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Richard D. Gandour - Publications

Affiliations: 
Chemistry Virginia Polytechnic Institute and State University, Blacksburg, VA, United States 
Area:
Organic Chemistry
Website:
https://chem.vt.edu/people/faculty/rgandour.html
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42 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2014 Savage AM, Li Y, Matolyak LE, Doncel GF, Turner SR, Gandour RD. Anti-HIV activities of precisely defined, semirigid, carboxylated alternating copolymers Journal of Medicinal Chemistry. 57: 6354-6363. PMID 25026140 DOI: 10.1021/Jm401913W  0.301
2013 Muckom RJ, Stanzione F, Gandour RD, Sum AK. Dendritic amphiphiles strongly affect the biophysical properties of DPPC bilayer membranes. The Journal of Physical Chemistry. B. 117: 1810-8. PMID 23330648 DOI: 10.1021/Jp310043A  0.332
2012 Falkinham JO, Macri RV, Maisuria BB, Actis ML, Sugandhi EW, Williams AA, Snyder AV, Jackson FR, Poppe MA, Chen L, Ganesh K, Gandour RD. Antibacterial activities of dendritic amphiphiles against nontuberculous mycobacteria. Tuberculosis (Edinburgh, Scotland). 92: 173-81. PMID 22209468 DOI: 10.1016/J.Tube.2011.12.002  0.754
2011 Maisuria BB, Actis ML, Hardrict SN, Falkinham JO, Cole MF, Cihlar RL, Peters SM, Macri RV, Sugandhi EW, Williams AA, Poppe MA, Esker AR, Gandour RD. Comparing micellar, hemolytic, and antibacterial properties of di- and tricarboxyl dendritic amphiphiles. Bioorganic & Medicinal Chemistry. 19: 2918-26. PMID 21493076 DOI: 10.1016/J.Bmc.2011.03.036  0.753
2009 Macri RV, Karlovská J, Doncel GF, Du X, Maisuria BB, Williams AA, Sugandhi EW, Falkinham JO, Esker AR, Gandour RD. Comparing anti-HIV, antibacterial, antifungal, micellar, and cytotoxic properties of tricarboxylato dendritic amphiphiles. Bioorganic & Medicinal Chemistry. 17: 3162-8. PMID 19307123 DOI: 10.1016/J.Bmc.2009.02.055  0.765
2007 Sugandhi EW, Slebodnick C, Falkinham JO, Gandour RD. Synthesis and antimicrobial evaluation of water-soluble, dendritic derivatives of epimeric 5alpha-cholestan-3-amines and 5alpha-cholestan-3-yl aminoethanoates. Steroids. 72: 615-26. PMID 17532019 DOI: 10.1016/J.Steroids.2007.04.001  0.77
2007 Sugandhi EW, Falkinham JO, Gandour RD. Synthesis and antimicrobial activity of symmetrical two-tailed dendritic tricarboxylato amphiphiles. Bioorganic & Medicinal Chemistry. 15: 3842-53. PMID 17400459 DOI: 10.1016/J.Bmc.2007.03.017  0.795
2007 Sugandhi EW, Macri RV, Williams AA, Kite BL, Slebodnick C, Falkinham JO, Esker AR, Gandour RD. Synthesis, critical micelle concentrations, and antimycobacterial properties of homologous, dendritic amphiphiles. Probing intrinsic activity and the "cutoff" effect. Journal of Medicinal Chemistry. 50: 1645-50. PMID 17346035 DOI: 10.1021/Jm061240D  0.723
2007 Williams AA, Sugandhi EW, Macri RV, Falkinham JO, Gandour RD. Antimicrobial activity of long-chain, water-soluble, dendritic tricarboxylato amphiphiles. The Journal of Antimicrobial Chemotherapy. 59: 451-8. PMID 17242037 DOI: 10.1093/Jac/Dkl503  0.746
