/0006-291X(86)91071-5  1
1986 Smith TL, Yamamura HI, Lee L. Effect of ethanol on receptor-stimulated phosphatidic acid and polyphosphoinositide metabolism in mouse brain. Life Sciences. 39: 1675-84. PMID 3022092 DOI: 10.1016/0024-3205(86)90165-7  1
1986 Gee KW, Lawrence LJ, Yamamura HI. Modulation of the chloride ionophore by benzodiazepine receptor ligands: influence of gamma-aminobutyric acid and ligand efficacy. Molecular Pharmacology. 30: 218-25. PMID 3018479  1
1986 Concas A, Gehlert DR, Wamsley JK, Yamamura HI. Effect of benzodiazepine binding site ligands on [35S] t-butylbicyclophosphorothionate ([35S]TBPS) binding to rat brain: an autoradiographic study. Advances in Biochemical Psychopharmacology. 41: 227-38. PMID 3017072  0.6
1986 Gulya K, Gehlert DR, Wamsley JK, Mosberg H, Hruby VJ, Yamamura HI. Light microscopic autoradiographic localization of delta opioid receptors in the rat brain using a highly selective bis-penicillamine cyclic enkephalin analog. The Journal of Pharmacology and Experimental Therapeutics. 238: 720-6. PMID 3016247  1
1986 Yamada S, Yamamura HI, Roeske WR. Effects of chemical sympathectomy with 6-hydroxydopamine on alpha- and beta-adrenoceptors and muscarinic cholinoceptors in rat kidney. European Journal of Pharmacology. 121: 345-53. PMID 3009209 DOI: 10.1016/0014-2999(86)90255-4  1
1986 Akiyama K, Vickroy TW, Watson M, Roeske WR, Reisine TD, Smith TL, Yamamura HI. Muscarinic cholinergic ligand binding to intact mouse pituitary tumor cells (AtT-20/D16-16) coupling with two biochemical effectors: adenylate cyclase and phosphatidylinositol turnover. The Journal of Pharmacology and Experimental Therapeutics. 236: 653-61. PMID 3005550  0.8
1986 Gulya K, Lui GK, Pelton JT, Kazmierski W, Hruby VJ, Yamamura HI. H-D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Pen-Thr-NH2: a potent and selective antagonist opioid receptors. Nida Research Monograph. 75: 209-12. PMID 2893264  1
1986 Pelton JT, Kazmierski W, Gulya K, Yamamura HI, Hruby VJ. Design and synthesis of conformationally constrained somatostatin analogues with high potency and specificity for mu opioid receptors. Journal of Medicinal Chemistry. 29: 2370-5. PMID 2878079 DOI: 10.1021/JM00161A037  1
1986 Gulya K, Pelton JT, Hruby VJ, Yamamura HI. Cyclic somatostatin octapeptide analogues with high affinity and selectivity toward mu opioid receptors. Life Sciences. 38: 2221-9. PMID 2872570 DOI: 10.1016/0024-3205(86)90574-6  1
1986 Obata T, Yamamura HI. The effect of benzodiazepines and beta-carbolines on GABA-stimulated chloride influx by membrane vesicles from the rat cerebral cortex. Biochemical and Biophysical Research Communications. 141: 1-6. PMID 2432889 DOI: 10.1016/S0006-291X(86)80325-4  1
1986 Sugg EE, Shook JE, Serra M, Korc M, Yamamura HI, Burks TF, Hruby VJ. Synthesis and biological evaluation of N alpha-hydroxysulfonyl-[Nle28,31]-CCK26-33. Life Sciences. 39: 1623-9. PMID 2430160 DOI: 10.1016/0024-3205(86)90158-X  1
1985 Gehlert DR, Dawson TM, Yamamura HI, Wamsley JK. Quantitative autoradiography of [3H]forskolin binding sites in the rat brain. Brain Research. 361: 351-60. PMID 4084804  0.6
1985 Brinton RE, Wamsley JK, Gehlert D, Wan YP, Yamamura HI. Vasopressin metabolite peptide (AVP-(4-9)) binding sites in rat kidney: distribution distinct from vasopressin binding sites. European Journal of Pharmacology. 108: 321-2. PMID 3987807  0.6
1985 Vickroy TW, Roeske WR, Gehlert DR, Wamsley JK, Yamamura HI. Quantitative light microscopic autoradiography of [3H]hemicholinium-3 binding sites in the rat central nervous system: a novel biochemical marker for mapping the distribution of cholinergic nerve terminals. Brain Research. 329: 368-73. PMID 3978459 DOI: 10.1016/0006-8993(85)90553-0  0.8
1985 Dawson TM, Gehlert DR, Yamamura HI, Barnett A, Wamsley JK. D-1 dopamine receptors in the rat brain: autoradiographic localization using [3H]SCH 23390. European Journal of Pharmacology. 108: 323-5. PMID 3886408  0.6
1985 Watson M, Vickroy TW, Roeske WR, Yamamura HI. Functional and biochemical basis for multiple muscarinic acetylcholine receptors. Progress in Neuro-Psychopharmacology & Biological Psychiatry. 9: 569-74. PMID 3841401 DOI: 10.1016/0278-5846(85)90018-1  1
1985 Evans RA, Watson M, Yamamura HI, Roeske WR. Differential ontogeny of putative M1 and M2 muscarinic receptor binding sites in the murine cerebral cortex and heart. The Journal of Pharmacology and Experimental Therapeutics. 235: 612-8. PMID 3841156  0.8
1985 Vickroy TW, Watson M, Leventer SM, Roeske WR, Hanin I, Yamamura HI. Regional differences in ethylcholine mustard aziridinium ion (AF64A)-induced deficits in presynaptic cholinergic markers for the rat central nervous system. The Journal of Pharmacology and Experimental Therapeutics. 235: 577-82. PMID 3841155  0.8
1985 Watson M, Vickroy TW, Fibiger HC, Roeske WR, Yamamura HI. Effects of bilateral ibotenate-induced lesions of the nucleus basalis magnocellularis upon selective cholinergic biochemical markers in the rat anterior cerebral cortex. Brain Research. 346: 387-91. PMID 3840399 DOI: 10.1016/0006-8993(85)90876-5  1
1985 Smith TL, Yamamura HI. Carbachol stimulation of phosphatidic acid synthesis: competitive inhibition by pirenzepine in synaptosomes from rat cerebral cortex. Biochemical and Biophysical Research Communications. 130: 282-5. PMID 3839668 DOI: 10.1016/0006-291X(85)90414-0  1
1985 Yamamura HI, Vickroy TW, Gehlert DR, Wamsley JK, Roeske WR. Autoradiographic localization of muscarinic agonist binding sites in the rat central nervous system with (+)-cis-[3H]methyldioxolane. Brain Research. 325: 340-4. PMID 3838491 DOI: 10.1016/0006-8993(85)90336-1  0.8
1985 Lee HR, Jaros JA, Roeske WR, Wiech NL, Ursillo R, Yamamura HI. Potent enhancement of [3H]nitrendipine binding in rat cerebral cortical and cardiac homogenates: a putative mechanism for the action of MDL 12,330A. The Journal of Pharmacology and Experimental Therapeutics. 233: 611-6. PMID 3159884  0.8
1985 Yamamura HI, Gehlert DR, Gee KW, Wamsley JK, Horst WD, Roeske WR. Specific high-affinity [3H]Ro5-4864 Ro5-4864 benzodiazepine binding sites in the brain and periphery. Progress in Clinical and Biological Research. 192: 187-96. PMID 3001751  1
1985 Lawrence LJ, Palmer CJ, Gee KW, Wang X, Yamamura HI, Casida JE. t-[3H]butylbicycloorthobenzoate: new radioligand probe for the gamma-aminobutyric acid-regulated chloride ionophore. Journal of Neurochemistry. 45: 798-804. PMID 2993514 DOI: 10.1111/j.1471-4159.1985.tb04063.x  1
1985 Gulya K, Gehlert DR, Wamsley JK, Mosberg HI, Hruby VJ, Duckles SP, Yamamura HI. Autoradiographic localization of delta opioid receptors in the rat brain using a highly selective bis-penicillamine cyclic enkephalin analog. European Journal of Pharmacology. 111: 285-6. PMID 2990955 DOI: 10.1016/0014-2999(85)90770-8  1
