| Year |
Citation |
Score |
| 2022 |
Bhandare RR, Sigalapalli DK, Shaik AB, Canney DJ, Blass BE. Selectivity profile comparison for certain γ-butyrolactone and oxazolidinone-based ligands on a sigma 2 receptor over sigma 1: a molecular docking approach. Rsc Advances. 12: 20096-20109. PMID 35919619 DOI: 10.1039/d2ra03497b |
0.75 |
|
| 2017 |
Padhariya K, Bhandare RR, Canney D, Velingkar V. Cardiovascular Concern of 5-HT2B Receptor and Recent Vistas in the Development of Its Antagonists. Cardiovascular & Hematological Disorders Drug Targets. PMID 28676029 DOI: 10.2174/1871529X17666170703115111 |
0.684 |
|
| 2016 |
Annadurai S, Zhang M, Gabriel JL, Bencheriff M, Canney DJ. Ether and carbamate derivatives of 3-quinuclidinol and 3-hydroxymethylquinuclidine: synthesis and evaluation as nicotinic ligands. Medicinal Chemistry (Shariqah (United Arab Emirates)). PMID 26833074 DOI: 10.2174/1573406412666160201121133 |
0.766 |
|
| 2015 |
Canney D, Gao R, Fan R. Synthesis of β,β-Disubstituted γ-Butyrolactones by Chemoselective Oxidation of 1,4-Diols and γ-Hydroxy Olefins with RuCl3/NaIO4 Synlett. 26: 661-665. DOI: 10.1055/S-0034-1379614 |
0.378 |
|
| 2014 |
Bhandare RR, Canney DJ. Bioisosteric replacement and related analogs in the design, synthesis and evaluation of ligands for muscarinic acetylcholine receptors. Medicinal Chemistry (ShāRiqah (United Arab Emirates)). 10: 361-75. PMID 24021160 DOI: 10.2174/15734064113096660043 |
0.776 |
|
| 2013 |
Gao R, Bhandare RR, Canney DJ. Homologation as a lead modification approach en route to a series of lactone-based muscarinic ligands Medicinal Chemistry Research. 23: 1023-1030. DOI: 10.1007/S00044-013-0692-3 |
0.77 |
|
| 2012 |
Annadurai S, Martinez R, Canney DJ, Eidem T, Dunman PM, Abou-Gharbia M. Design and synthesis of 2-aminothiazole based antimicrobials targeting MRSA. Bioorganic & Medicinal Chemistry Letters. 22: 7719-25. PMID 23116888 DOI: 10.1016/J.Bmcl.2012.09.095 |
0.746 |
|
| 2012 |
Iwuchukwu OF, Sharan S, Canney DJ, Nagar S. Analytical method development for synthesized conjugated metabolites of trans-resveratrol, and application to pharmacokinetic studies. Journal of Pharmaceutical and Biomedical Analysis. 63: 1-8. PMID 22342060 DOI: 10.1016/J.Jpba.2011.12.006 |
0.333 |
|
| 2012 |
Nantogmah S, Desai S, Bhandare R, Gabriel J, Soprano D, Canney DJ. Synthesis and preliminary evaluation of affinity to retinoic acid receptors for new organosilicon-based retinoids Pharmaceutical Chemistry Journal. 45: 612-621. DOI: 10.1007/S11094-012-0692-5 |
0.771 |
|
| 2010 |
Gao R, Canney DJ. A versatile and practical microwave-assisted synthesis of sterically hindered N-arylpiperazines. The Journal of Organic Chemistry. 75: 7451-3. PMID 20863109 DOI: 10.1021/Jo101478C |
0.335 |
|
| 2010 |
Bhandare RR, Canney DJ. Modifications to five-substituted 3,3-diethyl-4,5-dihydro-2(3H)-furanones en route to novel muscarinic receptor ligands Medicinal Chemistry Research. 20: 558-565. DOI: 10.1007/S00044-010-9349-7 |
0.785 |
|
| 2010 |
CANNEY DJ, HOLLAND KD, LEVINE JA, MCKEON AC, FERRENDELLI JA, COVEY DF. ChemInform Abstract: Synthesis and Structure-Activity Studies of Alkyl-Substituted γ- Butyrolactones and γ-Thiobutyrolactones: Ligands for the Picrotoxin Receptor. Cheminform. 22: no-no. DOI: 10.1002/chin.199144152 |
0.587 |
|
| 2010 |
CANNEY DJ, LEVINE JA, LU H, COVEY DF. ChemInform Abstract: Facile Synthesis of α,β- and/or γ-Alkyl-Substituted . gamma.-Butyrolactones Using Readily Prepared Olefinic Esters. Cheminform. 22: no-no. DOI: 10.1002/chin.199109177 |
0.441 |
|
| 2009 |
Sun W, Carroll PJ, Soprano DR, Canney DJ. Identification of a chromone-based retinoid containing a polyolefinic side chain via facile synthetic routes. Bioorganic & Medicinal Chemistry Letters. 19: 4339-42. PMID 19502054 DOI: 10.1016/J.Bmcl.2009.05.081 |
0.707 |
|
| 2009 |
Gao R, Canney DJ. A modified Prins reaction for the facile synthesis of structurally diverse substituted 5-(2-hydroxyethyl)-3,3-dihydrofurane-2(3H)-ones Tetrahedron Letters. 50: 5914-5916. DOI: 10.1016/J.Tetlet.2009.08.016 |
0.452 |
|
| 2008 |
