Year |
Citation |
Score |
2022 |
Xu J, Grosslight S, Mack KA, Nguyen SC, Clagg K, Lim NK, Timmerman JC, Shen J, White NA, Sirois LE, Han C, Zhang H, Sigman MS, Gosselin F. Atroposelective Negishi Coupling Optimization Guided by Multivariate Linear Regression Analysis: Asymmetric Synthesis of KRAS G12C Covalent Inhibitor GDC-6036. Journal of the American Chemical Society. PMID 36326518 DOI: 10.1021/jacs.2c09917 |
0.315 |
|
2021 |
Zell D, Kingston C, Jermaks J, Smith SR, Seeger N, Wassmer J, Sirois LE, Han C, Zhang H, Sigman MS, Gosselin F. Stereoconvergent and -divergent Synthesis of Tetrasubstituted Alkenes by Nickel-Catalyzed Cross-Couplings. Journal of the American Chemical Society. 143: 19078-19090. PMID 34735129 DOI: 10.1021/jacs.1c08399 |
0.322 |
|
2020 |
Lavernhe R, Alexy EJ, Zhang H, Stoltz BM. Palladium-Catalyzed Enantioselective Decarboxylative Allylic Alkylation of Protected Benzoin-Derived Enol Carbonates. Advanced Synthesis & Catalysis. 362: 344-347. PMID 33692657 DOI: 10.1002/adsc.201901281 |
0.55 |
|
2020 |
Fulton TJ, Cusumano AQ, Alexy EJ, Du YE, Zhang H, Houk KN, Stoltz BM. Global Diastereoconvergence in the Ireland-Claisen Rearrangement of Isomeric Enolates: Synthesis of Tetrasubstituted α-Amino Acids. Journal of the American Chemical Society. PMID 33320668 DOI: 10.1021/jacs.0c11480 |
0.494 |
|
2020 |
Lavernhe R, Alexy EJ, Zhang H, Stoltz BM. Palladium-Catalyzed Enantioselective Decarboxylative Allylic Alkylation of Acyclic α--Pyrrolyl/Indolyl Ketones. Organic Letters. PMID 32422045 DOI: 10.1021/Acs.Orglett.0C01303 |
0.565 |
|
2019 |
Fulton TJ, Wu B, Alexy EJ, Zhang H, Stoltz BM. Palladium-catalyzed α,β-dehydrogenation of acyclic ester equivalents promoted by a novel electron deficient phosphinooxazoline ligand. Tetrahedron. 75: 4104-4109. PMID 32255844 DOI: 10.1016/J.Tet.2019.05.065 |
0.524 |
|
2019 |
Alexy EJ, Fulton TJ, Zhang H, Stoltz BM. Palladium-catalyzed enantioselective decarboxylative allylic alkylation of fully substituted -acyl indole-derived enol carbonates. Chemical Science. 10: 5996-6000. PMID 31360407 DOI: 10.1039/C9Sc01726G |
0.545 |
|
2018 |
Zhang H, Li BX, Wong B, Stumpf A, Sowell CG, Gosselin F. Convergent Synthesis of PI3K Inhibitor GDC-0908 Featuring Palladium-Catalyzed Direct C‒H Arylation toward Dihydrobenzothienooxepines. The Journal of Organic Chemistry. PMID 30543748 DOI: 10.1021/Acs.Joc.8B02751 |
0.335 |
|
2018 |
Wolfard J, Xu J, Zhang H, Chung CK. Synthesis of Chiral Tryptamines via a Regioselective Indole Alkylation. Organic Letters. PMID 30130113 DOI: 10.1021/acs.orglett.8b02335 |
0.34 |
|
2018 |
Alexy EJ, Zhang H, Stoltz BM. Catalytic Enantioselective Synthesis of Acyclic Quaternary Centers: Palladium-Catalyzed Decarboxylative Allylic Alkylation of Fully Substituted Acyclic Enol Carbonates. Journal of the American Chemical Society. PMID 30049213 DOI: 10.1021/Jacs.8B05560 |
0.557 |
|
2018 |
Dalziel ME, Deichert JA, Carrera DE, Beaudry D, Han C, Zhang H, Angelaud R. Magnesium Ethoxide Promoted Conversion of Nitriles to Amidines and Its Application in 5,6-Dihydroimidazobenzoxazepine Synthesis. Organic Letters. PMID 29687714 DOI: 10.1021/Acs.Orglett.8B00824 |
