Joel Bockaert - Related publications

Affiliations: 
Centre CNRS INSERM Pharmacology & Endocrinology University of Montpellier, France, Montpellier, Occitanie, France 
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50 most relevant papers in past 60 days:
Year Citation  Score
2020 Glaser T, Andrejew R, Oliveira-Giacomelli Á, Ribeiro DE, Bonfim Marques L, Ye Q, Ren WJ, Semyanov A, Illes P, Tang Y, Ulrich H. Purinergic Receptors in Basal Ganglia Diseases: Shared Molecular Mechanisms between Huntington's and Parkinson's Disease. Neuroscience Bulletin. PMID 33026587 DOI: 10.1007/s12264-020-00582-8   
2020 Shin D, Cho KH, Joo K, Rhie DJ. Layer-specific serotonergic induction of long-term depression in the prefrontal cortex of rats. The Korean Journal of Physiology & Pharmacology : Official Journal of the Korean Physiological Society and the Korean Society of Pharmacology. 24: 517-527. PMID 33093273 DOI: 10.4196/kjpp.2020.24.6.517   
2020 Rodriguez Araujo N, Fabiani C, Mazzarini Dimarco A, Bouzat C, Corradi J. Orthosteric and Allosteric Activation of Human 5-HTA Receptors. Biophysical Journal. PMID 32946769 DOI: 10.1016/j.bpj.2020.08.029   
2020 Abad IPL, Fam RL, Nguyen DT, Nowell CJ, Trinh PNH, Manallack DT, Freihat LA, Chakrabarti J, Jamil A, Exintaris B, Yaakob NS, Irving HR. Visualising functional 5-HT receptors containing A and C subunits at or near the cell surface. Biomedicine & Pharmacotherapy = Biomedecine & Pharmacotherapie. 132: 110860. PMID 33059258 DOI: 10.1016/j.biopha.2020.110860   
2020 Nebrisi EE, Prytkova T, Lorke DE, Howarth L, Alzaabi AH, Yang KS, Howarth FC, Oz M. Capsaicin Is a Negative Allosteric Modulator of the 5-HT Receptor. Frontiers in Pharmacology. 11: 1274. PMID 32982728 DOI: 10.3389/fphar.2020.01274   
2020 Belliveau S, Kang W, Bovaird S, Hamadjida A, Bédard D, Dancause N, Stroh T, Huot P. Stereological investigation of 5-HT receptors in the substantia nigra and dorsal raphe nucleus in the rat. Journal of Chemical Neuroanatomy. 101881. PMID 33160048 DOI: 10.1016/j.jchemneu.2020.101881   
2020 Seitz BM, Fink GD, Watts SW. Activation of the 5-HT receptor but not nitric oxide synthase is necessary for chronic 5-hydroxytryptamine-induced hypotension. Experimental Physiology. PMID 33052620 DOI: 10.1113/EP088919   
2020 Symeonidis D, Lazaris A, Zizi Zerbetzoglou A, Christodoulou P, Kavantzas N, Tsavaris N, Thomopoulou GE. Correlation between LGR5 stem cells and location of tumor as well as age, sex and metastasis in colon adenocarcinoma. Journal of B.U.On. : Official Journal of the Balkan Union of Oncology. 25: 1827-1831. PMID 33099920   
2020 Watabe M, Yoshimura H, Arjunan SNV, Kaizu K, Takahashi K. Signaling activations through G-protein-coupled-receptor aggregations. Physical Review. E. 102: 032413. PMID 33076007 DOI: 10.1103/PhysRevE.102.032413   
2020 Chen H, Wang F, Ni X, Rigui Y, Bai Y, Xu L, Yang J, Zhang X, Deng J, Li J, Yin X, Ao W, Kwok KWH, Dong W. Aconitine disrupts serotonin neurotransmission via 5-hydroxytryptamine receptor in zebrafish embryo. Journal of Applied Toxicology : Jat. PMID 33085127 DOI: 10.1002/jat.4059   
2020 Ye N, Qin W, Tian S, Xu Q, Wold EA, Zhou J, Zhen XC. Small Molecules Selectively Targeting Sigma-1 Receptor for the Treatment of Neurological Diseases. Journal of Medicinal Chemistry. PMID 33111525 DOI: 10.1021/acs.jmedchem.0c01192   
