| Year |
Citation |
Score |
| 2020 |
Wnuk SF, Mudgal MM, Nowak I, Robins MJ. Model Substrate/Inactivation Reactions for MoaA and Ribonucleotide Reductases: Loss of Bromo, Chloro, or Tosylate Groups from C2 of 1,5-Dideoxyhomoribofuranoses upon Generation of an α-Oxy Radical at C3. Molecules (Basel, Switzerland). 25. PMID 32486052 DOI: 10.3390/Molecules25112539 |
0.373 |
|
| 2014 |
Rayala R, Theard P, Ortiz H, Yao S, Young JD, Balzarini J, Robins MJ, Wnuk SF. Synthesis of purine and 7-deazapurine nucleoside analogues of 6-N-(4-Nitrobenzyl)adenosine; inhibition of nucleoside transport and proliferation of cancer cells. Chemmedchem. 9: 2186-92. PMID 24788480 DOI: 10.1002/Cmdc.201402047 |
0.349 |
|
| 2012 |
Balzarini J, Gago F, Kulik W, van Kuilenburg AB, Karlsson A, Peterson MA, Robins MJ. Introduction of a fluorine atom at C3 of 3-deazauridine shifts its antimetabolic activity from inhibition of CTP synthetase to inhibition of orotidylate decarboxylase, an early event in the de novo pyrimidine nucleotide biosynthesis pathway. The Journal of Biological Chemistry. 287: 30444-54. PMID 22730407 DOI: 10.1074/Jbc.M112.378091 |
0.307 |
|
| 2011 |
Nowak I, Damaraju VL, Cass CE, Young JD, Robins MJ. Autofluorescent fused-pyrimidine nucleosides: Synthesis and evaluation as permeants and inhibitors of human nucleoside transporters Collection of Czechoslovak Chemical Communications. 76: 1395-1412. DOI: 10.1135/Cccc2011061 |
0.376 |
|
| 2010 |
Robins MJ, Peng Y, Damaraju VL, Mowles D, Barron G, Tackaberry T, Young JD, Cass CE. Improved syntheses of 5'-S-(2-aminoethyl)-6-N-(4-nitrobenzyl)-5'-thioadenosine (SAENTA), analogues, and fluorescent probe conjugates: analysis of cell-surface human equilibrative nucleoside transporter 1 (hENT1) levels for prediction of the antitumor efficacy of gemcitabine. Journal of Medicinal Chemistry. 53: 6040-53. PMID 20718495 DOI: 10.1021/Jm100432W |
0.337 |
|
| 2010 |
Robins MJ, Doboszewski B, Timoshchuk VA, Peterson MA. ChemInform Abstract: Nucleic Acid Related Compounds. Part 111. Glucose-Derived 3′-(Carboxymethyl)-3′-deoxyribonucleosides and 2′,3′-Lactones as Synthetic Precursors for Amide-Linked Oligonucleotide Analogues. Cheminform. 31: no-no. DOI: 10.1002/chin.200035202 |
0.311 |
|
| 2010 |
Peterson MA, Nilsson BL, Sarker S, Doboszewski B, Zhang W, Robins MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 110. Amide-Linked Ribonucleoside Dimers Derived from 5′-Amino-5′-deoxy- and 3′-(Carboxymethyl)-3′-deoxynucleoside Precursors. Cheminform. 31: no-no. DOI: 10.1002/chin.200007202 |
0.328 |
|
| 2010 |
MILES RW, SAMANO V, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 87. Nucleophilic Functionalization of Cytidine and 2′-Deoxycytidine Derivatives via Elaboration of the 4-Amino Group into a Readily Displaced 1,2,4- Triazol-4-yl Substituent. Cheminform. 27: no-no. DOI: 10.1002/chin.199611275 |
0.314 |
|
| 2010 |
MILES RW, SAMANO V, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 86. Nucleophilic Functionalization of Adenine, Adenosine, Tubercidin, and Formycin Derivatives via Elaboration of the Heterocyclic Amino Group into a Readily Displaced 1,2,4-Triazol-4-yl Substituen Cheminform. 26: no-no. DOI: 10.1002/chin.199540244 |
0.304 |
|
| 2010 |
SAMANO V, MILES RW, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 85. Efficient Conversion of 6- Aminopurines and Nucleosides into 6-Substituted Analogues via Novel 6-( 1,2,4-Triazol-4-yl)purine Derivatives. Cheminform. 26: no-no. DOI: 10.1002/chin.199517033 |
0.332 |
|
| 2010 |
WNUK SF, STOECKLER JD, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 82. Conversions of Adenosine to Inosine 5′-Thioether Derivatives with Aspergillus oryzae Adenosine Deaminase or Alkyl Nitrites. Substrate and Inhibitory Activities of Inosine 5′-Thioether Derivativ Cheminform. 26: no-no. DOI: 10.1002/chin.199502185 |
