☰

Jean-Philippe Pin - Publications

Affiliations: 
Institute for Functional Genomics, Montpellier, Occitanie, France 
Area:
Neuropharmacology, mGlu and GABAB receptors
Website:
http://www.igf.cnrs.fr/english/dept2e.php
Tree Info Grants Similar researchers PubMed Report error

287/379 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2024 Philibert CE, Disdier C, Lafon PA, Bouyssou A, Oosterlaken M, Galant S, Pizzoccaro A, Tuduri P, Ster J, Liu J, Kniazeff J, Pin JP, Rondard P, Marin P, Vandermoere F. TrkB receptor interacts with mGlu receptor and mediates antipsychotic-like effects of mGlu receptor activation in the mouse. Science Advances. 10: eadg1679. PMID 38277461 DOI: 10.1126/sciadv.adg1679  0.408
2024 Staudt M, Liu N, Malhaire F, Doroudian Y, Prézeau L, Renard E, Hasanpour Z, Pin JP, Bunch L. Synthesis and pharmacological characterization of conformationally restricted 2-amino-Adipic acid analogs and carboxycyclopropyl glycines as selective metabotropic glutamate 2 receptor agonists. European Journal of Medicinal Chemistry. 266: 116157. PMID 38245976 DOI: 10.1016/j.ejmech.2024.116157  0.387
2024 Liu N, Eshak F, Malhaire F, Brabet I, Prézeau L, Renard E, Pin JP, Acher FC, Staudt M, Bunch L. Design, Synthesis, Pharmacology, and In Silico Studies of (1,2,3)-2-(()-Amino(carboxy)methyl)-3-(carboxymethyl)cyclopropane-1-carboxylic Acid (LBG30300): A Picomolar Potency Subtype-Selective mGlu Receptor Agonist. Journal of Medicinal Chemistry. PMID 38170918 DOI: 10.1021/acs.jmedchem.3c01811  0.458
2023 Alexander SPH, Christopoulos A, Davenport AP, Kelly E, Mathie AA, Peters JA, Veale EL, Armstrong JF, Faccenda E, Harding SD, Davies JA, Abbracchio MP, Abraham G, Agoulnik A, Alexander W, ... ... Pin JP, et al. The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors. British Journal of Pharmacology. S23-S144. PMID 38123151 DOI: 10.1111/bph.16177  0.609
2023 Lecat-Guillet N, Quast RB, Liu H, Bourrier E, Møller TC, Rovira X, Soldevila S, Lamarque L, Trinquet E, Liu J, Pin JP, Rondard P, Margeat E. Concerted conformational changes control metabotropic glutamate receptor activity. Science Advances. 9: eadf1378. PMID 37267369 DOI: 10.1126/sciadv.adf1378  0.365
2023 Liu L, Lin L, Shen C, Rondard P, Pin JP, Xu C, Liu J. Asymmetric activation of GABA and metabotropic glutamate receptors. American Journal of Physiology. Cell Physiology. PMID 37184233 DOI: 10.1152/ajpcell.00150.2022  0.538
2023 Rem PD, Sereikaite V, Fernández-Fernández D, Reinartz S, Ulrich D, Fritzius T, Trovo L, Roux S, Chen Z, Rondard P, Pin JP, Schwenk J, Fakler B, Gassmann M, Barkat TR, et al. Soluble amyloid-β precursor peptide does not regulate GABA receptor activity. Elife. 12. PMID 36688536 DOI: 10.7554/eLife.82082  0.603
2022 Liu J, Tang H, Xu C, Zhou S, Zhu X, Li Y, Prézeau L, Xu T, Pin JP, Rondard P, Ji W, Liu J. Biased signaling due to oligomerization of the G protein-coupled platelet-activating factor receptor. Nature Communications. 13: 6365. PMID 36289206 DOI: 10.1038/s41467-022-34056-4  0.362
2022 Meng J, Xu C, Lafon PA, Roux S, Mathieu M, Zhou R, Scholler P, Blanc E, Becker JAJ, Le Merrer J, González-Maeso J, Chames P, Liu J, Pin JP, Rondard P. Nanobody-based sensors reveal a high proportion of mGlu heterodimers in the brain. Nature Chemical Biology. PMID 35681029 DOI: 10.1038/s41589-022-01050-2  0.305
2022 Fang W, Yang F, Xu C, Ling S, Lin L, Zhou Y, Sun W, Wang X, Liu P, Rondard P, Shi P, Pin JP, Tian C, Liu J. Structural basis of the activation of metabotropic glutamate receptor 3. Cell Research. PMID 35236939 DOI: 10.1038/s41422-022-00623-z  0.427
2022 Acher FC, Cabayé A, Eshak F, Goupil-Lamy A, Pin JP. Metabotropic glutamate receptor orthosteric ligands and their binding sites. Neuropharmacology. 204: 108886. PMID 34813860 DOI: 10.1016/j.neuropharm.2021.108886  0.389
2021 Gazdarica M, Noda J, Durydivka O, Novosadova V, Mackie K, Pin JP, Prezeau L, Blahos J. SGIP1 modulates kinetics and interactions of the cannabinoid receptor 1 and G protein-coupled receptor kinase 3 signalosome. Journal of Neurochemistry. PMID 34970999 DOI: 10.1111/jnc.15569  0.474
2021 Liu L, Fan Z, Rovira X, Xue L, Roux S, Brabet I, Xin M, Pin JP, Rondard P, Liu J. Allosteric ligands control the activation of a class C GPCR heterodimer by acting at the transmembrane interface. Elife. 10. PMID 34866572 DOI: 10.7554/eLife.70188  0.459
2021 Wang Y, Gai S, Zhang W, Huang X, Ma S, Huo Y, Wu Y, Tu H, Pin JP, Rondard P, Xu C, Liu J. The GABA receptor mediates neuroprotection by coupling to G. Science Signaling. 14: eaaz4112. PMID 34665640 DOI: 10.1126/scisignal.aaz4112  0.424
2021 Alexander SP, Christopoulos A, Davenport AP, Kelly E, Mathie A, Peters JA, Veale EL, Armstrong JF, Faccenda E, Harding SD, Pawson AJ, Southan C, Davies JA, Abbracchio MP, Alexander W, ... ... Pin JP, et al. THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein-coupled receptors. British Journal of Pharmacology. 178: S27-S156. PMID 34529832 DOI: 10.1111/bph.15538  0.606
2021 Cao AM, Quast RB, Fatemi F, Rondard P, Pin JP, Margeat E. Allosteric modulators enhance agonist efficacy by increasing the residence time of a GPCR in the active state. Nature Communications. 12: 5426. PMID 34521824 DOI: 10.1038/s41467-021-25620-5  0.439
2021 Nasrallah C, Cannone G, Briot J, Rottier K, Berizzi AE, Huang CY, Quast RB, Hoh F, Banères JL, Malhaire F, Berto L, Dumazer A, Font-Ingles J, Gómez-Santacana X, Catena J, ... ... Pin JP, et al. Agonists and allosteric modulators promote signaling from different metabotropic glutamate receptor 5 conformations. Cell Reports. 36: 109648. PMID 34469715 DOI: 10.1016/j.celrep.2021.109648  0.467
2021 Haubrich J, Font J, Quast RB, Goupil-Lamy A, Scholler P, Nevoltris D, Acher F, Chames P, Rondard P, Prézeau L, Pin JP. A nanobody activating metabotropic glutamate receptor 4 discriminates between homo- and heterodimers. Proceedings of the National Academy of Sciences of the United States of America. 118. PMID 34385321 DOI: 10.1073/pnas.2105848118  0.515
2021 Du J, Wang D, Fan H, Xu C, Tai L, Lin S, Han S, Tan Q, Wang X, Xu T, Zhang H, Chu X, Yi C, Liu P, Wang X, ... ... Pin JP, et al. Structures of human mGlu2 and mGlu7 homo- and heterodimers. Nature. PMID 34135509 DOI: 10.1038/s41586-021-03641-w  0.497
2021 Zindel D, Mensat P, Vol C, Homayed Z, Charrier-Savournin F, Trinquet E, Banères JL, Pin JP, Pannequin J, Roux T, Dupuis E, Prézeau L. G protein-coupled receptors can control the Hippo/YAP pathway through Gq signaling. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 35: e21668. PMID 34114695 DOI: 10.1096/fj.202002159R  0.383
2021 Shen C, Mao C, Xu C, Jin N, Zhang H, Shen DD, Shen Q, Wang X, Hou T, Chen Z, Rondard P, Pin JP, Zhang Y, Liu J. Structural basis of GABA receptor-G protein coupling. Nature. PMID 33911284 DOI: 10.1038/s41586-021-03507-1  0.477
2020 Zhang S, Xue L, Liu X, Zhang XC, Zhou R, Zhao H, Shen C, Pin JP, Rondard P, Liu J. Structural basis for distinct quality control mechanisms of GABA receptor during evolution. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. PMID 33058267 DOI: 10.1096/fj.202001355RR  0.399
2020 Liu H, Yi P, Zhao W, Wu Y, Acher F, Pin JP, Liu J, Rondard P. Illuminating the allosteric modulation of the calcium-sensing receptor. Proceedings of the National Academy of Sciences of the United States of America. PMID 32817431 DOI: 10.1073/Pnas.1922231117  0.483
2020 Shaye H, Ishchenko A, Lam JH, Han GW, Xue L, Rondard P, Pin JP, Katritch V, Gati C, Cherezov V. Structural basis of the activation of a metabotropic GABA receptor. Nature. PMID 32555460 DOI: 10.1038/S41586-020-2408-4  0.511
2019 Poirel O, Mamer LE, Herman MA, Arnulf-Kempcke M, Kervern M, Potier B, Miot S, Wang J, Favre-Besse FC, Brabet I, Laras Y, Bertrand HO, Acher F, Pin JP, Puel JL, et al. LSP5-2157 a new inhibitor of vesicular glutamate transporters. Neuropharmacology. 107902. PMID 31811873 DOI: 10.1016/J.Neuropharm.2019.107902  0.382
2019 Xue L, Sun Q, Zhao H, Rovira X, Gai S, He Q, Pin JP, Liu J, Rondard P. Rearrangement of the transmembrane domain interfaces associated with the activation of a GPCR hetero-oligomer. Nature Communications. 10: 2765. PMID 31235691 DOI: 10.1038/S41467-019-10834-5  0.459
2019 Hajj M, De Vita T, Vol C, Renassia C, Bologna JC, Brabet I, Cazade M, Pastore M, Blahos J, Labesse G, Pin JP, Prezeau L. Non-classical ligand-independent regulation of Go protein by an orphan Class C GPCR. Molecular Pharmacology. PMID 31189666 DOI: 10.1124/mol.118.113019  0.467
2019 Heuninck J, Perpina Viciano C, Işbilir A, Caspar B, Capoferri D, Briddon SJ, Durroux T, Hill SJ, Lohse MJ, Milligan G, Pin JP, Hoffmann C. Context-dependent signalling of CXC chemokine receptor 4 (CXCR4) and atypical chemokine receptor 3 (ACKR3). Molecular Pharmacology. PMID 31092552 DOI: 10.1124/Mol.118.115477  0.65
2019 Heuninck J, Hounsou C, Dupuis E, Trinquet E, Mouillac B, Pin JP, Bonnet D, Durroux T. Time-Resolved FRET-Based Assays to Characterize G Protein-Coupled Receptor Hetero-oligomer Pharmacology. Methods in Molecular Biology (Clifton, N.J.). 1947: 151-168. PMID 30969415 DOI: 10.1007/978-1-4939-9121-1_8  0.492
2019 Pin JP, Kniazeff J, Prézeau L, Liu JF, Rondard P. GPCR interaction as a possible way for allosteric control between receptors. Molecular and Cellular Endocrinology. PMID 30849406 DOI: 10.1016/J.Mce.2019.02.019  0.538
2019 Dötsch V, Pin J. Decision letter: The orphan receptor GPR88 blunts the signaling of opioid receptors and multiple striatal GPCRs Elife. DOI: 10.7554/Elife.50519.Sa1  0.467
2019 Acher F, Battaglia G, Bräuner-Osborne H, Conn PJ, Duvoisin R, Ferraguti F, Flor PJ, Goudet C, Gregory KJ, Hampson D, Johnson MP, Kubo Y, Monn J, Nakanishi S, Nicoletti F, ... ... Pin J, et al. Metabotropic glutamate receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database Iuphar/Bps Guide to Pharmacology Cite. 2019. DOI: 10.2218/gtopdb/f40/2019.4  0.743
2019 Bettler B, Bowery NG, Cryan JF, Enna SJ, Farb DH, Foestl W, Kaupmann K, Pin J. GABAB receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database Iuphar/Bps Guide to Pharmacology Cite. 2019. DOI: 10.2218/gtopdb/f26/2019.4  0.703
2018 Tora AS, Rovira X, Cao AM, Cabayé A, Olofsson L, Malhaire F, Scholler P, Baik H, Van Eeckhaut A, Smolders I, Rondard P, Margeat E, Acher F, Pin JP, Goudet C. Chloride ions stabilize the glutamate-induced active state of the metabotropic glutamate receptor 3. Neuropharmacology. 140: 275-286. PMID 30102917 DOI: 10.1016/J.Neuropharm.2018.08.011  0.537
2018 Belhocine A, Veglianese P, Hounsou C, Dupuis E, Acher F, Durroux T, Goudet C, Pin JP. Profiling of orthosteric and allosteric group-III metabotropic glutamate receptor ligands on various G protein-coupled receptors with Tag-lite assays. Neuropharmacology. 140: 233-245. PMID 30099051 DOI: 10.1016/j.neuropharm.2018.07.032  0.584
2018 Møller TC, Hottin J, Clerté C, Zwier JM, Durroux T, Rondard P, Prézeau L, Royer CA, Pin JP, Margeat E, Kniazeff J. Oligomerization of a G protein-coupled receptor in neurons controlled by its structural dynamics. Scientific Reports. 8: 10414. PMID 29991736 DOI: 10.1038/S41598-018-28682-6  0.593
2018 Nasrallah C, Rottier K, Marcellin R, Compan V, Font J, Llebaria A, Pin JP, Banères JL, Lebon G. Direct coupling of detergent purified human mGlureceptor to the heterotrimeric G proteins Gq and Gs. Scientific Reports. 8: 4407. PMID 29535347 DOI: 10.1038/s41598-018-22729-4  0.47
2018 Chelliah S, Lemasson IA, Brabet I, Oueslati N, Karaman B, Cabaye A, Tora AEL, Commare B, Courtiol T, Cesarini S, McCort-Tranchepain I, Rigault D, Mony L, Bessiron T, McLean H, ... ... Pin JP, et al. Increased potency and selectivity for group-III metabotropic glutamate receptor agonists binding at dual sites. Journal of Medicinal Chemistry. PMID 29397723 DOI: 10.1021/Acs.Jmedchem.7B01438  0.498
2018 Font J, López-Cano M, Notartomaso S, Scarselli P, Di Prieto P, Bresolí-Obach R, Battaglia G, Malhaire F, Rovira X, Catena J, Giraldo J, Pin JP, Fernández-Dueñas V, Goudet C, Nonell S, et al. Correction: Optical control of pain in vivo with a photoactive mGlu5 receptor negative allosteric modulator. Elife. 7. PMID 29313801 DOI: 10.7554/Elife.34752  0.366
2018 Stewart GD, Comps-Agrar L, Nørskov-Lauritsen LB, Pin JP, Kniazeff J. Allosteric interactions between GABAB1 subunits control orthosteric binding sites occupancy within GABAB oligomers. Neuropharmacology. PMID 29305121 DOI: 10.1016/j.neuropharm.2017.12.042  0.457
2017 Møller TC, Moreno-Delgado D, Pin JP, Kniazeff J. Class C G protein-coupled receptors: reviving old couples with new partners. Biophysics Reports. 3: 57-63. PMID 29238742 DOI: 10.1007/s41048-017-0036-9  0.558
2017 Hounsou C, Baehr C, Gasparik V, Alili D, Belhocine A, Rodriguez T, Dupuis E, Roux T, Mann A, Heissler D, Pin JP, Durroux T, Bonnet D, Hibert M. From the Promiscuous Asenapine to Potent Fluorescent Ligands Acting at a Series of Aminergic G Protein Coupled Receptors. Journal of Medicinal Chemistry. PMID 29219316 DOI: 10.1021/acs.jmedchem.7b01220  0.486
2017 Scholler P, Nevoltris D, de Bundel D, Bossi S, Moreno-Delgado D, Rovira X, Møller TC, El Moustaine D, Mathieu M, Blanc E, McLean H, Dupuis E, Mathis G, Trinquet E, Daniel H, ... ... Pin JP, et al. Allosteric nanobodies uncover a role of hippocampal mGlu2 receptor homodimers in contextual fear consolidation. Nature Communications. 8: 1967. PMID 29213077 DOI: 10.1038/S41467-017-01489-1  0.529
