Year |
Citation |
Score |
2023 |
Pakula RJ, Raffel DM, Koeppe RA, Winton WP, Stauff J, Bohnen NI, Albin RL, Scott PJH, Shao X. Automated production of [C]butyrate for keto body PET imaging. Nuclear Medicine and Biology. 108315. PMID 36680983 DOI: 10.1016/j.nucmedbio.2023.108315 |
0.368 |
|
2023 |
Mhanna K, Qian W, Zhong Z, Brooks AF, Ouchi E, Stauff J, Arteaga J, Papachristou M, Datseris IE, Liu B, Shao X, Scott PJH. Preparation and Evaluation of Cu-Radiolabled Dual-Ligand Multifunctional Gold Nanoparticles for Tumor Theragnosis. Pharmaceuticals (Basel, Switzerland). 16. PMID 36678568 DOI: 10.3390/ph16010071 |
0.703 |
|
2022 |
Jackson IM, Buccino PJ, Azevedo EC, Carlson ML, Luo ASZ, Deal EM, Kalita M, Reyes ST, Shao X, Beinat C, Nagy SC, Chaney AM, Anders DA, Scott PJH, Smith M, et al. Radiosynthesis and initial preclinical evaluation of [C]AZD1283 as a potential P2Y12R PET radiotracer. Nuclear Medicine and Biology. PMID 35680502 DOI: 10.1016/j.nucmedbio.2022.05.001 |
0.312 |
|
2021 |
Lindberg A, Mossine AV, Aliaga A, Hopewell R, Massarweh G, Rosa-Neto P, Shao X, Bernard-Gauthier V, Scott PJH, Vasdev N. Preliminary Evaluations of [C]Verubulin: Implications for Microtubule Imaging With PET. Frontiers in Neuroscience. 15: 725873. PMID 34566568 DOI: 10.3389/fnins.2021.725873 |
0.367 |
|
2020 |
Zhao AY, Brooks AF, Raffel DM, Stauff J, Arteaga J, Scott PJH, Shao X. Fully Automated Radiosynthesis of [C]Guanidines for Cardiac PET Imaging. Acs Medicinal Chemistry Letters. 11: 2325-2330. PMID 33214848 DOI: 10.1021/acsmedchemlett.0c00479 |
0.327 |
|
2020 |
Brooks AF, Mufarreh AJ, Shao X, Kaur T, Stauff J, Arteaga J, Kilbourn MR, Scott PJH. Improved Synthesis of [C]COU and [C]PHXY, Evaluation of Neurotoxicity, and Imaging of MAOs in Rodent Heart. Acs Medicinal Chemistry Letters. 11: 2300-2304. PMID 33214844 DOI: 10.1021/Acsmedchemlett.0C00419 |
0.57 |
|
2020 |
Jackson IM, Lee SJ, Sowa AR, Rodnick ME, Bruton L, Clark M, Preshlock S, Rothley J, Rogers VE, Botti LE, Henderson BD, Hockley BG, Torres J, Raffel DM, Brooks AF, ... ... Shao X, et al. Use of 55 PET radiotracers under approval of a Radioactive Drug Research Committee (RDRC). Ejnmmi Radiopharmacy and Chemistry. 5: 24. PMID 33175263 DOI: 10.1186/s41181-020-00110-z |
0.731 |
|
2020 |
Hill JR, Shao X, Massey NL, Stauff J, Sherman PS, Robertson AAB, Scott PJH. Synthesis and evaluation of NLRP3-inhibitory sulfonylurea [C]MCC950 in healthy animals. Bioorganic & Medicinal Chemistry Letters. 127186. PMID 32312583 DOI: 10.1016/J.Bmcl.2020.127186 |
0.364 |
|
2020 |
Scott PJH, Koeppe RA, Shao X, Rodnick ME, Sowa AR, Henderson BD, Stauff J, Sherman PS, Arteaga J, Carlo DJ, Moss RB. The Effects of Intramuscular Naloxone Dose on Mu Receptor Displacement of Carfentanil in Rhesus Monkeys. Molecules (Basel, Switzerland). 25. PMID 32192089 DOI: 10.3390/Molecules25061360 |
0.708 |
|
2019 |
Bernard-Gauthier V, Mossine AV, Knight A, Patnaik D, Zhao W, Cheng C, Krishnan HS, Xuan LL, Chindavong PS, Reis SA, Chen JM, Shao X, Stauff J, Arteaga J, Sherman PS, et al. Structural Basis for Achieving GSK-3 Inhibition with High Potency, Selectivity and Brain Exposure for PET Imaging and Drug Discovery. Journal of Medicinal Chemistry. PMID 31535859 DOI: 10.1021/Acs.Jmedchem.9B01030 |
0.318 |