1985 Gehlert DR, Yamamura HI, Wamsley JK. gamma-Aminobutyric acidB receptors in the rat brain: quantitative autoradiographic localization using [3H](-)-baclofen. Neuroscience Letters. 56: 183-8. PMID 2989740 DOI: 10.1016/0304-3940(85)90126-0  1
1985 Roeske WR, Lee HR, Yamamura HI, Schoemaker H. Identification of calcium-channel receptors in intact animals. Advances in Myocardiology. 6: 71-82. PMID 2986265  1
1985 Akiyama K, Gee KW, Mosberg HI, Hruby VJ, Yamamura HI. Characterization of [3H][2-D-penicillamine, 5-D-penicillamine]-enkephalin binding to delta opiate receptors in the rat brain and neuroblastoma--glioma hybrid cell line (NG 108-15). Proceedings of the National Academy of Sciences of the United States of America. 82: 2543-7. PMID 2986120  0.56
1985 Gehlert DR, Yamamura HI, Wamsley JK. Autoradiographic localization of "peripheral-type" benzodiazepine binding sites in the rat brain, heart and kidney. Naunyn-Schmiedeberg's Archives of Pharmacology. 328: 454-60. PMID 2986017 DOI: 10.1007/BF00692915  1
1985 Richter JA, Yamamura HI. Effects of pentobarbital on t-[35S]butylbicyclophosphorothionate and [3H]flunitrazepam binding to membrane-bound and solubilized preparations from rat forebrain. The Journal of Pharmacology and Experimental Therapeutics. 233: 125-33. PMID 2984410  1
1985 Wamsley JK, Golden JS, Yamamura HI, Barnett A. Quazepam, a sedative-hypnotic selective for the benzodiazepine type 1 receptor: autoradiographic localization in rat and human brain. Clinical Neuropharmacology. 8: S26-40. PMID 2874881  1
1985 Wamsley JK, Golden JS, Yamamura HI, Barnett A. Autoradiographic demonstration of the selectivity of two 1-N-trifluoroethyl benzodiazepines for the BZD-1 receptors in the rat brain. Pharmacology, Biochemistry, and Behavior. 23: 973-8. PMID 2867566 DOI: 10.1016/0091-3057(85)90103-0  1
1985 Pelton JT, Gulya K, Hruby VJ, Duckles S, Yamamura HI. Somatostatin analogs with affinity for opiate receptors in rat brain binding assay. Peptides. 6: 159-63. PMID 2864680 DOI: 10.1016/0196-9781(85)90026-9  1
1985 Gulya K, Wamsley JK, Gehlert D, Pelton JT, Duckles SP, Hruby VJ, Yamamura HI. Light microscopic autoradiographic localization of somatostatin receptors in the rat brain. The Journal of Pharmacology and Experimental Therapeutics. 235: 254-8. PMID 2864434  1
1985 Pelton JT, Gulya K, Hruby VJ, Duckles SP, Yamamura HI. Conformationally restricted analogs of somatostatin with high mu-opiate receptor specificity. Proceedings of the National Academy of Sciences of the United States of America. 82: 236-9. PMID 2857488 DOI: 10.1073/pnas.82.1.236  1
1985 Darman PS, Landis GC, Smits JR, Hirning LD, Gulya K, Yamamura HI, Burks TF, Hruby VJ. Conformationally restricted cyclic analogues of substance P: insight into the receptor binding process. Biochemical and Biophysical Research Communications. 127: 656-62. PMID 2579658 DOI: 10.1016/S0006-291X(85)80211-4  1
1985 Lee HR, Watson M, Yamamura HI, Roeske WR. Decreased [3H]nitrendipine binding in the brainstem of deoxycorticosterone-NaCl hypertensive rats. Life Sciences. 37: 971-7. PMID 2412086 DOI: 10.1016/0024-3205(85)90534-X  1
1985 Lawrence LJ, Gee KW, Yamamura HI. Interactions of pyrethroid insecticides with chloride ionophore-associated binding sites. Neurotoxicology. 6: 87-98. PMID 2410833  1
1985 Tivol E, Halonen M, Yamamura HI. Characterization of muscarinic cholinergic receptor sites in the rabbit peripheral lung using radiolabeled pirenzepine Federation Proceedings. 44.  1
1985 Yamamura HI, Akiyama K, Gee KW. Tritium (D-pen2,D-pen5)enkephalin, a highly selective radioligand for the identification and characterization of the delta opioid receptor Federation Proceedings. 44.  1
1985 Watson M, Lee HR, Yamamura HI, Roeske WR. [3H]Pirenzepine and [3H](-)quinuclidinylbenzilate binding to putative M1 And M2 muscarinic sites in deoxycorticosterone-NACL hypertensive rats Federation Proceedings. 44.  1
1985 Gee KW, Lawrence LJ, Yamamura HI. Differential modulation of 35S-t-butylbicyclophosphorothionate (35S-TBPS) binding in rat brain by benzodiazepine (BZ) receptor ligands: Effect of GABA and ligand efficacy Federation Proceedings. 44.  1
1984 Boles RG, Yamamura HI, Schoemaker H, Roeske WR. Temperature-dependent modulation of [3H]nitrendipine binding by the calcium channel antagonists verapamil and diltiazem in rat brain synaptosomes. The Journal of Pharmacology and Experimental Therapeutics. 229: 333-9. PMID 6716261  1
1984 Wilkes BC, Hruby VJ, Yamamura HI, Akiyama K, Castrucci AM, Hadley ME, Andrews JR, Wan YP. Synthesis of tritium labeled Ac-[Nle4, D-Phe7]-alpha-MSH4-11-NH2: a superpotent melanotropin with prolonged biological activity. Life Sciences. 34: 977-84. PMID 6608041  0.8
1984 Yamamura HI, Watson M, Wamsley JK, Johnson PC, Roeske WR. Light microscopic autoradiographic localization of [3H]pirenzepine and [3H](-)quinuclidinyl benzilate binding in human stellate ganglia. Life Sciences. 35: 753-7. PMID 6547993  0.8
1984 Wamsley JK, Gehlert DR, Roeske WR, Yamamura HI. Muscarinic antagonist binding site heterogeneity as evidenced by autoradiography after direct labeling with [3H]-QNB and [3H]-pirenzepine. Life Sciences. 34: 1395-402. PMID 6546776  0.8
1984 Akiyama K, Watson M, Roeske WR, Yamamura HI. High-affinity [3H]pirenzepine binding to putative M1 muscarinic sites in the neuroblastoma x glioma hybrid cell line (NG 108-15). Biochemical and Biophysical Research Communications. 119: 289-97. PMID 6546688  0.8
1984 Watson M, Roeske WR, Johnson PC, Yamamura HI. [3H]Pirenzepine identifies putative M1 muscarinic receptors in human stellate ganglia. Brain Research. 290: 179-82. PMID 6546354 DOI: 10.1016/0006-8993(84)90751-0  0.8
1984 Gehlert DR, Dawson TM, Yamamura HI, Wamsley JK. Localization of [3H]forskolin binding sites in the rat brain using quantitative autoradiography. European Journal of Pharmacology. 106: 223-5. PMID 6543336  0.6
1984 Akiyama K, Yamamura HI, Wilkes BC, Cody WL, Hruby VJ, Castrucci AM, Hadley ME. Relative stability of alpha-melanotropin and related analogues to rat brain homogenates. Peptides. 5: 1191-5. PMID 6531272  0.8
1984 Vickroy TW, Roeske WR, Yamamura HI. Sodium-dependent high-affinity binding of [3H]hemicholinium-3 in the rat brain: a potentially selective marker for presynaptic cholinergic sites. Life Sciences. 35: 2335-43. PMID 6503616  0.8
1984 Vickroy TW, Fibiger HC, Roeske WR, Yamamura HI. Reduced density of sodium-dependent [3H]hemicholinium-3 binding sites in the anterior cerebral cortex of rats following chemical destruction of the nucleus basalis magnocellularis. European Journal of Pharmacology. 102: 369-70. PMID 6479222 DOI: 10.1016/0014-2999(84)90271-1  1