0.303 |
|
2018 |
Sandoval C, Lim NK, Zhang H. Two-Step Synthesis of 3,4-Dihydropyrrolopyrazinones from Ketones and Piperazin-2-ones. Organic Letters. PMID 29406723 DOI: 10.1021/acs.orglett.8b00197 |
0.365 |
|
2017 |
Chen AY, Lu Q, Fu Y, Sarpong R, Stoltz BM, Zhang H. Isocanthine Synthesis via Rh(III)-Catalyzed Intramolecular C-H Functionalization. The Journal of Organic Chemistry. PMID 29182872 DOI: 10.1021/Acs.Joc.7B02731 |
0.665 |
|
2017 |
Lim NK, Weiss P, Li BX, McCulley CH, Hare SR, Bensema BL, Palazzo TA, Tantillo DJ, Zhang H, Gosselin F. Synthesis of Highly Stereodefined Tetrasubstituted Acyclic All-Carbon Olefins via a Syn-Elimination Approach. Organic Letters. PMID 29115843 DOI: 10.1021/Acs.Orglett.7B03141 |
0.339 |
|
2017 |
Li BX, Le DN, Mack KA, McClory A, Lim NK, Cravillion T, Savage S, Han C, Collum DB, Zhang H, Gosselin F. Highly Stereoselective Synthesis of Tetrasubstituted Acyclic All-carbon Olefins via Enol Tosylation and Suzuki‒Miyaura Coupling. Journal of the American Chemical Society. PMID 28715208 DOI: 10.1021/Jacs.7B05071 |
0.361 |
|
2016 |
Yao T, Zhang H, Zhao Y. Synthesis of 9,10-Phenanthrenes via Palladium-Catalyzed Aryne Annulation by o-Halostyrenes and Formal Synthesis of (±)-Tylophorine. Organic Letters. PMID 27188401 DOI: 10.1021/acs.orglett.6b00558 |
0.589 |
|
2016 |
Pushkarskaya E, Wong B, Han C, Capomolla S, Gu C, Stoltz BM, Zhang H. Single-step synthesis of 3-hydroxycarbazoles by annulation of electron-rich anilines and quinones Tetrahedron Letters. 57: 5653-5657. DOI: 10.1016/J.Tetlet.2016.11.009 |
0.48 |
|
2015 |
Shen J, Wong B, Gu C, Zhang H. Negishi Approach to 1,5-Disubstituted 3-Amino-1H-1,2,4-triazoles. Organic Letters. PMID 26381464 DOI: 10.1021/acs.orglett.5b02021 |
0.3 |
|
2014 |
Zhang H, Bednarz MS, Lim NK, Hernandez G, Wu W. One-pot synthesis of 4-substituted 3-amino-2-cyanothiophenes involving O-ethyl thioformate. Organic Letters. 16: 2522-5. PMID 24746285 DOI: 10.1021/ol500895t |
0.314 |
|
2010 |
Bagdanoff JT, Donoviel MS, Nouraldeen A, Carlsen M, Jessop TC, Tarver J, Aleem S, Dong L, Zhang H, Boteju L, Hazelwood J, Yan J, Bednarz M, Layek S, Owusu IB, et al. Inhibition of sphingosine 1-phosphate lyase for the treatment of rheumatoid arthritis: discovery of (E)-1-(4-((1R,2S,3R)-1,2,3,4-tetrahydroxybutyl)-1H-imidazol-2-yl)ethanone oxime (LX2931) and (1R,2S,3R)-1-(2-(isoxazol-3-yl)-1H-imidazol-4-yl)butane-1,2,3,4-tetraol (LX2932). Journal of Medicinal Chemistry. 53: 8650-62. PMID 21090716 DOI: 10.1021/jm101183p |
0.656 |
|
2010 |
Roesch KR, Zhang H, Larock RC. ChemInform Abstract: Synthesis of Isoquinolines and Pyridines by the Palladium-Catalyzed Iminoannulation of Internal Alkynes. Cheminform. 33: no-no. DOI: 10.1002/chin.200223161 |
0.369 |
|
2010 |
Zhang H, Larock RC. ChemInform Abstract: Synthesis of β- and γ-Carbolines by the Palladium-Catalyzed Iminoannulation of Internal Alkynes. Cheminform. 33: no-no. DOI: 10.1002/chin.200204166 |
0.48 |
|
2009 |