|
2018 |
Yang L, Brooks AF, Makaravage KJ, Zhang H, Sanford MS, Scott PJH, Shao X. Radiosynthesis of [C]LY2795050 for Preclinical and Clinical PET Imaging Using Cu(II)-Mediated Cyanation. Acs Medicinal Chemistry Letters. 9: 1274-1279. PMID 30613339 DOI: 10.1021/Acsmedchemlett.8B00460 |
0.376 |
|
2018 |
Tanzey SS, Shao X, Stauff J, Arteaga J, Sherman P, Scott PJH, Mossine AV. Synthesis and Initial In Vivo Evaluation of [C]AZ683-A Novel PET Radiotracer for Colony Stimulating Factor 1 Receptor (CSF1R). Pharmaceuticals (Basel, Switzerland). 11. PMID 30551596 DOI: 10.3390/ph11040136 |
0.383 |
|
2018 |
Brooks AF, Drake LR, Shao X, Zhao A, Scott PJH, Kilbourn MR. Evaluation of Enzyme Substrate Radiotracers as PET/MRS Hybrid Imaging Agents. Acs Medicinal Chemistry Letters. 9: 1140-1143. PMID 30429959 DOI: 10.1021/Acsmedchemlett.8B00402 |
0.536 |
|
2018 |
Drake LR, Brooks AF, Mufarreh AJ, Pham JM, Koeppe RA, Shao X, Scott PJH, Kilbourn MR. Deuterium Kinetic Isotope Effect Studies of a Potential In Vivo Metabolic Trapping Agent for Monoamine Oxidase-B. Acs Chemical Neuroscience. PMID 30074755 DOI: 10.1021/Acschemneuro.8B00219 |
0.562 |
|
2018 |
Sowa AR, Brooks AF, Shao X, Henderson BD, Sherman PS, Arteaga J, Stauff J, Lee AC, Koeppe RA, Scott PJH, Kilbourn MR. Development of Positron Emission Tomography (PET) Radiotracers for the GABA Transporter 1 (GAT-1). Acs Chemical Neuroscience. PMID 29763549 DOI: 10.1021/Acschemneuro.8B00183 |
0.557 |
|
2017 |
Bernard-Gauthier V, Mossine AV, Mahringer A, Aliaga A, Bailey JJ, Shao X, Stauff J, Arteaga J, Sherman PS, Grand'Maison M, Rochon PL, Wängler B, Wängler C, Bartenstein P, Kostikov A, et al. Identification of 18FTRACK, a Fluorine-18-Labeled Tropomyosin Receptor Kinase (Trk) Inhibitor for PET Imaging. Journal of Medicinal Chemistry. PMID 29257860 DOI: 10.1021/Acs.Jmedchem.7B01607 |
0.345 |
|
2017 |
Bernard-Gauthier V, Bailey JJ, Mossine AV, Lindner SK, Vomacka L, Aliaga A, Shao X, Quesada CA, Sherman PS, Mahringer A, Kostikov A, Grand'Maison M, Rosa-Neto P, Soucy JP, Thiel A, et al. A Kinome-Wide Selective Radiolabeled TrkB/C Inhibitor for in Vitro and in Vivo Neuroimaging: Synthesis, Preclinical Evaluation and First-in-Human. Journal of Medicinal Chemistry. PMID 28696690 DOI: 10.1021/Acs.Jmedchem.7B00396 |
0.311 |
|
2017 |
Blecha JE, Henderson BD, Hockley BG, VanBrocklin HF, Zubieta JK, DaSilva AF, Kilbourn MR, Koeppe RA, Scott PJH, Shao X. An Updated Synthesis of [(11) C]Carfentanil for Positron Emission Tomography (PET) Imaging of the μ-Opioid Receptor. Journal of Labelled Compounds & Radiopharmaceuticals. PMID 28419528 DOI: 10.1002/Jlcr.3513 |
0.588 |
|
2017 |
Piert M, Shao X, Raffel DM, Davenport MS, Montgomery J, Kunju L, Hockley BG, Siddiqui J, Scott PJ, Chinnaiyan A, Rajandiran T. Preclinical evaluation of (11)C-sarcosine as a substrate of proton-coupled amino acid transporters and first human application in prostate cancer. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. PMID 28302759 DOI: 10.2967/jnumed.116.173179 |
0.529 |
|
2016 |
Saccone PA, Lindsey AM, Koeppe RA, Zelenock KA, Shao X, Sherman P, Quesada CA, Woods JH, Scott PJ. Intranasal opioid administration in rhesus monkeys: PET imaging and antinociception. The Journal of Pharmacology and Experimental Therapeutics. PMID 27625351 DOI: 10.1124/Jpet.116.235192 |