1984 Vickroy TW, Watson M, Yamamura HI, Roeske WR. Agonist binding to multiple muscarinic receptors. Federation Proceedings. 43: 2785-90. PMID 6383872  1
1984 Ehlert FJ, Yamamura HI. A comparison of the effects of cinnarizine and related compounds on [3H]nitrendipine binding in the brain, heart and ileum. Life Sciences. 34: 2347-55. PMID 6328164 DOI: 10.1016/0024-3205(84)90421-1  1
1984 Buck SH, Maurin Y, Burks TF, Yamamura HI. High-affinity 3H-substance P binding to longitudinal muscle membranes of the guinea pig small intestine. Life Sciences. 34: 497-507. PMID 6319946 DOI: 10.1016/0024-3205(84)90506-X  1
1984 Vickroy TW, Watson M, Yamamura HI, Roeske WR. Differential regulation of putative M1/M2 muscarinic receptors: implications for different receptor-effector coupling mechanisms. Advances in Experimental Medicine and Biology. 175: 99-114. PMID 6208760  1
1984 Gehlert DR, Yamamura HI, Wamsley JK. Use of autoradiographic techniques for the localization of neurotransmitter receptors in brain and periphery: recent applications. Advances in Experimental Medicine and Biology. 175: 255-70. PMID 6208759  0.6
1984 Maurin Y, Buck SH, Wamsley JK, Burks TF, Yamamura HI. Light microscopic autoradiographic localization of [3H] substance P binding sites in rat thoracic spinal cord. Life Sciences. 34: 1713-6. PMID 6203003  0.6
1984 Vickroy TW, Roeske WR, Yamamura HI. Pharmacological differences between the high-affinity muscarinic agonist binding states of the rat heart and cerebral cortex labeled with (+)-[3H]cismethyldioxolane. The Journal of Pharmacology and Experimental Therapeutics. 229: 747-55. PMID 6202869  1
1984 Mimaki T, Yabuuchi H, Laird H, Yamamura HI. Effects of seizures and antiepileptic drugs on benzodiazepine receptors in rat brain. Pediatric Pharmacology (New York, N.Y.). 4: 205-11. PMID 6097863  1
1984 Brinton RE, Gee KW, Wamsley JK, Davis TP, Yamamura HI. Regional distribution of putative vasopressin receptors in rat brain and pituitary by quantitative autoradiography. Proceedings of the National Academy of Sciences of the United States of America. 81: 7248-52. PMID 6095279 DOI: 10.1073/pnas.81.22.7248  1
1984 Lawrence LJ, Gee KW, Yamamura HI. Benzodiazepine anticonvulsant action: gamma-aminobutyric acid-dependent modulation of the chloride ionophore. Biochemical and Biophysical Research Communications. 123: 1130-7. PMID 6091648 DOI: 10.1016/S0006-291X(84)80250-8  1
1984 Gee KW, Yamamura SH, Roeske WR, Yamamura HI. Benzodiazepine receptor heterogeneity: possible molecular basis and functional significance. Federation Proceedings. 43: 2767-72. PMID 6090222  1
1984 Brinton RE, Wamsley JK, Gee KW, Wan YP, Yamamura HI. [3H]oxytocin binding sites in the rat brain demonstrated by quantitative light microscopic autoradiography. European Journal of Pharmacology. 102: 365-7. PMID 6090165 DOI: 10.1016/0014-2999(84)90270-X  1
1984 Lee HR, Roeske WR, Yamamura HI. High affinity specific [3H](+)PN 200-110 binding to dihydropyridine receptors associated with calcium channels in rat cerebral cortex and heart. Life Sciences. 35: 721-32. PMID 6088927 DOI: 10.1016/0024-3205(84)90340-0  1
1984 Richter JA, Yamamura HI. Differential effects of pentobarbital on solubilized picrotoxin/barbiturate and benzodiazepine binding sites Federation Proceedings. 43.  1
1984 Fleisher JH, Pinnas JL, Yamamura HI. In vitro studies of bronchodilator drugs Federation Proceedings. 43.  1
1983 Brinton RE, Deshmukh PP, Chen A, Davis TP, Hsiao S, Yamamura HI. A non-equilibrium 24-hour vasopressin radioimmunoassay: development and basal levels in the rat brain. Brain Research. 266: 344-7. PMID 6871669 DOI: 10.1016/0006-8993(83)90667-4  1
1983 Schoemaker H, Lee HR, Roeske WR, Yamamura HI. In vivo identification of calcium antagonist binding sites using [3H]nitrendipine European Journal of Pharmacology. 88: 275-276. PMID 6852115 DOI: 10.1016/0014-2999(83)90019-5  1
1983 Yamamura HI, Watson M, Roeske WR. [3H]pirenzepine specifically labels a high affinity muscarinic receptor in the rat cerebral cortex Advances in Biochemical Psychopharmacology. 37: 331-336. PMID 6688917  1
1983 Yamamura HI, Wamsley JK, Deshmukh P, Roeske WR. Differential light microscopic autoradiographic localization of muscarinic cholinergic receptors in the brainstem and spinal cord of the rat using [3H]pirenzepine European Journal of Pharmacology. 91: 147-149. PMID 6688587 DOI: 10.1016/0014-2999(83)90379-5  1
1983 Watson M, Yamamura HI, Roeske WR. A unique regulatory profile and regional distribution of [3H]pirenzepine binding in the rat provide evidence for distinct M1 and M2 muscarinic receptor subtypes Life Sciences. 32: 3001-3011. PMID 6688111 DOI: 10.1016/0024-3205(83)90652-5  1
1983 Lee HR, Roeske WR, Yamamura HI. The measurement of free nitrendipine in human serum by an equilibrium dialysis - radioreceptor assay. Life Sciences. 33: 1821-9. PMID 6645780 DOI: 10.1016/0024-3205(83)90690-2  1
1983 Erman RD, Yamamura HI, Roeske WR. The ontogeny of specific binding sites for the calcium channel antagonist, nitrendipine, in mouse heart and brain. Brain Research. 278: 327-31. PMID 6640324  0.8
1983 Vickroy TW, Yamamura HI, Roeske WR. Differential regulation of high-affinity agonist binding to muscarinic sites in the rat heart, cerebellum, and cerebral cortex. Biochemical and Biophysical Research Communications. 116: 284-90. PMID 6639662  0.8
1983 Mosberg HI, Hurst R, Hruby VJ, Gee K, Akiyama K, Yamamura HI, Galligan JJ, Burks TF. Cyclic penicillamine containing enkephalin analogs display profound delta receptor selectivities. Life Sciences. 33: 447-50. PMID 6319901 DOI: 10.1016/0024-3205(83)90538-6  1
1983 Gehlert DR, Yamamura HI, Wamsley JK. Autoradiographic localization of 'peripheral' benzodiazepine binding sites in the rat brain and kidney using [3H]RO5-4864. European Journal of Pharmacology. 95: 329-30. PMID 6317419 DOI: 10.1016/0014-2999(83)90658-1  1
1983 Wamsley JK, Gee KW, Yamamura HI. Comparison of the distribution of convulsant/barbiturate and benzodiazepine receptors using light microscopic autoradiography. Life Sciences. 33: 2321-9. PMID 6316061 DOI: 10.1016/0024-3205(83)90266-7  1
1983 Smith TL, Vickers AE, Brendel K, Yamamura HI. Influence of chronic ethanol treatment on alpha1-adrenergic and vasopressin receptor-stimulated phosphatidylinositol synthesis in isolated rat hepatocytes. Biochemical Pharmacology. 32: 3059-62. PMID 6315016 DOI: 10.1016/0006-2952(83)90249-6  1
1983 Gee KW, Yamamura HI. Photoaffinity labeling of benzodiazepine receptors in rat brain with flunitrazepam alters the affinity of benzodiazepine receptor agonist but not antagonist binding. Journal of Neurochemistry. 41: 1407-13. PMID 6311986 DOI: 10.1111/j.1471-4159.1983.tb00839.x  1
1983 Ehlert FJ, Roeske WR, Gee KW, Yamamura HI. An allosteric model for benzodiazepine receptor function Biochemical Pharmacology. 32: 2375-2383. PMID 6311215 DOI: 10.1016/0006-2952(83)90679-2  1
