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Scott R. Gilbertson, Ph.D. - Publications

Affiliations: 
1990-2003 Chemistry Washington University, Saint Louis, St. Louis, MO 
 2003- Chemistry University of Houston, Houston, TX, United States 
Area:
Organic synthesis
Website:
http://www.chem.uh.edu/people/faculty/Gilbertson/index.php

82 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2021 Li J, Gilbertson SR. Diastereoselective Rhodium Catalyzed [4 + 2] Cycloisomerization of Allenes. Organic Letters. PMID 33783221 DOI: 10.1021/acs.orglett.1c00554  0.307
2019 Abbasgholizadeh R, Zhang H, Craft JW, Bryan RM, Bark SJ, Briggs JM, Fox RO, Agarkov A, Zimmer WE, Gilbertson SR, Schwartz RJ. Discovery of vascular Rho kinase (ROCK) inhibitory peptides. Experimental Biology and Medicine (Maywood, N.J.). 1535370219849581. PMID 31132884 DOI: 10.1177/1535370219849581  0.754
2018 Tao Y, Gilbertson SR. Diastereoselective synthesis of 1,3-disubstituted isoindolines and sultams via bronsted acid catalysis. Chemical Communications (Cambridge, England). PMID 30232479 DOI: 10.1039/C8Cc04946G  0.406
2018 Gilbertson SR, Chen YC, Soto CA, Yang Y, Rice KC, Cunningham KA, Anastasio NC. Synthesis and activity of functionalizable derivatives of the serotonin (5-HT) 5-HTreceptor (5-HTR) antagonist M100907. Bioorganic & Medicinal Chemistry Letters. PMID 29555153 DOI: 10.1016/J.Bmcl.2018.02.058  0.358
2017 Soto CA, Shashack MJ, Fox RG, Bubar MJ, Rice KC, Watson CS, Cunningham KA, Gilbertson SR, Anastasio NC. Novel Bivalent 5-HT2A Receptor Antagonists Exhibit High Affinity and Potency in Vitro and Efficacy in Vivo. Acs Chemical Neuroscience. PMID 29111677 DOI: 10.1021/Acschemneuro.7B00309  0.313
2017 Chen YC, Hartley RM, Anastasio NC, Cunningham KA, Gilbertson SR. Synthesis and structure-activity relationships of tools based on WAY163909, a 5-HT2c receptor agonist. Acs Chemical Neuroscience. PMID 28414422 DOI: 10.1021/Acschemneuro.6B00439  0.316
2017 Zhang W, Gilbertson SR. Diastereoselective synthesis of N-sulfinyl α-aminophosphine sulfides and phosphines Tetrahedron Letters. 58: 2175-2177. DOI: 10.1016/J.Tetlet.2017.03.067  0.393
2016 Do HT, Zhang N, Pati D, Gilbertson SR. Synthesis and activity of benzimidazole-1,3-dioxide inhibitors of separase. Bioorganic & Medicinal Chemistry Letters. PMID 27530289 DOI: 10.1016/J.Bmcl.2016.07.080  0.313
2015 Do H, Kang CW, Cho JH, Gilbertson SR. Enantioselective Synthesis of (-)-Dysiherbaine. Organic Letters. 17: 3972-4. PMID 26258884 DOI: 10.1021/Acs.Orglett.5B01821  0.544
2015 Do H, Kang CW, Cho JH, Gilbertson SR. Enantioselective Synthesis of (-)-Dysiherbaine Organic Letters. 17: 3972-3974. DOI: 10.1021/acs.orglett.5b01821  0.483
2015 Demerzhan S, Gilbertson SR. Palladium-NHC catalyzed formation of cyclopenta[b]benzofurans and their subsequent modification Tetrahedron Letters. DOI: 10.1016/J.Tetlet.2015.01.192  0.372
2014 Canlas GM, Gilbertson SR. [4+2+2] Cycloaddition catalyzed by a new cationic rhodium-bisphosphine monooxide complex. Chemical Communications (Cambridge, England). 50: 5007-10. PMID 24706156 DOI: 10.1039/C4Cc01320D  0.357
