Year |
Citation |
Score |
2017 |
Li S, Jin F, Viji M, Jo H, Sim J, Kim HS, Lee H, Jung J. A novel cyclization/oxidation strategy for a two-step synthesis of (Z)-aurone Tetrahedron Letters. 58: 1417-1420. DOI: 10.1016/J.Tetlet.2017.02.074 |
0.307 |
|
2012 |
Mallik SK, Li da Y, Cui M, Song HO, Park H, Kim HS. Synthesis and evaluation of peptidyl α,β-unsaturated carbonyl derivatives as anti-malarial calpain inhibitors. Archives of Pharmacal Research. 35: 469-79. PMID 22477194 DOI: 10.1007/S12272-012-0310-9 |
0.308 |
|
2009 |
Park PH, Kim HS, Hur J, Jin XY, Jin YL, Sohn DH. YL-I-108, a synthetic chalcone derivative, inhibits lipopolysaccharide-stimulated nitric oxide production in RAW 264.7 murine macrophages: involvement of heme oxygenase-1 induction and blockade of activator protein-1. Archives of Pharmacal Research. 32: 79-89. PMID 19183880 DOI: 10.1007/S12272-009-1121-5 |
0.32 |
|
2009 |
Kim SA, Jin YL, Kim HS. Structure-activity relationship studies of novel oxygen-incorporated SAHA analogues. Archives of Pharmacal Research. 32: 15-21. PMID 19183872 DOI: 10.1007/S12272-009-1113-5 |
0.31 |
|
2009 |
Park PH, Kim HS, Jin XY, Jin F, Hur J, Ko G, Sohn DH. KB-34, a newly synthesized chalcone derivative, inhibits lipopolysaccharide-stimulated nitric oxide production in RAW 264.7 macrophages via heme oxygenase-1 induction and blockade of activator protein-1. European Journal of Pharmacology. 606: 215-24. PMID 19174156 DOI: 10.1016/J.Ejphar.2008.12.034 |
0.309 |
|
2008 |
Jin YL, Jin XY, Jin F, Sohn DH, Kim HS. Structure activity relationship studies of anti-inflammatory TMMC derivatives: 4-dimethylamino group on the B ring responsible for lowering the potency. Archives of Pharmacal Research. 31: 1145-52. PMID 18806957 DOI: 10.1007/S12272-001-1281-7 |
0.32 |
|
2008 |
Jin YL, Kim S, Kim YS, Kim S, Kim HS. The first total synthesis of glycyrol Tetrahedron Letters. 49: 6835-6837. DOI: 10.1016/J.Tetlet.2008.09.070 |
0.332 |
|
2007 |
Jin F, Jin XY, Jin YL, Sohn DW, Kim SA, Sohn DH, Kim YC, Kim HS. Structural requirements of 2',4',6'-tris(methoxymethoxy) chalcone derivatives for anti-inflammatory activity: the importance of a 2'-hydroxy moiety. Archives of Pharmacal Research. 30: 1359-67. PMID 18087801 DOI: 10.1007/Bf02977357 |
0.301 |
|
2007 |
Kim H, Kim S, Lee H, Ryu J. Synthesis of Conformationally Locked Methanocarba-uridine as a Precursor for Nucleotides Agonizing P2Y6 Receptor Synlett. 2007: 1055-1058. DOI: 10.1055/S-2007-973902 |
0.374 |
|
2006 |
Kim S, Jacobson KA, Kim HS. New Synthetic Approach to the Bicyclo[3.1.0]hexane Ring System from (+)-(1R,4R)-4-(Benzyloxymethyl)-4-(hydroxymethyl)cyclopent-2-enol. Cheminform. 37. DOI: 10.5012/Bkcs.2005.26.10.1503 |
0.358 |
|
2005 |
Jeong BS, Choi NS, Ahn SK, Bae H, Kim HS, Kim D. Total synthesis and antiangiogenic activity of cyclopentane analogues of fumagillol. Bioorganic & Medicinal Chemistry Letters. 15: 3580-3. PMID 15978809 DOI: 10.1016/J.Bmcl.2005.05.065 |
0.345 |
|
2005 |
Kim D, Ahn SK, Bae H, Kim HS. A stereoselective asymmetric synthesis of antibiotic (-)-fumagillol using claisen rearrangement and intramolecular ester enolate alkylation as key steps. Archives of Pharmacal Research. 28: 129-41. PMID 15789740 DOI: 10.1007/Bf02977704 |
0.315 |
|
2004 |
Dunn PM, Kim HS, Jacobson KA, Burnstock G. Northern Ring Conformation of Methanocarba-Adenosine 5'-Triphosphate Required for Activation of P2X Receptors. Drug Development Research. 61: 227-232. PMID 22833693 DOI: 10.1002/Ddr.10381 |