1983 Davis TP, Schoemaker H, Culling AJ, Yamamura HI. Isolation and characterization of in vitro central beta-endorphin metabolism in schizophrenia. Proceedings of the Western Pharmacology Society. 26: 89-94. PMID 6310636  1
1983 Chen AD, Davis TP, Yamamura HI. Demonstration and partial characterization of a bovine cerebral cortical factor which interacts competitively at the benzodiazepine receptor. Proceedings of the Western Pharmacology Society. 26: 225-30. PMID 6310627  1
1983 Schoemaker H, Boles RG, Roeske WR, Yamamura HI. Allosteric modulation by diltiazem and verapamil of [3H]nitrendipine binding to calcium channel sites in rat brain Proceedings of the Western Pharmacology Society. 219-224. PMID 6310626  1
1983 Mosberg HI, Hurst R, Hruby VJ, Gee K, Yamamura HI, Galligan JJ, Burks TF. Bis-penicillamine enkephalins possess highly improved specificity toward delta opioid receptors. Proceedings of the National Academy of Sciences of the United States of America. 80: 5871-4. PMID 6310598  1
1983 Gee KW, Wamsley JK, Yamamura HI. Light microscopic autoradiographic identification of picrotoxin/barbiturate binding sites in rat brain with [35S]t-butyl-bicyclophosphathionate European Journal of Pharmacology. 89: 323-324. PMID 6307715 DOI: 10.1016/0014-2999(83)90516-2  1
1983 Ehlert FJ, Roeske WR, Yamamura SH, Yamamura HI. The benzodiazepine receptor: complex binding properties and the influence of GABA Advances in Biochemical Psychopharmacology. 36: 209-220. PMID 6305148  1
1983 Mosberg HI, Hurst R, Hruby VJ, Galligan JJ, Burks TF, Gee K, Yamamura HI. Conformationally constrained cyclic enkephalin analogs with pronounced delta opioid receptor agonist selectivity. Life Sciences. 32: 2565-9. PMID 6304440 DOI: 10.1016/0024-3205(83)90239-4  1
1983 Gee KW, Brinton RE, Yamamura HI. PK 8165 and PK 9084, two quinoline derivatives with anxiolytic properties, antagonize the anticonvulsant effects of diazepam Brain Research. 264: 168-172. PMID 6303496 DOI: 10.1016/0006-8993(83)91138-1  1
1983 Yamamura HI, Gee KW, Brinton RE, Davis TP, Hadley M, Wamsley JK. Light microscopic autoradiographic visualization of [3H]-arginine vasopressin binding sites in rat brain. Life Sciences. 32: 1919-24. PMID 6300592 DOI: 10.1016/0024-3205(83)90072-3  1
1983 Gee KW, Ehlert FJ, Yamamura HI. Differential effect of γ-aminobutyric acid on benzodiazepine receptor subtypes labeled by [3H]propyl β-carboline-3-carboxylate in rat brain Journal of Pharmacology and Experimental Therapeutics. 225: 132-137. PMID 6300371  1
1983 Gee KW, Brinton RE, Yamamura HI. CL 218872 antagonism of diazepam induced loss of righting reflex: Evidence for partial agonistic activity at the benzodiazepine receptor Life Sciences. 32: 1037-1040. PMID 6298552 DOI: 10.1016/0024-3205(83)90936-0  1
1983 Schoemaker H, Smith TL, Yamamura HI. Effect of chronic ethanol consumption on central and peripheral type benzodiazepine binding sites in the mouse brain Brain Research. 258: 347-350. PMID 6297665 DOI: 10.1016/0006-8993(83)91164-2  1
1983 Hynes MR, Culling AJ, Galligan JJ, Burks TF, Schoemaker H, Yamamura HI, Davis TP. Processing of beta-endorphin in the dog intestine: regional specificity. Proceedings of the Western Pharmacology Society. 26: 95-9. PMID 6193534  0.48
1983 Gee KW, Yamamura HI. Selective anxiolytics: are the actions related to partial "agonist" activity or a preferential affinity for benzodiazepine receptor subtypes? Advances in Biochemical Psychopharmacology. 38: 1-9. PMID 6142598  1
1983 Schoemaker H, Boles RG, Horst WD, Yamamura HI. Specific high-affinity binding sites for [3H]Ro 5-4864 in rat brain and kidney Journal of Pharmacology and Experimental Therapeutics. 225: 61-69. PMID 6132001  1
1983 Brinton RE, Gee KW, Yamamura HI. CL 218872, PK 8165 and PK 9084: Selective anxiolytics that may act as partial agonist at the benzodiazepine receptor Federation Proceedings. 42.  1
1982 Schoemaker H, Chen A, Davis TP, Yamamura HI. A study of the metabolism of des-tyrosine-gamma-endorphin using an improved HPLC system. Psychopharmacology Bulletin. 18: 144-8. PMID 7156277  1
1982 Deshmukh PP, Nelson DL, Yamamura HI. Autoradiographic localization of 5-HT1 receptor subtypes in rat brain Proceedings of the Western Pharmacology Society. 83-86. PMID 7122545  1
1982 Ehlert FJ, Roeske WR, Itoga E, Yamamura HI. The binding of [3H]nitrendipine to receptors for calcium channel antagonists in the heart, cerebral cortex, and ileum of rats Life Sciences. 30: 2191-2202. PMID 7109844 DOI: 10.1016/0024-3205(82)90293-4  1
1982 Ehlert FJ, Itoga E, Roeske WR, Yamamura HI. The interaction of [3H]nitrendipine with receptors for calcium antagonists in the cerebral cortex and heart of rats Biochemical and Biophysical Research Communications. 104: 937-943. PMID 7073736 DOI: 10.1016/0006-291X(82)91339-0  1
1982 Barritt D, Yamamura HI, Roeske WR. Muscarinic receptor binding in the mouse heart: the selective modulatory effect of fluoride ion on agonist binding Life Sciences. 30: 875-877. PMID 7070200 DOI: 10.1016/0024-3205(82)90602-6  1
1982 Watson M, Roeske WR, Yamamura HI. [3H] pirenzepine selectively identifies a high affinity population of muscarinic cholinergic receptors in the rat cerebral cortex Life Sciences. 31: 2019-2023. PMID 6897437 DOI: 10.1016/0024-3205(82)90041-8  1
1982 Gee KW, Yamamura HI. Regional heterogeneity of benzodiazepine receptors at 37°C: An in vitro study in various regions of the rat brain Life Sciences. 31: 1939-1945. PMID 6294423 DOI: 10.1016/0024-3205(82)90032-7  1
1982 Yamamura HI, Schoemaker H, Boles RG, Roeske WR. Diltiazem enhancement of [3H]nitrendipine binding to calcium channel associated drug receptor sites in rat brain synaptosomes Biochemical and Biophysical Research Communications. 108: 640-646. PMID 6293498 DOI: 10.1016/0006-291X(82)90877-4  1
1982 Yamada S, Yamamura HI, Roeske WR. Characterization of postsynaptic β-adrenergic receptors and presynaptic muscarinic cholinergic receptors in the rat spleen Life Sciences. 31: 1161-1170. PMID 6292605 DOI: 10.1016/0024-3205(82)90091-1  1
1982 Schoemaker H, Morelli M, Deshmukh P, Yamamura HI. [3H]Ro5-4864 benzodiazepine binding in the kainate lesioned striatum and Huntington's diseased basal ganglia Brain Research. 248: 396-401. PMID 6291702 DOI: 10.1016/0006-8993(82)90602-3  1
1982 Gee KW, Yamamura HI. Differentiation of benzodiazepine receptor agonist and antagonist: Sparing of [3H]benzodiazepine antagonist binding following the photolabelling of benzodiazepine receptors European Journal of Pharmacology. 82: 239-241. PMID 6290239 DOI: 10.1016/0014-2999(82)90521-0  1
1982 Yamada S, Yamamura HI, Roeske WR. An increase in cardiac alpha1-adrenoceptors following chronic clonidine treatment Naunyn-Schmiedeberg's Archives of Pharmacology. 320: 115-118. PMID 6289138 DOI: 10.1007/BF00506311  1