0.332 |
|
| 2010 |
SAMANO V, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 83. Synthesis of 3′- Deoxyadenosine-3′-spirocyclopropane, 3′-Deoxyuridine-3′- spirocyclopropane, and 5′-Deoxy-4′,5′-methanoadenosine. Cheminform. 25: no-no. DOI: 10.1002/chin.199442254 |
0.306 |
|
| 2010 |
ROBINS MJ, WNUK SF, MULLAH KB, DALLEY NK, YUAN C, LEE Y, BORCHARDT RT. ChemInform Abstract: Nucleic Acid Related Compounds. Part 80. Synthesis of 5′-S-(Alkyl and aryl)-5′-fluoro-5′-thioadenosines with Xenon Difluoride or ( Diethylamido)sulfur Trifluoride, Hydrolysis in Aqueous Buffer, and inhibition of S-Adenosyl-L-homocyste Cheminform. 25: no-no. DOI: 10.1002/chin.199426263 |
0.322 |
|
| 2010 |
WNUK SF, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 78. Stereocontrolled Syntheses of 6′(E and Z)-Halovinyl Analogues from Uridine-Derived Vinylsulfones via Vinyltin Intermediates. Cheminform. 24: no-no. DOI: 10.1002/chin.199330281 |
0.302 |
|
| 2010 |
SAMANO V, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 77. 2′,3′-Didehydro-2′,3′-dideoxy- 2′(and 3′)-methylnucleosides via (3.3)-Sigmatropic Rearrangements of 2′ (and 3′)-Methylene-3′(and 2′)-O-thiocarbonyl Derivatives and Radical Reduction of a 2′-Chl Cheminform. 24: no-no. DOI: 10.1002/chin.199330280 |
0.312 |
|
| 2010 |
WNUK SF, DALLEY NK, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 76. Synthesis of 5′(E- and Z)- Chloro-4′,5′-didehydro-5′-deoxyadenosines via Chlorination and Thermolysis of Adenosine 5′-Sulfoxides. Mechanism-Based Inhibition of S-Adenosyl-L-homocysteine Hydrola Cheminform. 24: no-no. DOI: 10.1002/chin.199321232 |
0.306 |
|
| 2010 |
ROBINS MJ, MULLAH KB, WNUK SF, DALLEY NK. ChemInform Abstract: Nucleic Acid Related Compounds. Part 73. Fluorination of Uridine 2′-Thioethers with Xenon Difluoride or (Diethylamino)sulfur Trifluoride. Synthesis of Stable 2′-(Alkyl(or Aryl)sulfonyl)-2′-deoxy-2′-fluorouridines. Cheminform. 23: no-no. DOI: 10.1002/chin.199234297 |
0.35 |
|
| 2010 |
SAMANO V, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 75. Synthesis and Radical-Induced Ring-Opening Reactions of 2′-Deoxyadenosine-2′-spirocyclopropane and Its Uridine Analogue. Mechanistic Probes for Ribonucleotide Reductases. Cheminform. 23: no-no. DOI: 10.1002/chin.199234295 |
0.338 |
|
| 2010 |
WNUK SF, DALLEY NK, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 67. Synthesis of 5′-Amino and 5′-Methylthio Chain-Extended Nucleosides from Uridine. Cheminform. 23: no-no. DOI: 10.1002/chin.199227268 |
0.305 |
|
| 2010 |
SAMANO MC, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 69. Efficient Reduction of Azides to Amines with Tributylstannane. High-Yield Synthesis of Amino and Diamino Deoxynucleosides. Cheminform. 23: no-no. DOI: 10.1002/chin.199226284 |
0.311 |
|
| 2010 |
SAMANO V, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 70. Synthesis of 2′(and 3′)-Deoxy- 2′(and 3′)-methyleneadenosines and Bis(methylene)furan 4′,5′-Didehydro- 5′-deoxy-2′(and 3′)-methyleneadenosines. Inhibitors of S-Adenosyl-L- homocysteine Hydrolas Cheminform. 23: no-no. DOI: 10.1002/chin.199222243 |
0.305 |
|
| 2010 |
ROBINS MJ, WNUK SF, MULLAH KB, DALLEY NK. ChemInform Abstract: Nucleic Acid Related Compounds. Part 68. Fluorination of C5′ of Nucleoside 5′-Thioethers with DAST/Antimony(III) Chloride or Xenon Difluoride to give 5′-S-Aryl-5′-fluoro-5′-thiouridines. Cheminform. 23: no-no. DOI: 10.1002/chin.199218275 |
0.314 |
|
| 2010 |
ROBINS MJ, HANSSKE F, WNUK SF, KANAI T. ChemInform Abstract: Nucleic Acid Related Compounds. Part 66. Improved Syntheses of 5′- Chloro-5′-deoxy- and 5′-S-Aryl(or Alkyl)-5′-thionucleosides. Cheminform. 23: no-no. DOI: 10.1002/chin.199206280 |