2007 Karlovská J, Williams AA, Macri RV, Gandour RD, Funari SS, Uhríková D, Balgavý P. Synchrotron SAX and WAX diffraction study of a hydrated very long-chain, dendritic amphiphile + DPPC mixture. Colloids and Surfaces. B, Biointerfaces. 54: 160-4. PMID 17134885 DOI: 10.1016/J.Colsurfb.2006.10.009  0.763
2005 Savle PS, Neptune NE, Yang Y, Rouden JH, Kite BL, Sugandhi EW, Macri RV, Kashfi K, Gandour RD. Comparison of (+)- and (-)-hemipalmitoylcarnitinium as inhibitors of hepatic mitochondrial carnitine palmitoyltransferases in diabetic rats. Medicinal Chemistry (ShāRiqah (United Arab Emirates)). 1: 445-53. PMID 16787328 DOI: 10.2174/1573406054864115  0.694
2005 Gandour RD. Toward a design of affordable, topical microbicides: acylcarnitine analogues. Current Pharmaceutical Design. 11: 3757-67. PMID 16305510 DOI: 10.2174/138161205774580705  0.309
2005 Williams AA, Day BS, Kite BL, McPherson MK, Slebodnick C, Morris JR, Gandour RD. Homologous, long-chain alkyl dendrons form homologous thin films on silver oxide surfaces. Chemical Communications (Cambridge, England). 5053-5. PMID 16220168 DOI: 10.1039/B506710C  0.734
2002 Wong YL, Hubieki MP, Curfman CL, Doncel GF, Dudding TC, Savle PS, Gandour RD. A structure-activity study of spermicidal and anti-HIV properties of hydroxylated cationic surfactants. Bioorganic & Medicinal Chemistry. 10: 3599-608. PMID 12213475 DOI: 10.1016/S0968-0896(02)00245-6  0.632
2002 Wong YL, Curfman CL, Doncel GF, Patricia Hubieki M, Dudding TC, Savle PS, Gandour RD. Spermicidal, anti-HIV, and micellar properties of di- and trihydroxylated cationic surfactants Tetrahedron. 58: 45-54. DOI: 10.1016/S0040-4020(01)01114-0  0.639
2002 Ramsay RR, Gandour RD. Selective Modulation of Carnitine Long-chain Acyltransferase Activities Advances in Experimental Medicine and Biology. 466: 103-109. DOI: 10.1007/0-306-46818-2_11  0.31
2000 Savle PS, Shelton TE, Meadows CA, Potts M, Gandour RD, Kennelly PJ. N-(cyclohexanecarboxyl)-O-phospho-l-serine, a minimal substrate for the dual-specificity protein phosphatase IphP. Archives of Biochemistry and Biophysics. 376: 439-48. PMID 10775432 DOI: 10.1006/Abbi.2000.1750  0.303
1999 Savle PS, Pande SV, Lee TS, Gandour RD. Stereoisomeric acylamidomorpholinium carnitine analogues: Selective inhibitors of carnitine palmitoyltransferase I and II Bioorganic and Medicinal Chemistry Letters. 9: 3099-3102. PMID 10560732 DOI: 10.1016/S0960-894X(99)00543-0  0.319
1999 Savle PS, Doncel GF, Bryant SD, Hubieki MP, Robinette RG, Gandour RD. Acylcarnitine analogues as topical, microbicidal spermicides Bioorganic and Medicinal Chemistry Letters. 9: 2545-2548. PMID 10498205 DOI: 10.1016/S0960-894X(99)00423-0  0.413
1998 Savle PS, Medhekar RA, Kelley EL, May JG, Watkins SF, Fronczek FR, Quinn DM, Gandour RD. Change in the mode of inhibition of acetylcholinesterase by (4-nitrophenyl)sulfonoxyl derivatives of conformationally constrained choline analogues. Chemical Research in Toxicology. 11: 19-25. PMID 9477222 DOI: 10.1021/Tx970019O  0.373
