Year |
Citation |
Score |
2021 |
Li J, Gilbertson SR. Diastereoselective Rhodium Catalyzed [4 + 2] Cycloisomerization of Allenes. Organic Letters. PMID 33783221 DOI: 10.1021/acs.orglett.1c00554 |
0.307 |
|
2019 |
Abbasgholizadeh R, Zhang H, Craft JW, Bryan RM, Bark SJ, Briggs JM, Fox RO, Agarkov A, Zimmer WE, Gilbertson SR, Schwartz RJ. Discovery of vascular Rho kinase (ROCK) inhibitory peptides. Experimental Biology and Medicine (Maywood, N.J.). 1535370219849581. PMID 31132884 DOI: 10.1177/1535370219849581 |
0.754 |
|
2018 |
Tao Y, Gilbertson SR. Diastereoselective synthesis of 1,3-disubstituted isoindolines and sultams via bronsted acid catalysis. Chemical Communications (Cambridge, England). PMID 30232479 DOI: 10.1039/C8Cc04946G |
0.406 |
|
2018 |
Gilbertson SR, Chen YC, Soto CA, Yang Y, Rice KC, Cunningham KA, Anastasio NC. Synthesis and activity of functionalizable derivatives of the serotonin (5-HT) 5-HTreceptor (5-HTR) antagonist M100907. Bioorganic & Medicinal Chemistry Letters. PMID 29555153 DOI: 10.1016/J.Bmcl.2018.02.058 |
0.358 |
|
2017 |
Soto CA, Shashack MJ, Fox RG, Bubar MJ, Rice KC, Watson CS, Cunningham KA, Gilbertson SR, Anastasio NC. Novel Bivalent 5-HT2A Receptor Antagonists Exhibit High Affinity and Potency in Vitro and Efficacy in Vivo. Acs Chemical Neuroscience. PMID 29111677 DOI: 10.1021/Acschemneuro.7B00309 |
0.313 |
|
2017 |
Chen YC, Hartley RM, Anastasio NC, Cunningham KA, Gilbertson SR. Synthesis and structure-activity relationships of tools based on WAY163909, a 5-HT2c receptor agonist. Acs Chemical Neuroscience. PMID 28414422 DOI: 10.1021/Acschemneuro.6B00439 |
0.316 |
|
2017 |
Zhang W, Gilbertson SR. Diastereoselective synthesis of N-sulfinyl α-aminophosphine sulfides and phosphines Tetrahedron Letters. 58: 2175-2177. DOI: 10.1016/J.Tetlet.2017.03.067 |
0.393 |
|
2016 |
Do HT, Zhang N, Pati D, Gilbertson SR. Synthesis and activity of benzimidazole-1,3-dioxide inhibitors of separase. Bioorganic & Medicinal Chemistry Letters. PMID 27530289 DOI: 10.1016/J.Bmcl.2016.07.080 |
0.313 |
|
2015 |
Do H, Kang CW, Cho JH, Gilbertson SR. Enantioselective Synthesis of (-)-Dysiherbaine. Organic Letters. 17: 3972-4. PMID 26258884 DOI: 10.1021/Acs.Orglett.5B01821 |
0.544 |
|
2015 |
Do H, Kang CW, Cho JH, Gilbertson SR. Enantioselective Synthesis of (-)-Dysiherbaine Organic Letters. 17: 3972-3974. DOI: 10.1021/acs.orglett.5b01821 |
0.483 |
|
2015 |
Demerzhan S, Gilbertson SR. Palladium-NHC catalyzed formation of cyclopenta[b]benzofurans and their subsequent modification Tetrahedron Letters. DOI: 10.1016/J.Tetlet.2015.01.192 |
0.372 |
|
2014 |
Canlas GM, Gilbertson SR. [4+2+2] Cycloaddition catalyzed by a new cationic rhodium-bisphosphine monooxide complex. Chemical Communications (Cambridge, England). 50: 5007-10. PMID 24706156 DOI: 10.1039/C4Cc01320D |
0.357 |
|
2014 |
Zhao Y, Gilbertson SR. Synthesis of proline-based N-heterocyclic carbene ligands. Organic Letters. 16: 1033-5. PMID 24495075 DOI: 10.1021/Ol403465D |
0.497 |
|
2013 |
De S, Chen L, Zhang S, Gilbertson SR. Synthesis of a 2(1H)-pyridone library via rhodium-catalyzed formation of isomunchones. Acs Combinatorial Science. 15: 340-3. PMID 23742807 DOI: 10.1021/Co400067Q |