2020 Kim JH, Marton J, Ametamey SM, Cumming P. A Review of Molecular Imaging of Glutamate Receptors. Molecules (Basel, Switzerland). 25. PMID 33081223 DOI: 10.3390/molecules25204749   
2020 Pollok S, Reiner A. Subunit-selective iGluR antagonists can potentiate heteromeric receptor responses by blocking desensitization. Proceedings of the National Academy of Sciences of the United States of America. 117: 25851-25858. PMID 32999066 DOI: 10.1073/pnas.2007471117   
2020 Ramesh S, Park S, Call MJ, Im W, Call ME. Experimentally Guided Computational Methods Yield Highly Accurate Insights into Transmembrane Interactions within the T Cell Receptor Complex. The Journal of Physical Chemistry. B. PMID 33030343 DOI: 10.1021/acs.jpcb.0c06403   
2020 Pandey S, Saha S, Shukla AK. Transmitting the Signal: Structure of the β1-Adrenergic Receptor-Gs Protein Complex. Molecular Cell. 80: 3-5. PMID 33007256 DOI: 10.1016/j.molcel.2020.09.016   
2020 Pandey S, Saha S, Shukla AK. Transmitting the Signal: Structure of the β1-Adrenergic Receptor-Gs Protein Complex. Molecular Cell. 80: 3-5. PMID 33007256 DOI: 10.1016/j.molcel.2020.09.016   
2020 Kurtz R, Steinberg LG, Betcher M, Fowler D, Shepard BD. The Sensing Liver: Localization and Ligands for Hepatic Murine Olfactory and Taste Receptors. Frontiers in Physiology. 11: 574082. PMID 33123030 DOI: 10.3389/fphys.2020.574082   
2020 Jin Y, Qiu CY, Wei S, Han L, Liu TT, Hu WP. Potentiation of P2X3 receptor mediated currents by endothelin-1 in rat dorsal root ganglion neurons. Neuropharmacology. 108356. PMID 33069757 DOI: 10.1016/j.neuropharm.2020.108356   
2020 Navarro G, Gonzalez A, Campanacci S, Rivas-Santisteban R, Reyes-Resina I, Casajuana-Martin N, Cordomí A, Pardo L, Franco R. Experimental and computational analysis of biased agonism on full-length and a C-terminally truncated adenosine A receptor. Computational and Structural Biotechnology Journal. 18: 2723-2732. PMID 33101610 DOI: 10.1016/j.csbj.2020.09.028   
2020 Liu YP, Wu X, Meng JH, Yao J, Wang BJ. Functional Analysis of the 3' Untranslated Region of the Human Gene in Regulating Gene Expression in vitro. Neuropsychiatric Disease and Treatment. 16: 2361-2370. PMID 33116535 DOI: 10.2147/NDT.S268753   
2020 Yang LK, Tao YX. Alanine Scanning Mutagenesis of the DRYxxI Motif and Intracellular Loop 2 of Human Melanocortin-4 Receptor. International Journal of Molecular Sciences. 21. PMID 33076233 DOI: 10.3390/ijms21207611   
2020 Dasgupta P, Günther T, Reinscheid RK, Zaveri NT, Schulz S. Rapid assessment of G protein signaling of four opioid receptors using a real-time fluorescence-based membrane potential assay. European Journal of Pharmacology. 173640. PMID 33045198 DOI: 10.1016/j.ejphar.2020.173640   
2020 Dasgupta P, Günther T, Reinscheid RK, Zaveri NT, Schulz S. Rapid assessment of G protein signaling of four opioid receptors using a real-time fluorescence-based membrane potential assay. European Journal of Pharmacology. 173640. PMID 33045198 DOI: 10.1016/j.ejphar.2020.173640   
2020 Cheng Q, Feng X, Meng Q, Li Y, Chen S, Wang G, Nie K. [6]-Gingerol Ameliorates Cisplatin-Induced Pica by Regulating the TPH/MAO-A/SERT/5-HT/5-HT Receptor System in Rats. Drug Design, Development and Therapy. 14: 4085-4099. PMID 33061309 DOI: 10.2147/DDDT.S270185   
2020 Leung SW. The vascular impact of IP-TP receptor interactions. Acta Physiologica (Oxford, England). e13577. PMID 33135294 DOI: 10.1111/apha.13577   