2017 Liu J, Zhang Z, Moreno-Delgado D, Dalton JA, Rovira X, Trapero A, Goudet C, Llebaria A, Giraldo J, Yuan Q, Rondard P, Huang S, Liu J, Pin JP. Allosteric control of an asymmetric transduction in a G protein-coupled receptor heterodimer. Elife. 6. PMID 28829739 DOI: 10.7554/Elife.26985  0.541
2017 Dalton JAR, Pin JP, Giraldo J. Analysis of positive and negative allosteric modulation in metabotropic glutamate receptors 4 and 5 with a dual ligand. Scientific Reports. 7: 4944. PMID 28694498 DOI: 10.1038/s41598-017-05095-5  0.497
2017 Moreno Delgado D, Møller TC, Ster J, Giraldo J, Maurel D, Rovira X, Scholler P, Zwier JM, Perroy J, Durroux T, Trinquet E, Prezeau L, Rondard P, Pin JP. Pharmacological evidence for a metabotropic glutamate receptor heterodimer in neuronal cells. Elife. 6. PMID 28661401 DOI: 10.7554/Elife.25233  0.482
2017 Ayoub MA, Crépieux P, Koglin M, Parmentier M, Pin JP, Poupon A, Reiter E, Smit M, Steyaert J, Watier H, Wilkinson T. Antibodies targeting G protein-coupled receptors: Recent advances and therapeutic challenges. Mabs. 0. PMID 28475474 DOI: 10.1080/19420862.2017.1325052  0.427
2017 Font J, López-Cano M, Notartomaso S, Scarselli P, Di Pietro P, Bresolí-Obach R, Battaglia G, Malhaire F, Rovira X, Catena J, Giraldo J, Pin JP, Fernández-Dueñas V, Goudet C, Nonell S, et al. Optical control of pain in vivo with a photoactive mGlu5 receptor negative allosteric modulator. Elife. 6. PMID 28395733 DOI: 10.7554/Elife.23545  0.306
2017 Lecat-Guillet N, Monnier C, Rovira X, Kniazeff J, Lamarque L, Zwier JM, Trinquet E, Pin JP, Rondard P. FRET-Based Sensors Unravel Activation and Allosteric Modulation of the GABAB Receptor. Cell Chemical Biology. PMID 28286129 DOI: 10.1016/J.Chembiol.2017.02.011  0.565
2017 Gómez-Santacana X, Pittolo S, Rovira X, Lopez M, Zussy C, Dalton JA, Faucherre A, Jopling C, Pin JP, Ciruela F, Goudet C, Giraldo J, Gorostiza P, Llebaria A. Illuminating Phenylazopyridines To Photoswitch Metabotropic Glutamate Receptors: From the Flask to the Animals. Acs Central Science. 3: 81-91. PMID 28149957 DOI: 10.1021/Acscentsci.6B00353  0.466
2017 Scholler P, Moreno-Delgado D, Lecat-Guillet N, Doumazane E, Monnier C, Charrier-Savournin F, Fabre L, Chouvet C, Soldevila S, Lamarque L, Donsimoni G, Roux T, Zwier JM, Trinquet E, Rondard P, ... Pin JP, et al. HTS-compatible FRET-based conformational sensors clarify membrane receptor activation. Nature Chemical Biology. PMID 28135236 DOI: 10.1038/Nchembio.2286  0.524
2017 Gómez-Santacana X, Dalton JA, Rovira X, Pin JP, Goudet C, Gorostiza P, Giraldo J, Llebaria A. Positional isomers of bispyridine benzene derivatives induce efficacy changes on mGlu5 negative allosteric modulation. European Journal of Medicinal Chemistry. 127: 567-576. PMID 28109949 DOI: 10.1016/j.ejmech.2017.01.013  0.353
2017 Liu J, Zhang Z, Moreno-Delgado D, Dalton JA, Rovira X, Trapero A, Goudet C, Llebaria A, Giraldo J, Yuan Q, Rondard P, Huang S, Liu J, Pin J. Author response: Allosteric control of an asymmetric transduction in a G protein-coupled receptor heterodimer Elife. DOI: 10.7554/Elife.26985.025  0.491
2017 Delgado DM, Møller TC, Ster J, Giraldo J, Maurel D, Rovira X, Scholler P, Zwier JM, Perroy J, Durroux T, Trinquet E, Prezeau L, Rondard P, Pin J. Author response: Pharmacological evidence for a metabotropic glutamate receptor heterodimer in neuronal cells Elife. DOI: 10.7554/Elife.25233.032  0.453
2017 Cao A, Fatemi F, Oloffson L, Felekyan S, Seidel C, Rondard P, Pin J, Margeat E. Structural Dynamics of Single Metabotropic Glutamate Receptors in Solution Biophysical Journal. 112: 328a. DOI: 10.1016/J.Bpj.2016.11.1774  0.557
2016 Pin JP, Bettler B. Organization and functions of mGlu and GABAB receptor complexes. Nature. 540: 60-68. PMID 27905440 DOI: 10.1038/Nature20566  0.74
2016 ZIndel D, Engel S, Bottrill AR, Pin JP, Prézeau L, Tobin AB, Bünemann M, Krasel C, Butcher AJ. Identification of key phosphorylation sites in PTH1R which determine arrestin3 binding and fine tune receptor signaling. The Biochemical Journal. PMID 27623777 DOI: 10.1042/Bcj20160740  0.52
2016 Rovira X, Trapero A, Pittolo S, Zussy C, Faucherre A, Jopling C, Giraldo J, Pin JP, Gorostiza P, Goudet C, Llebaria A. OptoGluNAM4.1, a Photoswitchable Allosteric Antagonist for Real-Time Control of mGlu4 Receptor Activity. Cell Chemical Biology. PMID 27478159 DOI: 10.1016/j.chembiol.2016.06.013  0.54
2016 Huynh TH, Erichsen MN, Tora AS, Goudet C, Sagot E, Assaf Z, Thomsen C, Brodbeck R, Stensbøl TB, Bjørn-Yoshimoto WE, Nielsen B, Pin JP, Gefflaut T, Bunch L. New 4-Functionalized Glutamate Analogues Are Selective Agonists at Metabotropic Glutamate Receptor Subtype 2 or Selective Agonists at Metabotropic Glutamate Receptor Group III. Journal of Medicinal Chemistry. PMID 26814576 DOI: 10.1021/acs.jmedchem.5b01333  0.466
2016 Sun B, Chen L, Liu L, Xia Z, Pin JP, Nan F, Liu J. A negative allosteric modulator modulates GABAB receptor signaling through GB2 subunits. The Biochemical Journal. PMID 26772870 DOI: 10.1042/BJ20150979  0.58
2016 Cao A, Fatemi F, Rondard P, Pin J, Margeat E. Structural Dynamics of the Full-Length Metabotropic Glutamate Receptors by Single-Molecule FRET Biophysical Journal. 110: 637a. DOI: 10.1016/J.Bpj.2015.11.3408  0.588
2015 Dalton JA, Lans I, Rovira X, Malhaire F, Santacana XG, Pittolo S, Gorostiza P, Llebaria A, Goudet C, Pin JP, Giraldo J. Shining Light On An mGlu5 Photoswitchable NAM: A Theoretical Perspective. Current Neuropharmacology. PMID 26391742 DOI: 10.2174/1570159X13666150407231417  0.395
2015 Vischer HF, Castro M, Pin JP. G Protein-Coupled Receptor Multimers: A Question Still Open Despite the Use of Novel Approaches. Molecular Pharmacology. 88: 561-71. PMID 26138074 DOI: 10.1124/mol.115.099440  0.395
2015 Tora AS, Rovira X, Dione I, Bertrand HO, Brabet I, De Koninck Y, Doyon N, Pin JP, Acher F, Goudet C. Allosteric modulation of metabotropic glutamate receptors by chloride ions. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 29: 4174-88. PMID 26116702 DOI: 10.1096/Fj.14-269746  0.474
2015 Zhang Z, Zhang W, Huang S, Sun Q, Wang Y, Hu Y, Sun N, Zhang Y, Jiang Z, Minato N, Pin JP, Su L, Liu J. GABAB receptor promotes its own surface expression by recruiting a Rap1-dependent signaling cascade. Journal of Cell Science. 128: 2302-13. PMID 25967549 DOI: 10.1242/jcs.167056  0.453
2015 Ivashkin P, Lemonnier G, Tora AS, Pin JP, Goudet C, Jubault P, Pannecoucke X. Synthesis and studies on the mGluR agonist activity of FAP4 stereoisomers. Bioorganic & Medicinal Chemistry Letters. 25: 2523-6. PMID 25958247 DOI: 10.1016/j.bmcl.2015.04.043  0.468
2015 Faklaris O, Cottet M, Falco A, Villier B, Laget M, Zwier JM, Trinquet E, Mouillac B, Pin JP, Durroux T. Multicolor time-resolved Förster resonance energy transfer microscopy reveals the impact of GPCR oligomerization on internalization processes. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 29: 2235-46. PMID 25690655 DOI: 10.1096/Fj.14-260059  0.363
2015 Oueslati N, Hounsou C, Belhocine A, Rodriguez T, Dupuis E, Zwier JM, Trinquet E, Pin JP, Durroux T. Time-resolved FRET strategy to screen GPCR ligand library. Methods in Molecular Biology (Clifton, N.J.). 1272: 23-36. PMID 25563174 DOI: 10.1007/978-1-4939-2336-6_2  0.454
2015 Isberg V, de Graaf C, Bortolato A, Cherezov V, Katritch V, Marshall FH, Mordalski S, Pin JP, Stevens RC, Vriend G, Gloriam DE. Generic GPCR residue numbers - aligning topology maps while minding the gaps. Trends in Pharmacological Sciences. 36: 22-31. PMID 25541108 DOI: 10.1016/J.Tips.2014.11.001  0.377
2015 Rondard P, Pin JP. Dynamics and modulation of metabotropic glutamate receptors. Current Opinion in Pharmacology. 20: 95-101. PMID 25529199 DOI: 10.1016/J.Coph.2014.12.001  0.547
2015 Xue L, Rovira X, Scholler P, Zhao H, Liu J, Pin JP, Rondard P. Major ligand-induced rearrangement of the heptahelical domain interface in a GPCR dimer. Nature Chemical Biology. 11: 134-40. PMID 25503927 DOI: 10.1038/Nchembio.1711  0.548
2015 Commare B, Rigault D, Lemasson IA, Deschamps P, Tomas A, Roussel P, Brabet I, Goudet C, Pin JP, Leroux FR, Colobert F, Acher FC. Determination of the absolute configuration of phosphinic analogues of glutamate. Organic & Biomolecular Chemistry. 13: 1106-12. PMID 25417857 DOI: 10.1039/C4Ob01960A  0.467
2015 Fernández-Dueñas V, Taura JJ, Cottet M, Gómez-Soler M, López-Cano M, Ledent C, Watanabe M, Trinquet E, Pin JP, Luján R, Durroux T, Ciruela F. Untangling dopamine-adenosine receptor-receptor assembly in experimental parkinsonism in rats. Disease Models & Mechanisms. 8: 57-63. PMID 25398851 DOI: 10.1242/Dmm.018143  0.315
2015 Hounsou C, Margathe JF, Oueslati N, Belhocine A, Dupuis E, Thomas C, Mann A, Ilien B, Rognan D, Trinquet E, Hibert M, Pin JP, Bonnet D, Durroux T. Time-resolved FRET binding assay to investigate hetero-oligomer binding properties: proof of concept with dopamine D1/D3 heterodimer. Acs Chemical Biology. 10: 466-74. PMID 25350273 DOI: 10.1021/cb5007568  0.449
2015 Rovira X, Malhaire F, Scholler P, Rodrigo J, Gonzalez-Bulnes P, Llebaria A, Pin JP, Giraldo J, Goudet C. Overlapping binding sites drive allosteric agonism and positive cooperativity in type 4 metabotropic glutamate receptors. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 29: 116-30. PMID 25342125 DOI: 10.1096/fj.14-257287  0.511
2014 Olofsson L, Felekyan S, Doumazane E, Scholler P, Fabre L, Zwier JM, Rondard P, Seidel CA, Pin JP, Margeat E. Fine tuning of sub-millisecond conformational dynamics controls metabotropic glutamate receptors agonist efficacy. Nature Communications. 5: 5206. PMID 25323157 DOI: 10.1038/Ncomms6206  0.555
2014 Rovira X, Harrak Y, Trapero A, González-Bulnes P, Malhaire F, Pin JP, Goudet C, Giraldo J, Llebaria A. Exploring the active conformation of cyclohexane carboxylate positive allosteric modulators of the type 4 metabotropic glutamate receptor. Chemmedchem. 9: 2685-98. PMID 25196639 DOI: 10.1002/cmdc.201402190  0.466
2014 Pittolo S, Gómez-Santacana X, Eckelt K, Rovira X, Dalton J, Goudet C, Pin JP, Llobet A, Giraldo J, Llebaria A, Gorostiza P. An allosteric modulator to control endogenous G protein-coupled receptors with light. Nature Chemical Biology. 10: 813-5. PMID 25173999 DOI: 10.1038/Nchembio.1612  0.535
2014 Armando S, Quoyer J, Lukashova V, Maiga A, Percherancier Y, Heveker N, Pin JP, Prézeau L, Bouvier M. The chemokine CXC4 and CC2 receptors form homo- and heterooligomers that can engage their signaling G-protein effectors and βarrestin. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 28: 4509-23. PMID 25053617 DOI: 10.1096/Fj.13-242446  0.466
2014 Christopoulos A, Changeux JP, Catterall WA, Fabbro D, Burris TP, Cidlowski JA, Olsen RW, Peters JA, Neubig RR, Pin JP, Sexton PM, Kenakin TP, Ehlert FJ, Spedding M, Langmead CJ. International Union of Basic and Clinical Pharmacology. XC. multisite pharmacology: recommendations for the nomenclature of receptor allosterism and allosteric ligands. Pharmacological Reviews. 66: 918-47. PMID 25026896 DOI: 10.1124/Pr.114.008862  0.428
2014 Ayoub MA, Trebaux J, Vallaghe J, Charrier-Savournin F, Al-Hosaini K, Gonzalez Moya A, Pin JP, Pfleger KD, Trinquet E. Homogeneous time-resolved fluorescence-based assay to monitor extracellular signal-regulated kinase signaling in a high-throughput format. Frontiers in Endocrinology. 5: 94. PMID 25002860 DOI: 10.3389/fendo.2014.00094  0.434
2014 Sbai O, Monnier C, Dodé C, Pin JP, Hardelin JP, Rondard P. Biased signaling through G-protein-coupled PROKR2 receptors harboring missense mutations. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 28: 3734-44. PMID 24830383 DOI: 10.1096/Fj.13-243402  0.502
2014 Xu C, Zhang W, Rondard P, Pin JP, Liu J. Complex GABAB receptor complexes: how to generate multiple functionally distinct units from a single receptor. Frontiers in Pharmacology. 5: 12. PMID 24575041 DOI: 10.3389/Fphar.2014.00012  0.506
2014 Ferré S, Casadó V, Devi LA, Filizola M, Jockers R, Lohse MJ, Milligan G, Pin JP, Guitart X. G protein-coupled receptor oligomerization revisited: functional and pharmacological perspectives. Pharmacological Reviews. 66: 413-34. PMID 24515647 DOI: 10.1124/Pr.113.008052  0.653
2014 Gómez-Santacana X, Rovira X, Dalton JA, Goudet C, Pin JP, Gorostiza P, Giraldo J, Llebaria A. A double effect molecular switch leads to a novel potent negative allosteric modulator of metabotropic glutamate receptor 5 Medchemcomm. 5: 1548-1554. DOI: 10.1039/c4md00208c  0.389
2014 Olofsson L, Felekyan s, Doumazane E, Scholler P, Fabre L, Zwier J, Pin J, Seidel C, Rondard P, Margeat E. Specific Regulation of Transition Rates between Active and Inactive States of the Metabotropic Glutamate Receptor Determines Agonist Efficacy Biophysical Journal. 106: 100a-101a. DOI: 10.1016/J.Bpj.2013.11.627  0.537
2013 Alexander SP, Benson HE, Faccenda E, Pawson AJ, Sharman JL, McGrath JC, Catterall WA, Spedding M, Peters JA, Harmar AJ, Abul-Hasn N, Anderson CM, Anderson CM, Araiksinen MS, ... ... Pin JP, et al. The Concise Guide to PHARMACOLOGY 2013/14: overview. British Journal of Pharmacology. 170: 1449-58. PMID 24528237 DOI: 10.1111/Bph.12444  0.308
2013 Ayoub MA, Pin JP. Interaction of Protease-Activated Receptor 2 with G Proteins and β-Arrestin 1 Studied by Bioluminescence Resonance Energy Transfer. Frontiers in Endocrinology. 4: 196. PMID 24391627 DOI: 10.3389/fendo.2013.00196  0.376