0.553 |
|
2016 |
Scott PJ, Shao X, Desmond TJ, Hockley BG, Sherman P, Quesada CA, Frey KA, Koeppe RA, Kilbourn MR, Bohnen NI. Investigation of Proposed Activity of Clarithromycin at GABAA Receptors Using [(11)C]Flumazenil PET. Acs Medicinal Chemistry Letters. 7: 746-50. PMID 27563397 DOI: 10.1021/Acsmedchemlett.5B00435 |
0.651 |
|
2016 |
Mossine AV, Brooks AF, Jackson IM, Quesada CA, Sherman PS, Cole EL, Donnelly D, Scott PJ, Shao X. Synthesis of Diverse (11)C-Labelled PET Radiotracers via Direct Incorporation of [(11)C]CO 2. Bioconjugate Chemistry. PMID 27043721 DOI: 10.1021/Acs.Bioconjchem.6B00163 |
0.71 |
|
2015 |
Brooks AF, Shao X, Quesada CA, Sherman P, Scott PJ, Kilbourn MR. In Vivo Metabolic Trapping Radiotracers for Imaging Monoamine Oxidase-A and -B Enzymatic Activity. Acs Chemical Neuroscience. PMID 26393369 DOI: 10.1021/Acschemneuro.5B00223 |
0.657 |
|
2015 |
Brooks AF, Jackson IM, Shao X, Kropog GW, Sherman P, Quesada CA, Scott PJ. Synthesis and evaluation of [(11)C]PBD150, a radiolabeled glutaminyl cyclase inhibitor for the potential detection of Alzheimer's disease prior to amyloid β aggregation. Medchemcomm. 6: 1065-1068. PMID 26101580 DOI: 10.1039/C5Md00148J |
0.598 |
|
2015 |
Li L, Shao X, Cole EL, Ohnmacht SA, Ferrari V, Hong YT, Williamson DJ, Fryer TD, Quesada CA, Sherman P, Riss PJ, Scott PJ, Aigbirhio FI. Synthesis and Initial in Vivo Studies with [(11)C]SB-216763: The First Radiolabeled Brain Penetrative Inhibitor of GSK-3. Acs Medicinal Chemistry Letters. 6: 548-52. PMID 26005531 DOI: 10.1021/acsmedchemlett.5b00044 |
0.613 |
|
2015 |
Cary BP, Brooks AF, Fawaz MV, Shao X, Desmond TJ, Carpenter GM, Sherman P, Quesada CA, Albin RL, Scott PJ. Targeting Metal-Aβ Aggregates with Bifunctional Radioligand [(11)C]L2-b and a Fluorine-18 Analogue [(18)F]FL2-b. Acs Medicinal Chemistry Letters. 6: 112-116. PMID 25705326 DOI: 10.1021/Ml500413D |
0.509 |
|
2014 |
Fawaz MV, Brooks AF, Rodnick ME, Carpenter GM, Shao X, Desmond TJ, Sherman P, Quesada CA, Hockley BG, Kilbourn MR, Albin RL, Frey KA, Scott PJ. High affinity radiopharmaceuticals based upon lansoprazole for PET imaging of aggregated tau in Alzheimer's disease and progressive supranuclear palsy: synthesis, preclinical evaluation, and lead selection. Acs Chemical Neuroscience. 5: 718-30. PMID 24896980 DOI: 10.1021/Cn500103U |
0.744 |
|
2014 |
Cole EL, Shao X, Sherman P, Quesada C, Fawaz MV, Desmond TJ, Scott PJ. Synthesis and evaluation of [(11)C]PyrATP-1, a novel radiotracer for PET imaging of glycogen synthase kinase-3β (GSK-3β). Nuclear Medicine and Biology. 41: 507-12. PMID 24768148 DOI: 10.1016/j.nucmedbio.2014.03.025 |
0.512 |
|
2014 |
Rodnick ME, Shao X, Kozloff KM, Scott PJ, Kilbourn MR. Carbon-11 labeled cathepsin K inhibitors: syntheses and preliminary in vivo evaluation. Nuclear Medicine and Biology. 41: 384-9. PMID 24637099 DOI: 10.1016/J.Nucmedbio.2014.02.004 |
0.706 |
|
2014 |
Shao X, Fawaz MV, Jang K, Scott PJ. Ethanolic carbon-11 chemistry: the introduction of green radiochemistry. Applied Radiation and Isotopes : Including Data, Instrumentation and Methods For Use in Agriculture, Industry and Medicine. 89: 125-9. PMID 24631743 DOI: 10.1016/J.Apradiso.2014.01.033 |