0.325 |
|
| 2010 |
SAMANO V, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 62. Stereoselective Addition of a Wittig Reagent to Give a Single Nucleoside Oxaphosphetane Diastereomer. Synthesis of 2′(and 3′)-Deoxy-2′(and 3′)-methyleneuridine (and - cytidine) Derivatives from Cheminform. 22: no-no. DOI: 10.1002/chin.199144292 |
0.353 |
|
| 2010 |
CHEN YJ, HANSSKE F, JANDA KD, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 64. Synthesis of 2′,3′-Diazido-2′, 3′-dideoxyadenosine and 2′,3′-Diamino-2′,3′-dideoxyadenosine from 9-(. beta.-D-Arabinofuranosyl)adenine. Cheminform. 22: no-no. DOI: 10.1002/chin.199139245 |
0.31 |
|
| 2010 |
WNUK SF, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 63. Synthesis of 5′-Deoxy-5′- methyleneadenosine and Related Wittig-Extended Nucleosides. Cheminform. 22: no-no. DOI: 10.1002/chin.199128231 |
0.321 |
|
| 2010 |
SAMANO V, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 60. Mild Periodinane Oxidation of Protected Nucleosides to give 2′- and 3′-Keto Nucleosides. The First Isolation of a Purine 2′-Deoxy 3′-Keto Nucleoside Derivative. Cheminform. 22: no-no. DOI: 10.1002/chin.199106286 |
0.314 |
|
| 2009 |
Robins MJ, Yang H, Miranda K, Peterson MA, De Clercq E, Balzarini J. Synthesis and biological evaluation of 3,3-difluoropyridine-2,4(1H,3H)-dione and 3-deaza-3-fluorouracil base and nucleoside derivatives. Journal of Medicinal Chemistry. 52: 3018-27. PMID 19378989 DOI: 10.1021/Jm900203H |
0.385 |
|
| 2009 |
Miles DW, Inskeep WH, Robins MJ, Winkley MW, Robins RK, Eyring H. Circular dichroism of nucleoside derivatives. VII. The electronic structure and spectra of some simple nucleoside derivatives International Journal of Quantum Chemistry. 3: 129-145. DOI: 10.1002/Qua.560030718 |
0.357 |
|
| 2007 |
Robins MJ, Nowak I, Wnuk SF, Hansske F, Madej D. Deoxygenative [1,2]-hydride shift rearrangements in nucleoside and sugar chemistry: analogy with the [1,2]-electron shift in the deoxygenation of ribonucleotides by ribonucleotide reductases. The Journal of Organic Chemistry. 72: 8216-21. PMID 17918996 DOI: 10.1021/Jo071102B |
0.374 |
|
| 2007 |
Robins MJ, Nowak I, Rajwanshi VK, Miranda K, Cannon JF, Peterson MA, Andrei G, Snoeck R, De Clercq E, Balzarini J. Synthesis and antiviral evaluation of 6-(alkyl-heteroaryl)furo[2,3-d]pyrimidin-2(3H)-one nucleosides and analogues with ethynyl, ethenyl, and ethyl spacers at C6 of the furopyrimidine core. Journal of Medicinal Chemistry. 50: 3897-905. PMID 17622128 DOI: 10.1021/Jm070210N |
0.419 |
|
| 2007 |
Liu J, Robins MJ. S(N)Ar displacements with 6-(fluoro, chloro, bromo, iodo, and alkylsulfonyl)purine nucleosides: synthesis, kinetics, and mechanism1. Journal of the American Chemical Society. 129: 5962-8. PMID 17439120 DOI: 10.1021/Ja070021U |
0.637 |
|
| 2007 |
Nowak I, Robins MJ. Synthesis of 3'-deoxynucleosides with 2-oxabicyclo[3.1.0]hexane sugar moieties: addition of difluorocarbene to a 3',4'-unsaturated uridine derivative and 1,2-dihydrofurans derived from D- and L-xylose1. The Journal of Organic Chemistry. 72: 3319-25. PMID 17385920 DOI: 10.1021/Jo062614D |
0.381 |
|
| 2007 |
Nowak I, Cannon JF, Robins MJ. Addition of difluorocarbene to 3',4'-unsaturated nucleosides: synthesis of 2'-deoxy analogues with a 2-oxabicyclo[3.1.0]hexane framework. The Journal of Organic Chemistry. 72: 532-7. PMID 17221971 DOI: 10.1021/Jo061965P |
0.403 |
|
| 2006 |
Zhong M, Robins MJ. Regiospecific N9 alkylation of 6-(heteroaryl)purines: shielding of N7 by a proximal heteroaryl C-H1. The Journal of Organic Chemistry. 71: 8901-6. PMID 17081021 DOI: 10.1021/Jo061759H |
0.565 |
|
| 2006 |
