Year |
Citation |
Score |
2011 |
Tommasi RA, Weiler S, Mcquire LW, Rogel O, Chambers M, Clark K, Doughty J, Fang J, Ganu V, Grob J, Goldberg R, Goldstein R, Lavoie S, Kulathila R, Macchia W, ... ... Shultz M, et al. Potent and selective 2-naphthylsulfonamide substituted hydroxamic acid inhibitors of matrix metalloproteinase-13 Bioorganic and Medicinal Chemistry Letters. 21: 6440-6445. PMID 21937229 DOI: 10.1016/J.Bmcl.2011.08.087 |
0.308 |
|
2011 |
Shultz M, Fan J, Chen C, Cho YS, Davis N, Bickford S, Buteau K, Cao X, Holmqvist M, Hsu M, Jiang L, Liu G, Lu Q, Patel C, Suresh JR, et al. The design, synthesis and structure-activity relationships of novel isoindoline-based histone deacetylase inhibitors. Bioorganic & Medicinal Chemistry Letters. 21: 4909-12. PMID 21742496 DOI: 10.1016/J.Bmcl.2011.06.015 |
0.326 |
|
2010 |
Cho YS, Whitehead L, Li J, Chen CHT, Jiang L, Vögtle M, Francotte E, Richert P, Wagner T, Traebert M, Lu Q, Cao X, Dumotier B, Fejzo J, Rajan S, ... ... Shultz M, et al. Conformational refinement of hydroxamate-based histone deacetylase inhibitors and exploration of 3-piperidin-3-ylindole analogues of dacinostat (LAQ824) Journal of Medicinal Chemistry. 53: 2952-2963. PMID 20205394 DOI: 10.1021/Jm100007M |
0.367 |
|
2010 |
ZUTSHI R, SHULTZ MD, ULYSSE L, LUTGRING R, BISHOP P, SCHWEITZER B, VOGEL K, FRANCISKOVICH J, WILSON M, CHMIELEWSKI J. ChemInform Abstract: Inhibiting the Dimerization of HIV-1 Protease Cheminform. 29: no-no. DOI: 10.1002/CHIN.199852336 |
0.715 |
|
2004 |
Shultz MD, Ham YW, Lee SG, Davis DA, Brown C, Chmielewski J. Small-molecule dimerization inhibitors of wild-type and mutant HIV protease: a focused library approach. Journal of the American Chemical Society. 126: 9886-7. PMID 15303839 DOI: 10.1021/Ja048139N |
0.821 |
|
2003 |
Zhao L, O'Reilly MK, Shultz MD, Chmielewski J. Interfacial peptide inhibitors of HIV-1 integrase activity and dimerization Bioorganic and Medicinal Chemistry Letters. 13: 1175-1177. PMID 12643937 DOI: 10.1016/S0960-894X(03)00040-4 |
0.748 |
|
2000 |
Shultz M, Bowman M, Ham Y, Zhao X, Tora G, Chmielewski J. Small-Molecule Inhibitors of HIV-1 Protease Dimerization Derived from Cross-Linked Interfacial Peptides Angewandte Chemie. 112: 2822-2825. DOI: 10.1002/1521-3757(20000804)112:15<2822::Aid-Ange2822>3.0.Co;2-1 |
0.824 |
|
1999 |
Shultz MD, Chmielewski J. Probing the role of interfacial residues in a dimerization inhibitor of HIV-1 protease Bioorganic and Medicinal Chemistry Letters. 9: 2431-2436. PMID 10476882 DOI: 10.1016/S0960-894X(99)00400-X |
0.746 |
|
1998 |
Zutshi R, Shultz MD, Ulysse L, Lutgring R, Bishop P, Schweitzer B, Vogel K, Franciskovich J, Wilson M, Chmielewski J. Inhibiting the Dimerization of HIV-1 Protease Synlett. 1998: 1040-1044. DOI: 10.1055/S-1998-1854 |
0.617 |
|
1997 |
Zutshi R, Franciskovich J, Shultz M, Schweitzer B, Bishop P, Wilson M, Chmielewski J. Targeting the dimerization interface of HIV-1 protease: Inhibition with cross-linked interfacial peptides Journal of the American Chemical Society. 119: 4841-4845. DOI: 10.1021/Ja962496J |
0.778 |
|
1997 |
Shultz MD, Chmielewski J. Hydrophobicity versus activity in crosslinked interfacial peptide inhibitors of HIV-1 protease Tetrahedron Asymmetry. 8: 3881-3886. DOI: 10.1016/S0957-4166(97)00572-7 |
0.733 |
|
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