2014 Zhao Y, Gilbertson SR. Synthesis of proline-based N-heterocyclic carbene ligands. Organic Letters. 16: 1033-5. PMID 24495075 DOI: 10.1021/Ol403465D  0.497
2013 De S, Chen L, Zhang S, Gilbertson SR. Synthesis of a 2(1H)-pyridone library via rhodium-catalyzed formation of isomunchones. Acs Combinatorial Science. 15: 340-3. PMID 23742807 DOI: 10.1021/Co400067Q  0.572
2013 Anastasio NC, Gilbertson SR, Bubar MJ, Agarkov A, Stutz SJ, Jeng Y, Bremer NM, Smith TD, Fox RG, Swinford SE, Seitz PK, Charendoff MN, Craft JW, Laezza FM, Watson CS, et al. Peptide inhibitors disrupt the serotonin 5-HT2C receptor interaction with phosphatase and tensin homolog to allosterically modulate cellular signaling and behavior. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 33: 1615-30. PMID 23345234 DOI: 10.1523/Jneurosci.2656-12.2013  0.744
2012 Gilbertson SR. Chemistry. Relay reactions that trap organometallic intermediates. Science (New York, N.Y.). 338: 1432-3. PMID 23239726 DOI: 10.1126/Science.1231509  0.386
2012 Chen D, Ma L, Kanalas JJ, Gao J, Pawlik J, Jimenez ME, Walter MA, Peterson JW, Gilbertson SR, Schein CH. Structure-based redesign of an edema toxin inhibitor. Bioorganic & Medicinal Chemistry. 20: 368-76. PMID 22154558 DOI: 10.1016/J.Bmc.2011.10.091  0.319
2011 Khalaf J, Estrella-Jimenez ME, Shashack MJ, Phatak SS, Zhang S, Gilbertson SR. Design, synthesis, and diversification of 3,5-substituted enone library. Acs Combinatorial Science. 13: 351-6. PMID 21648460 DOI: 10.1021/Co200070M  0.46
2010 Prasad BA, Buechele AE, Gilbertson SR. Pd-NHC catalyzed cyclopentannulation of diazabicyclic alkenes with ortho-aryl halides. Organic Letters. 12: 5422-5. PMID 21043477 DOI: 10.1021/Ol102270R  0.346
2010 Tanifum EA, Gilbertson SR. Design, synthesis, and diversification of 5,5-dimethyl cyclohexen-1,4-dione library. Journal of Combinatorial Chemistry. 12: 318-20. PMID 20387791 DOI: 10.1021/Cc100030H  0.455
2009 Prasad BA, Gilbertson SR. One-pot synthesis of unsymmetrical N-heterocyclic carbene ligands from N-(2-iodoethyl)arylamine salts. Organic Letters. 11: 3710-3. PMID 19624103 DOI: 10.1021/Ol901189M  0.402
2009 Tanifum EA, Kots AY, Choi BK, Murad F, Gilbertson SR. Novel pyridopyrimidine derivatives as inhibitors of stable toxin a (STa) induced cGMP synthesis. Bioorganic & Medicinal Chemistry Letters. 19: 3067-71. PMID 19409779 DOI: 10.1016/J.Bmcl.2009.04.024  0.374
2008 Agarkov A, Gilbertson SR. Preparation of a library of unsymmetrical ureas based on 8-azabicyclo[3.2.1]octane scaffold. Journal of Combinatorial Chemistry. 10: 655-7. PMID 18611055 DOI: 10.1021/Cc800068K  0.794
2008 Jimenez ME, Bush K, Pawlik J, Sower L, Peterson JW, Gilbertson SR. Synthesis and screening of small molecule inhibitors of anthrax edema factor. Bioorganic & Medicinal Chemistry Letters. 18: 4215-8. PMID 18539457 DOI: 10.1016/J.Bmcl.2008.05.059  0.36
2008 Drew ME, Banerjee R, Uffman EW, Gilbertson S, Rosenthal PJ, Goldberg DE. Plasmodium food vacuole plasmepsins are activated by falcipains. The Journal of Biological Chemistry. 283: 12870-6. PMID 18308731 DOI: 10.1074/Jbc.M708949200  0.751
