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Jon C. Antilla, Ph.D. - Publications

Affiliations: 
Chemistry Department University of South Florida, Tampa, FL, United States 
Area:
Organic Chemistry, Chiral Organocatalysis, Metal-Catalysis, New Stereoselective Reaction Methodology, Drug Discovery
Website:
http://chemistry.usf.edu/faculty/antilla/
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72 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 He H, Shen X, Ding X, Antilla JC. Enantioselective Mukaiyama-Michael Reaction of β,γ-Unsaturated α-Keto Esters with Silyl Ketene Acetals Catalyzed by a Chiral Magnesium Phosphate. Organic Letters. 25: 782-787. PMID 36700837 DOI: 10.1021/acs.orglett.2c04277  0.483
2022 He H, Tummalapalli KSS, Zhu L, Chen M, Krishnamurthy S, Antilla JC. Asymmetric Rubottom-type Oxidation Catalyzed by Chiral Calcium Phosphates. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 36541518 DOI: 10.1002/chem.202203720  0.406
2022 Wu Z, He H, Chen M, Zhu L, Zheng W, Cao Y, Antilla JC. Asymmetric Reductive Amination with Pinacolborane Catalyzed by Chiral SPINOL Borophosphates. Organic Letters. 24: 9436-9441. PMID 36519791 DOI: 10.1021/acs.orglett.2c03866  0.606
2022 Yuan J, Jain P, Antilla JC. Chiral Phosphoric Acid-Catalyzed Enantio- and Diastereoselective Allylboration of Aldehydes with β,γ-Substituted Allylboronates. The Journal of Organic Chemistry. 87: 8256-8266. PMID 35657081 DOI: 10.1021/acs.joc.2c00764  0.685
2022 Wu Z, Krishnamurthy S, Tummalapalli KSS, Antilla JC. Chiral Calcium Phosphate-Catalyzed Enantioselective Amination of 3-Aryl-2-oxindoles with Dibenzyl Azodicarboxylate. The Journal of Organic Chemistry. 87: 8203-8212. PMID 35621216 DOI: 10.1021/acs.joc.2c00432  0.466
2022 Wu Z, Krishnamurthy S, Tummalapalli KSS, Xu J, Yue C, Antilla JC. Enantioselective amination of β-keto esters catalyzed by chiral calcium phosphates. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 35508801 DOI: 10.1002/chem.202200907  0.483
2022 Li HL, Yang DF, Jing HQ, Antilla JC, Kuninobu Y. Palladium-Catalyzed Enantioselective C(sp)-H Arylation of 2-Propyl Azaaryls Enabled by an Amino Acid Ligand. Organic Letters. 24: 1286-1291. PMID 35142219 DOI: 10.1021/acs.orglett.1c04215  0.428
2021 He H, Cao Y, Xu J, Antilla JC. Catalytic Asymmetric C-7 Friedel-Crafts Alkylation/-Hemiacetalization of 4-Aminoindoles. Organic Letters. PMID 33792336 DOI: 10.1021/acs.orglett.1c00699  0.546
2021 He H, Tang X, Cao Y, Antilla JC. Catalytic Asymmetric Reduction of α-Trifluoromethylated Imines with Catecholborane by BINOL-Derived Boro-phosphates. The Journal of Organic Chemistry. PMID 33586987 DOI: 10.1021/acs.joc.0c03009  0.453
2020 Liu R, Krishnamurthy S, Wu Z, Tummalapalli KSS, Antilla JC. Chiral Calcium Phosphate Catalyzed Enantioselective Amination of 3-Aryl-2-benzofuranones. Organic Letters. 22: 8101-8105. PMID 32969228 DOI: 10.1021/acs.orglett.0c03059  0.547
2020 Yuan J, Jain P, Antilla JC. Bi(cyclopentyl)diol-Derived Boronates in Highly Enantioselective Chiral Phosphoric Acid-Catalyzed Allylation, Propargylation and Crotylation of Aldehydes. The Journal of Organic Chemistry. PMID 32960066 DOI: 10.1021/Acs.Joc.0C01646  0.751
2020 Na F, Lopez SS, Beauseigneur A, Hernandez LW, Sun Z, Antilla JC. Catalytic Asymmetric Transfer Hydrogenation of -Chalcone Derivatives Using BINOL-derived Boro-phosphates. Organic Letters. PMID 32692927 DOI: 10.1021/acs.orglett.0c02042  0.428