2020 Zhu C, Li X, Peng W, Fu W. Discovery of Novel Indolealkylpiperazine Derivatives as Potent 5-HT Receptor Agonists for the Potential Future Treatment of Depression. Molecules (Basel, Switzerland). 25. PMID 33139658 DOI: 10.3390/molecules25215078   
2020 Devenish SO, Winters BL, Anderson LL, Arnold JC, McGregor IS, Vaughan CW, Chebib M, Absalom NL. The anticonvulsant zonisamide positively modulates recombinant and native glycine receptors at clinically relevant concentrations. Neuropharmacology. 108371. PMID 33122032 DOI: 10.1016/j.neuropharm.2020.108371   
2020 Haruta-Tsukamoto A, Miyahara Y, Funahashi H, Nishimori T, Ishida Y. Perampanel attenuates scratching behavior induced by acute or chronic pruritus in mice. Biochemical and Biophysical Research Communications. PMID 33028486 DOI: 10.1016/j.bbrc.2020.09.109   
2020 Pieterse L, van der Walt MM, Terre'Blanche G. C2-substituted quinazolinone derivatives exhibit A and/or A adenosine receptor affinities in the low micromolar range. Bioorganic & Medicinal Chemistry Letters. 30: 127274. PMID 32631506 DOI: 10.1016/j.bmcl.2020.127274   
2020 Williams CA, Miller KE, Williams NP, Portfors CV, Perkel DJ. Distribution and co-expression of adrenergic receptor-encoding mRNA in the mouse inferior colliculus. The Journal of Comparative Neurology. PMID 33067825 DOI: 10.1002/cne.25053   
2020 Touma AM, Malik RU, Gupte T, Sivaramakrishnan S. Allosteric modulation of adenosine A1 and cannabinoid 1 receptor signaling by G-peptides. Pharmacology Research & Perspectives. 8: e00673. PMID 33124765 DOI: 10.1002/prp2.673   
2020 Li M, Huang C, Wu X, Ding F, Hu Z, Zhu Y, Zhao L, Hou L, Chen H, Wang H, Xu J, Tang D. The optimization of a novel selective antagonist for human M muscarinic acetylcholine receptor. Bioorganic & Medicinal Chemistry Letters. 30: 127632. PMID 33132116 DOI: 10.1016/j.bmcl.2020.127632   
2020 Di Giovanni G, De Deurwaerdère P. Serotonin research: Crossing scales and boundaries. Neuropharmacology. 181: 108340. PMID 33007358 DOI: 10.1016/j.neuropharm.2020.108340   
2020 Toneatti R, Shin JM, Shah UH, Mayer CR, Saunders JM, Fribourg M, Arsenovic PT, Janssen WG, Sealfon SC, López-Giménez JF, Benson DL, Conway DE, González-Maeso J. Interclass GPCR heteromerization affects localization and trafficking. Science Signaling. 13. PMID 33082287 DOI: 10.1126/scisignal.aaw3122   
2020 Reeh K, Summers PA, Gould IR, Woscholski R, Vilar R. Design, synthesis and evaluation of a tripodal receptor for phosphatidylinositol phosphates. Scientific Reports. 10: 18450. PMID 33116198 DOI: 10.1038/s41598-020-75484-w   
2020 Fernandes RA, Su L, Nishiga Y, Ren J, Bhuiyan AM, Cheng N, Kuo CJ, Picton LK, Ohtsuki S, Majzner RG, Rietberg SP, Mackall CL, Yin Q, Ali LR, Yang X, et al. Immune receptor inhibition through enforced phosphatase recruitment. Nature. PMID 33087934 DOI: 10.1038/s41586-020-2851-2   
2020 Jakubík J, Randáková A, Chetverikov N, El-Fakahany EE, Doležal V. The operational model of allosteric modulation of pharmacological agonism. Scientific Reports. 10: 14421. PMID 32879329 DOI: 10.1038/s41598-020-71228-y   
2020 Rajan R, Schepmann D, Schreiber JA, Seebohm G, Wünsch B. Synthesis of GluN2A-selective NMDA receptor antagonists with an electron-rich aromatic B-ring. European Journal of Medicinal Chemistry. 112939. PMID 33162207 DOI: 10.1016/j.ejmech.2020.112939   