0.572 |
|
2013 |
Anastasio NC, Gilbertson SR, Bubar MJ, Agarkov A, Stutz SJ, Jeng Y, Bremer NM, Smith TD, Fox RG, Swinford SE, Seitz PK, Charendoff MN, Craft JW, Laezza FM, Watson CS, et al. Peptide inhibitors disrupt the serotonin 5-HT2C receptor interaction with phosphatase and tensin homolog to allosterically modulate cellular signaling and behavior. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 33: 1615-30. PMID 23345234 DOI: 10.1523/Jneurosci.2656-12.2013 |
0.744 |
|
2012 |
Gilbertson SR. Chemistry. Relay reactions that trap organometallic intermediates. Science (New York, N.Y.). 338: 1432-3. PMID 23239726 DOI: 10.1126/Science.1231509 |
0.386 |
|
2012 |
Chen D, Ma L, Kanalas JJ, Gao J, Pawlik J, Jimenez ME, Walter MA, Peterson JW, Gilbertson SR, Schein CH. Structure-based redesign of an edema toxin inhibitor. Bioorganic & Medicinal Chemistry. 20: 368-76. PMID 22154558 DOI: 10.1016/J.Bmc.2011.10.091 |
0.319 |
|
2011 |
Khalaf J, Estrella-Jimenez ME, Shashack MJ, Phatak SS, Zhang S, Gilbertson SR. Design, synthesis, and diversification of 3,5-substituted enone library. Acs Combinatorial Science. 13: 351-6. PMID 21648460 DOI: 10.1021/Co200070M |
0.46 |
|
2010 |
Prasad BA, Buechele AE, Gilbertson SR. Pd-NHC catalyzed cyclopentannulation of diazabicyclic alkenes with ortho-aryl halides. Organic Letters. 12: 5422-5. PMID 21043477 DOI: 10.1021/Ol102270R |
0.346 |
|
2010 |
Tanifum EA, Gilbertson SR. Design, synthesis, and diversification of 5,5-dimethyl cyclohexen-1,4-dione library. Journal of Combinatorial Chemistry. 12: 318-20. PMID 20387791 DOI: 10.1021/Cc100030H |
0.455 |
|
2009 |
Prasad BA, Gilbertson SR. One-pot synthesis of unsymmetrical N-heterocyclic carbene ligands from N-(2-iodoethyl)arylamine salts. Organic Letters. 11: 3710-3. PMID 19624103 DOI: 10.1021/Ol901189M |
0.402 |
|
2009 |
Tanifum EA, Kots AY, Choi BK, Murad F, Gilbertson SR. Novel pyridopyrimidine derivatives as inhibitors of stable toxin a (STa) induced cGMP synthesis. Bioorganic & Medicinal Chemistry Letters. 19: 3067-71. PMID 19409779 DOI: 10.1016/J.Bmcl.2009.04.024 |
0.374 |
|
2008 |
Agarkov A, Gilbertson SR. Preparation of a library of unsymmetrical ureas based on 8-azabicyclo[3.2.1]octane scaffold. Journal of Combinatorial Chemistry. 10: 655-7. PMID 18611055 DOI: 10.1021/Cc800068K |
0.794 |
|
2008 |
Jimenez ME, Bush K, Pawlik J, Sower L, Peterson JW, Gilbertson SR. Synthesis and screening of small molecule inhibitors of anthrax edema factor. Bioorganic & Medicinal Chemistry Letters. 18: 4215-8. PMID 18539457 DOI: 10.1016/J.Bmcl.2008.05.059 |
0.36 |
|
2008 |
Drew ME, Banerjee R, Uffman EW, Gilbertson S, Rosenthal PJ, Goldberg DE. Plasmodium food vacuole plasmepsins are activated by falcipains. The Journal of Biological Chemistry. 283: 12870-6. PMID 18308731 DOI: 10.1074/Jbc.M708949200 |
0.751 |
|
2008 |
Agarkov A, Chauhan S, Lory PJ, Gilbertson SR, Motin VL. Substrate specificity and screening of the integral membrane protease Pla. Bioorganic & Medicinal Chemistry Letters. 18: 427-31. PMID 17981463 DOI: 10.1016/J.Bmcl.2007.09.104 |
