| Year |
Citation |
Score |
| 2017 |
Liu X, Khadtare N, Patel H, Stephani R, Cantor J. Time-dependent effects of HJP272, an endothelin receptor antagonist, in bleomycin-induced pulmonary fibrosis. Pulmonary Pharmacology & Therapeutics. PMID 28619646 DOI: 10.1016/J.Pupt.2017.06.003 |
0.305 |
|
| 2017 |
Khadtare N, Stephani R, Korlipara V. Design, synthesis and evaluation of 1,3,6-trisubstituted-4-oxo-1,4-dihydroquinoline-2-carboxylic acid derivatives as ETA receptor selective antagonists using FRET assay. Bioorganic & Medicinal Chemistry Letters. PMID 28462837 DOI: 10.1016/J.Bmcl.2017.04.049 |
0.349 |
|
| 2015 |
Patel HJ, Patel PD, Ochiana SO, Yan P, Sun W, Patel MR, Shah SK, Tramentozzi E, Brooks J, Bolaender A, Shrestha L, Stephani R, Finotti P, Leifer C, Li Z, et al. Structure-activity relationship in a purine-scaffold compound series with selectivity for the endoplasmic reticulum Hsp90 paralog Grp94. Journal of Medicinal Chemistry. 58: 3922-43. PMID 25901531 DOI: 10.1021/Acs.Jmedchem.5B00197 |
0.521 |
|
| 2014 |
Patel S, Liu X, Liu M, Stephani R, Patel H, Cantor J. HJP272, a novel endothelin receptor antagonist, attenuates lipopolysaccharide-induced acute lung injury in hamsters. Lung. 192: 803-10. PMID 25087133 DOI: 10.1007/S00408-014-9628-Z |
0.487 |
|
| 2013 |
Patel PD, Yan P, Seidler PM, Patel HJ, Sun W, Yang C, Que NS, Taldone T, Finotti P, Stephani RA, Gewirth DT, Chiosis G. Paralog-selective Hsp90 inhibitors define tumor-specific regulation of HER2. Nature Chemical Biology. 9: 677-84. PMID 23995768 DOI: 10.1038/Nchembio.1335 |
0.416 |
|
| 2012 |
Sadarangani IR, Bhatia S, Amarante D, Lengyel I, Stephani RA. Synthesis, resolution and anticonvulsant activity of chiral N-1'-ethyl,N-3'-(1-phenylethyl)-(R,S)-2'H,3H,5'H-spiro-(2-benzofuran-1,4'-imidazolidine)-2',3,5'-trione diastereomers. Bioorganic & Medicinal Chemistry Letters. 22: 2507-9. PMID 22401865 DOI: 10.1016/J.Bmcl.2012.02.005 |
0.589 |
|
| 2010 |
Patel HJ, Olgun N, Lengyel I, Reznik S, Stephani RA. Synthesis and pharmacological activity of 1,3,6-trisubstituted-4-oxo-1,4-dihydroquinoline-2-carboxylic acids as selective ET(A) antagonists. Bioorganic & Medicinal Chemistry Letters. 20: 6840-4. PMID 20932745 DOI: 10.1016/J.Bmcl.2010.08.074 |
0.505 |
|
| 2010 |
Olgun NS, Patel HJ, Stephani R, Lengyel I, Reznik SE. Blockade of endothelin-1 with a novel series of 1,3,6-trisubstituted-2-carboxy-quinol-4-ones controls infection-associated preterm birth. The American Journal of Pathology. 177: 1929-35. PMID 20802183 DOI: 10.2353/Ajpath.2010.100281 |
0.513 |
|
| 2010 |
DEVITO SC, STEPHANI RA. ChemInform Abstract: Synthesis and Pharmacological Evaluation of Some Novel 13-(N,N- Dialkylamino-alkyl)benzo(g)(2)benzopyrano(4,3-b)indol-5(13H)ones. Cheminform. 22: no-no. DOI: 10.1002/chin.199145168 |
0.308 |
|
| 2008 |
Bhavsar T, Liu XJ, Patel H, Stephani R, Cantor JO. Preferential recruitment of neutrophils by endothelin-1 in acute lung inflammation induced by lipopolysaccharide or cigarette smoke. International Journal of Chronic Obstructive Pulmonary Disease. 3: 477-81. PMID 18990977 DOI: 10.2147/Copd.S2837 |
0.47 |
|
| 2008 |
Olgun N, Patel HJ, Stephani R, Wang W, Yen H, Reznik SE. Effect of the putative novel selective ETA-receptor antagonist HJP272, a 1,3,6-trisubstituted-2-carboxy-quinol-4-one, on infection-mediated premature delivery. Canadian Journal of Physiology and Pharmacology. 86: 571-5. PMID 18758506 DOI: 10.1139/Y08-057 |
0.463 |
|
| 2007 |
Lengyei I, Patel HJ, Stephani RA. The preparation and characterization of nineteen new phthalidyl spirohydantoins Heterocycles. 73: 349-375. DOI: 10.3987/Com-07-S(U)9 |
0.543 |
|
| 2006 |
Patel HJ, Sarra J, Caruso F, Rossi M, Doshi U, Stephani RA. Synthesis and anticonvulsant activity of new N-1',N-3'-disubstituted-2'H,3H,5'H-spiro-(2-benzofuran-1,4'-imidazolidine)-2',3,5'-triones. Bioorganic & Medicinal Chemistry Letters. 16: 4644-7. PMID 16793262 DOI: 10.1016/J.Bmcl.2006.05.102 |
0.559 |
|
| 2002 |
Stephani R, Cesare V, Sadarangani I, Lengyel I. Synthesis of new optically active and racemic phenylsuccinamic acids Synthesis. 47-52. DOI: 10.1055/S-2002-19294 |
0.574 |
|
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