Nowak I, Robins MJ. Addition of difluorocarbene to 4',5'-unsaturated nucleosides: synthesis and deoxygenation reactions of difluorospirocyclopropane nucleosides. The Journal of Organic Chemistry. 71: 8876-83. PMID 17081018 DOI: 10.1021/Jo061606U |
0.423 |
|
| 2006 |
Zhong M, Nowak I, Robins MJ. Regiospecific and highly stereoselective coupling of 6-(substituted-imidazol-1-yl)purines with 2-deoxy-3,5-di-O-(p-toluoyl)-alpha-D-erythro-pentofuranosyl chloride. Sodium-salt glycosylation in binary solvent mixtures: improved synthesis of cladribine. The Journal of Organic Chemistry. 71: 7773-9. PMID 16995685 DOI: 10.1021/Jo061282+ |
0.604 |
|
| 2006 |
Nowak I, Cannon JF, Robins MJ. N-oxides of adenosine-type nucleosides undergo pyrimidine ring opening and closure to give 5-amino-4-(1,2,4-oxadiazol-3-yl)imidazole derivatives. Organic Letters. 8: 4565-8. PMID 16986951 DOI: 10.1021/Ol061715V |
0.416 |
|
| 2006 |
Zhang J, Smith KM, Tackaberry T, Sun X, Carpenter P, Slugoski MD, Robins MJ, Nielsen LP, Nowak I, Baldwin SA, Young JD, Cass CE. Characterization of the transport mechanism and permeant binding profile of the uridine permease Fui1p of Saccharomyces cerevisiae. The Journal of Biological Chemistry. 281: 28210-21. PMID 16854981 DOI: 10.1074/Jbc.M605129200 |
0.303 |
|
| 2006 |
Zhong M, Nowak I, Cannon JF, Robins MJ. Structure and synthesis of 6-(substituted-imidazol-1-yl)purines: versatile substrates for regiospecific alkylation and glycosylation at N9. The Journal of Organic Chemistry. 71: 4216-21. PMID 16709063 DOI: 10.1021/Jo060340O |
0.623 |
|
| 2006 |
Nowak I, Jones CT, Robins MJ. Selective removal of the 2'- and 3'-O-acyl groups from 2',3',5'-tri-O-acylribonucleoside derivatives with lithium trifluoroethoxide. The Journal of Organic Chemistry. 71: 3077-81. PMID 16599602 DOI: 10.1021/Jo0600104 |
0.317 |
|
| 2006 |
Robins MJ, Miranda K, Rajwanshi VK, Peterson MA, Andrei G, Snoeck R, De Clercq E, Balzarini J. Synthesis and biological evaluation of 6-(alkyn-1-yl)furo[2,3-d]pyrimidin-2(3H)-one base and nucleoside derivatives. Journal of Medicinal Chemistry. 49: 391-8. PMID 16392824 DOI: 10.1021/Jm050867D |
0.383 |
|
| 2006 |
Janeba Z, Maklad N, Robins MJ. Synthesis of 6-(alkoxymethyl)- and 6-(alkylsulfanylmethyl)furo[2,3-d] pyrimidin-2(3H)-one analogues Canadian Journal of Chemistry. 84: 561-568. DOI: 10.1139/V06-042 |
0.362 |
|
| 2006 |
Janeba Z, Balzarini J, Andrei G, Snoeck R, De Clercq E, Robins MJ. Synthesis and biological evaluation of 5-(alkyn-1-yl)-1-(p-toluenesulfonyl) uracil derivatives Canadian Journal of Chemistry. 84: 580-586. DOI: 10.1139/V06-041 |
0.407 |
|
| 2006 |
Lin X, Robins MJ. Nucleic acid related compounds. 136. Synthesis of 2-amino- and 2,6-diaminopurine derivatives via inverse-electron-demand Diels-Alder reactions Collection of Czechoslovak Chemical Communications. 71: 1029-1041. DOI: 10.1135/Cccc20061029 |
0.578 |
|
| 2005 |
Robins MJ, Wnuk SF. Reduction of ribonucleosides to 2'-deoxyribonucleosides. Current Protocols in Nucleic Acid Chemistry / Edited by Serge L. Beaucage ... [Et Al.]. Unit 1.11. PMID 18428933 DOI: 10.1002/0471142700.Nc0111S21 |
0.389 |
|
| 2005 |
Janeba Z, Maklad N, Robins MJ. An efficient alternative route to 3,6-disubstituted-furo[2,3-d]pyrimidin-2-one analogues. Nucleosides, Nucleotides & Nucleic Acids. 24: 1729-43. PMID 16438044 DOI: 10.1080/10810730500265757 |
0.432 |
|
| 2005 |
Nowak I, Robins MJ. Hydrothermal deamidation of 4-N-acylcytosine nucleoside derivatives: efficient synthesis of uracil nucleoside esters. Organic Letters. 7: 4903-5. PMID 16235918 DOI: 10.1021/Ol0518378 |
0.413 |
|
| 2005 |
Zhong M, Nowak I, Robins MJ. 6-(2-Alkylimidazol-1-yl)purines undergo regiospecific glycosylation at N9. Organic Letters. 7: 4601-3. PMID 16209489 DOI: 10.1021/Ol051573P |
0.558 |
|
| 2005 |