1982 Gee KW, Ehlert FJ, Yamamura HI. The influence of temperature and gamma-aminobutyric acid on benzodiazepine receptor subtypes in the hippocampus of the rat Biochemical and Biophysical Research Communications. 106: 1134-1140. PMID 6288041 DOI: 10.1016/0006-291X(82)91230-X  1
1982 Morelli M, Gee KW, Yamamura HI. The effect of GABA on in vitro binding of two novel non-benzodiazepines, PK 8165 and CGS 8216, to benzodiazepine receptors in the rat brain Life Sciences. 31: 77-81. PMID 6287150 DOI: 10.1016/0024-3205(82)90403-9  1
1982 Gee KW, Yamamura HI. A novel pyrazoloquinoline that interacts with brain benzodiazepine receptors: Characterization of some in vitro and in vivo properties of CGS 9896 Life Sciences. 30: 2245-2252. PMID 6287145 DOI: 10.1016/0024-3205(82)90251-X  1
1982 Mosberg HI, Hurst R, Hruby VJ, Galligan JJ, Burks TF, Gee K, Yamamura HI. [D-Pen2, L-Cys5]enkephalinamide and[D-Pen2, D-Cys5] enkephalinamide, conformationally constrained cyclic enkephalinamide analogs with delta receptor specificity. Biochemical and Biophysical Research Communications. 106: 506-12. PMID 6285922 DOI: 10.1016/0006-291X(82)91139-1  1
1982 Fon Chiu Mia Chen, Yamamura HI, Roeske WR. Adenylate cyclase and beta adrenergic receptor development in the mouse heart Journal of Pharmacology and Experimental Therapeutics. 222: 7-13. PMID 6283073  1
1982 Davis TP, Schoemaker H, Chen A, Yamamura HI. I. High performance liquid chromatography of pharmacologically active amines and peptides in biological materials Life Sciences. 30: 971-987. PMID 6280002 DOI: 10.1016/0024-3205(82)90515-X  1
1982 Buck SH, Walsh JH, Yamamura HI, Burks TF. Neuropeptides in sensory neurons Life Sciences. 30: 1857-1866. PMID 6180272 DOI: 10.1016/0024-3205(82)90465-9  1
1982 Buck SH, Burks TF, Yamamura HI. Neuropeptide alterations in the central nervous system in aging Gerontology. 28: 25-34. PMID 6177585 DOI: 10.1159/000212571  1
1982 Schoemaker H, Davis TP, Pedigo NW, Chen A, Berens ES, Ragan P, Ling NC, Yamamura HI. Identification of beta-endorphin-6(16-17) as the principal metabolite of des-tyrosin-gamma-endorphin (DTgammaE) in vitro and assessment of its activity in neurotransmitter receptor binding assays. European Journal of Pharmacology. 81: 459-68. PMID 6126374 DOI: 10.1016/0014-2999(82)90111-X  1
1982 Gee KW, Morelli M, Yamamura HI. The effect of temperature on CL 218872 and propyl beta-carboline-3-carboxylate inhibition of [3H]-flunitrazepam binding in rat brain Biochemical and Biophysical Research Communications. 105: 1532-1537. PMID 6125147 DOI: 10.1016/0006-291X(82)90962-7  1
1982 Gee KW, Horst WD, O'Brien R, Yamamura HI. High affinity inhibition of [3H]-Flunitrazepam binding to brain benzodiazepine receptors by CGS 9896, a novel pyrazoloquinoline Biochemical and Biophysical Research Communications. 105: 457-461. PMID 6124246 DOI: 10.1016/0006-291X(82)91456-5  1
1982 Schoemaker H, Morelli M, Yamamura HI. 3H-Ro5-4864 benzodiazepine binding in the kainic acid lesioned rat striatum and in Huntington's disease Federation Proceedings. 41.  1
1982 Morelli M, Dichiara G, Yamamura HI. The role of the dorsal mesencephalic reticular formation and deep layers of the superior colliculus in the turning behavior originating from the corpus striatum Proceedings of the Western Pharmacology Society. 433-436.  1
1982 Yamanaka K, Yamamura HI, Roeske WR. Antagonist affinity states of cardiac α-adrenoceptors and their regulation Federation Proceedings. 41: 6047.  1
1982 Morelli M, Ehlert F, Roeske W, Yamamura HI. The GABA shift: A predictor of anxiolytic efficacy Federation Proceedings. 41: 7987.  1
1982 Ehlert FJ, Roeske WR, Chen A, Yamamura HI. Correlation between pharmacological activity and the influence of GABA on the binding of flunitrazepam and the specific benzodiazepine antagonist, Ro 15-1788 Psychopharmacology Bulletin. 18: 100-101.  1
1982 Ehlert FJ, Roeske WR, Yamamura HI. Complex binding properties of the benzodiazepine receptor Federation Proceedings. 41.  1
1982 Deshmukh PP, Nelson DL, Yamamura HI. Localization of 5-HT1 receptor subtypes in rat brain by autoradiography Federation Proceedings. 41.  1
1981 Pedigo NW, Yamamura HI, Nelson DL. Discrimination of multiple [3H]5-hydroxytryptamine binding sites by the neuroleptic spiperone in rat brain Journal of Neurochemistry. 36: 220-226. PMID 7463047 DOI: 10.1111/j.1471-4159.1981.tb02397.x  1
1981 Nelson DL, Pedigo NW, Yamamura HI. Multiple 3H-5-hydroxytryptamine binding sites in rat brain Journal De Physiologie. 77: 369-372. PMID 7288652  1
1981 Ehlert FJ, Roeske WR, Yamamura HI. Dopaminergic regulation of muscarinic receptor binding in the corpus striatum Proceedings of the Western Pharmacology Society. 93-95. PMID 7255494  1
1981 Overstreet DH, Driscoll P, Martin JR, Yamamura HI. Brain muscarinic cholinergic receptor binding in Roman high- and low-avoidance rats Psychopharmacology. 72: 143-145. PMID 6782603 DOI: 10.1007/BF00431647  1
1981 Mimaki T, Yamamura HI. Modulation of benzodiazepine receptor binding by antiepileptic drugs and seizures Medical Journal of Osaka University. 32: 15-24. PMID 6285156  1
1981 Pedigo NW, Schoemaker H, Morelli M, McDougal JN, Malick JB, Burks TF, Yamamura HI. Benzodiazepine receptor binding in young, mature and senescent rat brain and kidney Neurobiology of Aging. 2: 83-88. PMID 6272144 DOI: 10.1016/0197-4580(81)90003-8  1
1981 Ehlert FJ, Roeske WR, Yamamura HI. Multiple benzodiazepine receptors and their regulation by γ-aminobutyric Life Sciences. 29: 235-248. PMID 6270491 DOI: 10.1016/0024-3205(81)90239-3  1
1981 Schoemaker H, Bliss M, Yamamura HI. Specific high-affinity saturable binding of [3H] Ro5-4864 To benzodiazepine binding sites in the rat cerebral cortex European Journal of Pharmacology. 71: 173-175. PMID 6263650 DOI: 10.1016/0014-2999(81)90405-2  1
1981 Lippa AS, Critchett DJ, Ehlert F, Yamamura HI, Enna SJ, Bartus RT. Age-related alterations in neurotransmitter receptors: an electrophysiological and biochemical analysis. Neurobiology of Aging. 2: 3-8. PMID 6115325 DOI: 10.1016/0197-4580(81)90052-X  1
1981 Regan JW, Yamamura HI, Yamada S, Roeske WR. High affinity renal [3H]flunitrazepam binding: Characterization, localization, and alteration in hypertension Life Sciences. 28: 991-998. PMID 6111733 DOI: 10.1016/0024-3205(81)90744-X  1
1981 Johnson RW, Yamamura HI. Fractionation of murine brain homogenates by isopycnic centrifugation: Evidence for benzodiazepine receptor heterogeneity Federation Proceedings. 40: 440.  1
1981 Yamamura HI, Schoemaker H, Yamamura S, Bliss M. Specific high affinity saturable binding of 3H-Ro5-4864 to benzodiazepine binding sites in the rat cerebral cortex Pharmacologist. 23.  1
