Year |
Citation |
Score |
2020 |
Yamano MM, Kelleghan AV, Shao Q, Giroud M, Simmons BJ, Li B, Chen S, Houk KN, Garg NK. Intercepting fleeting cyclic allenes with asymmetric nickel catalysis. Nature. PMID 32846425 DOI: 10.1038/S41586-020-2701-2 |
0.576 |
|
2019 |
Dander JE, Giroud M, Racine S, Darzi ER, Alvizo O, Entwistle D, Garg NK. Chemoenzymatic conversion of amides to enantioenriched alcohols in aqueous medium. Communications Chemistry. 2. PMID 32042928 DOI: 10.1038/s42004-019-0182-8 |
0.473 |
|
2018 |
Picazo E, Anthony SM, Giroud M, Simon A, Miller MA, Houk KN, Garg NK. Arynes and Cyclic Alkynes as Synthetic Building Blocks for Stereodefined Quaternary Centers. Journal of the American Chemical Society. PMID 29716194 DOI: 10.1021/Jacs.8B02875 |
0.609 |
|
2018 |
Giroud M, Kuhn B, Saint-Auret S, Kuratli C, Martin RE, Schuler F, Diederich F, Kaiser M, Brun R, Schirmeister T, Haap W. 2H-1,2,3-Triazole-Based Dipeptidyl Nitriles: Potent, Selective, and Trypanocidal Rhodesain Inhibitors by Structure-Based Design. Journal of Medicinal Chemistry. PMID 29590751 DOI: 10.1021/Acs.Jmedchem.7B01870 |
0.442 |
|
2018 |
Giroud M, Dietzel U, Anselm L, Banner D, Kuglstatter A, Benz J, Blanc JB, Gaufreteau D, Liu H, Lin X, Stich A, Kuhn B, Schuler F, Kaiser M, Brun R, et al. Repurposing a Library of Human Cathepsin L Ligands: Identification of Macrocyclic Lactams as Potent Rhodesain and Trypanosoma brucei Inhibitors. Journal of Medicinal Chemistry. PMID 29590750 DOI: 10.1021/Acs.Jmedchem.7B01869 |
0.426 |
|
2017 |
Kuhn B, Tichý M, Wang L, Robinson S, Martin RE, Kuglstatter A, Benz J, Giroud M, Schirmeister T, Abel R, Diederich F, Hert J. Prospective Evaluation of Free Energy Calculations for the Prioritization of Cathepsin L Inhibitors. Journal of Medicinal Chemistry. PMID 28287264 DOI: 10.1021/Acs.Jmedchem.6B01881 |
0.449 |
|
2016 |
Giroud M, Ivkovic J, Martignoni M, Fleuti M, Trapp N, Haap W, Kuglstatter A, Benz J, Kuhn B, Schirmeister T, Diederich F. Inhibition of the Cysteine Protease Human Cathepsin L by Triazine Nitriles: Amide···Heteroarene π-Stacking Interactions and Chalcogen Bonding in the S3 Pocket. Chemmedchem. PMID 27992115 DOI: 10.1002/Cmdc.201600563 |
0.491 |
|
2016 |
Giroud M, Harder M, Kuhn B, Haap W, Trapp N, Schweizer WB, Schirmeister T, Diederich F. Fluorine Scan of Inhibitors of the Cysteine Protease Human Cathepsin L: Dipolar and Quadrupolar Effects in the π-Stacking of Fluorinated Phenyl Rings on Peptide Amide Bonds. Chemmedchem. PMID 27095165 DOI: 10.1002/Cmdc.201600132 |
0.495 |
|
2015 |
Barandun LJ, Ehrmann FR, Zimmerli D, Immekus F, Giroud M, Grünenfelder C, Schweizer WB, Bernet B, Betz M, Heine A, Klebe G, Diederich F. Replacement of water molecules in a phosphate binding site by furanoside-appended lin-benzoguanine ligands of tRNA-guanine transglycosylase (TGT). Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 126-35. PMID 25483606 DOI: 10.1002/Chem.201405764 |
0.47 |
|
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