0.773 |
|
2007 |
Lory PM, Estrella-Jimenez ME, Shashack MJ, Lokesh GL, Natarajan A, Gilbertson SR. Synthesis and screening of 3-substituted thioxanthen-9-one-10,10-dioxides. Bioorganic & Medicinal Chemistry Letters. 17: 5940-3. PMID 17826998 DOI: 10.1016/J.Bmcl.2007.07.103 |
0.359 |
|
2007 |
DeBoef B, Counts WR, Gilbertson SR. Rhodium-catalyzed synthesis of eight-membered rings. The Journal of Organic Chemistry. 72: 799-804. PMID 17253798 DOI: 10.1021/Jo0620462 |
0.772 |
|
2006 |
Agarkov A, Greenfield S, Xie D, Pawlick R, Starkey G, Gilbertson SR. Synthesis of phosphine containing amino acids: utilization of peptide synthesis in ligand design. Biopolymers. 84: 48-73. PMID 16235230 DOI: 10.1002/Bip.20395 |
0.776 |
|
2006 |
Lory PMJ, Agarkov A, Gilbertson SR. An expedient route to 3-chlorothioxanthen-9-one-10,10-dioxide and derivation by palladium-catalyzed coupling Synlett. 3045-3048. DOI: 10.1055/S-2006-951520 |
0.796 |
|
2005 |
Xu G, Gilbertson SR. Development of building blocks for the synthesis of N-heterocyclic carbene ligands. Organic Letters. 7: 4605-8. PMID 16209490 DOI: 10.1021/Ol0516521 |
0.525 |
|
2005 |
Agarkov A, Gilbertson SR. Coordination mode for turn-based phosphine ligands: The origin of selectivity in Pd catalysis Tetrahedron Letters. 46: 181-183. DOI: 10.1016/J.Tetlet.2004.10.096 |
0.809 |
|
2004 |
Agarkov A, Greenfield SJ, Ohishi T, Collibee SE, Gilbertson SR. Catalysis with phosphine-containing amino acids in various "turn" motifs. The Journal of Organic Chemistry. 69: 8077-85. PMID 15527293 DOI: 10.1021/Jo049103G |
0.773 |
|
2004 |
Gilbertson SR, Yamada S. A study of catalyst selectivity with polymer bound palladium phosphine complexes on various solid phase synthesis supports Tetrahedron Letters. 45: 3917-3920. DOI: 10.1016/J.Tetlet.2004.03.110 |
0.447 |
|
2003 |
Greenfield SJ, Agarkov A, Gilbertson SR. High asymmetric induction with beta-turn-derived palladium phosphine complexes. Organic Letters. 5: 3069-72. PMID 12916983 DOI: 10.1021/Ol035097J |
0.794 |
|
2003 |
Agarkov A, Uffman EW, Gilbertson SR. Parallel approach to selective catalysts for palladium-catalyzed desymmetrization of 2,4-cyclopentenediol. Organic Letters. 5: 2091-4. PMID 12790536 DOI: 10.1021/Ol034548X |
0.773 |
|
2003 |
Xu G, Gilbertson SR. Asymmetric hydrogenation of aromatic olefins catalyzed by iridium complexes of proline derived phosphine-oxazoline ligands Tetrahedron Letters. 44: 953-955. DOI: 10.1016/S0040-4039(02)02747-8 |
0.458 |
|
2003 |
DeBoef B, Gilbertson SR. C-C bond formation via C-H bond activation: Synthesis of the core of teleocidin B4 Chemtracts. 16: 249-253. |
0.628 |
|
2002 |
Gilbertson SR, DeBoef B. Rhodium catalyzed [4 + 2 + 2] cycloaddition and alkyne insertion: a new route to eight-membered rings. Journal of the American Chemical Society. 124: 8784-5. PMID 12137517 DOI: 10.1021/Ja026536X |
0.732 |
|
2002 |
Gilbertson SR, Lan P. Solid-phase synthesis of phosphine-oxazoline peptides Tetrahedron Letters. 43: 6961-6965. DOI: 10.1016/S0040-4039(02)01596-4 |
0.605 |
|
2002 |