2020 Calderón-Zamora L, Canizalez-Román A, León-Sicairos N, Aguilera-Mendez A, Huang F, Hong E, Villafaña S. Changes in expression of orphan receptors GPR99 and GPR107 during the development and establishment of hypertension in spontaneously hypertensive rats. Journal of Receptor and Signal Transduction Research. 1-8. PMID 33121311 DOI: 10.1080/10799893.2020.1835959   
2020 Jones EM, Lubock NB, Venkatakrishnan AJ, Wang J, Tseng AM, Paggi JM, Latorraca NR, Cancilla D, Satyadi M, Davis JE, Babu MM, Dror RO, Kosuri S. Structural and functional characterization of G protein-coupled receptors with deep mutational scanning. Elife. 9. PMID 33084570 DOI: 10.7554/eLife.54895   
2020 Béchade C, D'Andrea I, Etienne F, Verdonk F, Moutkine I, Banas SM, Kolodziejczak M, Diaz SL, Parkhurst CN, Gan WB, Maroteaux L, Roumier A. The serotonin 2B receptor is required in neonatal microglia to limit neuroinflammation and sickness behavior in adulthood. Glia. PMID 33095507 DOI: 10.1002/glia.23918   
2020 Yeliseev A, van den Berg A, Zoubak L, Hines K, Stepnowski S, Williston K, Yan W, Gawrisch K, Zmuda J. Thermostability of a recombinant G protein-coupled receptor expressed at high level in mammalian cell culture. Scientific Reports. 10: 16805. PMID 33033368 DOI: 10.1038/s41598-020-73813-7   
2020 Holze J, Bermudez M, Pfeil EM, Kauk M, Bödefeld T, Irmen M, Matera C, Dallanoce C, De Amici M, Holzgrabe U, König GM, Tränkle C, Wolber G, Schrage R, Mohr K, et al. Ligand-Specific Allosteric Coupling Controls G-Protein-Coupled Receptor Signaling. Acs Pharmacology & Translational Science. 3: 859-867. PMID 33073186 DOI: 10.1021/acsptsci.0c00069   
2020 Kukkonen JP. Allosteric interactions via the orthosteric ligand binding sites in a constitutive G-protein-coupled receptor homodimer. Pharmacological Research. 105116. PMID 32783977 DOI: 10.1016/j.phrs.2020.105116   
2020 Lyons EL, Leone-Kabler S, Kovach AL, Thomas BF, Howlett AC. Cannabinoid receptor subtype influence on neuritogenesis in human SH-SY5Y cells. Molecular and Cellular Neurosciences. 103566. PMID 33049367 DOI: 10.1016/j.mcn.2020.103566   
2020 Gao N, Tiliwaerde M, Zheng W, Xiong J, Li XR, Jin Z. Neuropharmacological and antidepressant-like effects of ZY-1408: A novel serotonin/norepinephrine reuptake inhibitor and serotonin receptor 2C antagonist. Neuropharmacology. 108376. PMID 33122031 DOI: 10.1016/j.neuropharm.2020.108376   
2020 Chen J, Cai X, Yan M, Wang Z, Lv Z, Wang C. A method for identifying G protein-coupled receptor dimers and their interfaces. Biochimica Et Biophysica Acta. Molecular Cell Research. 118887. PMID 33075383 DOI: 10.1016/j.bbamcr.2020.118887   
2020 Paudel P, Shrestha S, Park SE, Seong SH, Fauzi FM, Jung HA, Choi JS. Emodin Derivatives as Multi-Target-Directed Ligands Inhibiting Monoamine Oxidase and Antagonizing Vasopressin V Receptors. Acs Omega. 5: 26720-26731. PMID 33110998 DOI: 10.1021/acsomega.0c03649   
2020 Velard F, Chatron-Colliet A, Côme D, Ah-Kioon MD, Lin H, Hafsia N, Cohen-Solal M, Ea HK, Lioté F. Adrenomedullin and truncated peptide adrenomedullin(22-52) affect chondrocyte response to apoptotis in vitro: downregulation of FAS protects chondrocyte from cell death. Scientific Reports. 10: 16740. PMID 33028903 DOI: 10.1038/s41598-020-73924-1   
2020 King BF. Burnstock and the legacy of the inhibitory junction potential and P2Y1 receptors. Purinergic Signalling. PMID 33125617 DOI: 10.1007/s11302-020-09747-6