2020 Cao R, Antilla JC. Imine Amidation Catalyzed by a Chiral VAPOL Calcium Phosphate. Organic Letters. PMID 32663015 DOI: 10.1021/acs.orglett.0c02048  0.548
2019 Tang X, He H, Fang X, Chang Z, Antilla JC. Design and synthesis of new alkyl-based chiral phosphoric acid catalysts. Chirality. PMID 31197898 DOI: 10.1002/chir.23101  0.511
2019 Bai Y, Yuan J, Hu X, Antilla JC. Catalytic Enantioselective Diels-Alder Reactions of Benzoquinones and Vinylindoles with Chiral Magnesium Phosphate Complexes. Organic Letters. PMID 31150254 DOI: 10.1021/acs.orglett.9b01437  0.56
2019 Fang X, Deng Z, Zheng W, Antilla JC. Catalytic One-Pot Double Asymmetric Cascade Reaction: Synthesis of Chlorinated Oxindoles and Geminal Diamines Acs Catalysis. 9: 1748-1752. DOI: 10.1021/acscatal.8b05019  0.544
2018 Yue C, Na F, Fang X, Yang C, Antilla J. Chiral phosphoric acid-catalyzed asymmetric synthesis of hetero-triarylmethanes from racemic indolyl alcohols. Angewandte Chemie (International Ed. in English). PMID 29968269 DOI: 10.1002/anie.201804330  0.581
2017 Nimmagadda SK, Mallojjala SC, Woztas L, Wheeler SE, Antilla JC. Enantioselective Synthesis of Chiral Oxime Ethers: Desymmetrization and Dynamic Kinetic Resolution of Substituted Cyclohexanones. Angewandte Chemie (International Ed. in English). PMID 28111889 DOI: 10.1002/Anie.201611602  0.815
2014 Fan YS, Jiang YJ, An D, Sha D, Antilla JC, Zhang S. H8-BINOL chiral imidodiphosphoric acids catalyzed enantioselective synthesis of dihydroindolo-/-pyrrolo[1,2-a]quinoxalines. Organic Letters. 16: 6112-5. PMID 25415871 DOI: 10.1021/Ol502965P  0.627
2014 Ingle G, Mormino MG, Antilla JC. Lithium BINOL phosphate catalyzed desymmetrization of meso-epoxides with aromatic thiols. Organic Letters. 16: 5548-51. PMID 25317934 DOI: 10.1021/Ol502527Q  0.737
2014 Liang T, Li G, Wojtas L, Antilla JC. Chiral metal phosphate catalysis: highly asymmetric hetero-Diels-Alder reactions. Chemical Communications (Cambridge, England). 50: 14187-90. PMID 25283964 DOI: 10.1039/C4Cc06520D  0.564
2014 Nimmagadda SK, Zhang Z, Antilla JC. Asymmetric one-pot synthesis of 1,3-oxazolidines and 1,3-oxazinanes via hemiaminal intermediates. Organic Letters. 16: 4098-101. PMID 25075467 DOI: 10.1021/Ol501789C  0.852
2013 Zhang Z, Ji YR, Wojtas L, Gao WY, Ma S, Zaworotko MJ, Antilla JC. Two homochiral organocatalytic metal organic materials with nanoscopic channels. Chemical Communications (Cambridge, England). 49: 7693-5. PMID 23884019 DOI: 10.1039/C3Cc43801E  0.369
2013 Li G, Liang T, Wojtas L, Antilla JC. An asymmetric Diels-Alder reaction catalyzed by chiral phosphate magnesium complexes: highly enantioselective synthesis of chiral spirooxindoles. Angewandte Chemie (International Ed. in English). 52: 4628-32. PMID 23519960 DOI: 10.1002/Anie.201209295  0.639
2013 Wang H, Jain P, Antilla JC, Houk KN. Origins of stereoselectivities in chiral phosphoric acid catalyzed allylborations and propargylations of aldehydes. The Journal of Organic Chemistry. 78: 1208-15. PMID 23298338 DOI: 10.1021/Jo302787M  0.641
2013 Behensky AA, Cortes-Salva M, Seminerio MJ, Matsumoto RR, Antilla JC, Cuevas J. In vitro evaluation of guanidine analogs as sigma receptor ligands for potential anti-stroke therapeutics. The Journal of Pharmacology and Experimental Therapeutics. 344: 155-66. PMID 23065135 DOI: 10.1124/Jpet.112.199513  0.743