2008 Agarkov A, Chauhan S, Lory PJ, Gilbertson SR, Motin VL. Substrate specificity and screening of the integral membrane protease Pla. Bioorganic & Medicinal Chemistry Letters. 18: 427-31. PMID 17981463 DOI: 10.1016/J.Bmcl.2007.09.104  0.773
2007 Lory PM, Estrella-Jimenez ME, Shashack MJ, Lokesh GL, Natarajan A, Gilbertson SR. Synthesis and screening of 3-substituted thioxanthen-9-one-10,10-dioxides. Bioorganic & Medicinal Chemistry Letters. 17: 5940-3. PMID 17826998 DOI: 10.1016/J.Bmcl.2007.07.103  0.359
2007 DeBoef B, Counts WR, Gilbertson SR. Rhodium-catalyzed synthesis of eight-membered rings. The Journal of Organic Chemistry. 72: 799-804. PMID 17253798 DOI: 10.1021/Jo0620462  0.772
2006 Agarkov A, Greenfield S, Xie D, Pawlick R, Starkey G, Gilbertson SR. Synthesis of phosphine containing amino acids: utilization of peptide synthesis in ligand design. Biopolymers. 84: 48-73. PMID 16235230 DOI: 10.1002/Bip.20395  0.776
2006 Lory PMJ, Agarkov A, Gilbertson SR. An expedient route to 3-chlorothioxanthen-9-one-10,10-dioxide and derivation by palladium-catalyzed coupling Synlett. 3045-3048. DOI: 10.1055/S-2006-951520  0.796
2005 Xu G, Gilbertson SR. Development of building blocks for the synthesis of N-heterocyclic carbene ligands. Organic Letters. 7: 4605-8. PMID 16209490 DOI: 10.1021/Ol0516521  0.525
2005 Agarkov A, Gilbertson SR. Coordination mode for turn-based phosphine ligands: The origin of selectivity in Pd catalysis Tetrahedron Letters. 46: 181-183. DOI: 10.1016/J.Tetlet.2004.10.096  0.809
2004 Agarkov A, Greenfield SJ, Ohishi T, Collibee SE, Gilbertson SR. Catalysis with phosphine-containing amino acids in various "turn" motifs. The Journal of Organic Chemistry. 69: 8077-85. PMID 15527293 DOI: 10.1021/Jo049103G  0.773
2004 Gilbertson SR, Yamada S. A study of catalyst selectivity with polymer bound palladium phosphine complexes on various solid phase synthesis supports Tetrahedron Letters. 45: 3917-3920. DOI: 10.1016/J.Tetlet.2004.03.110  0.447
2003 Greenfield SJ, Agarkov A, Gilbertson SR. High asymmetric induction with beta-turn-derived palladium phosphine complexes. Organic Letters. 5: 3069-72. PMID 12916983 DOI: 10.1021/Ol035097J  0.794
2003 Agarkov A, Uffman EW, Gilbertson SR. Parallel approach to selective catalysts for palladium-catalyzed desymmetrization of 2,4-cyclopentenediol. Organic Letters. 5: 2091-4. PMID 12790536 DOI: 10.1021/Ol034548X  0.773
2003 Xu G, Gilbertson SR. Asymmetric hydrogenation of aromatic olefins catalyzed by iridium complexes of proline derived phosphine-oxazoline ligands Tetrahedron Letters. 44: 953-955. DOI: 10.1016/S0040-4039(02)02747-8  0.458
2003 DeBoef B, Gilbertson SR. C-C bond formation via C-H bond activation: Synthesis of the core of teleocidin B4 Chemtracts. 16: 249-253.  0.628
2002 Gilbertson SR, DeBoef B. Rhodium catalyzed [4 + 2 + 2] cycloaddition and alkyne insertion: a new route to eight-membered rings. Journal of the American Chemical Society. 124: 8784-5. PMID 12137517 DOI: 10.1021/Ja026536X  0.732