2013 Vilar B, Busserolles J, Ling B, Laffray S, Ulmann L, Malhaire F, Chapuy E, Aissouni Y, Etienne M, Bourinet E, Acher F, Pin JP, Eschalier A, Goudet C. Alleviating pain hypersensitivity through activation of type 4 metabotropic glutamate receptor. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 33: 18951-65. PMID 24285900 DOI: 10.1523/Jneurosci.1221-13.2013  0.324
2013 Ivankova K, Turecek R, Fritzius T, Seddik R, Prezeau L, Comps-Agrar L, Pin JP, Fakler B, Besseyrias V, Gassmann M, Bettler B. Up-regulation of GABA(B) receptor signaling by constitutive assembly with the K+ channel tetramerization domain-containing protein 12 (KCTD12). The Journal of Biological Chemistry. 288: 24848-56. PMID 23843457 DOI: 10.1074/Jbc.M113.476770  0.69
2013 Davenport AP, Alexander SP, Sharman JL, Pawson AJ, Benson HE, Monaghan AE, Liew WC, Mpamhanga CP, Bonner TI, Neubig RR, Pin JP, Spedding M, Harmar AJ. International Union of Basic and Clinical Pharmacology. LXXXVIII. G protein-coupled receptor list: recommendations for new pairings with cognate ligands. Pharmacological Reviews. 65: 967-86. PMID 23686350 DOI: 10.1124/pr.112.007179  0.473
2013 Pin JP. Tuning synaptic activity with light-controlled GPCRs. Nature Neuroscience. 16: 377-9. PMID 23528934 DOI: 10.1038/nn.3363  0.357
2013 Doumazane E, Scholler P, Fabre L, Zwier JM, Trinquet E, Pin JP, Rondard P. Illuminating the activation mechanisms and allosteric properties of metabotropic glutamate receptors. Proceedings of the National Academy of Sciences of the United States of America. 110: E1416-25. PMID 23487753 DOI: 10.1073/Pnas.1215615110  0.581
2013 Cottet M, Faklaris O, Falco A, Trinquet E, Pin JP, Mouillac B, Durroux T. Fluorescent ligands to investigate GPCR binding properties and oligomerization. Biochemical Society Transactions. 41: 148-53. PMID 23356275 DOI: 10.1042/Bst20120237  0.431
2013 Scholler P, Zwier JM, Trinquet E, Rondard P, Pin JP, Prézeau L, Kniazeff J. Time-resolved Förster resonance energy transfer-based technologies to investigate G protein-coupled receptor machinery: high-throughput screening assays and future development. Progress in Molecular Biology and Translational Science. 113: 275-312. PMID 23244793 DOI: 10.1016/B978-0-12-386932-6.00007-7  0.391
2013 Amalric M, Lopez S, Goudet C, Fisone G, Battaglia G, Nicoletti F, Pin JP, Acher FC. Group III and subtype 4 metabotropic glutamate receptor agonists: discovery and pathophysiological applications in Parkinson's disease. Neuropharmacology. 66: 53-64. PMID 22664304 DOI: 10.1016/J.Neuropharm.2012.05.026  0.306
2012 Kniazeff J, Pin JP. [G-protein-coupled receptors dimers and oligomers: for which purpose? The GABA(B) receptor under investigation]. Mã©Decine Sciences : M/S. 28: 858-63. PMID 23067417 DOI: 10.1051/medsci/20122810014  0.608
2012 El Moustaine D, Granier S, Doumazane E, Scholler P, Rahmeh R, Bron P, Mouillac B, Banères JL, Rondard P, Pin JP. Distinct roles of metabotropic glutamate receptor dimerization in agonist activation and G-protein coupling. Proceedings of the National Academy of Sciences of the United States of America. 109: 16342-7. PMID 22988116 DOI: 10.1073/Pnas.1205838109  0.561
2012 Hlavackova V, Zabel U, Frankova D, Bätz J, Hoffmann C, Prezeau L, Pin JP, Blahos J, Lohse MJ. Sequential inter- and intrasubunit rearrangements during activation of dimeric metabotropic glutamate receptor 1. Science Signaling. 5: ra59. PMID 22894836 DOI: 10.1126/Scisignal.2002720  0.692
2012 Cottet M, Faklaris O, Maurel D, Scholler P, Doumazane E, Trinquet E, Pin JP, Durroux T. BRET and Time-resolved FRET strategy to study GPCR oligomerization: from cell lines toward native tissues. Frontiers in Endocrinology. 3: 92. PMID 22837753 DOI: 10.3389/fendo.2012.00092  0.376
2012 Lemonnier G, Lion C, Quirion JC, Pin JP, Goudet C, Jubault P. Α-amino-β-fluorocyclopropanecarboxylic acids as a new tool for drug development: synthesis of glutamic acid analogs and agonist activity towards metabotropic glutamate receptor 4. Bioorganic & Medicinal Chemistry. 20: 4716-26. PMID 22750138 DOI: 10.1016/j.bmc.2012.06.006  0.478
2012 Ayoub MA, Al-Senaidy A, Pin JP. Receptor-G protein interaction studied by bioluminescence resonance energy transfer: lessons from protease-activated receptor 1. Frontiers in Endocrinology. 3: 82. PMID 22737145 DOI: 10.3389/fendo.2012.00082  0.478
2012 Geng Y, Xiong D, Mosyak L, Malito DL, Kniazeff J, Chen Y, Burmakina S, Quick M, Bush M, Javitch JA, Pin JP, Fan QR. Structure and functional interaction of the extracellular domain of human GABA(B) receptor GBR2. Nature Neuroscience. 15: 970-8. PMID 22660477 DOI: 10.1038/Nn.3133  0.553
2012 Comps-Agrar L, Kniazeff J, Brock C, Trinquet E, Pin JP. Stability of GABAB receptor oligomers revealed by dual TR-FRET and drug-induced cell surface targeting. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 26: 3430-9. PMID 22613777 DOI: 10.1096/fj.12-203646  0.485
2012 Fazio F, Lionetto L, Molinaro G, Bertrand HO, Acher F, Ngomba RT, Notartomaso S, Curini M, Rosati O, Scarselli P, Di Marco R, Battaglia G, Bruno V, Simmaco M, Pin JP, et al. Cinnabarinic acid, an endogenous metabolite of the kynurenine pathway, activates type 4 metabotropic glutamate receptors. Molecular Pharmacology. 81: 643-56. PMID 22311707 DOI: 10.1124/Mol.111.074765  0.462
2012 Goudet C, Vilar B, Courtiol T, Deltheil T, Bessiron T, Brabet I, Oueslati N, Rigault D, Bertrand HO, McLean H, Daniel H, Amalric M, Acher F, Pin JP. A novel selective metabotropic glutamate receptor 4 agonist reveals new possibilities for developing subtype selective ligands with therapeutic potential. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 26: 1682-93. PMID 22223752 DOI: 10.1096/Fj.11-195941  0.537
2011 Tallet E, Fernandez I, Zhang C, Salsac M, Gregor N, Ayoub MA, Pin JP, Trinquet E, Goffin V. Investigation of prolactin receptor activation and blockade using time-resolved fluorescence resonance energy transfer. Frontiers in Endocrinology. 2: 29. PMID 22649370 DOI: 10.3389/fendo.2011.00029  0.371
2011 Huang S, Cao J, Jiang M, Labesse G, Liu J, Pin JP, Rondard P. Interdomain movements in metabotropic glutamate receptor activation. Proceedings of the National Academy of Sciences of the United States of America. 108: 15480-5. PMID 21896740 DOI: 10.1073/Pnas.1107775108  0.536
2011 Comps-Agrar L, Maurel D, Rondard P, Pin JP, Trinquet E, Prézeau L. Cell-surface protein-protein interaction analysis with time-resolved FRET and snap-tag technologies: application to G protein-coupled receptor oligomerization. Methods in Molecular Biology (Clifton, N.J.). 756: 201-14. PMID 21870227 DOI: 10.1007/978-1-61779-160-4_10  0.519
2011 Cottet M, Albizu L, Comps-Agrar L, Trinquet E, Pin JP, Mouillac B, Durroux T. Time resolved FRET strategy with fluorescent ligands to analyze receptor interactions in native tissues: application to GPCR oligomerization. Methods in Molecular Biology (Clifton, N.J.). 746: 373-87. PMID 21607869 DOI: 10.1007/978-1-61779-126-0_21  0.489
2011 Comps-Agrar L, Kniazeff J, Nørskov-Lauritsen L, Maurel D, Gassmann M, Gregor N, Prézeau L, Bettler B, Durroux T, Trinquet E, Pin JP. The oligomeric state sets GABA(B) receptor signalling efficacy. The Embo Journal. 30: 2336-49. PMID 21552208 DOI: 10.1038/Emboj.2011.143  0.687
2011 Kniazeff J, Prézeau L, Rondard P, Pin JP, Goudet C. Dimers and beyond: The functional puzzles of class C GPCRs. Pharmacology & Therapeutics. 130: 9-25. PMID 21256155 DOI: 10.1016/J.Pharmthera.2011.01.006  0.576
2011 Pellissier LP, Barthet G, Gaven F, Cassier E, Trinquet E, Pin JP, Marin P, Dumuis A, Bockaert J, Banères JL, Claeysen S. G protein activation by serotonin type 4 receptor dimers: evidence that turning on two protomers is more efficient. The Journal of Biological Chemistry. 286: 9985-97. PMID 21247891 DOI: 10.1074/Jbc.M110.201939  0.496
2011 Monnier C, Tu H, Bourrier E, Vol C, Lamarque L, Trinquet E, Pin JP, Rondard P. Trans-activation between 7TM domains: implication in heterodimeric GABAB receptor activation. The Embo Journal. 30: 32-42. PMID 21063387 DOI: 10.1038/Emboj.2010.270  0.574
2011 Nicoletti F, Bockaert J, Collingridge GL, Conn PJ, Ferraguti F, Schoepp DD, Wroblewski JT, Pin JP. Metabotropic glutamate receptors: from the workbench to the bedside. Neuropharmacology. 60: 1017-41. PMID 21036182 DOI: 10.1016/J.Neuropharm.2010.10.022  0.524
2011 Doumazane E, Scholler P, Zwier JM, Trinquet E, Rondard P, Pin JP. A new approach to analyze cell surface protein complexes reveals specific heterodimeric metabotropic glutamate receptors. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 25: 66-77. PMID 20826542 DOI: 10.1096/Fj.10-163147  0.558
2011 Rondard P, Goudet C, Kniazeff J, Pin JP, Prézeau L. The complexity of their activation mechanism opens new possibilities for the modulation of mGlu and GABAB class C G protein-coupled receptors. Neuropharmacology. 60: 82-92. PMID 20713070 DOI: 10.1016/J.Neuropharm.2010.08.009  0.609
2011 Acher FC, Selvam C, Pin JP, Goudet C, Bertrand HO. A critical pocket close to the glutamate binding site of mGlu receptors opens new possibilities for agonist design. Neuropharmacology. 60: 102-7. PMID 20621106 DOI: 10.1016/J.Neuropharm.2010.07.002  0.5
2011 Cottet M, Faklaris O, Zwier JM, Trinquet E, Pin JP, Durroux T. Original fluorescent ligand-based assays open new perspectives in G-protein coupled receptor drug screening Pharmaceuticals. 4: 202-214. DOI: 10.3390/ph4010202  0.372
2011 Prézeau L, Rondard P, Goudet C, Kniazeff J, Pin JP. Class C receptor activation mechanisms illustrated by mGlu and GABA B receptors. A review. Flavour and Fragrance Journal. 26: 218-222. DOI: 10.1002/Ffj.2044  0.602
2010 Albizu L, Cottet M, Kralikova M, Stoev S, Seyer R, Brabet I, Roux T, Bazin H, Bourrier E, Lamarque L, Breton C, Rives ML, Newman A, Javitch J, Trinquet E, ... ... Pin JP, et al. Time-resolved FRET between GPCR ligands reveals oligomers in native tissues. Nature Chemical Biology. 6: 587-94. PMID 20622858 DOI: 10.1038/Nchembio.396  0.527
2010 Khelashvili G, Dorff K, Shan J, Camacho-Artacho M, Skrabanek L, Vroling B, Bouvier M, Devi LA, George SR, Javitch JA, Lohse MJ, Milligan G, Neubig RR, Palczewski K, Parmentier M, ... Pin JP, et al. GPCR-OKB: the G Protein Coupled Receptor Oligomer Knowledge Base. Bioinformatics (Oxford, England). 26: 1804-5. PMID 20501551 DOI: 10.1093/Bioinformatics/Btq264  0.618
2010 Ayoub MA, Trinquet E, Pfleger KD, Pin JP. Differential association modes of the thrombin receptor PAR1 with Galphai1, Galpha12, and beta-arrestin 1. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 24: 3522-35. PMID 20410441 DOI: 10.1096/fj.10-154997  0.48
2010 Martín R, Durroux T, Ciruela F, Torres M, Pin JP, Sánchez-Prieto J. The metabotropic glutamate receptor mGlu7 activates phospholipase C, translocates munc-13-1 protein, and potentiates glutamate release at cerebrocortical nerve terminals. The Journal of Biological Chemistry. 285: 17907-17. PMID 20375012 DOI: 10.1074/Jbc.M109.080838  0.521
2010 Selvam C, Oueslati N, Lemasson IA, Brabet I, Rigault D, Courtiol T, Cesarini S, Triballeau N, Bertrand HO, Goudet C, Pin JP, Acher FC. A virtual screening hit reveals new possibilities for developing group III metabotropic glutamate receptor agonists. Journal of Medicinal Chemistry. 53: 2797-813. PMID 20218620 DOI: 10.1021/Jm901523T  0.566
2010 Tu H, Xu C, Zhang W, Liu Q, Rondard P, Pin JP, Liu J. GABAB receptor activation protects neurons from apoptosis via IGF-1 receptor transactivation. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 30: 749-59. PMID 20071540 DOI: 10.1523/Jneurosci.2343-09.2010  0.564
2010 Rovira X, Pin JP, Giraldo J. The asymmetric/symmetric activation of GPCR dimers as a possible mechanistic rationale for multiple signalling pathways. Trends in Pharmacological Sciences. 31: 15-21. PMID 19963287 DOI: 10.1016/j.tips.2009.10.008  0.471
2010 Prezeau L, Rives ML, Comps-Agrar L, Maurel D, Kniazeff J, Pin JP. Functional crosstalk between GPCRs: with or without oligomerization. Current Opinion in Pharmacology. 10: 6-13. PMID 19962942 DOI: 10.1016/j.coph.2009.10.009  0.584
2009 Miller J, Agarwal A, Devi LA, Fontanini K, Hamilton JA, Pin JP, Shields DC, Spek CA, Sakmar TP, Kuliopulos A, Hunt SW. Insider access: pepducin symposium explores a new approach to GPCR modulation. Annals of the New York Academy of Sciences. 1180: E1-12. PMID 19925639 DOI: 10.1111/J.1749-6632.2009.05326.X  0.506
2009 Pin JP, Comps-Agrar L, Maurel D, Monnier C, Rives ML, Trinquet E, Kniazeff J, Rondard P, Prézeau L. G-protein-coupled receptor oligomers: two or more for what? Lessons from mGlu and GABAB receptors. The Journal of Physiology. 587: 5337-44. PMID 19723778 DOI: 10.1113/Jphysiol.2009.179978  0.536
2009 Ayoub MA, Damian M, Gespach C, Ferrandis E, Lavergne O, De Wever O, Banères JL, Pin JP, Prévost GP. Inhibition of heterotrimeric G protein signaling by a small molecule acting on Galpha subunit. The Journal of Biological Chemistry. 284: 29136-45. PMID 19648112 DOI: 10.1074/jbc.M109.042333  0.51
2009 Rives ML, Vol C, Fukazawa Y, Tinel N, Trinquet E, Ayoub MA, Shigemoto R, Pin JP, Prézeau L. Crosstalk between GABAB and mGlu1a receptors reveals new insight into GPCR signal integration. The Embo Journal. 28: 2195-208. PMID 19590495 DOI: 10.1038/emboj.2009.177  0.585
2009 Beurrier C, Lopez S, Révy D, Selvam C, Goudet C, Lhérondel M, Gubellini P, Kerkerian-LeGoff L, Acher F, Pin JP, Amalric M. Electrophysiological and behavioral evidence that modulation of metabotropic glutamate receptor 4 with a new agonist reverses experimental parkinsonism. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 23: 3619-28. PMID 19525404 DOI: 10.1096/fj.09-131789  0.549