Bagdanoff JT, Donoviel MS, Nouraldeen A, Tarver J, Fu Q, Carlsen M, Jessop TC, Zhang H, Hazelwood J, Nguyen H, Baugh SD, Gardyan M, Terranova KM, Barbosa J, Yan J, et al. Inhibition of sphingosine-1-phosphate lyase for the treatment of autoimmune disorders. Journal of Medicinal Chemistry. 52: 3941-53. PMID 19489538 DOI: 10.1021/jm900278w |
0.666 |
|
2009 |
Ferreira EM, Zhang H, Stoltz BM. Oxidative Heck-Type Reactions (Fujiwara-Moritani Reactions) The Mizoroki-Heck Reaction. 345-382. DOI: 10.1002/9780470716076.ch9 |
0.62 |
|
2008 |
Ferreira EM, Zhang H, Stoltz BM. C-H Bond Functionalizations with Palladium(II): Intramolecular Oxidative Annulations of Arenes. Tetrahedron. 64: 5987-6001. PMID 18587498 DOI: 10.1016/J.Tet.2008.01.052 |
0.661 |
|
2007 |
Campo MA, Zhang H, Yao T, Ibdah A, McCulla RD, Huang Q, Zhao J, Jenks WS, Larock RC. Aryl to aryl palladium migration in the Heck and Suzuki coupling of o-halobiaryls. Journal of the American Chemical Society. 129: 6298-307. PMID 17451243 DOI: 10.1021/Ja069238Z |
0.687 |
|
2004 |
Zhang H, Ferreira EM, Stoltz BM. Direct oxidative Heck cyclizations: intramolecular Fujiwara-Moritani arylations for the synthesis of functionalized benzofurans and dihydrobenzofurans. Angewandte Chemie (International Ed. in English). 43: 6144-8. PMID 15549760 DOI: 10.1002/Anie.200461294 |
0.666 |
|
2003 |
Zhang H, Larock RC. Synthesis of annulated gamma-carbolines and heteropolycycles by the palladium-catalyzed intramolecular annulation of alkynes. The Journal of Organic Chemistry. 68: 5132-8. PMID 12816467 DOI: 10.1021/Jo0343228 |
0.582 |
|
2003 |
Zhang H, Larock RC. Synthesis of β- and γ-Carbolines by the Palladium-Catalyzed Iminoannulation of Alkynes. Cheminform. 34. DOI: 10.1002/chin.200320169 |
0.476 |
|
2002 |
Zhang H, Larock RC. Synthesis of beta- and gamma-carbolines by the palladium-catalyzed iminoannulation of alkynes. The Journal of Organic Chemistry. 67: 9318-30. PMID 12492334 DOI: 10.1021/Jo026317U |
0.562 |
|
2002 |
Zhang H, Larock RC. Synthesis of beta- and gamma-carbolines by the palladium/copper-catalyzed coupling and cyclization of terminal acetylenes. The Journal of Organic Chemistry. 67: 7048-56. PMID 12353999 DOI: 10.1021/Jo0258857 |
0.527 |
|
2002 |
Zhang H, Larock RC. Synthesis of annulated gamma-carbolines by palladium-catalyzed intramolecular iminoannulation. Organic Letters. 4: 3035-8. PMID 12201710 DOI: 10.1021/Ol026255U |
0.603 |
|
2002 |
Zhang H, Larock RC. Synthesis of β- and γ-carbolines by the palladium/copper-catalyzed coupling and copper-catalyzed or thermal cyclization of terminal acetylenes Tetrahedron Letters. 43: 1359-1362. DOI: 10.1016/S0040-4039(02)00005-9 |
0.543 |
|
2001 |
Zhang H, Larock RC. Synthesis of beta- and gamma-carbolines by the palladium-catalyzed iminoannulation of internal alkynes. Organic Letters. 3: 3083-6. PMID 11574000 DOI: 10.1021/Ol010124W |
0.548 |
|
2000 |
Zhang Y, Gong X, Zhang H, Larock RC, Yeung ES. Combinatorial screening of homogeneous catalysis and reaction optimization based on multiplexed capillary electrophoresis Journal of Combinatorial Chemistry. 2: 450-2. PMID 11029169 DOI: 10.1021/Cc000043B |
0.448 |
|
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