Xu G, Gilbertson SR. Facile synthesis of proline based phosphine-oxazoline ligands by formation of a P-N bond Tetrahedron Letters. 43: 2811-2814. DOI: 10.1016/S0040-4039(02)00346-5 |
0.437 |
|
2002 |
Uffman EW, Gilbertson SR. A novel peptide-based encoding system for "one-bead one-compound" peptidomimetic and small molecule combinatorial libraries Chemtracts. 15: 606-610. |
0.774 |
|
2001 |
Gilbertson SR, Xie D, Fu Z. Proline-based P, N ligands in asymmetric allylation and the Heck reaction. The Journal of Organic Chemistry. 66: 7240-6. PMID 11681933 DOI: 10.1021/Jo0158231 |
0.469 |
|
2001 |
Gilbertson SR, Lan P. Kinetic resolution in palladium-catalyzed asymmetric allylic alkylations by a P,O ligand system. Organic Letters. 3: 2237-40. PMID 11440588 DOI: 10.1021/Ol0161256 |
0.576 |
|
2001 |
Gilbertson SR, Fu Z. Chiral P,N-ligands based on ketopinic acid in the asymmetric Heck reaction. Organic Letters. 3: 161-4. PMID 11430024 DOI: 10.1021/Ol006747B |
0.497 |
|
2001 |
Greenfield SJ, Gilbertson SR. Preparation of diphenylphosphinoserine and synthesis of other phosphine containing amino acids using zinc/copper reagents Synthesis. 2337-2340. DOI: 10.1055/S-2001-18431 |
0.8 |
|
2001 |
Gilbertson SR, Fu Z, Xie D. Proline derived phosphine-oxazoline ligands in the asymmetric Heck reaction Tetrahedron Letters. 42: 365-368. DOI: 10.1016/S0040-4039(00)01938-9 |
0.47 |
|
2000 |
Gilbertson SR, Genov DG, Rheingold AL. Synthesis of new bicyclic P-N ligands and their application in asymmetric Pd-catalyzed pi-allyl alkylation and Heck reaction. Organic Letters. 2: 2885-8. PMID 10964390 DOI: 10.1021/Ol006323H |
0.688 |
|
2000 |
Gilbertson SR, Collibee SE, Agarkov A. Asymmetric catalysis with libraries of palladium β-turn phosphine complexes [18] Journal of the American Chemical Society. 122: 6522-6523. DOI: 10.1021/Ja992306F |
0.773 |
|
1999 |
Gilbertson SR, Lopez OD. Kinetic Resolution of Diiron Acyl Complexes-An Approach to Asymmetric Bicyclic β-Lactams. Angewandte Chemie (International Ed. in English). 38: 1116-9. PMID 25138514 DOI: 10.1002/(Sici)1521-3773(19990419)38:8<1116::Aid-Anie1116>3.0.Co;2-M |
0.429 |
|
1999 |
Gilbertson SR, Xie D. Proline-Based P,N Ligands in Palladium-Catalyzed Asymmetric pi-Allyl Additions. Angewandte Chemie (International Ed. in English). 38: 2750-2752. PMID 10508370 DOI: 10.1002/(Sici)1521-3773(19990917)38:18<2750::Aid-Anie2750>3.0.Co;2-5 |
0.414 |
|
1999 |
Gilbertson SR, Fu Z, Starkey GW. Palladium-catalyzed synthesis of vinyl phosphines from ketones Tetrahedron Letters. 40: 8509-8512. DOI: 10.1016/S0040-4039(99)01819-5 |
0.786 |
|
1999 |
Gilbertson SR, Wang X. The parallel synthesis of peptide based phosphine ligands Tetrahedron. 55: 11609-11618. DOI: 10.1016/S0040-4020(99)00682-1 |
0.488 |
|
1998 |
Gilbertson SR, Hoge GS, Genov DG. Rhodium-catalyzed asymmetric [4 + 2] cycloisomerization reactions Journal of Organic Chemistry. 63: 10077-10080. DOI: 10.1021/Jo981870Q |
0.646 |
|
1998 |
Gilbertson SR, Chang CWT. Synthesis of phosphino oxazoline ligand libraries from amino acid and phosphino carboxylate building blocks Journal of Organic Chemistry. 63: 8424-8431. DOI: 10.1021/Jo981420Y |
0.485 |
|
1998 |