0.483 |
|
2013 |
Shao X, Schnau PL, Fawaz MV, Scott PJ. Enhanced radiosyntheses of [¹¹C]raclopride and [¹¹C]DASB using ethanolic loop chemistry. Nuclear Medicine and Biology. 40: 109-16. PMID 23123138 DOI: 10.1016/j.nucmedbio.2012.09.008 |
0.463 |
|
2012 |
Shao X, Carpenter GM, Desmond TJ, Sherman P, Quesada CA, Fawaz M, Brooks AF, Kilbourn MR, Albin RL, Frey KA, Scott PJ. Evaluation of [(11)C]N-Methyl Lansoprazole as a Radiopharmaceutical for PET Imaging of Tau Neurofibrillary Tangles. Acs Medicinal Chemistry Letters. 3: 936-41. PMID 24900410 DOI: 10.1021/Ml300216T |
0.692 |
|
2012 |
Hoareau R, Shao X, Henderson BD, Scott PJ. Fully automated radiosynthesis of [¹¹C]PBR28, a radiopharmaceutical for the translocator protein (TSPO) 18 kDa, using a GE TRACERlab FXC-Pro. Applied Radiation and Isotopes : Including Data, Instrumentation and Methods For Use in Agriculture, Industry and Medicine. 70: 1779-83. PMID 22503515 DOI: 10.1016/j.apradiso.2012.03.006 |
0.596 |
|
2011 |
Shao X, Hoareau R, Hockley BG, Tluczek LJ, Henderson BD, Padgett HC, Scott PJ. Highlighting the Versatility of the Tracerlab Synthesis Modules. Part 1: Fully Automated Production of [F]Labelled Radiopharmaceuticals using a Tracerlab FX(FN). Journal of Labelled Compounds & Radiopharmaceuticals. 54: 292-307. PMID 21769163 DOI: 10.1002/Jlcr.1865 |
0.498 |
|
2011 |
Runkle AC, Shao X, Tluczek LJ, Henderson BD, Hockley BG, Scott PJ. Automated production of [11C]acetate and [11C]palmitate using a modified GE Tracerlab FX(C-Pro). Applied Radiation and Isotopes : Including Data, Instrumentation and Methods For Use in Agriculture, Industry and Medicine. 69: 691-8. PMID 21256039 DOI: 10.1016/j.apradiso.2011.01.002 |
0.55 |
|
2011 |
Shao X, Hockley BG, Hoareau R, Schnau PL, Scott PJ. Fully automated preparation of [11C]choline and [18F]fluoromethylcholine using TracerLab synthesis modules and facilitated quality control using analytical HPLC. Applied Radiation and Isotopes : Including Data, Instrumentation and Methods For Use in Agriculture, Industry and Medicine. 69: 403-9. PMID 21115355 DOI: 10.1016/j.apradiso.2010.09.022 |
0.547 |
|
2009 |
Shao X, Kilbourn MR. A simple modification of GE tracerlab FX C Pro for rapid sequential preparation of [11C]carfentanil and [11C]raclopride Applied Radiation and Isotopes. 67: 602-605. PMID 19162491 DOI: 10.1016/J.Apradiso.2008.12.013 |
0.513 |
|
2005 |
Shao X, Koeppe RA, Butch ER, Kilbourn MR, Snyder SE. Evaluation of 18F-labeled acetylcholinesterase substrates as PET radiotracers Bioorganic and Medicinal Chemistry. 13: 869-875. PMID 15653352 DOI: 10.1016/J.Bmc.2004.10.034 |
0.658 |
|
2003 |
Shao X, Butch ER, Kilbourn MR, Snyder SE. N-[18F]fluoroethylpiperidinyl, N-[18F]fluoroethylpiperidinemethyl and N-[18F]fluoroethylpyrrolidinyl esters as radiotracers for acetylcholinesterase Nuclear Medicine and Biology. 30: 491-500. PMID 12831986 DOI: 10.1016/S0969-8051(03)00031-3 |
0.632 |
|
2003 |
Shao X, Lisi JM, Butch ER, Kilbourn MR, Snyder SE. N-methylpiperidinemethyl, N-methylpyrrolidyl and N-methylpyrrolidinemethyl esters as PET radiotracers for acetylcholinesterase activity Nuclear Medicine and Biology. 30: 293-302. PMID 12745021 DOI: 10.1016/S0969-8051(02)00438-9 |
0.629 |
|
Show low-probability matches. |