2012 Zhang Z, Antilla JC. Enantioselective construction of pyrroloindolines catalyzed by chiral phosphoric acids: total synthesis of (-)-debromoflustramine B. Angewandte Chemie (International Ed. in English). 51: 11778-82. PMID 22987616 DOI: 10.1002/Anie.201203553  0.564
2012 Jain P, Wang H, Houk KN, Antilla JC. Brønsted acid catalyzed asymmetric propargylation of aldehydes. Angewandte Chemie (International Ed. in English). 51: 1391-4. PMID 22223476 DOI: 10.1002/Anie.201107407  0.741
2011 Zhang Z, Jain P, Antilla JC. Asymmetric reduction of ketones by phosphoric acid derived catalysts. Angewandte Chemie (International Ed. in English). 50: 10961-4. PMID 21948631 DOI: 10.1002/Anie.201103883  0.735
2011 Cui S, Wojtas L, Antilla JC. Pd-catalyzed C4-olefination of oxazoles via C-H bond activation: divergent synthesis of functionalized amino alcohol and amino acid derivatives. Organic Letters. 13: 5040-3. PMID 21861479 DOI: 10.1021/Ol201865H  0.426
2011 Ingle GK, Mormino MG, Wojtas L, Antilla JC. Chiral phosphoric acid-catalyzed addition of thiols to N-acyl imines: access to chiral N,S-acetals. Organic Letters. 13: 4822-5. PMID 21842841 DOI: 10.1021/Ol201899C  0.779
2011 He Y, Lin M, Li Z, Liang X, Li G, Antilla JC. Direct synthesis of chiral 1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazines via a catalytic asymmetric intramolecular aza-Friedel-Crafts reaction. Organic Letters. 13: 4490-3. PMID 21834569 DOI: 10.1021/Ol2018328  0.704
2011 Cui S, Wojtas L, Antilla JC. Palladium-catalyzed tunable functionalization of allylic imidates: regioselective aminodiacetoxylation and aziridination. Angewandte Chemie (International Ed. in English). 50: 8927-30. PMID 21834109 DOI: 10.1002/Anie.201103500  0.506
2011 Larson SE, Li G, Rowland GB, Junge D, Huang R, Woodcock HL, Antilla JC. Catalytic asymmetric aza-Darzens reaction with a vaulted biphenanthrol magnesium phosphate salt. Organic Letters. 13: 2188-91. PMID 21476598 DOI: 10.1021/Ol200407R  0.85
2011 Ingle GK, Liang Y, Mormino MG, Li G, Fronczek FR, Antilla JC. Chiral magnesium BINOL phosphate-catalyzed phosphination of imines: access to enantioenriched α-amino phosphine oxides. Organic Letters. 13: 2054-7. PMID 21413695 DOI: 10.1021/Ol200456Y  0.745
2011 Zheng W, Zhang Z, Kaplan MJ, Antilla JC. Chiral calcium VAPOL phosphate mediated asymmetric chlorination and Michael reactions of 3-substituted oxindoles. Journal of the American Chemical Society. 133: 3339-41. PMID 21341790 DOI: 10.1021/Ja109824X  0.599
2011 Zhang Z, Zheng W, Antilla JC. Highly enantioselective catalytic benzoyloxylation of 3-aryloxindoles using chiral VAPOL calcium phosphate. Angewandte Chemie (International Ed. in English). 50: 1135-8. PMID 21268212 DOI: 10.1002/Anie.201006595  0.569
2011 Cortes-Salva M, Garvin C, Antilla JC. Ligand-free copper-catalyzed arylation of amidines. The Journal of Organic Chemistry. 76: 1456-9. PMID 21250705 DOI: 10.1021/Jo102235U  0.824
2011 Larson SE, Li GL, Rowland GB, Junge D, Huang RC, Woodcock HL, Antilla JC. Asymmetric Aza-Darzens Reaction Catalyzed by Mg PhosphateSalt Synfacts. 2011: 862-862. DOI: 10.1055/S-0030-1260744  0.813
2011 Ingle GK, Liang Y, Mormino M, Li G, Fronczek FR, Antilla JC. Magnesium BINOL Phosphate Catalyzed Phosphination of Imines Synfacts. 2011: 735-735. DOI: 10.1055/S-0030-1260647  0.514
2010 Liang T, Zhang Z, Antilla JC. Chiral Brønsted acid catalyzed pinacol rearrangement. Angewandte Chemie (International Ed. in English). 49: 9734-6. PMID 21077074 DOI: 10.1002/Anie.201004778  0.59