1981 Schoemaker H, Bliss M, Yamamura SH, Yamamura HI. High affinity benzodiazepine binding sites for 3H-RO5-4864 in rat cerebral cortex and kidney Neuroscience Letters. 24.  1
1981 Barritt D, Roeske WR, Yamamura S, Yamamura HI. Postnatal development and regulation of the muscarinic receptor in the mouse heart using the agonist [3H]CIS methyldioxolane Federation Proceedings. 40: 488.  1
1981 Ehlert FJ, Roeske WR, Yamamura SH, Yamamura HI. Bnezodiazepine Benzodiazepine binding using [3H]propyl β-carboline-3-carboxylate Federation Proceedings. 40: 437.  1
1981 Yamamura HI, Ehlert F, Mimaki T. Benzodiazepine receptor binding studies in rat brain using two novel nonbenzodiazepines Neuroendocrinology Letters. 3: 67.  1
1981 Roeske WR, Yamamura HI, Yamada S. Post-synaptic β-adrenergic receptors increase and pre-synaptic muscarinic receptors decrease in splenic tissue after 6-hydroxydopamine treatment Federation Proceedings. 40: 136.  1
1981 Yamamura HI, Mimaki T, Horst D, O'Brien R. [3H]CL 218,872: a novel triazolopyridazine which labels the benzodiazepine receptor Federation Proceedings. 40: 438.  1
1981 Buck SH, Yamamura HI, Burks TF. Capsaicin is a potent depletor of primary afferent substance P (SP) producing long-lasting thermal and chemogenic analgesia in guinea pigs Pharmacologist. 23.  1
1980 Regan JW, Yamamura HI, Yamada S, Roeske WR. Renal benzodiazepine binding increases during deoxycorticosterone/salt hypertension in rats European Journal of Pharmacology. 67: 167-168. PMID 7418732 DOI: 10.1016/0014-2999(80)90029-1  1
1980 Schallert T, Overstreet DH, Yamamura HI. Muscarinic receptor binding and behavioral effects of atropoine following chronic catecholamine depletion or acetylcholinesterase inhibition in rats. Pharmacology, Biochemistry, and Behavior. 13: 187-92. PMID 7413689 DOI: 10.1016/0091-3057(80)90071-4  1
1980 Ehlert FJ, Dumont Y, Roeske WR, Yamamura HI. Muscarinic receptor binding in rat brain using the agonist, [3H]cis methyldioxolane Life Sciences. 26: 961-967. PMID 7392777 DOI: 10.1016/0024-3205(80)90117-4  1
1980 Rosenberger LB, Yamamura HI, Roeske WR. Cardiac muscarinic cholinergic receptor binding is regulated by Na+ and guanyl nucleotides Journal of Biological Chemistry. 255: 820-823. PMID 7356659  1
1980 Ehlert FJ, Roeske WR, Yamamura HI. Regulation of muscarinic receptor binding by guanine nucleotides and N-ethylmaleimide Journal of Supramolecular and Cellular Biochemistry. 14: 149-162. PMID 7230804  1
1980 Yamada S, Yamamura HI, Roeske WR. Alterations in central and peripheral adrenergic receptors in deoxycorticosterone/salt hypertensive rats Life Sciences. 27: 2405-2416. PMID 6259480 DOI: 10.1016/0024-3205(80)90512-3  1
1980 Yamada S, Yamamura HI, Roeske WR. Ontogeny of mammalian cardiac α1-adrenergic recpeptors European Journal of Pharmacology. 68: 217-221. PMID 6258929  1
1980 Mimaki T, Deshmukh PP, Yamamura HI. Decreased benzodiazepine receptor density in rat cerebellum following neurotoxic doses of phenytoin Journal of Neurochemistry. 35: 1473-1475. PMID 6255101  1
1980 Yamada S, Yamamura HI, Roeske WR. Alterations in cardiac autonomic receptors following 6-hydroxydopamine treatment in rats Molecular Pharmacology. 18: 185-192. PMID 6252437  1
1980 Olsen RW, Reisine TD, Yamamura HI. Neurotransmitter receptors - biochemistry and alterations in neuropsychiatric disorders Life Sciences. 27: 801-808. PMID 6251327 DOI: 10.1016/0024-3205(80)90073-9  1
1980 Martin AR, Paradkar VM, Peng GW, Speth RC, Yamamura HI, Horn AS. Conformationally restricted tricyclic antidepressants. 1. Octahydrodibenzazepinonaphthyridines as rigid imipramine analogues. Journal of Medicinal Chemistry. 23: 865-73. PMID 6249933 DOI: 10.1021/JM00182A011  1
1980 Yamada S, Yamamura HI, Roeske WR. The regulation of cardiac α1-adrenergic receptors by guanine nucleotides and by muscarinic cholinergic agonists European Journal of Pharmacology. 63: 239-241. PMID 6247169 DOI: 10.1016/0014-2999(80)90455-0  1
1980 U'Prichard DC, Reisine TD, Yamamura S, Mason ST, Fibiger HC, Ehlert F, Yamamura HI. Differential supersensitivity of beta-receptor subtypes in rat cortex and cerebellum after central noradrenergic denervation. Life Sciences. 26: 355-64. PMID 6245317 DOI: 10.1016/0024-3205(80)90151-4  0.36
1980 U'Prichard DC, Reisine TD, Mason ST, Fibiger HC, Yamamura HI. Modulation of rat brain alpha- and beta-adrenergic receptor populations by lesion of the dorsal noradrenergic bundle. Brain Research. 187: 143-54. PMID 6244065 DOI: 10.1016/0006-8993(80)90500-4  0.36
1980 Nagy JI, Vincent SR, Staines WA, Fibiger HC, Reisine TD, Yamamura HI. Neurotoxic action of capsaicin on spinal substance P neurons. Brain Research. 186: 435-44. PMID 6153557 DOI: 10.1016/0006-8993(80)90987-7  1
1980 Yamada S, Yamamura HI, Roeske WR. Characterization of alpha-1 adrenergic receptors in the heart using [sup 3H]WB4101: Effect of 6-hydroxydopamine treatment Journal of Pharmacology and Experimental Therapeutics. 215: 176-185. PMID 6109014  1
1980 Reisine TD, Overstreet D, Gale K, Rossor M, Iversen L, Yamamura HI. Benzodiazepine receptors: the effect of GABA on their characteristics in human brain and their alteration in Huntington's disease. Brain Research. 199: 79-88. PMID 6105905 DOI: 10.1016/0006-8993(80)90231-0  0.36
1980 Martin AR, Kim SH, Yamamura HI, Horn AS. Conformationally restricted phenothiazine neuroleptics. 1. 3-(Dimethylamino)-1,2,3,4-tetrahydroazepino[3,2,1-kl]phenothiazine. Journal of Medicinal Chemistry. 23: 938-41. PMID 6105219 DOI: 10.1021/JM00182A022  0.44
1980 Regan JW, Roeske WR, Yamamura HI. 3H-flunitrazepam binding to bovine retina and the effect of GABA thereon Neuropharmacology. 19: 413-414. PMID 6104311 DOI: 10.1016/0028-3908(80)90195-1  1
1980 U'Prichard DC, Yamamura HI, Reisine TD. Characterization and differential in vivo regulation of brain adrenergic receptor subtypes Advances in Biochemical Psychopharmacology. 21: 213-221. PMID 6103648  1
1980 Regan JW, Roeske WR, Yamamura HI. The effect of GABA on the binding of 3H-flunitrazepam in mouse brains during development Brain Research Bulletin. 5: 857-860. DOI: 10.1016/0361-9230(80)90144-6  1
1980 Yamamura HI, Reisine TD, Beaumont K. Huntington's disease: Alterations in GABA and benzodiazepine receptors in the human brain Brain Research Bulletin. 5: 773-775. DOI: 10.1016/0361-9230(80)90128-8  1
1980 Mimaki T, Deshmukh PP, Yamamura HI. Decreased benzodiazepine receptor density in rat brain following chronic phenytoin administration Annals of Neurology. 8: 230.  1
1980 Yamada S, Yamamura HI, Roeske WR. Alterations in central and peripheral receptors (R) in salt deoxycorticosterone (DOCA) treated rats Circulation. 62.  1
1980 Mimaki T, Deshmukh PP, Yamamura HI. An interaction of phenytoin (DPH) with benzodiazepine receptor in rat brain Pharmacologist. 22: 141.  1