Nowak I, Conda-Sheridan M, Robins MJ. Nucleic acid related compounds. 127. Selective N-deacylation of N,O-peracylated nucleosides in superheated methanol. The Journal of Organic Chemistry. 70: 7455-8. PMID 16122277 DOI: 10.1021/Jo051256W |
0.367 |
|
| 2005 |
Janeba Z, Balzarini J, Andrei G, Snoeck R, De Clercq E, Robins MJ. Synthesis and biological evaluation of acyclic 3-[(2-hydroxyethoxy)methyl] analogues of antiviral furo- and pyrrolo[2,3-d]pyrimidine nucleosides. Journal of Medicinal Chemistry. 48: 4690-6. PMID 16000005 DOI: 10.1021/Jm050291S |
0.363 |
|
| 2005 |
Liu J, Robins MJ. Fluoro, alkylsulfanyl, and alkylsulfonyl leaving groups in suzuki cross-coupling reactions of purine 2'-deoxynucleosides and nucleosides. Organic Letters. 7: 1149-51. PMID 15760161 DOI: 10.1021/Ol050063S |
0.628 |
|
| 2005 |
Nowak I, Robins MJ. New methodology for the deoxygenative difluoromethylenation of aldehydes and ketones; unexpected formation of tetrafluorocyclopropanes. Organic Letters. 7: 721-4. PMID 15704934 DOI: 10.1021/Ol047416S |
0.302 |
|
| 2004 |
Nowak I, Cannon JF, Robins MJ. Synthesis and properties of gem-(difluorocyclopropyl)amine derivatives of bicyclo[n.1.0]alkanes. Organic Letters. 6: 4767-70. PMID 15575681 DOI: 10.1021/Ol047943B |
0.374 |
|
| 2004 |
Liu J, Robins MJ. Azoles as Suzuki cross-coupling leaving groups: syntheses of 6-arylpurine 2'-deoxynucleosides and nucleosides from 6-(imidazol-1-yl)- and 6-(1,2,4-triazol-4-yl)purine derivatives. Organic Letters. 6: 3421-3. PMID 15355067 DOI: 10.1021/Ol048490D |
0.665 |
|
| 2004 |
Liu J, Janeba Z, Robins MJ. SNAr iodination of 6-chloropurine nucleosides: aromatic Finkelstein reactions at temperatures below -40 degrees C. Organic Letters. 6: 2917-9. PMID 15330647 DOI: 10.1021/Ol048987N |
0.63 |
|
| 2004 |
Janeba Z, Lin X, Robins MJ. Functionalization of guanosine and 2'-deoxyguanosine at C6: a modified Appel process and S(N)Ar displacement of imidazole. Nucleosides, Nucleotides & Nucleic Acids. 23: 137-47. PMID 15043142 DOI: 10.1081/Ncn-120027823 |
0.548 |
|
| 2003 |
Nowak I, Robins MJ. Protection of the amino group of adenosine and guanosine derivatives by elaboration into a 2,5-dimethylpyrrole moiety. Organic Letters. 5: 3345-8. PMID 12943423 DOI: 10.1021/Ol035264F |
0.362 |
|
| 2003 |
Janeba Z, Francom P, Robins MJ. Efficient syntheses of 2-chloro-2'-deoxyadenosine (cladribine) from 2'-deoxyguanosine(1). The Journal of Organic Chemistry. 68: 989-92. PMID 12558425 DOI: 10.1021/Jo020644K |
0.402 |
|
| 2003 |
Francom P, Robins MJ. Nucleic acid related compounds. 118. Nonaqueous diazotization of aminopurine derivatives. Convenient access to 6-halo- and 2,6-dihalopurine nucleosides and 2'-deoxynucleosides with acyl or silyl halides. The Journal of Organic Chemistry. 68: 666-9. PMID 12530909 DOI: 10.1021/Jo020625A |
0.424 |
|
| 2003 |
Zhong M, Robins MJ. Regioisomers in Vorbrüggen's guanine nucleoside synthesis; N9 selectivity with a glucosamine derivative and 2-N-acetyl-6-O- diphenylcarbamoylguanine Tetrahedron Letters. 44: 9327-9330. DOI: 10.1016/J.Tetlet.2003.10.070 |
0.557 |
|
| 2002 |
Wnuk SF, Companioni DR, Neschadimenko V, Robins MJ. The beta-fluorine effect. Electronic versus steric effects in radical deoxygenations of fluorine-containing pentofuranose nucleosides. The Journal of Organic Chemistry. 67: 8794-7. PMID 12467391 DOI: 10.1021/Jo020428B |
0.326 |
|
| 2002 |
Miles RW, Nielsen LP, Ewing GJ, Yin D, Borchardt RT, Robins MJ. S-homoadenosyl-L-cysteine and S-homoadenosyl-L-homocysteine. Synthesis and binding studies of hon-hydrolyzed substrate analogues with S-adenosyl-L-homocysteine hydrolase. The Journal of Organic Chemistry. 67: 8258-60. PMID 12423165 DOI: 10.1021/Jo020478G |
0.303 |
|
| 2002 |