2009 Cuomo D, Martella G, Barabino E, Platania P, Vita D, Madeo G, Selvam C, Goudet C, Oueslati N, Pin JP, Acher F, Pisani A, Beurrier C, Melon C, Kerkerian-Le Goff L, et al. Metabotropic glutamate receptor subtype 4 selectively modulates both glutamate and GABA transmission in the striatum: implications for Parkinson's disease treatment. Journal of Neurochemistry. 109: 1096-105. PMID 19519781 DOI: 10.1111/j.1471-4159.2009.06036.x  0.343
2009 Ahier A, Rondard P, Gouignard N, Khayath N, Huang S, Trolet J, Donoghue DJ, Gauthier M, Pin JP, Dissous C. A new family of receptor tyrosine kinases with a venus flytrap binding domain in insects and other invertebrates activated by aminoacids. Plos One. 4: e5651. PMID 19461966 DOI: 10.1371/Journal.Pone.0005651  0.508
2009 Ferré S, Baler R, Bouvier M, Caron MG, Devi LA, Durroux T, Fuxe K, George SR, Javitch JA, Lohse MJ, Mackie K, Milligan G, Pfleger KD, Pin JP, Volkow ND, et al. Building a new conceptual framework for receptor heteromers. Nature Chemical Biology. 5: 131-4. PMID 19219011 DOI: 10.1038/Nchembio0309-131  0.533
2009 Goudet C, Magnaghi V, Landry M, Nagy F, Gereau RW, Pin JP. Metabotropic receptors for glutamate and GABA in pain. Brain Research Reviews. 60: 43-56. PMID 19146876 DOI: 10.1016/J.Brainresrev.2008.12.007  0.711
2009 Harmar AJ, Hills RA, Rosser EM, Jones M, Buneman OP, Dunbar DR, Greenhill SD, Hale VA, Sharman JL, Bonner TI, Catterall WA, Davenport AP, Delagrange P, Dollery CT, Foord SM, ... ... Pin JP, et al. IUPHAR-DB: the IUPHAR database of G protein-coupled receptors and ion channels. Nucleic Acids Research. 37: D680-5. PMID 18948278 DOI: 10.1093/Nar/Gkn728  0.321
2009 Monnier C, Dodé C, Fabre L, Teixeira L, Labesse G, Pin JP, Hardelin JP, Rondard P. PROKR2 missense mutations associated with Kallmann syndrome impair receptor signalling activity. Human Molecular Genetics. 18: 75-81. PMID 18826963 DOI: 10.1093/Hmg/Ddn318  0.449
2008 Kumpost J, Syrova Z, Kulihova L, Frankova D, Bologna JC, Hlavackova V, Prezeau L, Kralikova M, Hruskova B, Pin JP, Blahos J. Surface expression of metabotropic glutamate receptor variants mGluR1a and mGluR1b in transfected HEK293 cells. Neuropharmacology. 55: 409-18. PMID 18627772 DOI: 10.1016/j.neuropharm.2008.06.073  0.508
2008 Damian M, Mary S, Martin A, Pin JP, Banères JL. G protein activation by the leukotriene B4 receptor dimer. Evidence for an absence of trans-activation. The Journal of Biological Chemistry. 283: 21084-92. PMID 18490452 DOI: 10.1074/jbc.M710419200  0.532
2008 Maurel D, Comps-Agrar L, Brock C, Rives ML, Bourrier E, Ayoub MA, Bazin H, Tinel N, Durroux T, Prézeau L, Trinquet E, Pin JP. Cell-surface protein-protein interaction analysis with time-resolved FRET and snap-tag technologies: application to GPCR oligomerization. Nature Methods. 5: 561-7. PMID 18488035 DOI: 10.1038/nmeth.1213  0.508
2008 Rondard P, Huang S, Monnier C, Tu H, Blanchard B, Oueslati N, Malhaire F, Li Y, Trinquet E, Labesse G, Pin JP, Liu J. Functioning of the dimeric GABA(B) receptor extracellular domain revealed by glycan wedge scanning. The Embo Journal. 27: 1321-32. PMID 18388862 DOI: 10.1038/Emboj.2008.64  0.481
2008 Rovira X, Roche D, Serra J, Kniazeff J, Pin JP, Giraldo J. Modeling the binding and function of metabotropic glutamate receptors. The Journal of Pharmacology and Experimental Therapeutics. 325: 443-56. PMID 18287211 DOI: 10.1124/jpet.107.133967  0.544
2008 Chen Y, Goudet C, Pin JP, Conn PJ. N-{4-Chloro-2-[(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)methyl]phenyl}-2-hydroxybenzamide (CPPHA) acts through a novel site as a positive allosteric modulator of group 1 metabotropic glutamate receptors. Molecular Pharmacology. 73: 909-18. PMID 18056795 DOI: 10.1124/mol.107.040097  0.438
2008 Goudet C, Chapuy E, Alloui A, Acher F, Pin JP, Eschalier A. Group III metabotropic glutamate receptors inhibit hyperalgesia in animal models of inflammation and neuropathic pain. Pain. 137: 112-24. PMID 17900808 DOI: 10.1016/j.pain.2007.08.020  0.38
2008 Pin JP, Ayoub MA, Maurel D, Perroy J, Trinquet E. Energy Transfer Technologies to Monitor the Dynamics and Signaling Properties of G-Protein-Coupled Receptors in Living Cells Biophysical Analysis of Membrane Proteins: Investigating Structure and Function. 309-334. DOI: 10.1002/9783527621224.ch13  0.313
2007 Pin JP, Prézeau L. Allosteric modulators of GABA(B) receptors: mechanism of action and therapeutic perspective. Current Neuropharmacology. 5: 195-201. PMID 19305802 DOI: 10.2174/157015907781695919  0.495
2007 Brock C, Oueslati N, Soler S, Boudier L, Rondard P, Pin JP. Activation of a dimeric metabotropic glutamate receptor by intersubunit rearrangement. The Journal of Biological Chemistry. 282: 33000-8. PMID 17855348 DOI: 10.1074/Jbc.M702542200  0.591
2007 Selvam C, Goudet C, Oueslati N, Pin JP, Acher FC. L-(+)-2-Amino-4-thiophosphonobutyric acid (L-thioAP4), a new potent agonist of group III metabotropic glutamate receptors: increased distal acidity affords enhanced potency. Journal of Medicinal Chemistry. 50: 4656-64. PMID 17722902 DOI: 10.1021/jm070400y  0.4
2007 Sibille P, Lopez S, Brabet I, Valenti O, Oueslati N, Gaven F, Goudet C, Bertrand HO, Neyton J, Marino MJ, Amalric M, Pin JP, Acher FC. Synthesis and biological evaluation of 1-amino-2-phosphonomethylcyclopropanecarboxylic acids, new group III metabotropic glutamate receptor agonists. Journal of Medicinal Chemistry. 50: 3585-95. PMID 17602546 DOI: 10.1021/Jm070262C  0.527
2007 Tu H, Rondard P, Xu C, Bertaso F, Cao F, Zhang X, Pin JP, Liu J. Dominant role of GABAB2 and Gbetagamma for GABAB receptor-mediated-ERK1/2/CREB pathway in cerebellar neurons. Cellular Signalling. 19: 1996-2002. PMID 17582742 DOI: 10.1016/J.Cellsig.2007.05.004  0.449
2007 Skrabanek L, Murcia M, Bouvier M, Devi L, George SR, Lohse MJ, Milligan G, Neubig R, Palczewski K, Parmentier M, Pin JP, Vriend G, Javitch JA, Campagne F, Filizola M. Requirements and ontology for a G protein-coupled receptor oligomerization knowledge base. Bmc Bioinformatics. 8: 177. PMID 17537266 DOI: 10.1186/1471-2105-8-177  0.585
2007 Pin JP, Neubig R, Bouvier M, Devi L, Filizola M, Javitch JA, Lohse MJ, Milligan G, Palczewski K, Parmentier M, Spedding M. International Union of Basic and Clinical Pharmacology. LXVII. Recommendations for the recognition and nomenclature of G protein-coupled receptor heteromultimers. Pharmacological Reviews. 59: 5-13. PMID 17329545 DOI: 10.1124/Pr.59.1.5  0.63
2007 Binet V, Duthey B, Lecaillon J, Vol C, Quoyer J, Labesse G, Pin JP, Prézeau L. Common structural requirements for heptahelical domain function in class A and class C G protein-coupled receptors. The Journal of Biological Chemistry. 282: 12154-63. PMID 17310064 DOI: 10.1074/Jbc.M611071200  0.555
2007 Chen Y, Nong Y, Goudet C, Hemstapat K, de Paulis T, Pin JP, Conn PJ. Interaction of novel positive allosteric modulators of metabotropic glutamate receptor 5 with the negative allosteric antagonist site is required for potentiation of receptor responses. Molecular Pharmacology. 71: 1389-98. PMID 17303702 DOI: 10.1124/mol.106.032425  0.428
2007 Ayoub MA, Maurel D, Binet V, Fink M, Prézeau L, Ansanay H, Pin JP. Real-time analysis of agonist-induced activation of protease-activated receptor 1/Galphai1 protein complex measured by bioluminescence resonance energy transfer in living cells. Molecular Pharmacology. 71: 1329-40. PMID 17267663 DOI: 10.1124/Mol.106.030304  0.523
2007 Frauli M, Hubert N, Schann S, Triballeau N, Bertrand HO, Acher F, Neuville P, Pin JP, Prézeau L. Amino-pyrrolidine tricarboxylic acids give new insight into group III metabotropic glutamate receptor activation mechanism. Molecular Pharmacology. 71: 704-12. PMID 17167031 DOI: 10.1124/Mol.106.030254  0.575
2006 Damian M, Martin A, Mesnier D, Pin JP, Banères JL. Asymmetric conformational changes in a GPCR dimer controlled by G-proteins. The Embo Journal. 25: 5693-702. PMID 17139258 DOI: 10.1038/sj.emboj.7601449  0.566
2006 Trinquet E, Fink M, Bazin H, Grillet F, Maurin F, Bourrier E, Ansanay H, Leroy C, Michaud A, Durroux T, Maurel D, Malhaire F, Goudet C, Pin JP, Naval M, et al. D-myo-inositol 1-phosphate as a surrogate of D-myo-inositol 1,4,5-tris phosphate to monitor G protein-coupled receptor activation. Analytical Biochemistry. 358: 126-35. PMID 16965760 DOI: 10.1016/j.ab.2006.08.002  0.39
2006 Masdeu C, Faure H, Coulombe J, Schoenfelder A, Mann A, Brabet I, Pin JP, Traiffort E, Ruat M. Identification and characterization of Hedgehog modulator properties after functional coupling of Smoothened to G15. Biochemical and Biophysical Research Communications. 349: 471-9. PMID 16945339 DOI: 10.1016/J.Bbrc.2006.07.216  0.508
2006 Albizu L, Balestre MN, Breton C, Pin JP, Manning M, Mouillac B, Barberis C, Durroux T. Probing the existence of G protein-coupled receptor dimers by positive and negative ligand-dependent cooperative binding. Molecular Pharmacology. 70: 1783-91. PMID 16926282 DOI: 10.1124/Mol.106.025684  0.474
2006 Rondard P, Liu J, Huang S, Malhaire F, Vol C, Pinault A, Labesse G, Pin JP. Coupling of agonist binding to effector domain activation in metabotropic glutamate-like receptors. The Journal of Biological Chemistry. 281: 24653-61. PMID 16787923 DOI: 10.1074/Jbc.M602277200  0.576
2006 Frauli M, Neuville P, Vol C, Pin JP, Prézeau L. Among the twenty classical L-amino acids, only glutamate directly activates metabotropic glutamate receptors. Neuropharmacology. 50: 245-53. PMID 16310227 DOI: 10.1016/j.neuropharm.2005.09.016  0.542
2005 Davenport AP, Bonner TI, Foord SM, Harmar AJ, Neubig RR, Pin JP, Spedding M, Kojima M, Kangawa K. International Union of Pharmacology. LVI. Ghrelin receptor nomenclature, distribution, and function. Pharmacological Reviews. 57: 541-6. PMID 16382107 DOI: 10.1124/pr.57.4.1  0.453
2005 Brock C, Boudier L, Maurel D, Blahos J, Pin JP. Assembly-dependent surface targeting of the heterodimeric GABAB Receptor is controlled by COPI but not 14-3-3. Molecular Biology of the Cell. 16: 5572-8. PMID 16176975 DOI: 10.1091/mbc.E05-05-0400  0.461
2005 Pin JP, Kniazeff J, Liu J, Binet V, Goudet C, Rondard P, Prézeau L. Allosteric functioning of dimeric class C G-protein-coupled receptors. The Febs Journal. 272: 2947-55. PMID 15955055 DOI: 10.1111/J.1742-4658.2005.04728.X  0.468
2005 Foord SM, Bonner TI, Neubig RR, Rosser EM, Pin JP, Davenport AP, Spedding M, Harmar AJ. International Union of Pharmacology. XLVI. G protein-coupled receptor list. Pharmacological Reviews. 57: 279-88. PMID 15914470 DOI: 10.1124/pr.57.2.5  0.43
2005 Goudet C, Kniazeff J, Hlavackova V, Malhaire F, Maurel D, Acher F, Blahos J, Prézeau L, Pin JP. Asymmetric functioning of dimeric metabotropic glutamate receptors disclosed by positive allosteric modulators. The Journal of Biological Chemistry. 280: 24380-5. PMID 15863499 DOI: 10.1074/jbc.M502642200  0.632
2005 Triballeau N, Acher F, Brabet I, Pin JP, Bertrand HO. Virtual screening workflow development guided by the "receiver operating characteristic" curve approach. Application to high-throughput docking on metabotropic glutamate receptor subtype 4. Journal of Medicinal Chemistry. 48: 2534-47. PMID 15801843 DOI: 10.1021/Jm049092J  0.366
2005 Hlavackova V, Goudet C, Kniazeff J, Zikova A, Maurel D, Vol C, Trojanova J, Prézeau L, Pin JP, Blahos J. Evidence for a single heptahelical domain being turned on upon activation of a dimeric GPCR. The Embo Journal. 24: 499-509. PMID 15660124 DOI: 10.1038/sj.emboj.7600557  0.581
2004 Binet V, Goudet C, Brajon C, Le Corre L, Acher F, Pin JP, Prézeau L. Molecular mechanisms of GABA(B) receptor activation: new insights from the mechanism of action of CGP7930, a positive allosteric modulator. Biochemical Society Transactions. 32: 871-2. PMID 15494037 DOI: 10.1042/BST0320871  0.365
2004 Pin JP, Kniazeff J, Binet V, Liu J, Maurel D, Galvez T, Duthey B, Havlickova M, Blahos J, Prézeau L, Rondard P. Activation mechanism of the heterodimeric GABA(B) receptor. Biochemical Pharmacology. 68: 1565-72. PMID 15451400 DOI: 10.1016/J.Bcp.2004.06.035  0.448
2004 Kniazeff J, Bessis AS, Maurel D, Ansanay H, Prézeau L, Pin JP. Closed state of both binding domains of homodimeric mGlu receptors is required for full activity. Nature Structural & Molecular Biology. 11: 706-13. PMID 15235591 DOI: 10.1038/nsmb794  0.579
2004 Pin JP, Kniazeff J, Goudet C, Bessis AS, Liu J, Galvez T, Acher F, Rondard P, Prézeau L. The activation mechanism of class-C G-protein coupled receptors. Biology of the Cell / Under the Auspices of the European Cell Biology Organization. 96: 335-42. PMID 15207901 DOI: 10.1016/J.Biolcel.2004.03.005  0.527
2004 Maurel D, Kniazeff J, Mathis G, Trinquet E, Pin JP, Ansanay H. Cell surface detection of membrane protein interaction with homogeneous time-resolved fluorescence resonance energy transfer technology. Analytical Biochemistry. 329: 253-62. PMID 15158484 DOI: 10.1016/j.ab.2004.02.013  0.342
2004 Binet V, Brajon C, Le Corre L, Acher F, Pin JP, Prézeau L. The heptahelical domain of GABA(B2) is activated directly by CGP7930, a positive allosteric modulator of the GABA(B) receptor. The Journal of Biological Chemistry. 279: 29085-91. PMID 15126507 DOI: 10.1074/jbc.M400930200  0.445