1980 Chen FCM, Yamamura HI, Roeske WR. β-Adrenergic receptor and adenyl cyclase development in the mouse heart Clinical Research. 28.  1
1979 Johnson RW, Yamamura HI. Photoaffinity labeling of the benzodiazepine receptor in bovine cerebral cortex Life Sciences. 25: 1613-1620. PMID 522618 DOI: 10.1016/0024-3205(79)90445-4  1
1979 Speth RC, Bresolin N, Yamamura HI. Acute diazepam administration produces rapid increases in brain benzodiazepine receptor density European Journal of Pharmacology. 59: 159-160. PMID 510397 DOI: 10.1016/0014-2999(79)90041-4  1
1979 Speth RC, Yamamura HI. On the ability of choline and its analogues to interact with muscarinic cholinergic receptors in the rat brain European Journal of Pharmacology. 58: 197-201. PMID 499350 DOI: 10.1016/0014-2999(79)90012-8  1
1979 Reisine TD, Nagy JI, Fibiger HC, Yamamura HI. Localization of dopamine receptors in rat brain. Brain Research. 169: 209-14. PMID 455093 DOI: 10.1016/0006-8993(79)90391-3  1
1979 Reisine TD, Nagy JI, Beaumont K, Fibiger HC, Yamamura HI. The localization of receptor binding sites in the substantia nigra and striatum of the rat. Brain Research. 177: 241-52. PMID 227532 DOI: 10.1016/0006-8993(79)90775-3  0.36
1979 Overstreet DH, Yamamura HI. Receptor alterations and drug tolerance Life Sciences. 25: 1865-1877. PMID 43446 DOI: 10.1016/0024-3205(79)90607-6  1
1979 Pedigo NW, Schallert T, Overstreet DH, Ling NC, Ragan P, Reisine TD, Yamamura HI. Inhibition of in vivo 3H-spiperone binding by the proposed antipsychotic Des-Tyr1-gamma-endorphin. European Journal of Pharmacology. 60: 359-64. PMID 43261 DOI: 10.1016/0014-2999(79)90242-5  1
1979 Speth RC, Yamamura HI. Alterations in benzodiazepine receptors in cerebella of mutant mice Federation Proceedings. 38.  1
1979 Roeske WR, Yamamura HI. Mechanisms of cardiac arrhythmias: Muscarinic cholinergic receptor alterations in the production of asystole Clinical Research. 27.  1
1978 Pedigo NW, Reisine TD, Fields JZ, Yamamura HI. 3H-spiroperidol binding to two receptor sites in both the corpus striatum and frontal cortex of rat brain European Journal of Pharmacology. 50: 451-453. PMID 699968 DOI: 10.1016/0014-2999(78)90154-1  1
1978 Kobayashi RM, Palkovits M, Hruska RE, Rothschild R, Yamamura HI. Regional distribution of muscarinic cholinergic receptors in rat brain. Brain Research. 154: 13-23. PMID 698807 DOI: 10.1016/0006-8993(78)91047-8  1
1978 Hruska RE, Schwarcz R, Coyle JT, Yamamura HI. Alterations of muscarinic cholinergic receptors in the rat striatum after kainic acid injections. Brain Research. 152: 620-5. PMID 687979 DOI: 10.1016/0006-8993(78)91120-4  0.36
1978 Roeske WR, Yamamura HI. Maturation of mammalian myocardial muscarinic cholinergic receptors Life Sciences. 23: 127-132. PMID 682873 DOI: 10.1016/0024-3205(78)90260-6  1
1978 Hruska RE, White R, Azari J, Yamamura HI. Muscarinic cholinergic receptors in mammalian retina Brain Research. 148: 493-498. PMID 656944 DOI: 10.1016/0006-8993(78)90736-9  1
1978 Fields JZ, Roeske WR, Morkin E, Yamamura HI. Cardiac muscarinic cholinergic receptors. Biochemical identification and characterization Journal of Biological Chemistry. 253: 3251-3258. PMID 641068  1
1978 Davis KL, Yamamura HI. Cholinergic underactivity in human memory disorders Life Sciences. 23: 1729-1733. PMID 364228 DOI: 10.1016/0024-3205(78)90100-5  1
1978 Reisine TD, Yamamura HI, Bird ED, Spokes E, Enna SJ. Pre- and postsynaptic neurochemical alterations in Alzheimer's disease. Brain Research. 159: 477-81. PMID 215272 DOI: 10.1016/0006-8993(78)90562-0  1
1978 Beaumont K, Chilton WS, Yamamura HI, Enna SJ. Muscimol binding in rat brain: association with synaptic GABA receptors. Brain Research. 148: 153-62. PMID 207386 DOI: 10.1016/0006-8993(78)90385-2  1
1978 Wastek GJ, Yamamura HI. Biochemical characterization of the muscarinic cholinergic receptor in human brain: Alterations in Huntington's disease Molecular Pharmacology. 14: 768-780. PMID 152407  1
1978 Beaumont K, Fields JZ, Reisine TD, Yamamura HI. 3H-kainic acid (KA) binding: Alterations after striatal KA lesions Pharmacologist. 20: 473.  1
1977 Harris LW, Kundig F, Yamamura HI. Partial purification and separation of retinal acetylcholinesterase from butyrylcholinesterase by affinity chromatography Biochemical Pharmacology. 26: 1441-1443. PMID 901558 DOI: 10.1016/0006-2952(77)90371-9  1
1977 Hruska RE, Huxtable RJ, Yamamura HI. Purification of [3H]taurine of high specific activity Analytical Biochemistry. 79: 568-570. PMID 869192 DOI: 10.1016/0003-2697(77)90431-6  1
1977 Yaksh TL, Yamamura HI. Depression by morphine of the resting and evoked release of [3H]-acetylcholine from the cat caudate nucleus in vivo Neuropharmacology. 16: 227-233. PMID 859683 DOI: 10.1016/0028-3908(77)90099-5  1
1977 Arregui A, Bennett JP, Bird ED, Yamamura HI, Iversen LL, Snyder SH. Huntington's chorea: selective depletion of activity of angiotensin coverting enzyme in the corpus striatum. Annals of Neurology. 2: 294-8. PMID 214022 DOI: 10.1002/ana.410020406  1
1977 Enna SJ, Stern LZ, Wastek GJ, Yamamura HI. Cerebrospinal fluid gamma-aminobutyric acid variations in neurological disorders. Archives of Neurology. 34: 683-5. PMID 143928 DOI: 10.1001/ARCHNEUR.1977.00500230053008  1
1977 Wastek GJ, Stern LZ, Yamamura HI. Recent advances in the neurochemistry of Huntington's disease Arizona Medicine. 34: 547-548. PMID 143259  1
1977 Snyder SH, Yamamura HI. Antidepressants and the muscarinic acetylcholine receptor. Archives of General Psychiatry. 34: 236-9. PMID 14603 DOI: 10.1001/archpsyc.1977.01770140126014  0.96
1977 Enna SJ, Bennett JP, Bylund DB, Creese I, Burt DR, Charness ME, Yamamura HI, Simantov R, Snyder SH. Neurotransmitter receptor binding: regional distribution in human brain. Journal of Neurochemistry. 28: 233-6. PMID 13155 DOI: 10.1111/j.1471-4159.1977.tb07733.x  1
1977 Speth RC, Chen FM, Lindstrom JM, Kobayashi RM, Yamamura HI. Nicotinic cholinergic receptors in rat brain identified by [125I] Naja naja siamensis α-toxin binding Brain Research. 131: 350-355. DOI: 10.1016/0006-8993(77)90527-3  1
1977 Hruska RE, Yamamura HI. Biochemical characterization of muscarinic cholinergic receptors in mammalian retina Pharmacologist. 19.  1
1977 Fields JZ, Roeske WR, Morkin E, Yamamura HI. Biochemical demonstration of muscarinic cholinergic receptors in mammalian heart Federation Proceedings. 36.  1
1976 Yamamura HI, Manian AA, Snyder SH. Muscarinic cholinergic receptor binding: influence of pimozide and chlorpromazine metabolites. Life Sciences. 18: 685-91. PMID 1263751 DOI: 10.1016/0024-3205(76)90179-X  1
1976 Enna SJ, Yamamura HI, Snyder SH. Development of muscarinic cholinergic and GABA receptor binding in chick embryo brain. Brain Research. 101: 177-83. PMID 1244218 DOI: 10.1016/0006-8993(76)91001-5  1