Francom P, Janeba Z, Shibuya S, Robins MJ. Nucleic acid related compounds. 116. Nonaqueous diazotization of aminopurine nucleosides. Mechanistic considerations and efficient procedures with tert-butyl nitrite or sodium nitrite. The Journal of Organic Chemistry. 67: 6788-96. PMID 12227811 DOI: 10.1021/Jo0204101 |
0.373 |
|
| 2002 |
Wnuk SF, Chowdhury SM, Garcia PI, Robins MJ. Stereodefined synthesis of O3'-labeled uracil nucleosides. 3'-[(17)O]-2'-Azido-2'-deoxyuridine 5'-diphosphate as a probe for the mechanism of inactivation of ribonucleotide reductases. The Journal of Organic Chemistry. 67: 1816-9. PMID 11895397 DOI: 10.1021/Jo010899I |
0.306 |
|
| 2001 |
Robins MJ, Miles RW, Samano MC, Kaspar RL. Syntheses of puromycin from adenosine and 7-deazapuromycin from tubercidin, and biological comparisons of the 7-aza/deaza pair. The Journal of Organic Chemistry. 66: 8204-10. PMID 11722226 DOI: 10.1021/Jo010935D |
0.457 |
|
| 2001 |
Robins MJ, Wilson JS, Madej D, Tyrrell DLJ, Gati WP, Lindmark RJ, Wnuk SF. Nucleic acid related compounds. 114. Synthesis of 2,6-(disubstituted)purine 2′,3′-dideoxynucleosides and selected cytotoxic, anti-hepatitis B, and adenosine deaminase substrate activities Journal of Heterocyclic Chemistry. 38: 1297-1306. DOI: 10.1002/Jhet.5570380609 |
0.461 |
|
| 2001 |
Kumarasinghe ES, Peterson MA, Robins MJ. ChemInform Abstract: Synthesis of 5,6-Bis(alkyn-1-yl)pyrimidines and Related Nucleosides. Cheminform. 32: no-no. DOI: 10.1002/chin.200109138 |
0.304 |
|
| 2000 |
Yang X, Yin D, Wnuk SF, Robins MJ, Borchardt RT. Mechanisms of inactivation of human S-adenosylhomocysteine hydrolase by 5',5',6',6'-tetradehydro-6'-deoxy-6'-halohomoadenosines. Biochemistry. 39: 15234-41. PMID 11106503 DOI: 10.1021/Bi0015055 |
0.332 |
|
| 2000 |
Lin X, Robins MJ. Mild and efficient functionalization at C6 of purine 2'-deoxynucleosides and ribonucleosides. Organic Letters. 2: 3497-9. PMID 11082018 DOI: 10.1021/Ol000255H |
0.492 |
|
| 2000 |
Robins MJ, Doboszewski B, Timoshchuk VA, Peterson MA. Glucose-derived 3'-(carboxymethyl)-3'-deoxyribonucleosides and 2', 3'-lactones as synthetic precursors for amide-linked oligonucleotide analogues. The Journal of Organic Chemistry. 65: 2939-45. PMID 10814181 DOI: 10.1021/Jo991399G |
0.399 |
|
| 2000 |
Robins MJ, Doboszewski B, Nilsson BL, Peterson MA. Synthesis of amide-linked [(3')CH2CO-NH(5')] nucleoside analogues of small oligonucleotides. Nucleosides, Nucleotides & Nucleic Acids. 19: 69-86. PMID 10772703 DOI: 10.1080/15257770008032997 |
0.406 |
|
| 2000 |
Wnuk SF, Valdez CA, Khan J, Moutinho P, Robins MJ, Yang X, Borchardt RT, Balzarini J, De Clercq E. Doubly homologated dihalovinyl and acetylene analogues of adenosine: synthesis, interaction with S-adenosyl-L-homocysteine hydrolase, and antiviral and cytostatic effects. Journal of Medicinal Chemistry. 43: 1180-6. PMID 10737751 DOI: 10.1021/Jm990486Y |
0.391 |
|
| 2000 |
Kumarasinghe ES, Peterson MA, Robins MJ. Synthesis of 5,6-bis(alkyn-1-yl)pyrimidines and related nucleosides Tetrahedron Letters. 41: 8741-8745. DOI: 10.1016/S0040-4039(00)01566-5 |
0.425 |
|
| 2000 |
Lin X, Robins MJ. Mild and efficient functionalization at C6 of purine 2′-deoxynucleosides and ribonucleosides Organic Letters. 2: 3497-3499. |
0.437 |
|
| 1999 |
Peterson MA, Nilsson BL, Sarker S, Doboszewski B, Zhang W, Robins MJ. Amide-Linked Ribonucleoside Dimers Derived from 5'-Amino-5'-deoxy- and 3'-(Carboxymethyl)-3'-deoxynucleoside Precursors(1). The Journal of Organic Chemistry. 64: 8183-8192. PMID 11674735 DOI: 10.1021/Jo9908647 |
0.435 |
|
| 1999 |
Giziewicz J, Wnuk SF, Robins MJ. Nucleic Acid Related Compounds. 107. Efficient Nitration of Uracil Base and Nucleoside Derivatives(1). The Journal of Organic Chemistry. 64: 2149-2151. PMID 11674318 DOI: 10.1021/Jo9822939 |
0.385 |
|
| 1999 |