1998 Savle PS, Lamoreaux MJ, Berry JF, Gandour RD. A convenient resolution of long-chain alkyl epoxides with Jacobsen's salen(Co)III(OAc) catalysts Tetrahedron Asymmetry. 9: 1843-1846. DOI: 10.1016/S0957-4166(98)00175-X  0.323
1995 Sun G, Fronczek FR, Gandour RD. Methyl (2S,6S:2R,6R)-6-(2-cyanoethyl)-4,6-dimethyl-2-morpholineacetate Acta Crystallographica, Section C: Crystal Structure Communications. 51. PMID 7779326 DOI: 10.1107/S0108270194003604  0.319
1994 Kumaravel G, Nic a' Bháird N, Fronczek FR, Ramsay RR, Ashendel CL, Gandour RD. Evaluation of (2S,4S)/(2R,4R) and (2S,4R)/(2R,4S) 6,6-N,N-dimethyl-2-methyl-2-oxo-1,3-dioxa-4-hexadecyl-6,aza-2-phosphacyc looctane bromide as inhibitors for protein kinase C, carnitine octanoyltransferase, and carnitine palmitoyltransferase Bioorganic and Medicinal Chemistry Letters. 4: 883-886. DOI: 10.1016/S0960-894X(01)80256-0  0.327
1993 Gandour RD, Leung OT, Greway AT, Ramsay RR, Nic A'Bháird N, Fronczek FR, Bellard BM, Kumaravel G. (+)-Hemipalmitoylcarnitinium strongly inhibits carnitine palmitoyltransferase-I in intact mitochondria Journal of Medicinal Chemistry. 36: 237-242. PMID 8423595 DOI: 10.1021/Jm00054A007  0.331
1992 Lee BH, Stelly TC, Colucci WJ, Garcia JG, Gandour RD, Quinn DM. Inhibition of acetylcholinesterase by hemicholiniums, conformationally constrained choline analogues. Evaluation of aryl and alkyl substituents. Comparisons with choline and (3-hydroxyphenyl)trimethylammonium. Chemical Research in Toxicology. 5: 411-8. PMID 1504265 DOI: 10.1021/Tx00027A015  0.331
1992 Sun G, Fronczek FR, Gandour RD. (R)‐(1‐Methyloxiranyl)methyl 4‐nitrobenzenesulfonate Acta Crystallographica Section C. 48: 758-760. DOI: 10.1107/S0108270191010995  0.305
1992 Gandour RD, Blackwell NL, Colucci WJ, Chung C, Bieber LL, Ramsay RR, Brass EP, Fronczek FR. Syntheses, structures, and enzymatic evaluations of hemiacylcarnitiniums, a new class of carnitine acyltransferase inhibitors The Journal of Organic Chemistry. 57: 3426-3431. DOI: 10.1021/Jo00038A035  0.305
1992 Garcia JG, Fronczek FR, Gandour RD. The structure of the products when α-bromoacetoarenones react with 3-(N,N-dimethylamino)propan-1-ol Bioorganic and Medicinal Chemistry Letters. 2: 157-160. DOI: 10.1016/S0960-894X(01)80441-8  0.345
1991 Brass EP, Gandour RD, Griffith OW. Effect of carnitine acetyltransferase inhibition on rat hepatocyte metabolism. Biochimica Et Biophysica Acta. 1095: 17-22. PMID 1932127 DOI: 10.1016/0167-4889(91)90039-Z  0.348
1991 Fronczek FR, Gandour RD, Fyles TM, Hocking PJ, McDermid SJ, Wotton PD. Polycarboxylate crown ethers from meso-tartaric acid Canadian Journal of Chemistry. 69: 12-19. DOI: 10.1139/V91-003  0.324
1988 Gandour RD, Colucci WJ, Stelly TC, Brady PS, Brady LJ. Hemipalmitoylcarnitinium, a strong competitive inhibitor of purified hepatic carnitine palmitoyltransferase Archives of Biochemistry and Biophysics. 267: 515-520. PMID 3214166 DOI: 10.1016/0003-9861(88)90058-6  0.302