Gilbertson SR, Hoge GS. Rhodium catalyzed intramolecular [4+2] cycloisomerization reactions Tetrahedron Letters. 39: 2075-2078. DOI: 10.1016/S0040-4039(98)00265-2 |
0.407 |
|
1997 |
Gilbertson SR, Chang CWT. A modular approach to ligands for asymmetric π-allyl palladium catalysed additions Chemical Communications. 975-976. DOI: 10.1039/A607200C |
0.475 |
|
1997 |
Gilbertson SR, Chen G, Kao J, Beatty A, Campana CF. Structure of Phosphorus-Containing Peptide Ligands. X-ray and NMR Structural Study of Free Ligand and Rhodium Complex Journal of Organic Chemistry. 62: 5557-5566. DOI: 10.1021/Jo970773E |
0.374 |
|
1997 |
Gilbertson SR, Lopez OD. Synthesis of and asymmetric cycloaddition with chiral diiron acyl complexes Journal of the American Chemical Society. 119: 3399-3400. DOI: 10.1021/Ja964195F |
0.426 |
|
1996 |
Gilbertson SR, Starkey GW. Palladium-Catalyzed Synthesis of Phosphine-Containing Amino Acids. The Journal of Organic Chemistry. 61: 2922-2923. PMID 11667143 DOI: 10.1021/Jo960077Z |
0.773 |
|
1996 |
Gilbertson SR, Wang X. Synthesis of (Dicyclohexylphosphino)serine, Its Incorporation into a Dodecapeptide, and the Coordination of Rhodium. The Journal of Organic Chemistry. 61: 434-435. PMID 11666953 DOI: 10.1021/Jo951327Z |
0.429 |
|
1996 |
Klug CA, Studelska DR, Chen G, Gilbertson SR, Schaefer J. Distance between phosphine-sulfide sidechains of a disubstituted peptide by DRAMA 31P NMR. Solid State Nuclear Magnetic Resonance. 7: 173-6. PMID 9050154 DOI: 10.1016/S0926-2040(96)01268-4 |
0.323 |
|
1996 |
Gilbertson SR, Wang X, Hoge GS, Klug CA, Schaefer J. Synthesis of phosphine-rhodium complexes attached to a standard peptide synthesis resin Organometallics. 15: 4678-4680. DOI: 10.1021/Om9606000 |
0.452 |
|
1996 |
Gilbertson SR, Wang X. The combinatorial synthesis of chiral phosphine ligands Tetrahedron Letters. 37: 6475-6478. DOI: 10.1016/0040-4039(96)01424-4 |
0.498 |
|
1996 |
Gilbertson SR, Pawlick RV. Synthesis of Thiophosphoryl Derivatives of Proline: Building Blocks for Phosphanyl-Substituted Peptides with β-Turns Angewandte Chemie (International Edition in English). 35: 902-904. DOI: 10.1002/Anie.199609021 |
0.728 |
|
1996 |
Gilbertson SR, Pawlick RV. Synthese von Thiophosphorylprolinen als Bausteine für phosphanylsubstituierte Peptide mit β-Turns† Angewandte Chemie. 108: 963-966. DOI: 10.1002/Ange.19961080819 |
0.314 |
|
1996 |
Gilbertson SR, Wang X. Synthesis of (dicyclohexylphosphino) serine, its incorporation into a dodecapeptide, and the coordination of rhodium Journal of Organic Chemistry. 61: 434-435. |
0.317 |
|
1995 |
Gilbertson SR, Chang CWT. Synthesis of new disugar phosphine ligands and their use in asymmetric hydrogenation Journal of Organic Chemistry. 60: 6226-6228. DOI: 10.1021/Jo00124A051 |
0.404 |
|
1995 |
Gilbertson SR, Dawson DP, Lopez OD, Marshall KL. Endo-Selective Reactions of .alpha.,.beta.-Unsaturated Hexacarbonyldiiron Bridging Acyl Complexes with Nitrones Journal of the American Chemical Society. 117: 4431-4432. DOI: 10.1021/Ja00120A039 |
0.319 |
|
1995 |
Gilbertson SR, Pawlick RV. The synthesis and conformation of dihydroxy-cyclo(d-Pro-l-Pro-d-Pro-l-Pro) Tetrahedron Letters. 36: 1229-1232. DOI: 10.1016/0040-4039(95)00022-5 |