2010 Jain P, Antilla JC. Chiral Brønsted acid-catalyzed allylboration of aldehydes. Journal of the American Chemical Society. 132: 11884-6. PMID 20690662 DOI: 10.1021/Ja104956S  0.762
2010 Zheng W, Wojtas L, Antilla JC. Chiral phosphoric acid catalyzed peroxidation of imines. Angewandte Chemie (International Ed. in English). 49: 6589-91. PMID 20661982 DOI: 10.1002/Anie.201002972  0.657
2010 Li G, Kaplan MJ, Wojtas L, Antilla JC. Chiral phosphoric acid catalyzed addition of dihydropyrans to N-acyl imines: stereocontrolled access to enantioenriched spirocyclic oxazoletetrahydropyrans with three contiguous stereocenters. Organic Letters. 12: 1960-3. PMID 20361794 DOI: 10.1021/Ol100378T  0.617
2010 Cortes-Salva M, Nguyen BL, Cuevas J, Pennypacker KR, Antilla JC. Copper-catalyzed guanidinylation of aryl iodides: the formation of N,N'-disubstituted guanidines. Organic Letters. 12: 1316-9. PMID 20170103 DOI: 10.1021/Ol1002175  0.811
2010 Antilla J, Liang T, Zhang Z. Brønsted Acid Catalyzed Asymmetric Pinacol Rearrangement Synfacts. 2011: 0094-0094. DOI: 10.1055/S-0030-1259192  0.558
2010 Antilla J, Zheng W, Wojtas L. Catalytic Asymmetric Peroxidation of Imines Synfacts. 2010: 1186-1186. DOI: 10.1055/s-0030-1258675  0.447
2010 Antilla J, Jain P. Allylboration of Aldehydes Synfacts. 2010: 1187-1187. DOI: 10.1055/S-0030-1258672  0.71
2010 Desai AA, Huang L, Wulff WD, Rowland GB, Antilla JC. Gram-scale preparation of VAPOL hydrogenphosphate: A structurally distinct chiral brønsted acid Synthesis. 2106-2109. DOI: 10.1055/S-0029-1218783  0.812
2009 Larson SE, Baso JC, Li G, Antilla JC. Chiral phosphoric acid-catalyzed desymmetrization of meso-aziridines with functionalized mercaptans. Organic Letters. 11: 5186-9. PMID 19905027 DOI: 10.1021/Ol902123H  0.812
2009 Li G, Antilla JC. Highly enantioselective hydrogenation of enamides catalyzed by chiral phosphoric acids. Organic Letters. 11: 1075-8. PMID 19199770 DOI: 10.1021/Ol802860U  0.616
2008 Li G, Fronczek FR, Antilla JC. Catalytic asymmetric addition of alcohols to imines: enantioselective preparation of chiral N,O-aminals. Journal of the American Chemical Society. 130: 12216-7. PMID 18722443 DOI: 10.1021/Ja8033334  0.592
2007 Liang Y, Rowland EB, Rowland GB, Perman JA, Antilla JC. VAPOL phosphoric acid catalysis: the highly enantioselective addition of imides to imines. Chemical Communications (Cambridge, England). 4477-9. PMID 17971961 DOI: 10.1039/B709276H  0.846
2007 Rowland EB, Rowland GB, Rivera-Otero E, Antilla JC. Brønsted acid-catalyzed desymmetrization of meso-aziridines. Journal of the American Chemical Society. 129: 12084-5. PMID 17877355 DOI: 10.1021/Ja0751779  0.855
2007 Li G, Rowland GB, Rowland EB, Antilla JC. Organocatalytic enantioselective Friedel-Crafts reaction of pyrrole derivatives with imines. Organic Letters. 9: 4065-8. PMID 17727293 DOI: 10.1021/Ol701881J  0.851
2007 Rowland GB, Rowland EB, Liang Y, Perman JA, Antilla JC. The highly enantioselective addition of indoles to N-acyl imines with use of a chiral phosphoric acid catalyst. Organic Letters. 9: 2609-11. PMID 17547413 DOI: 10.1021/Ol0703579  0.849
2007 Newman CA, Antilla JC, Chen P, Predeus AV, Fielding L, Wulff WD. Regulation of orthogonal functions in a dual catalyst system. Subservient role of a nonchiral Lewis acid in an asymmetric catalytic heteroatom Diels-Alder reaction. Journal of the American Chemical Society. 129: 7216-7. PMID 17503816 DOI: 10.1021/Ja069019D  0.86