1976 Coyle JT, Yamamura HI. Neurochemical aspects of the ontogenesis of cholinergic neurons in the rat brain Brain Research. 118: 429-440. PMID 1009427 DOI: 10.1016/0006-8993(76)90310-3  1
1976 Yamamura HI, Wastek G, Chang KJ, Snyder SH. Cholinergic receptors in the mammalian central nervous system. Proceedings of the Western Pharmacology Society. 19: 13-8. PMID 995977  1
1976 Kuhar MJ, Yamamura HI. Localization of cholinergic muscarinic receptors in rat brain by light microscopic radioautography Brain Research. 110: 229-243. PMID 938940 DOI: 10.1016/0006-8993(76)90399-1  1
1976 Enna SJ, Bird ED, Bennett JP, Bylund DB, Yamamura HI, Iversen LL, Snyder SH. Huntington's chorea. Changes in neurotransmitter receptors in the brain. The New England Journal of Medicine. 294: 1305-9. PMID 4733 DOI: 10.1056/NEJM197606102942402  1
1976 Speth R, Yamamura HI, Dettbarn WD. Prolonged cholinesterase inhibition and central muscarinic receptor activity Trans.Amer.Soc.Neurochem.. 7.  1
1975 Yaksh TL, Filbert MG, Harris LW, Yamamura HI. Acetylcholinesterase turnover in brain, cerebrospinal fluid and plasma. Journal of Neurochemistry. 25: 853-60. PMID 1206402 DOI: 10.1111/j.1471-4159.1975.tb04417.x  1
1975 Kuhar MJ, DeHaven RN, Yamamura HI, Rommel-Spacher H, Simon JR. Further evidence for cholinergic habenulo-interpeduncular neurons: Pharmacologic and functional characteristics Brain Research. 97: 265-275. PMID 1175046 DOI: 10.1016/0006-8993(75)90449-7  1
1975 Yaksh TL, Yamamura HI. The release in vivo of [3H]acetylcholine from cat caudate nucleus and cerebral cortex by atropine, pentylenetetrazol, K+ depolarization and electrical stimulation Journal of Neurochemistry. 25: 123-130. PMID 1141909  1
1975 Yaksh TL, Yamamura HI. Blockade by morphine of acetylcholine release from the caudate nucleus in the mid-pontine pretrigeminal cat Brain Research. 83: 520-524. PMID 1111819 DOI: 10.1016/0006-8993(75)90847-1  1
1975 Snyder SH, Chang KJ, Kuhar MJ, Yamamura HI. Biochemical indentification of the mammalian muscarinic cholinergic receptor. Federation Proceedings. 34: 1915-21. PMID 808430  1
1975 Guarnieri M, Krell LS, McKhann GM, Pasternak GW, Yamamura HI. The effects of cell isolation techniques on neuronal membrane receptors. Brain Research. 93: 337-42. PMID 169956 DOI: 10.1016/0006-8993(75)90355-8  0.4
1975 Yamamura HI, Snyder SH. Tricyclic antidepressants and the central cholinergic muscarinic receptor Pharmacologist. 17.  1
1974 Snyder SH, Banerjee SP, Yamamura HI, Greenberg D. Drugs, neurotransmitters, and schizophrenia. Science (New York, N.Y.). 184: 1243-53. PMID 17784215 DOI: 10.1126/science.184.4143.1243  1
1974 Yamamura HI, Snyder SH. Postsynaptic localization of muscarinic cholinergic receptor binding in rat hippocampus. Brain Research. 78: 320-6. PMID 4853717 DOI: 10.1016/0006-8993(74)90556-3  1
1974 Mulder AH, Yamamura HI, Kuhar MJ, Snyder SH. Release of acetylcholine from hippocampal slices by potassium depolarization: dependence on high affinity choline uptake. Brain Research. 70: 372-6. PMID 4825681 DOI: 10.1016/0006-8993(74)90329-1  1
1974 Yamamura HI, Kuhar MJ, Snyder SH. In vivo identification of muscarinic cholinergic receptor binding in rat brain. Brain Research. 80: 170-6. PMID 4421615 DOI: 10.1016/0006-8993(74)90738-0  1
1974 Yaksh TL, Yamamura HI. Factors affecting performance of the push pull cannula in brain Journal of Applied Physiology. 37: 428-434. PMID 4413416  1
1974 Snyder S, Greenberg D, Yamamura HI. Antischizophrenic Drugs and Brain Cholinergic Receptors: Affinity for Muscarinic Sites Predicts Extrapyramidal Effects Archives of General Psychiatry. 31: 58-61. PMID 4152054 DOI: 10.1001/archpsyc.1974.01760130040006  1
1974 Yamamura HI, Snyder SH. Muscarinic cholinergic binding in rat brain. Proceedings of the National Academy of Sciences of the United States of America. 71: 1725-9. PMID 4151898 DOI: 10.1073/pnas.71.5.1725  1
1974 Yaksh TL, Yamamura HI, Fedele LA. Appearance in cat cerebrospinal fluid of radiolabelled metabolites following intraventricular injection of [3H]choline Journal of Pharmacy and Pharmacology. 26: 65-67. PMID 4150939  1
1974 Yamamura HI, Kuhar MJ, Greenberg D, Snyder SH. Muscarinic cholinergic receptor binding: regional distribution in monkey brain Brain Research. 66: 541-546. DOI: 10.1016/0006-8993(74)90069-9  1
1974 Yaksh TL, Fedele LA, Yamamura HI. Recovery of cholinesterase activity in the cerebrospinal fluid, brainstem and plasma of the unanesthetized cat after irreversible cholinesterase inhibition Experientia. 30: 38-39. DOI: 10.1007/BF01921583  1
1974 Yamamura HI, Snyder SH. Muscarinic cholinergic receptor binding in the longitudinal muscle of the guinea pig ileum with ]:H]quinuclidinyl benzilate Molecular Pharmacology. 10: 861-867.  1
1974 Yamamura HI, Kuhar MJ, Snyder SH. Identification in vivo of muscarinic cholinergic receptor binding in rat brain Pharmacologist. 16.  1
1974 Snyder SH, Banerjee SP, Yamamura HI, Greenberg D. Drugs, neurotransmitters, and schizophrenia Science. 184: 1243-1253.  1
1974 Yamamura HI, Kuhar MJ, Snyder SH. Muscarinic cholinergic receptor binding in mammalian central and peripheral nervous system: demonstration in vitro and in vivo Trans.Amer.Soc.Neurochem.. 5.  1
1974 Yamamura HI, Broomfield CA, Snyder SH. Muscarinic cholinergic receptor binding in mammalian central and peripheral nervous system with (3H) quinuclidinyl benzilate Federation Proceedings. 33.  1
1973 Yamamura HI, Snyder SH. High affinity transport of choline into synaptosomes of rat brain. Journal of Neurochemistry. 21: 1355-74. PMID 4771436 DOI: 10.1111/j.1471-4159.1973.tb06022.x  1
1973 Yaksh TL, Fedele LA, Yamamura HI. Effects of repeated withdrawal of cerebrospinal fluid by cisternal puncture on cisternal protein levels in the unanesthetized cat Physiology and Behavior. 10: 149-151. PMID 4697008 DOI: 10.1016/0031-9384(73)90100-5  1
1973 Yaksh TL, Yamamura HI. The effect of morphine in vivo on resting and evoked release of 3H acetylcholine from the cat caudate nucleus Pharmacologist. 15: 261.  1
1972 Yamamura HI, Snyder SH. Choline: high-affinity uptake by rat brain synaptosomes. Science (New York, N.Y.). 178: 626-8. PMID 5086398 DOI: 10.1126/science.178.4061.626  1
1972 Adams GK, Yamamura HI, O'Leary JF. Spontaneous recovery of central respiratory function after an irreversible AChE inhibitor. European Journal of Pharmacology. 20: 377-80. PMID 4643460 DOI: 10.1016/0014-2999(72)90202-6  1
1971 Harris LW, Yamamura HI, Fleisher JH. De novo synthesis of acetylcholinesterase in guinea pig retina after inhibition by pinacolyl methyl-phosphonofluoridate Biochemical Pharmacology. 20: 2927-2930. PMID 5114524 DOI: 10.1016/0006-2952(71)90209-7  1
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