2002 Gilbertson SR, Lan P. Solid-phase synthesis of phosphine-oxazoline peptides Tetrahedron Letters. 43: 6961-6965. DOI: 10.1016/S0040-4039(02)01596-4  0.605
2002 Xu G, Gilbertson SR. Facile synthesis of proline based phosphine-oxazoline ligands by formation of a P-N bond Tetrahedron Letters. 43: 2811-2814. DOI: 10.1016/S0040-4039(02)00346-5  0.437
2002 Uffman EW, Gilbertson SR. A novel peptide-based encoding system for "one-bead one-compound" peptidomimetic and small molecule combinatorial libraries Chemtracts. 15: 606-610.  0.774
2001 Gilbertson SR, Xie D, Fu Z. Proline-based P, N ligands in asymmetric allylation and the Heck reaction. The Journal of Organic Chemistry. 66: 7240-6. PMID 11681933 DOI: 10.1021/Jo0158231  0.469
2001 Gilbertson SR, Lan P. Kinetic resolution in palladium-catalyzed asymmetric allylic alkylations by a P,O ligand system. Organic Letters. 3: 2237-40. PMID 11440588 DOI: 10.1021/Ol0161256  0.576
2001 Gilbertson SR, Fu Z. Chiral P,N-ligands based on ketopinic acid in the asymmetric Heck reaction. Organic Letters. 3: 161-4. PMID 11430024 DOI: 10.1021/Ol006747B  0.497
2001 Greenfield SJ, Gilbertson SR. Preparation of diphenylphosphinoserine and synthesis of other phosphine containing amino acids using zinc/copper reagents Synthesis. 2337-2340. DOI: 10.1055/S-2001-18431  0.8
2001 Gilbertson SR, Fu Z, Xie D. Proline derived phosphine-oxazoline ligands in the asymmetric Heck reaction Tetrahedron Letters. 42: 365-368. DOI: 10.1016/S0040-4039(00)01938-9  0.47
2000 Gilbertson SR, Genov DG, Rheingold AL. Synthesis of new bicyclic P-N ligands and their application in asymmetric Pd-catalyzed pi-allyl alkylation and Heck reaction. Organic Letters. 2: 2885-8. PMID 10964390 DOI: 10.1021/Ol006323H  0.688
2000 Gilbertson SR, Collibee SE, Agarkov A. Asymmetric catalysis with libraries of palladium β-turn phosphine complexes [18] Journal of the American Chemical Society. 122: 6522-6523. DOI: 10.1021/Ja992306F  0.773
1999 Gilbertson SR, Lopez OD. Kinetic Resolution of Diiron Acyl Complexes-An Approach to Asymmetric Bicyclic β-Lactams. Angewandte Chemie (International Ed. in English). 38: 1116-9. PMID 25138514 DOI: 10.1002/(Sici)1521-3773(19990419)38:8<1116::Aid-Anie1116>3.0.Co;2-M  0.429
1999 Gilbertson SR, Xie D. Proline-Based P,N Ligands in Palladium-Catalyzed Asymmetric pi-Allyl Additions. Angewandte Chemie (International Ed. in English). 38: 2750-2752. PMID 10508370 DOI: 10.1002/(Sici)1521-3773(19990917)38:18<2750::Aid-Anie2750>3.0.Co;2-5  0.414
1999 Gilbertson SR, Fu Z, Starkey GW. Palladium-catalyzed synthesis of vinyl phosphines from ketones Tetrahedron Letters. 40: 8509-8512. DOI: 10.1016/S0040-4039(99)01819-5  0.786
1999 Gilbertson SR, Wang X. The parallel synthesis of peptide based phosphine ligands Tetrahedron. 55: 11609-11618. DOI: 10.1016/S0040-4020(99)00682-1  0.488
1998 Gilbertson SR, Hoge GS, Genov DG. Rhodium-catalyzed asymmetric [4 + 2] cycloisomerization reactions Journal of Organic Chemistry. 63: 10077-10080. DOI: 10.1021/Jo981870Q  0.646
1998 Gilbertson SR, Chang CWT. Synthesis of phosphino oxazoline ligand libraries from amino acid and phosphino carboxylate building blocks Journal of Organic Chemistry. 63: 8424-8431. DOI: 10.1021/Jo981420Y  0.485