2004 Liu J, Maurel D, Etzol S, Brabet I, Ansanay H, Pin JP, Rondard P. Molecular determinants involved in the allosteric control of agonist affinity in the GABAB receptor by the GABAB2 subunit. The Journal of Biological Chemistry. 279: 15824-30. PMID 14736871 DOI: 10.1074/Jbc.M313639200  0.548
2004 Kniazeff J, Saintot PP, Goudet C, Liu J, Charnet A, Guillon G, Pin JP. Locking the dimeric GABA(B) G-protein-coupled receptor in its active state. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 24: 370-7. PMID 14724235 DOI: 10.1523/JNEUROSCI.3141-03.2004  0.57
2004 Goudet C, Gaven F, Kniazeff J, Vol C, Liu J, Cohen-Gonsaud M, Acher F, Prézeau L, Pin JP. Heptahelical domain of metabotropic glutamate receptor 5 behaves like rhodopsin-like receptors. Proceedings of the National Academy of Sciences of the United States of America. 101: 378-83. PMID 14691258 DOI: 10.1073/pnas.0304699101  0.519
2004 Mitri C, Parmentier ML, Pin JP, Bockaert J, Grau Y. Divergent evolution in metabotropic glutamate receptors. A new receptor activated by an endogenous ligand different from glutamate in insects. The Journal of Biological Chemistry. 279: 9313-20. PMID 14660580 DOI: 10.1074/Jbc.M310878200  0.566
2004 Goudet C, Binet V, Prezeau L, Pin J. Allosteric modulators of class-C G-protein-coupled receptors open new possibilities for therapeutic application Drug Discovery Today: Therapeutic Strategies. 1: 125-133. DOI: 10.1016/J.DDSTR.2004.08.017  0.584
2003 Galvez T, Pin JP. [How do G-protein-coupled receptors work? The case of metabotropic glutamate and GABA receptors]. Mã©Decine Sciences : M/S. 19: 559-65. PMID 12836389 DOI: 10.1051/medsci/2003195559  0.627
2003 Havlickova M, Blahos J, Brabet I, Liu J, Hruskova B, Prézeau L, Pin JP. The second intracellular loop of metabotropic glutamate receptors recognizes C termini of G-protein alpha-subunits. The Journal of Biological Chemistry. 278: 35063-70. PMID 12829705 DOI: 10.1074/jbc.M306555200  0.502
2003 Pin JP, Galvez T, Prézeau L. Evolution, structure, and activation mechanism of family 3/C G-protein-coupled receptors. Pharmacology & Therapeutics. 98: 325-54. PMID 12782243 DOI: 10.1016/S0163-7258(03)00038-X  0.592
2003 Bessis AS, Vadesne G, Bourrat E, Bertho G, Pin JP, Acher FC. 3-carboxy-4-phosphonocyclopentane amino acids: new metabotropic glutamate receptor ligands. Amino Acids. 24: 303-10. PMID 12707813 DOI: 10.1007/s00726-002-0405-6  0.337
2003 Vicogne J, Pin JP, Lardans V, Capron M, Noël C, Dissous C. An unusual receptor tyrosine kinase of Schistosoma mansoni contains a Venus Flytrap module. Molecular and Biochemical Parasitology. 126: 51-62. PMID 12554084 DOI: 10.1016/S0166-6851(02)00249-9  0.379
2003 Fourgeaud L, Bessis AS, Rossignol F, Pin JP, Olivo-Marin JC, Hémar A. The metabotropic glutamate receptor mGluR5 is endocytosed by a clathrin-independent pathway. The Journal of Biological Chemistry. 278: 12222-30. PMID 12529370 DOI: 10.1074/jbc.M205663200  0.499
2003 Galvez T, Pin J. Comment fonctionne un récepteur couplé aux protéines G? Le cas des récepteurs métabotropiques du glutamate et du GABA M S-Medecine Sciences. 19: 559-565. DOI: 10.7202/006625Ar  0.31
2003 Prezeau L, Parmentier M, Carroll F, Pin J. Inverse agonists to explore the mechanisms of metabotropic glutamate receptor activity International Congress Series. 1249: 235-244. DOI: 10.1016/S0531-5131(03)00601-0  0.45
2003 Fagni L, Ango F, Prezeau L, Worley PF, Pin J, Bockaert J. Control of constitutive activity of metabotropic glutamate receptors by Homer proteins International Congress Series. 1249: 245-251. DOI: 10.1016/S0531-5131(03)00600-9  0.436
2002 Pin JP, Acher F. The metabotropic glutamate receptors: structure, activation mechanism and pharmacology. Current Drug Targets. Cns and Neurological Disorders. 1: 297-317. PMID 12769621 DOI: 10.1016/B978-0-12-397032-9.00012-1  0.61
2002 Kniazeff J, Galvez T, Labesse G, Pin JP. No ligand binding in the GB2 subunit of the GABA(B) receptor is required for activation and allosteric interaction between the subunits. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 22: 7352-61. PMID 12196556 DOI: 10.1523/Jneurosci.22-17-07352.2002  0.509
2002 Bessis AS, Rondard P, Gaven F, Brabet I, Triballeau N, Prezeau L, Acher F, Pin JP. Closure of the Venus flytrap module of mGlu8 receptor and the activation process: Insights from mutations converting antagonists into agonists. Proceedings of the National Academy of Sciences of the United States of America. 99: 11097-102. PMID 12151600 DOI: 10.1073/Pnas.162138699  0.591
2002 Havlickova M, Prezeau L, Duthey B, Bettler B, Pin JP, Blahos J. The intracellular loops of the GB2 subunit are crucial for G-protein coupling of the heteromeric gamma-aminobutyrate B receptor. Molecular Pharmacology. 62: 343-50. PMID 12130687 DOI: 10.1124/Mol.62.2.343  0.712
2002 Bertrand HO, Bessis AS, Pin JP, Acher FC. Common and selective molecular determinants involved in metabotopic glutamate receptor agonist activity. Journal of Medicinal Chemistry. 45: 3171-83. PMID 12109902 DOI: 10.1021/Jm010323L  0.481
2002 Ango F, Robbe D, Tu JC, Xiao B, Worley PF, Pin JP, Bockaert J, Fagni L. Homer-dependent cell surface expression of metabotropic glutamate receptor type 5 in neurons. Molecular and Cellular Neurosciences. 20: 323-9. PMID 12093163 DOI: 10.1006/Mcne.2002.1100  0.434
2002 Parmentier ML, Prézeau L, Bockaert J, Pin JP. A model for the functioning of family 3 GPCRs. Trends in Pharmacological Sciences. 23: 268-74. PMID 12084632 DOI: 10.1016/S0165-6147(02)02016-3  0.595
2002 Perroy J, El Far O, Bertaso F, Pin JP, Betz H, Bockaert J, Fagni L. PICK1 is required for the control of synaptic transmission by the metabotropic glutamate receptor 7. The Embo Journal. 21: 2990-9. PMID 12065412 DOI: 10.1093/Emboj/Cdf313  0.408
2002 Gaillard I, Rouquier S, Pin JP, Mollard P, Richard S, Barnabé C, Demaille J, Giorgi D. A single olfactory receptor specifically binds a set of odorant molecules. The European Journal of Neuroscience. 15: 409-18. PMID 11876768 DOI: 10.1046/J.0953-816X.2001.01871.X  0.302
2002 Gasparini F, Kuhn R, Pin JP. Allosteric modulators of group I metabotropic glutamate receptors: novel subtype-selective ligands and therapeutic perspectives. Current Opinion in Pharmacology. 2: 43-9. PMID 11786307 DOI: 10.1016/S1471-4892(01)00119-9  0.563
2002 Duthey B, Caudron S, Perroy J, Bettler B, Fagni L, Pin JP, Prézeau L. A single subunit (GB2) is required for G-protein activation by the heterodimeric GABA(B) receptor. The Journal of Biological Chemistry. 277: 3236-41. PMID 11711539 DOI: 10.1074/jbc.M108900200  0.667
2001 Pin JP, Parmentier ML, Prézeau L. Positive allosteric modulators for gamma-aminobutyric acid(B) receptors open new routes for the development of drugs targeting family 3 G-protein-coupled receptors. Molecular Pharmacology. 60: 881-4. PMID 11641414 DOI: 10.1124/Mol.60.5.881  0.585
2001 Perroy J, Gutierrez GJ, Coulon V, Bockaert J, Pin JP, Fagni L. The C terminus of the metabotropic glutamate receptor subtypes 2 and 7 specifies the receptor signaling pathways. The Journal of Biological Chemistry. 276: 45800-5. PMID 11584003 DOI: 10.1074/Jbc.M106876200  0.472
2001 Ango F, Prézeau L, Muller T, Tu JC, Xiao B, Worley PF, Pin JP, Bockaert J, Fagni L. Agonist-independent activation of metabotropic glutamate receptors by the intracellular protein Homer. Nature. 411: 962-5. PMID 11418862 DOI: 10.1038/35082096  0.527
2001 Bessis AS, Bolte J, Pin JP, Acher F. New probes of the agonist binding site of metabotropic glutamate receptors. Bioorganic & Medicinal Chemistry Letters. 11: 1569-72. PMID 11412983 DOI: 10.1016/S0960-894X(01)00158-5  0.448
2001 Galvez T, Duthey B, Kniazeff J, Blahos J, Rovelli G, Bettler B, Prézeau L, Pin JP. Allosteric interactions between GB1 and GB2 subunits are required for optimal GABA(B) receptor function. The Embo Journal. 20: 2152-9. PMID 11331581 DOI: 10.1093/Emboj/20.9.2152  0.722
2001 Carroll FY, Stolle A, Beart PM, Voerste A, Brabet I, Mauler F, Joly C, Antonicek H, Bockaert J, Müller T, Pin JP, Prézeau L. BAY36-7620: a potent non-competitive mGlu1 receptor antagonist with inverse agonist activity. Molecular Pharmacology. 59: 965-73. PMID 11306677 DOI: 10.1124/Mol.59.5.965  0.513
2001 Costantino G, Maltoni K, Marinozzi M, Camaioni E, Prezeau L, Pin JP, Pellicciari R. Synthesis and biological evaluation of 2-(3'-(1H-tetrazol-5-yl) bicyclo[1.1.1]pent-1-yl)glycine (S-TBPG), a novel mGlu1 receptor antagonist. Bioorganic & Medicinal Chemistry. 9: 221-7. PMID 11249114 DOI: 10.1016/S0968-0896(00)00270-4  0.41
2001 Pagano A, Rovelli G, Mosbacher J, Lohmann T, Duthey B, Stauffer D, Ristig D, Schuler V, Meigel I, Lampert C, Stein T, Prezeau L, Blahos J, Pin J, Froestl W, et al. C-terminal interaction is essential for surface trafficking but not for heteromeric assembly of GABA(b) receptors. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 21: 1189-202. PMID 11160389 DOI: 10.1523/Jneurosci.21-04-01189.2001  0.62
2001 Blahos J, Fischer T, Brabet I, Stauffer D, Rovelli G, Bockaert J, Pin JP. A novel site on the Galpha -protein that recognizes heptahelical receptors. The Journal of Biological Chemistry. 276: 3262-9. PMID 11027680 DOI: 10.1074/Jbc.M004880200  0.488
2000 Bessis AS, Bertrand HO, Galvez T, De Colle C, Pin JP, Acher F. Three-dimensional model of the extracellular domain of the type 4a metabotropic glutamate receptor: new insights into the activation process. Protein Science : a Publication of the Protein Society. 9: 2200-9. PMID 11152130 DOI: 10.1110/Ps.9.11.2200  0.499
2000 Ango F, Pin JP, Tu JC, Xiao B, Worley PF, Bockaert J, Fagni L. Dendritic and axonal targeting of type 5 metabotropic glutamate receptor is regulated by homer1 proteins and neuronal excitation. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 20: 8710-6. PMID 11102477 DOI: 10.1523/Jneurosci.20-23-08710.2000  0.431
2000 Galvez T, Prezeau L, Milioti G, Franek M, Joly C, Froestl W, Bettler B, Bertrand HO, Blahos J, Pin JP. Mapping the agonist-binding site of GABAB type 1 subunit sheds light on the activation process of GABAB receptors. The Journal of Biological Chemistry. 275: 41166-74. PMID 10986293 DOI: 10.1074/jbc.M007848200  0.647
2000 Pagano A, Ruegg D, Litschig S, Stoehr N, Stierlin C, Heinrich M, Floersheim P, Prezèau L, Carroll F, Pin JP, Cambria A, Vranesic I, Flor PJ, Gasparini F, Kuhn R. The non-competitive antagonists 2-methyl-6-(phenylethynyl)pyridine and 7-hydroxyiminocyclopropan[b]chromen-1a-carboxylic acid ethyl ester interact with overlapping binding pockets in the transmembrane region of group I metabotropic glutamate receptors. The Journal of Biological Chemistry. 275: 33750-8. PMID 10934211 DOI: 10.1074/Jbc.M006230200  0.4
2000 De Colle C, Bessis AS, Bockaert J, Acher F, Pin JP. Pharmacological characterization of the rat metabotropic glutamate receptor type 8a revealed strong similarities and slight differences with the type 4a receptor. European Journal of Pharmacology. 394: 17-26. PMID 10771029 DOI: 10.1016/S0014-2999(00)00113-8  0.572
2000 Parmentier ML, Galvez T, Acher F, Peyre B, Pellicciari R, Grau Y, Bockaert J, Pin JP. Conservation of the ligand recognition site of metabotropic glutamate receptors during evolution. Neuropharmacology. 39: 1119-31. PMID 10760355 DOI: 10.1016/S0028-3908(99)00204-X  0.493
2000 Galvez T, Urwyler S, Prézeau L, Mosbacher J, Joly C, Malitschek B, Heid J, Brabet I, Froestl W, Bettler B, Kaupmann K, Pin JP. Ca(2+) requirement for high-affinity gamma-aminobutyric acid (GABA) binding at GABA(B) receptors: involvement of serine 269 of the GABA(B)R1 subunit. Molecular Pharmacology. 57: 419-26. PMID 10692480 DOI: 10.1124/Mol.57.3.419  0.602
2000 Dauban P, de Saint-Fuscien C, Acher F, Prézeau L, Brabet I, Pin JP, Dodd RH. First enantiospecific synthesis of a 3,4-dihydroxy-L-glutamic acid [(3S,4S)-DHGA], a new mGluR1 agonist. Bioorganic & Medicinal Chemistry Letters. 10: 129-33. PMID 10673095 DOI: 10.1016/S0960-894X(99)00641-1  0.43
1999 Franek M, Pagano A, Kaupmann K, Bettler B, Pin JP, Blahos J. The heteromeric GABA-B receptor recognizes G-protein alpha subunit C-termini. Neuropharmacology. 38: 1657-66. PMID 10587081 DOI: 10.1016/S0028-3908(99)00135-5  0.682
1999 Lafon-Cazal M, Viennois G, Kuhn R, Malitschek B, Pin JP, Shigemoto R, Bockaert J. mGluR7-like receptor and GABA(B) receptor activation enhance neurotoxic effects of N-methyl-D-aspartate in cultured mouse striatal GABAergic neurones. Neuropharmacology. 38: 1631-40. PMID 10530824 DOI: 10.1016/S0028-3908(99)00124-0  0.353
1999 Bessis AS, Jullian N, Coudert E, Pin JP, Acher F. Extended glutamate activates metabotropic receptor types 1, 2 and 4: selective features at mGluR4 binding site. Neuropharmacology. 38: 1543-51. PMID 10530816 DOI: 10.1016/S0028-3908(99)00096-9  0.419
1999 Ango F, Albani-Torregrossa S, Joly C, Robbe D, Michel JM, Pin JP, Bockaert J, Fagni L. A simple method to transfer plasmid DNA into neuronal primary cultures: functional expression of the mGlu5 receptor in cerebellar granule cells. Neuropharmacology. 38: 793-803. PMID 10465683 DOI: 10.1016/S0028-3908(99)00005-2  0.484
1999 Pfaff T, Malitschek B, Kaupmann K, Prézeau L, Pin JP, Bettler B, Karschin A. Alternative splicing generates a novel isoform of the rat metabotropic GABA(B)R1 receptor. The European Journal of Neuroscience. 11: 2874-82. PMID 10457184 DOI: 10.1046/J.1460-9568.1999.00704.X  0.658