1988 Arnold KA, Mallen J, Trafton JE, White BD, Fronczek FR, Gehrig LM, Gandour RD, Gokel GW. Ring-sidearm cooperativity in cation inclusion complexes of 12-membered ring lariat ethers: effect of sidearm chain length and a clarification of long-sidearm binding strengths The Journal of Organic Chemistry. 53: 5652-5657. DOI: 10.1021/Jo00259A008  0.342
1988 Arnold KA, Viscariello AM, Kim M, Gandour RD, Fronczek FR, Gokel GW. N,N'-Bis(subst1tuted)-4,13-diaza-18-crown-6 derivatives having pi-donor-group-sidearms: correlation of thermodynamics and solid state structures Tetrahedron Letters. 29: 3025-3028. DOI: 10.1016/0040-4039(88)85076-7  0.321
1987 Brady LJ, Brady PS, Gandour RD. Effect of methylglyoxal bis(guanylhydrazone) on hepatic, heart and skeletal muscle mitochondrial carnitine palmitoyltransferase and β-oxidation of fatty acids Biochemical Pharmacology. 36: 447-452. PMID 3827937 DOI: 10.1016/0006-2952(87)90349-2  0.34
1987 Colucci WJ, Turnbull SP, Gandour RD. Preparation of crystalline sodium norcarnitine: An easily handled precursor for the preparation of carnitine analogs and radiolabeled carnitine Analytical Biochemistry. 162: 459-462. PMID 3605609 DOI: 10.1016/0003-2697(87)90420-9  0.331
1987 Arnold KA, Echegoyen L, Fronczek FR, Gandour RD, Gatto VJ, White BD, Gokel GW. Evidence for cryptand-like behavior in bibracchial lariat ether (BiBLE) complexes obtained from x-ray crystallography and solution thermodynamic studies Journal of the American Chemical Society. 109: 3716-3721. DOI: 10.1021/Ja00246A032  0.307
1986 Gandour RD, Colucci WJ, Stelly TC, Brady PS, Brady LJ. Active-site probes of carnitine acyltransferases. Inhibition of carnitine acetyltransferase by hemiacetylcarnitinium, a reaction intermediate analogue Biochemical and Biophysical Research Communications. 138: 735-741. PMID 3741430 DOI: 10.1016/S0006-291X(86)80558-7  0.329
1986 Colucci WJ, Gandour RD, Mooberry EA. Conformational analysis of charged flexible molecules in water by application of a new karplus equation combined with MM2 computations: Conformations of carnitine and acetylcarnitine Journal of the American Chemical Society. 108: 7141-7147. DOI: 10.1021/Ja00283A001  0.301
1985 Tirado-Rives J, Fronczek FR, Gandour RD. (E)-1,2-Bis(2-methylphenyl)ethene, C16H16 Acta Crystallographica Section C Crystal Structure Communications. 41: 1327-1329. DOI: 10.1107/S0108270185007648  0.304
1975 Wang MS, Gandour RD, Rodgers J, Haslam JL, Schowen RL. Transition-state structure for a conformation change of ribonuclease Bioorganic Chemistry. 4: 392-406. DOI: 10.1016/0045-2068(75)90050-4  0.311
1972 Gandour RD, Schowen RL. Chapter 26. Intramolecular Catalysis in Medicinal Chemistry Annual Reports in Medicinal Chemistry. 7: 279-288. DOI: 10.1016/S0065-7743(08)60821-0  0.3
1971 Magid RM, Nieh EC, Gandour RD. Coupling reaction of phenyllithium with allylic chlorides. Influence of methyl substituents on the distribution of products Journal of Organic Chemistry. 36: 2099-2105. DOI: 10.1021/Jo00814A015  0.72
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