0.322 |
|
2004 |
Ohno M, Costanzi S, Kim HS, Kempeneers V, Vastmans K, Herdewijn P, Maddileti S, Gao ZG, Harden TK, Jacobson KA. Nucleotide analogues containing 2-oxa-bicyclo[2.2.1]heptane and l-alpha-threofuranosyl ring systems: interactions with P2Y receptors. Bioorganic & Medicinal Chemistry. 12: 5619-30. PMID 15465340 DOI: 10.1016/J.Bmc.2004.07.067 |
0.336 |
|
2003 |
Kim HS, Ohno M, Xu B, Kim HO, Choi Y, Ji XD, Maddileti S, Marquez VE, Harden TK, Jacobson KA. 2-Substitution of adenine nucleotide analogues containing a bicyclo[3.1.0]hexane ring system locked in a northern conformation: enhanced potency as P2Y1 receptor antagonists. Journal of Medicinal Chemistry. 46: 4974-87. PMID 14584948 DOI: 10.1021/Jm030127+ |
0.383 |
|
2003 |
Jacobson KA, Kim HS, Ravi G, Kim S, Lee K, Chen A, Chen W, Kim SG, Barak D, Liang BT, Gao Z. Engineering of A3 adenosine and P2Y nucleotide receptors and their ligands Drug Development Research. 58: 330-339. DOI: 10.1002/Ddr.10168 |
0.339 |
|
2002 |
Xu B, Stephens A, Kirschenheuter G, Greslin AF, Cheng X, Sennelo J, Cattaneo M, Zighetti ML, Chen A, Kim SA, Kim HS, Bischofberger N, Cook G, Jacobson KA. Acyclic analogues of adenosine bisphosphates as P2Y receptor antagonists: phosphate substitution leads to multiple pathways of inhibition of platelet aggregation. Journal of Medicinal Chemistry. 45: 5694-709. PMID 12477353 DOI: 10.1021/Jm020173U |
0.336 |
|
2002 |
Kim SA, Marshall MA, Melman N, Kim HS, Müller CE, Linden J, Jacobson KA. Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions. Journal of Medicinal Chemistry. 45: 2131-8. PMID 12014951 DOI: 10.1021/Jm0104318 |
0.357 |
|
2002 |
Kim HS, Ravi RG, Marquez VE, Maddileti S, Wihlborg AK, Erlinge D, Malmsjö M, Boyer JL, Harden TK, Jacobson KA. Methanocarba modification of uracil and adenine nucleotides: high potency of Northern ring conformation at P2Y1, P2Y2, P2Y4, and P2Y11 but not P2Y6 receptors. Journal of Medicinal Chemistry. 45: 208-18. PMID 11754592 DOI: 10.1021/Jm010369E |
0.355 |
|
2001 |
Kim HS, Barak D, Harden TK, Boyer JL, Jacobson KA. Acyclic and cyclopropyl analogues of adenosine bisphosphate antagonists of the P2Y1 receptor: structure-activity relationships and receptor docking. Journal of Medicinal Chemistry. 44: 3092-108. PMID 11543678 DOI: 10.1021/Jm010082H |
0.36 |
|
2001 |
Ravi G, Lee K, Ji X, Kim HS, Soltysiak KA, Marquez VE, Jacobson KA. Synthesis and purine receptor affinity of 6-oxopurine nucleosides and nucleotides containing (N)-methanocarba-pseudoribose rings. Bioorganic & Medicinal Chemistry Letters. 11: 2295-300. PMID 11527718 DOI: 10.1016/S0960-894X(01)00450-4 |
0.346 |
|
2001 |
Jacobson KA, Moro S, Hoffmann C, Kim YC, Kim HS, Ravi RG, Harden TK, Boyer JL. Structurally related nucleotides as selective agonists and antagonists at P2Y1 receptors. Farmaco (Società Chimica Italiana : 1989). 56: 71-5. PMID 11347970 DOI: 10.1016/S0014-827X(01)01023-0 |
0.321 |
|
1999 |
Li AH, Ji XD, Kim HS, Melman N, Jacobson KA. Pyran Template Approach to the Design of Novel A3 Adenosine Receptor Antagonists. Drug Development Research. 48: 171-177. PMID 27182099 DOI: 10.1002/(Sici)1098-2299(199912)48:4<171::Aid-Ddr4>3.0.Co;2-5 |
0.34 |
|
1997 |
Winkler JD, Kim HS, Kim S, Ando K, Houk KN. Stereoselective Synthesis of the Taxane Ring System via the Tandem Diels-Alder Cycloaddition. The Journal of Organic Chemistry. 62: 2957-2962. PMID 11671659 DOI: 10.1021/Jo961620E |
0.309 |
|
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