1999 Pin JP, De Colle C, Bessis AS, Acher F. New perspectives for the development of selective metabotropic glutamate receptor ligands. European Journal of Pharmacology. 375: 277-94. PMID 10443583 DOI: 10.1016/S0014-2999(99)00258-7  0.582
1999 Malitschek B, Schweizer C, Keir M, Heid J, Froestl W, Mosbacher J, Kuhn R, Henley J, Joly C, Pin JP, Kaupmann K, Bettler B. The N-terminal domain of gamma-aminobutyric Acid(B) receptors is sufficient to specify agonist and antagonist binding. Molecular Pharmacology. 56: 448-54. PMID 10419566 DOI: 10.1124/Mol.56.2.448  0.631
1999 Jullian N, Brabet I, Pin JP, Acher FC. Agonist selectivity of mGluR1 and mGluR2 metabotropic receptors: a different environment but similar recognition of an extended glutamate conformation. Journal of Medicinal Chemistry. 42: 1546-55. PMID 10229625 DOI: 10.1021/jm980571q  0.471
1999 Galvez T, Parmentier ML, Joly C, Malitschek B, Kaupmann K, Kuhn R, Bittiger H, Froestl W, Bettler B, Pin JP. Mutagenesis and modeling of the GABAB receptor extracellular domain support a venus flytrap mechanism for ligand binding. The Journal of Biological Chemistry. 274: 13362-9. PMID 10224098 DOI: 10.1074/Jbc.274.19.13362  0.685
1999 Bockaert J, Pin JP. Molecular tinkering of G protein-coupled receptors: an evolutionary success. The Embo Journal. 18: 1723-9. PMID 10202136 DOI: 10.1093/Emboj/18.7.1723  0.387
1999 Lafon-Cazal M, Fagni L, Guiraud MJ, Mary S, Lerner-Natoli M, Pin JP, Shigemoto R, Bockaert J. mGluR7-like metabotropic glutamate receptors inhibit NMDA-mediated excitotoxicity in cultured mouse cerebellar granule neurons. The European Journal of Neuroscience. 11: 663-72. PMID 10051767 DOI: 10.1046/J.1460-9568.1999.00475.X  0.374
1999 Litschig S, Gasparini F, Rueegg D, Stoehr N, Flor PJ, Vranesic I, Prézeau L, Pin JP, Thomsen C, Kuhn R. CPCCOEt, a noncompetitive metabotropic glutamate receptor 1 antagonist, inhibits receptor signaling without affecting glutamate binding. Molecular Pharmacology. 55: 453-61. PMID 10051528  0.479
1998 Corti C, Restituito S, Rimland JM, Brabet I, Corsi M, Pin JP, Ferraguti F. Cloning and characterization of alternative mRNA forms for the rat metabotropic glutamate receptors mGluR7 and mGluR8. The European Journal of Neuroscience. 10: 3629-41. PMID 9875342 DOI: 10.1046/j.1460-9568.1998.00371.x  0.783
1998 Pellicciari R, Costantino G, Giovagnoni E, Mattoli L, Brabet I, Pin JP. Synthesis and preliminary evaluation of (S)-2-(4'-carboxycubyl)glycine, a new selective mGluR1 antagonist. Bioorganic & Medicinal Chemistry Letters. 8: 1569-74. PMID 9873392 DOI: 10.1016/S0960-894X(98)00265-0  0.428
1998 Brabet I, Parmentier ML, De Colle C, Bockaert J, Acher F, Pin JP. Comparative effect of L-CCG-I, DCG-IV and gamma-carboxy-L-glutamate on all cloned metabotropic glutamate receptor subtypes. Neuropharmacology. 37: 1043-51. PMID 9833633 DOI: 10.1016/S0028-3908(98)00091-4  0.549
1998 Bockaert J, Pin JP. [Use of a G-protein-coupled receptor to communicate. An evolutionary success]. Comptes Rendus De L'Acadã©Mie Des Sciences. Sã©Rie Iii, Sciences De La Vie. 321: 529-51. PMID 9769853 DOI: 10.1016/S0764-4469(98)80455-1  0.497
1998 Copani A, Casabona G, Bruno V, Caruso A, Condorelli DF, Messina A, Di Giorgi Gerevini V, Pin JP, Kuhn R, Knöpfel T, Nicoletti F. The metabotropic glutamate receptor mGlu5 controls the onset of developmental apoptosis in cultured cerebellar neurons. The European Journal of Neuroscience. 10: 2173-84. PMID 9753103 DOI: 10.1046/j.1460-9568.1998.00230.x  0.417
1998 Blahos J, Mary S, Perroy J, de Colle C, Brabet I, Bockaert J, Pin JP. Extreme C terminus of G protein alpha-subunits contains a site that discriminates between Gi-coupled metabotropic glutamate receptors. The Journal of Biological Chemistry. 273: 25765-9. PMID 9748247 DOI: 10.1074/Jbc.273.40.25765  0.6
1998 Pin JP. Synaptic transmission. The two faces of glutamate. Nature. 394: 19-21. PMID 9665121 DOI: 10.1038/27771  0.401
1998 Tellier F, Acher F, Brabet I, Pin JP, Azerad R. Aminobicyclo[2.2.1.]heptane dicarboxylic acids (ABHD), rigid analogs of ACPD and glutamic acid: synthesis and pharmacological activity on metabotropic receptors mGluR1 and mGluR2. Bioorganic & Medicinal Chemistry. 6: 195-208. PMID 9547943 DOI: 10.1016/S0968-0896(97)10031-1  0.507
1998 Parmentier ML, Joly C, Restituito S, Bockaert J, Grau Y, Pin JP. The G protein-coupling profile of metabotropic glutamate receptors, as determined with exogenous G proteins, is independent of their ligand recognition domain. Molecular Pharmacology. 53: 778-86. PMID 9547371 DOI: 10.1124/Mol.53.4.778  0.816
1998 Mary S, Gomeza J, Prézeau L, Bockaert J, Pin JP. A cluster of basic residues in the carboxyl-terminal tail of the short metabotropic glutamate receptor 1 variants impairs their coupling to phospholipase C. The Journal of Biological Chemistry. 273: 425-32. PMID 9417099 DOI: 10.1074/Jbc.273.1.425  0.491
1997 Mary S, Stephan D, Gomeza J, Bockaert J, Pruss RM, Pin JP. The rat mGlu1d receptor splice variant shares functional properties with the other short isoforms of mGlu1 receptor. European Journal of Pharmacology. 335: 65-72. PMID 9371547 DOI: 10.1016/S0014-2999(97)01155-2  0.562
1997 Acher FC, Tellier FJ, Azerad R, Brabet IN, Fagni L, Pin JP. Synthesis and pharmacological characterization of aminocyclopentanetricarboxylic acids: new tools to discriminate between metabotropic glutamate receptor subtypes. Journal of Medicinal Chemistry. 40: 3119-29. PMID 9301676 DOI: 10.1021/jm970207b  0.393
1997 Conn PJ, Pin JP. Pharmacology and functions of metabotropic glutamate receptors. Annual Review of Pharmacology and Toxicology. 37: 205-37. PMID 9131252 DOI: 10.1146/annurev.pharmtox.37.1.205  0.47
1997 Todeschi N, Gharbi-Benarous J, Acher F, Larue V, Pin JP, Bockaert J, Azerad R, Girault JP. Conformational analysis of glutamic acid analogues as probes of glutamate receptors using molecular modelling and NMR methods. Comparison with specific agonists. Bioorganic & Medicinal Chemistry. 5: 335-52. PMID 9061198 DOI: 10.1016/S0968-0896(96)00252-0  0.467
1996 Gomeza J, Mary S, Brabet I, Parmentier ML, Restituito S, Bockaert J, Pin JP. Coupling of metabotropic glutamate receptors 2 and 4 to G alpha 15, G alpha 16, and chimeric G alpha q/i proteins: characterization of new antagonists. Molecular Pharmacology. 50: 923-30. PMID 8863838  0.728
1996 McCool BA, Pin JP, Brust PF, Harpold MM, Lovinger DM. Functional coupling of rat group II metabotropic glutamate receptors to an omega-conotoxin GVIA-sensitive calcium channel in human embryonic kidney 293 cells. Molecular Pharmacology. 50: 912-22. PMID 8863837  0.423
1996 Parmentier ML, Pin JP, Bockaert J, Grau Y. Cloning and functional expression of a Drosophila metabotropic glutamate receptor expressed in the embryonic CNS. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 16: 6687-94. PMID 8824309 DOI: 10.1523/Jneurosci.16-21-06687.1996  0.583
1996 Manahan-Vaughan D, Reiser M, Pin JP, Wilsch V, Bockaert J, Reymann KG, Riedel G. Physiological and pharmacological profile of trans-azetidine-2,4-dicarboxylic acid: metabotropic glutamate receptor agonism and effects on long-term potentiation. Neuroscience. 72: 999-1008. PMID 8735225 DOI: 10.1016/0306-4522(95)00594-3  0.376
1996 Flor PJ, Gomeza J, Tones MA, Kuhn R, Pin JP, Knöpfel T. The C-terminal domain of the mGluR1 metabotropic glutamate receptor affects sensitivity to agonists. Journal of Neurochemistry. 67: 58-63. PMID 8667026  0.376
1996 Prézeau L, Gomeza J, Ahern S, Mary S, Galvez T, Bockaert J, Pin JP. Changes in the carboxyl-terminal domain of metabotropic glutamate receptor 1 by alternative splicing generate receptors with differing agonist-independent activity. Molecular Pharmacology. 49: 422-9. PMID 8643081  0.46
1996 Gomeza J, Joly C, Kuhn R, Knöpfel T, Bockaert J, Pin JP. The second intracellular loop of metabotropic glutamate receptor 1 cooperates with the other intracellular domains to control coupling to G-proteins. The Journal of Biological Chemistry. 271: 2199-205. PMID 8567679 DOI: 10.1074/Jbc.271.4.2199  0.576
1995 Pin JP, Gomeza J, Joly C, Bockaert J. The metabotropic glutamate receptors: their second intracellular loop plays a critical role in the G-protein coupling specificity. Biochemical Society Transactions. 23: 91-6. PMID 7758811 DOI: 10.1042/Bst0230091  0.456
1995 Joly C, Gomeza J, Brabet I, Curry K, Bockaert J, Pin JP. Molecular, functional, and pharmacological characterization of the metabotropic glutamate receptor type 5 splice variants: comparison with mGluR1. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 15: 3970-81. PMID 7751958 DOI: 10.1523/Jneurosci.15-05-03970.1995  0.582
1995 Pin JP, Duvoisin R. The metabotropic glutamate receptors: structure and functions. Neuropharmacology. 34: 1-26. PMID 7623957 DOI: 10.1016/0028-3908(94)00129-G  0.72
1995 Pin JP, Bockaert J. Get receptive to metabotropic glutamate receptors. Current Opinion in Neurobiology. 5: 342-9. PMID 7580157 DOI: 10.1016/0959-4388(95)80047-6  0.586
1995 Tellier F, Acher F, Brabet I, Pin J, Bockaert J, Azerad R. Synthesis of conformationally-constrained stereospecific analogs of glutamic acid as antagonists of metabotropic receptors Bioorganic & Medicinal Chemistry Letters. 5: 2627-2632. DOI: 10.1016/0960-894X(95)00457-5  0.481
1994 Bockaert J, Pin J, Fagni L. Metabotropic glutamate receptors: an original family of G protein-coupled receptors. Fundamental & Clinical Pharmacology. 7: 473-85. PMID 8314195 DOI: 10.1111/j.1472-8206.1993.tb00252.x  0.577
1994 Pin JP, Joly C, Heinemann SF, Bockaert J. Domains involved in the specificity of G protein activation in phospholipase C-coupled metabotropic glutamate receptors. The Embo Journal. 13: 342-8. PMID 8313879  0.694
1994 Prézeau L, Carrette J, Helpap B, Curry K, Pin JP, Bockaert J. Pharmacological characterization of metabotropic glutamate receptors in several types of brain cells in primary cultures. Molecular Pharmacology. 45: 570-7. PMID 8183235  0.365
1994 Didier M, Mienville JM, Soubrié P, Bockaert J, Berman S, Bursztajn S, Pin JP. Plasticity of NMDA receptor expression during mouse cerebellar granule cell development. The European Journal of Neuroscience. 6: 1536-43. PMID 7850018 DOI: 10.1111/J.1460-9568.1994.Tb00544.X  0.412
1993 Didier M, Héaulme M, Gonalons N, Soubrié P, Bockaert J, Pin JP. 35 mM K(+)-stimulated 45Ca2+ uptake in cerebellar granule cell cultures mainly results from NMDA receptor activation. European Journal of Pharmacology. 244: 57-65. PMID 7678398 DOI: 10.1016/0922-4106(93)90059-I  0.396
1993 Bockaert J, Marin P, Lafon-Cazal M, Pin JP, Dumuis A. Arachidonic acid and nitric oxide production by glutamate receptors in cultured neurons Seminars in Neuroscience. 5: 181-188. DOI: 10.1016/S1044-5765(05)80051-X  0.404
1992 Pin JP, Waeber C, Prezeau L, Bockaert J, Heinemann SF. Alternative splicing generates metabotropic glutamate receptors inducing different patterns of calcium release in Xenopus oocytes. Proceedings of the National Academy of Sciences of the United States of America. 89: 10331-5. PMID 1438218 DOI: 10.1073/Pnas.89.21.10331  0.644
1992 Tapia-Arancibia L, Rage F, Récasens M, Pin JP. NMDA receptor activation stimulates phospholipase A2 and somatostatin release from rat cortical neurons in primary cultures. European Journal of Pharmacology. 225: 253-62. PMID 1355446 DOI: 10.1016/0922-4106(92)90027-S  0.391
1992 Sladeczek F, Manzoni O, Fagni L, Dumuis A, Pin JP, Sebben M, Bockaert J. The metabotropic glutamate receptor (MGR): pharmacology and subcellular location. Journal of Physiology, Paris. 86: 47-55. PMID 1343596 DOI: 10.1016/S0928-4257(05)80007-5  0.461
1991 Rage F, Pin JP, Tapia-Arancibia L. Phospholipase A and Somatostatin Release are Activated in Response to N-Methyl-D-Aspartate Receptor Stimulation in Hypothalamic Neurons in Primary Culture. Journal of Neuroendocrinology. 3: 515-22. PMID 19215501 DOI: 10.1111/j.1365-2826.1991.tb00312.x  0.383
1990 Manzoni O, Fagni L, Pin JP, Rassendren F, Poulat F, Sladeczek F, Bockaert J. (trans)-1-amino-cyclopentyl-1,3-dicarboxylate stimulates quisqualate phosphoinositide-coupled receptors but not ionotropic glutamate receptors in striatal neurons and Xenopus oocytes. Molecular Pharmacology. 38: 1-6. PMID 2164627  0.494
1990 Rassendren FA, Lory P, Pin JP, Nargeot J. Zinc has opposite effects on NMDA and non-NMDA receptors expressed in Xenopus oocytes. Neuron. 4: 733-40. PMID 2160837 DOI: 10.1016/0896-6273(90)90199-P  0.382
1990 Pin JP, Bockaert J. Omega-conotoxin GVIA and dihydropyridines discriminate two types of Ca2+ channels involved in GABA release from striatal neurons in culture. European Journal of Pharmacology. 188: 81-4. PMID 2155125 DOI: 10.1016/0922-4106(90)90250-2  0.303
1990 Bockaert J, Dumuis A, Manzoni O, Nargeot J, Oomagari K, Pin JP, Rassendren F, Sebben M, Sladeczek F. Intracellular messengers associated with excitatory amino acid (EAA) receptors. Advances in Experimental Medicine and Biology. 268: 79-91. PMID 1981654 DOI: 10.1007/978-1-4684-5769-8_10  0.322
1990 Charpentier N, Dumuis A, Sebben M, Bockaert J, Pin JP. On concanavalin A-treated striatal neurons quisqualate clearly behaves as a partial agonist of a receptor fully activated by kainate. European Journal of Pharmacology. 189: 241-51. PMID 1980646 DOI: 10.1016/0922-4106(90)90117-G  0.476
1990 Dumuis A, Pin JP, Oomagari K, Sebben M, Bockaert J. Arachidonic acid released from striatal neurons by joint stimulation of ionotropic and metabotropic quisqualate receptors. Nature. 347: 182-4. PMID 1975645 DOI: 10.1038/347182A0  0.413