2007 Li G, Liang Y, Antilla JC. A vaulted biaryl phosphoric acid-catalyzed reduction of alpha-imino esters: the highly enantioselective preparation of alpha-amino esters. Journal of the American Chemical Society. 129: 5830-1. PMID 17428058 DOI: 10.1021/Ja070519W  0.596
2007 Newman CA, Antilla JC, Chen P, Predeus AV, Fielding L, Wulff WD. Asymmetric Synthesis of Dihydropyridinones Synfacts. 2007: 921-921. DOI: 10.1055/S-2007-968911  0.667
2007 Antilla J, Li G, Liang Y. Phosphoric Acid Catalyzed Route to α-Amino Esters Synfacts. 2007: 0764-0764. DOI: 10.1055/s-2007-968632  0.353
2007 Zhang Z, Jain P, Antilla JC. Asymmetric Reduction of Ketones Synfacts. 2011: 1364-1364. DOI: 10.1055/S-0031-1289372  0.657
2006 Rowland GB, Rowland EB, Zhang Q, Antilla JC. Stereoselective aza-Diels-Alder reactions Current Organic Chemistry. 10: 981-1005. DOI: 10.2174/138527206777435463  0.8
2006 Rowland GB, Zhang H, Rowland EB, Chennamadhavuni S, Wang Y, Antilla JC. Broensted Acid Catalyzed Imine Amidation. Cheminform. 37. DOI: 10.1002/chin.200612083  0.805
2005 Rowland GB, Zhang H, Rowland EB, Chennamadhavuni S, Wang Y, Antilla JC. Brønsted acid-catalyzed imine amidation. Journal of the American Chemical Society. 127: 15696-7. PMID 16277499 DOI: 10.1055/S-2005-924799  0.84
2005 Antilla JC. Metal-Catalyzed Cross-Coupling Reactions, Second, Completely Revised and Enlarged Edition: Volumes 1 and 2 Edited by Armin de Meijere (George-August-Universität, Göttingen) and Francois Diederich (ETH, Zürich). Wiley-VCH Verlag GmbH & Co. KGaA: Weinheim, Germany. 2004. xxii + xxii + 916 pp. $450.00. ISBN 3-527-30518-1. Journal of the American Chemical Society. 127: 10121-10122. DOI: 10.1021/Ja059731V  0.421
2004 Antilla JC, Baskin JM, Barder TE, Buchwald SL. Copper-diamine-catalyzed N-arylation of pyrroles, pyrazoles, indazoles, imidazoles, and triazoles. The Journal of Organic Chemistry. 69: 5578-87. PMID 15307726 DOI: 10.1021/Jo049658B  0.841
2002 Antilla JC, Klapars A, Buchwald SL. The copper-catalyzed N-arylation of indoles. Journal of the American Chemical Society. 124: 11684-8. PMID 12296734 DOI: 10.1021/Ja027433H  0.568
2001 Klapars A, Antilla JC, Huang X, Buchwald SL. A general and efficient copper catalyst for the amidation of aryl halides and the N-arylation of nitrogen heterocycles. Journal of the American Chemical Society. 123: 7727-9. PMID 11481007 DOI: 10.1021/Ja016226Z  0.726
2001 Antilla JC, Buchwald SL. Copper-catalyzed coupling of arylboronic acids and amines. Organic Letters. 3: 2077-9. PMID 11418053 DOI: 10.1021/Ol0160396  0.648
2001 Antilla JC, Wulff WD. ChemInform Abstract: Catalytic Asymmetric Aziridination with Arylborate Catalysts Derived from VAPOL and VANOL Ligands. Cheminform. 32: no-no. DOI: 10.1002/chin.200115032  0.404
2000 Antilla JC, Wulff WD. Catalytic Asymmetric Aziridination with Arylborate Catalysts Derived from VAPOL and VANOL Ligands This work was supported by the National Institutes of Health and was performed at the University of Chicago. VAPOL=2,2'-diphenyl- Angewandte Chemie (International Ed. in English). 39: 4518-4521. PMID 11169656 DOI: 10.1002/1521-3773(20001215)39:24<4518::Aid-Anie4518>3.0.Co;2-J  0.624
1999 Antilla JC, Wulff WD. Catalytic asymmetric aziridination with a chiral VAPOL-boron Lewis acid Journal of the American Chemical Society. 121: 5099-5100. DOI: 10.1021/Ja9905187  0.743
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