Robins MJ. Mechanism-based inhibition of ribonucleotide reductases: new mechanistic considerations and promising biological applications. Nucleosides & Nucleotides. 18: 779-93. PMID 10432680 DOI: 10.1080/15257779908041565 |
0.301 |
|
| 1999 |
Robins MJ, Guo Z, Samano MC, Wnuk SF. Biomimetic simulation of free radical-initiated cascade reactions postulated to occur at the active site of ribonucleotide reductases Journal of the American Chemical Society. 121: X-1432. DOI: 10.1021/Ja983449P |
0.345 |
|
| 1999 |
Guo Z, Samano MC, Krzykawski JW, Wnuk SF, Ewing GJ, Robins MJ. Biomimetic modeling of the abstraction of H3' by ribonucleotide reductases. 1,5-Hydrogen atom transfer of H3 to aminyl and oxyl, but not thlyl, free radicals in homoribofuranose derivatives Tetrahedron. 55: 5705-5718. DOI: 10.1016/S0040-4020(99)00238-0 |
0.372 |
|
| 1998 |
Maeba I, Morishita N, Francom P, Robins MJ. Synthesis of (S)-5-(4,5-Dihydroxypentyl)uracil from Pseudouridine and Clarification of Stereochemistry(1). The Journal of Organic Chemistry. 63: 7539-7541. PMID 11672413 DOI: 10.1021/Jo980975Q |
0.317 |
|
| 1998 |
Robins MJ, Lewandowska E, Wnuk SF. Nucleic Acid Related Compounds. 105. Synthesis of 2',3'-Didehydro-2',3'-dideoxynucleosides from Ribonucleoside Cyclic 2',3'-(Sulfates or Phosphates) or 2',3'-Dimesylates via Reductive Elimination with Sodium Naphthalenide(1). The Journal of Organic Chemistry. 63: 7375-7381. PMID 11672386 DOI: 10.1021/Jo981013M |
0.427 |
|
| 1998 |
Robins MJ, Wnuk SF, Yang X, Yuan CS, Borchardt RT, Balzarini J, De Clercq E. Inactivation of S-adenosyl-L-homocysteine hydrolase and antiviral activity with 5',5',6',6'-tetradehydro-6'-deoxy-6'-halohomoadenosine analogues (4'-haloacetylene analogues derived from adenosine). Journal of Medicinal Chemistry. 41: 3857-64. PMID 9748360 DOI: 10.1021/Jm980163M |
0.407 |
|
| 1998 |
Wnuk SF, Yuan CS, Borchardt RT, Robins MJ. Synthesis of homologated halovinyl derivatives from aristeromycin and their inhibition of human placental S-adenosyl-L-homocysteine hydrolase. Nucleosides & Nucleotides. 17: 99-113. PMID 9708344 DOI: 10.1080/07328319808005161 |
0.353 |
|
| 1998 |
Wnuk SF, Mao Y, Yuan CS, Borchardt RT, Andrei G, Balzarini J, De Clercq E, Robins MJ. Discovery of type II (covalent) inactivation of S-adenosyl-L-homocysteine hydrolase involving its "hydrolytic activity": synthesis and evaluation of dihalohomovinyl nucleoside analogues derived from adenosine. Journal of Medicinal Chemistry. 41: 3078-83. PMID 9685247 DOI: 10.1021/Jm9801410 |
0.398 |
|
| 1998 |
Robins MJ, Neschadimenko V, Ro B, Yuan C, Borchardt RT, Wnuk SF. Nucleic Acid Related Compounds. 101.S-Adenosyl-l-homocysteine Hydrolase Does Not Hydrate (5‘-Fluoro)vinyl or (6‘-Halo)homovinyl Analogues Derived from 3‘-Deoxyadenosine or 3‘-(Chloro or Fluoro)-3‘-deoxyadenosine1 Journal of Organic Chemistry. 63: 1205-1211. DOI: 10.1021/Jo971741U |
0.384 |
|
| 1998 |
Robins MJ, Neschadimenko V, Ro BO, Yuan CS, Borchardt RT, Wnuk SF. Nucleic Acid Related Compounds. 101. S-Adenosyl-L-homocysteine Hydrolase Does Not Hydrate (5′-Fluoro)vinyl or (6′-Halo)homovinyl Analogues Derived from 3′-Deoxyadenosine or 3′-(Chloro or Fluoro)-3′-deoxyadenosine Journal of Organic Chemistry. 63: 1205-1211. |
0.305 |
|
| 1997 |
Wnuk SF, Yuan CS, Borchardt RT, Balzarini J, De Clercq E, Robins MJ. Anticancer and antiviral effects and inactivation of S-adenosyl-L-homocysteine hydrolase with 5'-carboxaldehydes and oximes synthesized from adenosine and sugar-modified analogues. Journal of Medicinal Chemistry. 40: 1608-18. PMID 9171871 DOI: 10.1021/Jm960828P |
0.414 |
|
| 1997 |
Robins MJ, Zou R, Hansske F, Wnuk SF. Synthesis of sugar-modified 2,6-diaminopurine and guanine nucleosides from guanosine via transformations of 2-aminoadenosine and enzymatic deamination with adenosine deaminase Canadian Journal of Chemistry. 75: 762-767. DOI: 10.1139/V97-092 |