1989 Pin JP, Bockaert J. Two distinct mechanisms, differentially affected by excitatory amino acids, trigger GABA release from fetal mouse striatal neurons in primary culture. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 9: 648-56. PMID 2918382 DOI: 10.1523/Jneurosci.09-02-00648.1989  0.339
1989 Didier M, Roux P, Piechaczyk M, Verrier B, Bockaert J, Pin JP. Cerebellar granule cell survival and maturation induced by K+ and NMDA correlate with c-fos proto-oncogene expression. Neuroscience Letters. 107: 55-62. PMID 2575730 DOI: 10.1016/0304-3940(89)90790-8  0.361
1989 Van Vliet BJ, Sebben M, Dumuis A, Gabrion J, Bockaert J, Pin JP. Endogenous amino acid release from cultured cerebellar neuronal cells: effect of tetanus toxin on glutamate release. Journal of Neurochemistry. 52: 1229-39. PMID 2564424 DOI: 10.1111/J.1471-4159.1989.Tb01870.X  0.317
1989 Pin JP, Van Vliet BJ, Bockaert J. Complex interaction between quisqualate and kainate receptors as revealed by measurement of GABA release from striatal neurons in primary culture. European Journal of Pharmacology. 172: 81-91. PMID 2541001 DOI: 10.1016/0922-4106(89)90047-3  0.466
1989 Rassendren FA, Lory P, Pin JP, Bockaert J, Nargeot J. A specific quisqualate agonist inhibits kainate responses induced in Xenopus oocytes injected with rat brain RNA. Neuroscience Letters. 99: 333-9. PMID 2471121 DOI: 10.1016/0304-3940(89)90469-2  0.455
1988 Pin JP, Van-Vliet BJ, Bockaert J. NMDA- and kainate-evoked GABA release from striatal neurones differentiated in primary culture: differential blocking by phencyclidine. Neuroscience Letters. 87: 87-92. PMID 2898115 DOI: 10.1016/0304-3940(88)90150-4  0.412
1988 Dumuis A, Sebben M, Haynes L, Pin JP, Bockaert J. NMDA receptors activate the arachidonic acid cascade system in striatal neurons. Nature. 336: 68-70. PMID 2847054 DOI: 10.1038/336068A0  0.396
1988 Pin JP, Yasumoto T, Bockaert J. Maitotoxin-evoked gamma-aminobutyric acid release is due not only to the opening of calcium channels. Journal of Neurochemistry. 50: 1227-32. PMID 2450172 DOI: 10.1111/J.1471-4159.1988.Tb10597.X  0.318
1987 Recasens M, Pin JP, Bockaert J. Chloride transport blockers inhibit the chloride-dependent glutamate binding to rat brain membranes. Neuroscience Letters. 74: 211-6. PMID 2883610 DOI: 10.1016/0304-3940(87)90151-0  0.584
1987 Pin JP, Rumigny JF, Bockaert J, Recasens M. Multiple Cl(-)-independent binding sites for the excitatory amino acids: glutamate, aspartate and cysteine sulfinate in rat brain membranes. Brain Research. 402: 11-20. PMID 2881598 DOI: 10.1016/0006-8993(87)91042-0  0.591
1987 Pin JP, Bockaert J. Multiple voltage-sensitive calcium channels are probably involved in endogenous GABA release from striatal neurones differentiated in primary culture. Naunyn-Schmiedeberg's Archives of Pharmacology. 336: 190-6. PMID 2446149 DOI: 10.1007/Bf00165804  0.305
1986 Bockaert J, Gabrion J, Sladeczek F, Pin JP, Recasens M, Sebben M, Kemp D, Dumuis A, Weiss S. Primary culture of striatal neurons: a model of choice for pharmacological and biochemical studies of neurotransmitter receptors. Journal De Physiologie. 81: 219-27. PMID 2883308  0.615
1986 Pin JP, Bockaert J, Recasens M. The binding of acidic amino acids to snail, Helix aspersa, periesophagic ring membranes reveals a single high-affinity glutamate/kainate site. Brain Research. 366: 290-9. PMID 2870764 DOI: 10.1016/0006-8993(86)91306-5  0.592
1985 Sladeczek F, Pin JP, Récasens M, Bockaert J, Weiss S. Glutamate stimulates inositol phosphate formation in striatal neurones. Nature. 317: 717-9. PMID 2865680 DOI: 10.1038/317717A0  0.469
Low-probability matches (unlikely to be authored by this person)
2016 Zussy C, Gómez-Santacana X, Rovira X, De Bundel D, Ferrazzo S, Bosch D, Asede D, Malhaire F, Acher F, Giraldo J, Valjent E, Ehrlich I, Ferraguti F, Pin JP, Llebaria A, et al. Dynamic modulation of inflammatory pain-related affective and sensory symptoms by optical control of amygdala metabotropic glutamate receptor 4. Molecular Psychiatry. PMID 27994221 DOI: 10.1038/Mp.2016.223  0.299
2018 Rivat C, Sar C, Mechaly I, Leyris JP, Diouloufet L, Sonrier C, Philipson Y, Lucas O, Mallié S, Jouvenel A, Tassou A, Haton H, Venteo S, Pin JP, Trinquet E, et al. Inhibition of neuronal FLT3 receptor tyrosine kinase alleviates peripheral neuropathic pain in mice. Nature Communications. 9: 1042. PMID 29531216 DOI: 10.1038/S41467-018-03496-2  0.296
1986 Pin JP, Weiss S, Sebben M, Kemp DE, Bockaert J. Release of endogenous amino acids from striatal neurons in primary culture. Journal of Neurochemistry. 47: 594-603. PMID 2426401 DOI: 10.1111/J.1471-4159.1986.Tb04541.X  0.295
1984 Pin JP, Bockaert J, Recasesn M. The Ca2+/C1- dependent L-[3H]glutamate binding: a new receptor or a particular transport process? Febs Letters. 175: 31-6. PMID 6090209 DOI: 10.1016/0014-5793(84)80563-3  0.281
1991 Oomagari K, Buisson B, Dumuis A, Bockaert J, Pin JP. Effect of Glutamate and Ionomycin on the Release of Arachidonic Acid, Prostaglandins and HETEs from Cultured Neurons and Astrocytes. The European Journal of Neuroscience. 3: 928-939. PMID 12106250 DOI: 10.1111/J.1460-9568.1991.Tb00028.X  0.279
2010 Magalhaes AC, Holmes KD, Dale LB, Comps-Agrar L, Lee D, Yadav PN, Drysdale L, Poulter MO, Roth BL, Pin JP, Anisman H, Ferguson SS. CRF receptor 1 regulates anxiety behavior via sensitization of 5-HT2 receptor signaling. Nature Neuroscience. 13: 622-9. PMID 20383137 DOI: 10.1038/Nn.2529  0.274
2021 Wei B, Zhu Y, Yang P, Han Y, Wang S, Wang X, Xia S, Song X, Zhang Z, Wang S, Rondard P, Pin JP, Jiang X, Liu J. GABA promotes the malignancy of human cancer cells by targeting the tyrosine phosphatase PTPN12. Iscience. 24: 103311. PMID 34778730 DOI: 10.1016/j.isci.2021.103311  0.27
1998 McCool BA, Pin JP, Harpold MM, Brust PF, Stauderman KA, Lovinger DM. Rat group I metabotropic glutamate receptors inhibit neuronal Ca2+ channels via multiple signal transduction pathways in HEK 293 cells. Journal of Neurophysiology. 79: 379-91. PMID 9425207 DOI: 10.1152/Jn.1998.79.1.379  0.265
2020 Sebastianutto I, Goyet E, Andreoli L, Font-Ingles J, Moreno-Delgado D, Bouquier N, Jahannault-Talignani C, Moutin E, Di Menna L, Maslava N, Pin JP, Fagni L, Nicoletti F, Ango F, Cenci MA, et al. D1-mGlu5 heteromers mediate noncanonical dopamine signaling in Parkinson's disease. The Journal of Clinical Investigation. PMID 32039920 DOI: 10.1172/Jci126361  0.265
1995 Brabet I, Mary S, Bockaert J, Pin JP. Phenylglycine derivatives discriminate between mGluR1- and mGluR5-mediated responses. Neuropharmacology. 34: 895-903. PMID 8532171 DOI: 10.1016/0028-3908(95)00079-L  0.265
2011 Cassier PA, Treilleux I, Bachelot T, Ray-Coquard I, Bendriss-Vermare N, Ménétrier-Caux C, Trédan O, Goddard-Léon S, Pin JJ, Mignotte H, Bathélémy-Dubois C, Caux C, Lebecque S, Blay JY. Prognostic value of the expression of C-Chemokine Receptor 6 and 7 and their ligands in non-metastatic breast cancer Bmc Cancer. 11. PMID 21624121 DOI: 10.1186/1471-2407-11-213  0.256
2019 Zindel D, Vol C, Lecha O, Bequignon I, Bilgic M, Vereecke M, Charrier-Savournin F, Romier M, Trinquet E, Pin JP, Pannequin J, Roux T, Dupuis E, Prézeau L. HTRF Total and Phospho-YAP (Ser127) Cellular Assays. Methods in Molecular Biology (Clifton, N.J.). 1893: 153-166. PMID 30565133 DOI: 10.1007/978-1-4939-8910-2_13  0.256
2005 Pin J. Moduler l’action du glutamate dans le cerveau: de nouvelles pistes ouvertes grâce aux récepteurs métabotropiques Psn. 3: 132-142. DOI: 10.1007/BF03005833  0.254
1988 Pares-Herbuté N, Bonet A, Peraldi S, Pin JP, Gabrion J, Astier H, Tapia-Arancibia L. The presence of non-neuronal cells influences somatostatin release from cultured cerebral cortical cells. Brain Research. 468: 89-97. PMID 2897872 DOI: 10.1016/0165-3806(88)90011-9  0.252
2017 Christensen SB, Hone AJ, Roux I, Kniazeff J, Pin JP, Upert G, Servent D, Glowatzki E, McIntosh JM. RgIA4 Potently Blocks Mouse α9α10 nAChRs and Provides Long Lasting Protection against Oxaliplatin-Induced Cold Allodynia. Frontiers in Cellular Neuroscience. 11: 219. PMID 28785206 DOI: 10.3389/Fncel.2017.00219  0.244
2011 Christov C, González-Bulnes P, Malhaire F, Karabencheva T, Goudet C, Pin JP, Llebaria A, Giraldo J. Integrated synthetic, pharmacological, and computational investigation of cis-2-(3,5-dichlorophenylcarbamoyl)cyclohexanecarboxylic acid enantiomers as positive allosteric modulators of metabotropic glutamate receptor subtype 4. Chemmedchem. 6: 131-40. PMID 21132834 DOI: 10.1002/cmdc.201000378  0.243
2015 Paoletti P, Pin JP. Editorial overview: neurosciences: targeting glutamatergic signaling in CNS diseases: new hopes? Current Opinion in Pharmacology. 20: iv-vi. PMID 25601440 DOI: 10.1016/J.Coph.2015.01.001  0.241
2002 Ango F, Prézeau L, Bockaert J, Pin J, Fagni L. Activation de récepteurs par une protéine intracellulaire : un nouveau concept et un nouveau type de cible pharmacologique MéDecine/Sciences. 18: 151-153. DOI: 10.1051/Medsci/2002182151  0.24
1992 Didier M, Roux P, Piechaczyk M, Mangeat P, Devilliers G, Bockaert J, Pin JP. Long-term expression of the c-fos protein during the in vitro differentiation of cerebellar granule cells induced by potassium or NMDA. Brain Research. Molecular Brain Research. 12: 249-58. PMID 1312204 DOI: 10.1016/0169-328X(92)90091-O  0.232
2023 Haubrich J, Zwier JM, Charrier-Savournin F, Prézeau L, Pin JP. Different EGF-induced receptor dimer conformations for signaling and internalization. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 38: e23356. PMID 38071470 DOI: 10.1096/fj.202301209R  0.223
2013 Toscano F, Estornes Y, Virard F, Garcia-Cattaneo A, Pierrot A, Vanbervliet B, Bonnin M, Ciancanelli MJ, Zhang SY, Funami K, Seya T, Matsumoto M, Pin JJ, Casanova JL, Renno T, et al. Cleaved/associated TLR3 represents the primary form of the signaling receptor Journal of Immunology. 190: 764-773. PMID 23255358 DOI: 10.4049/Jimmunol.1202173  0.221
2022 Derieux C, Léauté A, Brugoux A, Jaccaz D, Terrier C, Pin JP, Kniazeff J, Le Merrer J, Becker JAJ. Chronic sodium bromide treatment relieves autistic-like behavioral deficits in three mouse models of autism. Neuropsychopharmacology : Official Publication of the American College of Neuropsychopharmacology. PMID 35418620 DOI: 10.1038/s41386-022-01317-1  0.209
2011 Collingridge GL, Pin JP, Hubbard RE, Kiss JP, Spedding M. Introduction to the special issue on High Resolution Neuropharmacology. Neuropharmacology. 60: 1-2. PMID 20813115 DOI: 10.1016/J.Neuropharm.2010.08.020  0.196
2015 Mathis S, Pin JC, Pierre F, Ciron J, Iljicsov A, Lamy M, Neau JP. Anti-NMDA Receptor Encephalitis During Pregnancy: A Case Report. Medicine. 94: e1034. PMID 26131809 DOI: 10.1097/MD.0000000000001034  0.17
1990 Didier M, Heaulme M, Soubrié P, Bockaert J, Pin JP. Rapid, sensitive, and simple method for quantification of both neurotoxic and neurotrophic effects of NMDA on cultured cerebellar granule cells. Journal of Neuroscience Research. 27: 25-35. PMID 1979352 DOI: 10.1002/Jnr.490270105  0.164
2007 Bonnefont-Rebeix C, Marchal T, Bernaud J, Pin JJ, Leroux C, Lebecque S, Chabanne L, Rigal D. Toll-like receptor 3 (TLR3): A new marker of canine monocytes-derived dendritic cells (cMo-DC) Veterinary Immunology and Immunopathology. 118: 134-139. PMID 17521746 DOI: 10.1016/j.vetimm.2007.04.008  0.152
1986 Weiss S, Pin JP, Sebben M, Kemp DE, Sladeczek F, Gabrion J, Bockaert J. Synaptogenesis of cultured striatal neurons in serum-free medium: a morphological and biochemical study. Proceedings of the National Academy of Sciences of the United States of America. 83: 2238-42. PMID 3008155 DOI: 10.1073/pnas.83.7.2238  0.125
2024 Eshak F, Pion L, Scholler P, Nevoltris D, Chames P, Rondard P, Pin JP, Acher FC, Goupil-Lamy A. Epitope Identification of an mGlu5 Receptor Nanobody Using Physics-Based Molecular Modeling and Deep Learning Techniques. Journal of Chemical Information and Modeling. PMID 38423996 DOI: 10.1021/acs.jcim.3c01620  0.12
2010 Pin JP, Maurel D, Comps-Agrar L, Monnier C, Rives ML, Doumazane E, Rondard P, Durroux T, Prézeau L, Trinquet E. Time-resolved FRET approaches to study GPCR complexes G Protein-Coupled Receptors: Structure, Signaling, and Physiology. 67-89. DOI: 10.1017/CBO9780511760334.005  0.115
2006 Gautier G, de Saint-Vis B, Sénéchal B, Pin JJ, Bates EE, Caux C, Geissmann F, Garrone P. The class 6 semaphorin SEMA6A is induced by interferon-gamma and defines an activation status of langerhans cells observed in pathological situations. The American Journal of Pathology. 168: 453-65. PMID 16436660 DOI: 10.2353/ajpath.2006.050288  0.113
1992 Lafon-Cazal M, Bougault I, Steinberg R, Pin JP, Bockaert J. Measurement of gamma-enolase release, a new method for selective quantification of neurotoxicity independently from glial lysis. Brain Research. 593: 63-8. PMID 1458320 DOI: 10.1016/0006-8993(92)91264-F  0.112
2014 Bjordal M, Arquier N, Kniazeff J, Pin JP, Léopold P. Sensing of amino acids in a dopaminergic circuitry promotes rejection of an incomplete diet in Drosophila. Cell. 156: 510-21. PMID 24485457 DOI: 10.1016/j.cell.2013.12.024  0.111
2012 Vilar B, Busserolles J, Ling B, Malhaire F, Chapuy E, Acher F, Pin J, Eschalier A, Goudet C. Implication du récepteur métabotropique du glutamate de type 4 spinal dans la modulation de la douleur Douleurs : Evaluation - Diagnostic - Traitement. 13: A19-A20. DOI: 10.1016/j.douler.2012.08.055  0.103