0.68 |
|
1995 |
Gilbertson SR, Dawson DP, Lopez OD, Marshall KL. Endo-selective reactions of α,β-unsaturated hexacarbonyldiiron bridging acyl complexes with nitrones Journal of the American Chemical Society. 117: 4431-4432. |
0.629 |
|
1994 |
Gilbertson SR, Chen G, McLoughlin M. Versatile building block for the synthesis of phosphine-containing peptides: The sulfide of diphenylphosphinoserine Journal of the American Chemical Society. 116: 4481-4482. DOI: 10.1021/Ja00089A049 |
0.714 |
|
1993 |
Gilbertson SR, Zhao X, Dawson DP, Marshall KL. Exo-Selective Diels-Alder reactions of .alpha.,.beta.-unsaturated hexacarbonyl-diiron bridging acyl complexes Journal of the American Chemical Society. 115: 8517-8518. DOI: 10.1021/Ja00071A099 |
0.325 |
|
1993 |
Gilbertson SR, Zhao X, Dawson DP, Marshall KL. Exo-selective Diels-Alder reactions of α,β-unsaturated hexacarbonyl-diiron bridging acyl complexes Journal of the American Chemical Society. 115: 8517-8518. |
0.632 |
|
1989 |
Gilbertson SR, Wulff WD. Evaluation of the Cyclohexadienone Annulation of Chromium-Carbene Complexes for the Synthesis of Taxodione Synlett. 1989: 47-49. DOI: 10.1055/S-1989-34694 |
0.59 |
|
1988 |
Stuart McCallum J, Kunng FA, Gilbertson SR, Wulff WD. Mechanistic studies on the reaction of chromium carbene complexes with acetylenes: Furan formation and the dependence of the product distribution on the stereochemistry of reaction intermediates Organometallics. 7: 2346-2360. DOI: 10.1021/Om00101A015 |
0.575 |
|
1988 |
Gilbertson SR, Challener CA, Bos ME, Wulff WD. An examination of the coupling of vinyl and aryl triflates with stannyl cuprates for the purpose of providing regioselective access to vinyl lithiums Tetrahedron Letters. 29: 4795-4798. DOI: 10.1016/S0040-4039(00)80611-5 |
0.603 |
|
1986 |
Wulff WD, Gilbertson SR, Springer JP. Reactions of cobalt carbene complexes with alkynes. .eta.4-Vinylketene-complexed intermediates and a novel synthesis of bovolide. Journal of the American Chemical Society. 108: 520-2. PMID 22175480 DOI: 10.1021/Ja00263A035 |
0.619 |
|
1986 |
Wulff WD, Peterson GA, Bauta WE, Chan KS, Faron KL, Gilbertson SR, Kaesler RW, Yang DC, Murray CK. A regioselective entry to vinyllithiums from unsymmetrical ketones via enol triflates Journal of Organic Chemistry. 51: 277-279. DOI: 10.1002/Chin.198627244 |
0.794 |
|
1986 |
Wulff WD, Gilbertson SR, Springer JP. Reactions of cobalt carbene complexes with alkynes - η4-vinylketene complex intermediates and a novel synthesis of bovolide Journal of the American Chemical Society. 108: 520-522. DOI: 10.1002/Chin.198623282 |
0.619 |
|
1985 |
Wulff WD, Tang PC, Chan KS, McCallum JS, Yang DC, Gilbertson SR. Cycloadditions and annulations of transition metal carbene complexes Tetrahedron. 41: 5813-5832. DOI: 10.1016/S0040-4020(01)91421-8 |
0.64 |
|
1985 |
Wulff WD, Gilbertson SR. Aldol reactions of transition-metal carbene complexes Journal of the American Chemical Society. 107: 503-505. DOI: 10.1002/Chin.198521124 |
0.558 |
|
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