Desai S, Sun W, Gabriel J, Canney DJ. THE SYNTHESIS AND PRELIMINARY EVALUATION OF SUBSTITUTED CHROMONES, COUMARINS, CHROMANONES, AND BENZOPHENONES AS RETINOIC ACID RECEPTOR LIGANDS Heterocyclic Communications. 14. DOI: 10.1515/Hc.2008.14.3.129 |
0.76 |
|
| 2007 |
Sun W, Desai S, Piao H, Carroll P, Canney DJ. Wittig—Horner—Emmons Reactions of Triethyl 3-Methylphosphonocrotonate with 3-Formylchromones en route to Benzophenone-Based Retinoid Candidates. Cheminform. 38. DOI: 10.1002/CHIN.200730181 |
0.567 |
|
| 2005 |
Ahungena A, Canney DJ. Synthesis and Evaluation of Homologous Analogs of Anticonvulsant 5-Substituted 3,3-Diethyl-4,5-Dighdro-2(3H)-Furanones Medicinal Chemistry Research. 14: 404-428. DOI: 10.1007/S00044-006-0144-4 |
0.457 |
|
| 2005 |
Sun W, Blanton MP, Gabriel JL, Canney DJ. Bioisosteric replacement in the design and synthesis of ligands for nicotinic acetylcholine receptors Medicinal Chemistry Research. 14: 241-259. DOI: 10.1007/S00044-005-0137-8 |
0.71 |
|
| 1998 |
Canney DJ, Zhang M, Doukas PH, Massakowski C, Aronstam R, Gattu M, Buccafusco J. Characterization of ethyl (3-quinuclidinyl) acetate (EQA) as a ligand for acetylcholine receptors. Life Sciences. 63: PL329-36. PMID 9851313 DOI: 10.1016/S0024-3205(98)00502-5 |
0.353 |
|
| 1998 |
Canney DJ, Lu HF, McKeon AC, Yoon KW, Xu K, Holland KD, Rothman SM, Ferrendelli JA, Covey DF. Structure-activity studies of fluoroalkyl-substituted gamma-butyrolactone and gamma-thiobutyrolactone modulators of GABA(A) receptor function. Bioorganic & Medicinal Chemistry. 6: 43-55. PMID 9502104 DOI: 10.1016/S0968-0896(97)10006-2 |
0.606 |
|
| 1995 |
Canney DJ, Kung MP, Kung HF. Amino- and amido-tetrabenazine derivatives: Synthesis and evaluation as potential ligands for the vesicular monoamine transporter Nuclear Medicine and Biology. 22: 527-535. PMID 7550031 DOI: 10.1016/0969-8051(94)00118-4 |
0.488 |
|
| 1994 |
Kung MP, Canney DJ, Frederick D, Zhuang Z, Billings JJ, Kung HF. Binding of 125I-iodovinyltetrabenazine to CNS vesicular monoamine transport sites. Synapse (New York, N.Y.). 18: 225-32. PMID 7855735 DOI: 10.1002/Syn.890180308 |
0.332 |
|
| 1993 |
Canney DJ, Billings J, Francesconi LC, Guo YZ, Haggerty BS, Rheingold AL, Kung HF. Dicarboxylate diamide dimercaptide (N2S2) technetium-99m complexes: Synthesis and biological evaluation as potential renal radiopharmaceuticals Journal of Medicinal Chemistry. 36: 1032-1040. PMID 8478903 DOI: 10.1021/Jm00060A011 |
0.372 |
|
| 1993 |
Canney DJ, Covey DF, Evers AS. Direct observation of a fluorinated anticonvulsant in brain tissue using 19F-NMR techniques. Biochemical Pharmacology. 45: 949-59. PMID 8452571 DOI: 10.1016/0006-2952(93)90181-U |
0.477 |
|
| 1993 |
Holland KD, McKeon AC, Canney DJ, Covey DF, Ferrendelli JA. Relative anticonvulsant effects of GABAmimetic and GABA modulatory agents. Epilepsia. 33: 981-6. PMID 1334454 DOI: 10.1111/J.1528-1157.1992.Tb01747.X |
0.516 |
|
| 1993 |
Canney DJ, Guo Y‐, Kung M‐, Kung HF. Synthesis and preliminary evaluation of an iodovinyl‐tetrabenazine analog as a marker for the vesicular monoamine transporter Journal of Labelled Compounds and Radiopharmaceuticals. 33: 355-368. DOI: 10.1002/Jlcr.2580330413 |
0.325 |
|
| 1991 |
Canney DJ, Holland KD, Levine JA, McKeon AC, Ferrendelli JA, Covey DF. Synthesis and structure-activity studies of alkyl-substituted gamma-butyrolactones and gamma-thiobutyrolactones: ligands for the picrotoxin receptor. Journal of Medicinal Chemistry. 34: 1460-7. PMID 1849999 DOI: 10.1021/Jm00108A034 |
0.624 |
|
| 1990 |
Holland KD, Canney DJ, Rothman SM, Ferrendelli JA, Covey DF. Physiological modulation of the GABA receptor by convulsant and anticonvulsant barbiturates in cultured rat hippocampal neurons. Brain Research. 516: 147-50. PMID 2163720 DOI: 10.1016/0006-8993(90)90910-4 |
0.481 |
|
| 1990 |
Canney DJ, Levine JA, Lu H, Covey DF. Facile Synthesis of α, β, and/or γ-Alkyl-Substituted γ-Butyrolactones Using Readily Prepared Olefinic Esters Synthetic Communications. 20: 2065-2073. DOI: 10.1080/00397919008053138 |
0.531 |
|
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