2023 Tsitokana ME, Lafon PA, Prézeau L, Pin JP, Rondard P. Targeting the Brain with Single-Domain Antibodies: Greater Potential Than Stated So Far? International Journal of Molecular Sciences. 24. PMID 36768953 DOI: 10.3390/ijms24032632  0.074
2015 Pin JM, Sbirrazzuoli N, Mija A. From epoxidized linseed oil to bioresin: An overall approach of epoxy/anhydride cross-linking Chemsuschem. 8: 1232-1243. PMID 25754910 DOI: 10.1002/cssc.201403262  0.069
2013 Dawood R, Benjelloun F, Pin JJ, Kone A, Chanut B, Jospin F, Lucht F, Verrier B, Moog C, Genin C, Paul S. Generation of HIV-1 potent and broad neutralizing antibodies by immunization with postfusion HR1/HR2 complex Aids. 27: 717-730. PMID 23719346 DOI: 10.1097/QAD.0b013e32835cfca5  0.067
2011 Canard B, Vachon H, Fontaine T, Pin JJ, Paul S, Genin C, Mueller CG. Generation of anti-DC-SIGN monoclonal antibodies capable of blocking HIV-1 gp120 binding and reactive on formalin-fixed tissue Immunology Letters. 135: 165-172. PMID 21078343 DOI: 10.1016/j.imlet.2010.11.002  0.064
2019 Kansara M, Thomson K, Pang P, Dutour A, Mirabello L, Acher F, Pin JP, Demicco EG, Yan J, Teng MWL, Smyth MJ, Thomas DM. Infiltrating Myeloid Cells Drive Osteosarcoma Progression via GRM4 Regulation of IL23. Cancer Discovery. PMID 31527131 DOI: 10.1158/2159-8290.CD-19-0154  0.063
2010 Mougenot AL, Bétemps D, Hogeveen KN, Kovacs GG, Chouaf-Lakhdar L, Milhavet O, Lehmann S, Legastelois S, Pin JJ, Baron TG. Production of a monoclonal antibody, against human α-synuclein, in a subpopulation of C57BL/6J mice, presenting a deletion of the α-synuclein locus. Journal of Neuroscience Methods. 192: 268-76. PMID 20709102 DOI: 10.1016/j.jneumeth.2010.08.010  0.058
2008 Gómez AC, Guaiana G, Pin JE. When does partial commutative closure preserve regularity? Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 5126: 209-220. DOI: 10.1007/978-3-540-70583-3_18  0.057
2011 Biancheri-Mounicq I, Colombié M, Pin JC, Lecoanet A, Adam-Tariel F. Unexpected finding on I-123 FP-CIT SPECT leading to the diagnosis of cerebral meningioma Clinical Nuclear Medicine. 36: 156-157. PMID 21220989  0.052
2011 Rochereau N, Verrier B, Pin JJ, Genin C, Paul S. Phenotypic localization of distinct DC subsets in mouse Peyer Patch Vaccine. 29: 3655-3661. PMID 21439318 DOI: 10.1016/j.vaccine.2011.03.012  0.052
2014 Gehrke M, Krebs A, Pin JÉ. Ultrafilters on words for a fragment of logic Theoretical Computer Science. DOI: 10.1016/J.Tcs.2015.08.007  0.046
2015 Marins JA, Mija A, Pin JM, Giulieri F, Soares BG, Sbirrazzuoli N, Lançon P, Bossis G. Anisotropic reinforcement of epoxy-based nanocomposites with aligned magnetite-sepiolite hybrid nanofiller Composites Science and Technology. 112: 34-41. DOI: 10.1016/j.compscitech.2015.03.008  0.042
2015 Basold H, Hansen HH, Pin JÉ, Rutten J. Newton series, coinductively Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 9399: 91-109. DOI: 10.1007/978-3-319-25150-9_7  0.041
2016 Bonnefont-Rebeix C, Fournel-Fleury C, Ponce F, Belluco S, Watrelot D, Bouteille SE, Rapiteau S, Razanajaona-Doll D, Pin JJ, Leroux C, Marchal T. Characterization of a novel canine T-cell line established from a spontaneously occurring aggressive T-cell lymphoma with large granular cell morphology Immunobiology. 221: 12-22. DOI: 10.1016/j.imbio.2015.08.007  0.041
2009 Pin J, Xinyu D. RETRACTED ARTICLE: Principal and application for VRML explanatory character model display 2009 International Conference On E-Learning, E-Business, Enterprise Information Systems, and E-Government, Eeee 2009. 29-32. DOI: 10.1109/EEEE.2009.36  0.04
2010 Gehrke M, Grigorieff S, Pin JE. A topological approach to recognition Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 6199: 151-162. DOI: 10.1007/978-3-642-14162-1_13  0.04
2013 Mayen P, Pin JP. Building commitment among people undergoing APL (Accreditation of Prior Learning) | Conditions et processus de l'engagement en VAE Formation Emploi. 122: 13-29.  0.04
2011 Pin JE, Silva PV. On profinite uniform structures defined by varieties of finite monoids International Journal of Algebra and Computation. 21: 295-314. DOI: 10.1142/S0218196711006170  0.038
2008 Xinyu D, Pin J. Development and application of virtual avatar interactive technology Proceedings - 2008 International Conference On Advanced Computer Theory and Engineering, Icacte 2008. 286-289. DOI: 10.1109/ICACTE.2008.19  0.036
2014 Xun M, Jianjun D, Hongwei L, Jianqiang Y, Jinfeng L, Bing W, Yanling Q, Wenhui H, Lingyun W, Pin J, Hongtao L. Development of all-solid-state flash x-ray generator with photoconductive semiconductor switches. The Review of Scientific Instruments. 85: 093307. PMID 25273719 DOI: 10.1063/1.4895829  0.034
2014 Pin JE, Silva PV. A noncommutative extension of Mahler's theorem on interpolation series European Journal of Combinatorics. 36: 564-578. DOI: 10.1016/j.ejc.2013.09.009  0.03
2006 Golovkins M, Pin JE. Varieties generated by certain models of reversible finite automata Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 4112: 83-93.  0.029
2008 Pin JE, Silva PV. A Mahler's theorem for functions from words to integers Proceedings of the 25th International Symposium On Theoretical Aspects of Computer Science, Stacs 2008. 585-596.  0.027
2015 Ballester-Bolinches A, Pin JÉ, Soler-Escrivà X. Languages associated with saturated formations of groups Forum Mathematicum. 27: 1471-1505. DOI: 10.1515/forum-2012-0161  0.024
2009 Xinyu D, Pin J. Exploration of virtual avatar technology based on VRML and java Proceedings - 2009 2nd International Workshop On Knowledge Discovery and Data Mining, Wkkd 2009. 717-720. DOI: 10.1109/WKDD.2009.48  0.024
2006 Matsuyama A, Yasuda Y, Yasutake A, Xiaojie L, Pin J, Li L, Mei L, Yumin A, Liya Q. Detailed pollution map of an area highly contaminated by mercury containing wastewater from an organic chemical factory in People's Republic of China Bulletin of Environmental Contamination and Toxicology. 77: 82-87. PMID 16832759 DOI: 10.1007/s00128-006-1035-6  0.023
2007 Barthod M, Hayne B, Tébec JL, Pin JC. Experimental study of dynamic and noise produced by a gearing excited by a multi-harmonic excitation Applied Acoustics. 68: 982-1002. DOI: 10.1016/j.apacoust.2006.04.012  0.022
2007 Barthod M, Hayne B, Tébec JL, Pin JC. Experimental study of gear rattle excited by a multi-harmonic excitation Applied Acoustics. 68: 1003-1025. DOI: 10.1016/j.apacoust.2006.04.011  0.022
2014 Gehrke M, Krebs A, Pin JE. From ultrafilters on words to the expressive power of a fragment of logic Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 8614: 138-149. DOI: 10.1007/978-3-319-09704-6_13  0.022
2006 Chaubard L, Pin JE, Straubing H. Actions, wreath products of C-varieties and concatenation product Theoretical Computer Science. 356: 73-89. DOI: 10.1016/j.tcs.2006.01.039  0.021
2007 Wenhua J, Pin J, Yuanyuan M. Fast handover scheme for real-time applications in mobile WiMAX Ieee International Conference On Communications. 6038-6042. DOI: 10.1109/ICC.2007.1000  0.021
2011 Xinyu D, Pin J. Exploration to virtual reality 3D key techniques based on cosmo browser plug-in International Journal of Digital Content Technology and Its Applications. 5: 391-402. DOI: 10.4156/jdcta.vol5.issue6.46  0.021
2015 Pin JÉ. Newton’s forward difference equation for functions from words to words Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 9136: 71-82. DOI: 10.1007/978-3-319-20028-6_8  0.02
2014 Cipro R, Baron T, Martin M, Moeyaert J, David S, Gorbenko V, Bassani F, Bogumilowicz Y, Barnes JP, Rochat N, Loup V, Vizioz C, Allouti N, Chauvin N, Bao XY, ... ... Pin JB, et al. Low defect InGaAs quantum well selectively grown by metal organic chemical vapor deposition on Si(100) 300 mm wafers for next generation non planar devices Applied Physics Letters. 104. DOI: 10.1063/1.4886404  0.02
2013 Susaeta L, Pin JR, Idrovo S, Espejo A, Belizón M, Gallifa A, Aguirre M, Pedrozo EA. Generation or culture? Work attitude drivers: An analysis in Latin America and Iberian countries Cross Cultural Management. 20: 321-360. DOI: 10.1108/CCM-12-2011-0126  0.019
2008 Xinyu D, Baoqing G, Pin J. Concept and application of three dimension virtual study technology for academic e-learning Proceedings of the International Conference On Computer Science and Information Technology, Iccsit 2008. 741-744. DOI: 10.1109/ICCSIT.2008.116  0.018
2008 Gómez AC, Pin JE. A robust class of regular languages Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 5162: 36-51. DOI: 10.1007/978-3-540-85238-4_3  0.018
2006 Gomes GMS, Sezinando H, Pin JE. Presentations of the schützenberger product of n groups Communications in Algebra. 34: 1213-1235. DOI: 10.1080/00927870500454075  0.018
2013 Xinyu D, Pin J. Study exploration on three dimension virtual human energy body skeleton model Energy Education Science and Technology Part a: Energy Science and Research. 31: 239-242.  0.018
2009 Kogan Y, Pin J. Beginning the journey: The project approach with toddlers Early Childhood Research and Practice. 11.  0.017
2014 Ballester-Bolinches A, Pin JÉ, Soler-Escrivà X. Formations of finite monoids and formal languages: Eilenberg's variety theorem revisited Forum Mathematicum. 26: 1737-1761. DOI: 10.1515/forum-2012-0055  0.015
2013 Cano A, Guaiana G, Pin JE. Regular languages and partial commutations Information and Computation. 230: 76-96. DOI: 10.1016/j.ic.2013.07.003  0.015
2015 Pin JM, Guigo N, Vincent L, Sbirrazzuoli N, Mija A. Cationic Copolymerization as a Synergic Strategy to Combine Epoxidized Linseed Oil and Furfuryl Alcohol: Design of a Fully Bio-Based Thermoset Chemsuschem. DOI: 10.1002/cssc.201501566  0.014
2012 Cano A, Pin JE. Upper set monoids and length preserving morphisms Journal of Pure and Applied Algebra. 216: 1178-1183. DOI: 10.1016/j.jpaa.2011.10.022  0.014
2009 Pin JE. Profinite methods in automata theory Leibniz International Proceedings in Informatics, Lipics. 3: 31-50.  0.013
2008 Ma JH, Pin JH, Huang ZM, Gao YH, Lin T, Shi FW, Sun JL, Chu JH. Highly (h00) oriented growth of SrTiO3 thin films on Si(100) substrates by RF magnetron sputtering and their optical properties Proceedings of Spie - the International Society For Optical Engineering. 6984. DOI: 10.1117/12.792775  0.012
2010 Berstel J, Boasson L, Carton O, Pin JE, Restivo A. The expressive power of the shuffle product Information and Computation. 208: 1258-1272. DOI: 10.1016/j.ic.2010.06.002  0.012
2015 Pin JM, Guigo N, Vincent L, Sbirrazzuoli N, Mija A. Copolymerization as a Strategy to Combine Epoxidized Linseed Oil and Furfuryl Alcohol: The Design of a Fully Bio-Based Thermoset Chemsuschem. DOI: 10.1002/cssc.201501259  0.011
2006 Berstel J, Boasson L, Carton O, Petazzoni B, Pin JE. Operations preserving regular languages Theoretical Computer Science. 354: 405-420. DOI: 10.1016/j.tcs.2005.11.034  0.011
2008 Gehrke M, Grigorieff S, Pin JE. Duality and equational theory of regular languages Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 5126: 246-257. DOI: 10.1007/978-3-540-70583-3_21  0.011
2015 Almeida J, Cano A, Klíma O, Pin J. On fixed points of the lower set operator International Journal of Algebra and Computation. 25: 259-262. DOI: 10.1142/S021819671540010X  0.01
2015 Bogumilowicz Y, Hartmann JM, Cipro R, Alcotte R, Martin M, Bassani F, Moeyaert J, Baron T, Pin JB, Bao X, Ye Z, Sanchez E. Anti-phase boundaries-Free GaAs epilayers on "quasi-nominal" Ge-buffered silicon substrates Applied Physics Letters. 107. DOI: 10.1063/1.4935943  0.01
2014 Salleh H, Pin JGW, Wah ATK. Professional learning communities in the teacher internship program in Singapore Practical Knowledge in Teacher Education: Approaches to Teacher Internship Programmes. 195-209. DOI: 10.4324/9781315814056  0.01
2014 Pin JM, Guigo N, Mija A, Vincent L, Sbirrazzuoli N, Van Der Waal JC, De Jong E. Valorization of biorefinery side-stream products: Combination of humins with polyfurfuryl alcohol for composite elaboration Acs Sustainable Chemistry and Engineering. 2: 2182-2190. DOI: 10.1021/sc5003769  0.01
2013 Pin JE. An explicit formula for the intersection of two polynomials of regular languages Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 7907: 31-45. DOI: 10.1007/978-3-642-38771-5_5  0.01
2012 Pin JE. Equational descriptions of languages International Journal of Foundations of Computer Science. 23: 1227-1240. DOI: 10.1142/S0129054112400497  0.01
2011 Sharov I, Pin JC, Prat C, Jaafari N, Nkamhoua A, Devoize JL. [Cardiogenic shock in acute multiple sclerosis]. Zhurnal Nevrologii I Psikhiatrii Imeni S.S. Korsakova / Ministerstvo Zdravookhraneniia I Meditsinskoä­ Promyshlennosti Rossiä­Skoä­ Federatsii, Vserossiä­Skoe Obshchestvo Nevrologov [I] Vserossiä­Skoe Obshchestvo Psikhiatrov. 111: 72-5. PMID 21574517  0.01
2011 Pin JE. Theme and variations on the concatenation product Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 6742: 44-64. DOI: 10.1007/978-3-642-21493-6_3  0.01
2009 Branco MJJ, Pin JE. Equations defining the polynomial closure of a lattice of regular languages Lecture Notes in Computer Science (Including Subseries Lecture Notes in Artificial Intelligence and Lecture Notes in Bioinformatics). 5556: 115-126. DOI: 10.1007/978-3-642-02930-1_10  0.01
2006 Chaubard L, Pin JE, Straubing H. First order formulas with modular predicates Proceedings - Symposium On Logic in Computer Science. 211-220. DOI: 10.1109/LICS.2006.24  0.01
Hide low-probability matches.