1998 Gilbertson SR, Hoge GS. Rhodium catalyzed intramolecular [4+2] cycloisomerization reactions Tetrahedron Letters. 39: 2075-2078. DOI: 10.1016/S0040-4039(98)00265-2  0.407
1997 Gilbertson SR, Chang CWT. A modular approach to ligands for asymmetric π-allyl palladium catalysed additions Chemical Communications. 975-976. DOI: 10.1039/A607200C  0.475
1997 Gilbertson SR, Chen G, Kao J, Beatty A, Campana CF. Structure of Phosphorus-Containing Peptide Ligands. X-ray and NMR Structural Study of Free Ligand and Rhodium Complex Journal of Organic Chemistry. 62: 5557-5566. DOI: 10.1021/Jo970773E  0.374
1997 Gilbertson SR, Lopez OD. Synthesis of and asymmetric cycloaddition with chiral diiron acyl complexes Journal of the American Chemical Society. 119: 3399-3400. DOI: 10.1021/Ja964195F  0.426
1996 Gilbertson SR, Starkey GW. Palladium-Catalyzed Synthesis of Phosphine-Containing Amino Acids. The Journal of Organic Chemistry. 61: 2922-2923. PMID 11667143 DOI: 10.1021/Jo960077Z  0.773
1996 Gilbertson SR, Wang X. Synthesis of (Dicyclohexylphosphino)serine, Its Incorporation into a Dodecapeptide, and the Coordination of Rhodium. The Journal of Organic Chemistry. 61: 434-435. PMID 11666953 DOI: 10.1021/Jo951327Z  0.429
1996 Klug CA, Studelska DR, Chen G, Gilbertson SR, Schaefer J. Distance between phosphine-sulfide sidechains of a disubstituted peptide by DRAMA 31P NMR. Solid State Nuclear Magnetic Resonance. 7: 173-6. PMID 9050154 DOI: 10.1016/S0926-2040(96)01268-4  0.323
1996 Gilbertson SR, Wang X, Hoge GS, Klug CA, Schaefer J. Synthesis of phosphine-rhodium complexes attached to a standard peptide synthesis resin Organometallics. 15: 4678-4680. DOI: 10.1021/Om9606000  0.452
1996 Gilbertson SR, Wang X. The combinatorial synthesis of chiral phosphine ligands Tetrahedron Letters. 37: 6475-6478. DOI: 10.1016/0040-4039(96)01424-4  0.498
1996 Gilbertson SR, Pawlick RV. Synthesis of Thiophosphoryl Derivatives of Proline: Building Blocks for Phosphanyl-Substituted Peptides with β-Turns Angewandte Chemie (International Edition in English). 35: 902-904. DOI: 10.1002/Anie.199609021  0.728
1996 Gilbertson SR, Pawlick RV. Synthese von Thiophosphorylprolinen als Bausteine für phosphanylsubstituierte Peptide mit β-Turns† Angewandte Chemie. 108: 963-966. DOI: 10.1002/Ange.19961080819  0.314
1996 Gilbertson SR, Wang X. Synthesis of (dicyclohexylphosphino) serine, its incorporation into a dodecapeptide, and the coordination of rhodium Journal of Organic Chemistry. 61: 434-435.  0.317
1995 Gilbertson SR, Chang CWT. Synthesis of new disugar phosphine ligands and their use in asymmetric hydrogenation Journal of Organic Chemistry. 60: 6226-6228. DOI: 10.1021/Jo00124A051  0.404
1995 Gilbertson SR, Dawson DP, Lopez OD, Marshall KL. Endo-Selective Reactions of .alpha.,.beta.-Unsaturated Hexacarbonyldiiron Bridging Acyl Complexes with Nitrones Journal of the American Chemical Society. 117: 4431-4432. DOI: 10.1021/Ja00120A039  0.319
1995 Gilbertson SR, Pawlick RV. The synthesis and conformation of dihydroxy-cyclo(d-Pro-l-Pro-d-Pro-l-Pro) Tetrahedron Letters. 36: 1229-1232. DOI: 10.1016/0040-4039(95)00022-5  0.68
1995 Gilbertson SR, Dawson DP, Lopez OD, Marshall KL. Endo-selective reactions of α,β-unsaturated hexacarbonyldiiron bridging acyl complexes with nitrones Journal of the American Chemical Society. 117: 4431-4432.  0.629
1994 Gilbertson SR, Chen G, McLoughlin M. Versatile building block for the synthesis of phosphine-containing peptides: The sulfide of diphenylphosphinoserine Journal of the American Chemical Society. 116: 4481-4482. DOI: 10.1021/Ja00089A049  0.714
1993 Gilbertson SR, Zhao X, Dawson DP, Marshall KL. Exo-Selective Diels-Alder reactions of .alpha.,.beta.-unsaturated hexacarbonyl-diiron bridging acyl complexes Journal of the American Chemical Society. 115: 8517-8518. DOI: 10.1021/Ja00071A099  0.325
1993 Gilbertson SR, Zhao X, Dawson DP, Marshall KL. Exo-selective Diels-Alder reactions of α,β-unsaturated hexacarbonyl-diiron bridging acyl complexes Journal of the American Chemical Society. 115: 8517-8518.  0.632
1989 Gilbertson SR, Wulff WD. Evaluation of the Cyclohexadienone Annulation of Chromium-Carbene Complexes for the Synthesis of Taxodione Synlett. 1989: 47-49. DOI: 10.1055/S-1989-34694  0.59
1988 Stuart McCallum J, Kunng FA, Gilbertson SR, Wulff WD. Mechanistic studies on the reaction of chromium carbene complexes with acetylenes: Furan formation and the dependence of the product distribution on the stereochemistry of reaction intermediates Organometallics. 7: 2346-2360. DOI: 10.1021/Om00101A015  0.575
1988 Gilbertson SR, Challener CA, Bos ME, Wulff WD. An examination of the coupling of vinyl and aryl triflates with stannyl cuprates for the purpose of providing regioselective access to vinyl lithiums Tetrahedron Letters. 29: 4795-4798. DOI: 10.1016/S0040-4039(00)80611-5  0.603
1986 Wulff WD, Gilbertson SR, Springer JP. Reactions of cobalt carbene complexes with alkynes. .eta.4-Vinylketene-complexed intermediates and a novel synthesis of bovolide. Journal of the American Chemical Society. 108: 520-2. PMID 22175480 DOI: 10.1021/Ja00263A035  0.619
1986 Wulff WD, Peterson GA, Bauta WE, Chan KS, Faron KL, Gilbertson SR, Kaesler RW, Yang DC, Murray CK. A regioselective entry to vinyllithiums from unsymmetrical ketones via enol triflates Journal of Organic Chemistry. 51: 277-279. DOI: 10.1002/Chin.198627244  0.794
1986 Wulff WD, Gilbertson SR, Springer JP. Reactions of cobalt carbene complexes with alkynes - η4-vinylketene complex intermediates and a novel synthesis of bovolide Journal of the American Chemical Society. 108: 520-522. DOI: 10.1002/Chin.198623282  0.619
1985 Wulff WD, Tang PC, Chan KS, McCallum JS, Yang DC, Gilbertson SR. Cycloadditions and annulations of transition metal carbene complexes Tetrahedron. 41: 5813-5832. DOI: 10.1016/S0040-4020(01)91421-8  0.64
1985 Wulff WD, Gilbertson SR. Aldol reactions of transition-metal carbene complexes Journal of the American Chemical Society. 107: 503-505. DOI: 10.1002/Chin.198521124  0.558
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