0.403 |
|
| 1997 |
Lewandowska E, Neschadimenko V, Wnuk SF, Robins MJ. Efficient removal of sugar O-tosyl groups and heterocycle halogens from purine nucleosides with sodium naphthalenide Tetrahedron. 53: 6295-6302. DOI: 10.1016/S0040-4020(97)00313-X |
0.392 |
|
| 1997 |
Robins MJ, Sarker S, Samano V, Wnuk SF. Nucleic acid related compounds. 94. Remarkably high stereoselective reductions of 2'- and 3'-ketonucleoside derivatives to give arabino, ribo, and xylofuranosyl nucleosides with hydrogen isotopes at C2' and C3' Tetrahedron. 53: 447-456. DOI: 10.1016/S0040-4020(96)01035-6 |
0.442 |
|
| 1996 |
Wnuk SF, Liu S, Yuan CS, Borchardt RT, Robins MJ. Inactivation of S-adenosyl-L-homocysteine hydrolase by amide and ester derivatives of adenosine-5'-carboxylic acid. Journal of Medicinal Chemistry. 39: 4162-6. PMID 8863793 DOI: 10.1021/Jm960313Y |
0.36 |
|
| 1996 |
Robins MJ, Zou R, Guo Z, Wnuk SF. Nucleic acid related compounds. 93. A solution for the historic problem of regioselective sugar-base coupling to produce 9-glycosylguanines or 7-glycosylguanines Journal of Organic Chemistry. 61: 9207-9212. DOI: 10.1021/Jo9617023 |
0.412 |
|
| 1996 |
Xie M, Berges DA, Robins MJ. Efficient "dehomologation" of di-O-isopropylidenehexofuranose derivatives to give O-isopropylidenepentofuranoses by sequential treatment with periodic acid in ethyl acetate and sodium borohydride Journal of Organic Chemistry. 61: 5178-5179. DOI: 10.1021/Jo960355U |
0.336 |
|
| 1996 |
Robins MJ, Wnuk SF, Hernández-Thirring AE, Samano MC. Nucleic acid related compounds. 91. Biomimetic reactions are in harmony with loss of 2'-substituents as free radicals (not anions) during mechanism-based inactivation of ribonucleotide reductases. Differential interactions of azide, halogen, and alkylthio groups with tributylstannane and triphenylsilane Journal of the American Chemical Society. 118: 11341-11348. DOI: 10.1021/Ja962117M |
0.361 |
|
| 1996 |
Wnuk SF, Robins MJ. Stannyl Radical-Mediated Cleavage of π-Deficient Heterocyclic Sulfones. Synthesis of α-Fluoro Esters and the First Homonucleoside α-Fluoromethylene Phosphonate1 Journal of the American Chemical Society. 118: 2519-2520. DOI: 10.1021/Ja953513S |
0.316 |
|
| 1996 |
Yuan CS, Liu S, Wnuk SF, Robins MJ, Borchardt RT. Design and synthesis of S-adenosylhomocysteine hydrolase inhibitors as broad-spectrum antiviral agents Advances in Antiviral Drug Design. 2: 41-88. DOI: 10.1016/S1075-8593(96)80103-1 |
0.33 |
|
| 1996 |
Robins MJ, Sarker S, Xie M, Zhang W, Peterson MA. Synthesis of 2',3'-fused (3.3.0) γ-butyrolactone-nucleosides and coupling with amino-nucleosides to give amide-linked nucleotide-dimer analogues Tetrahedron Letters. 37: 3921-3924. DOI: 10.1016/0040-4039(96)00715-0 |
0.439 |
|
| 1995 |
Robins M, Samano M, Samano V. Ribonucleotide Reductase Targets for Chemotherapy; Mechanistic Aspects and Biologically Active Agents Nucleosides, Nucleotides and Nucleic Acids. 14: 485-493. DOI: 10.1080/15257779508012411 |
0.311 |
|
| 1995 |
Robins MJ, Wilson JS, Madej D, Low NH, Hansske F, Wnuk SF. Nucleic Acid-Related Compounds. 88. Efficient Conversions of Ribonucleosides into Their 2',3'-Anhydro, 2'(and 3')-Deoxy, 2',3'-Didehydro-2',3'-dideoxy, and 2',3'-Dideoxynucleoside Analogs The Journal of Organic Chemistry. 60: 7902-7908. DOI: 10.1021/Jo00129A034 |
0.446 |
|
| 1995 |
Miles RW, Samano V, Robins MJ. Nucleic Acid Related Compounds. 87. Nucleophilic Functionalization of Cytidine and 2'-Deoxycytidine Derivatives via Elaboration of the 4-Amino Group into a Readily Displaced 1,2,4-Triazol-4-yl Substituent The Journal of Organic Chemistry. 60: 7066-7069. DOI: 10.1021/Jo00126A078 |
0.401 |
|
| 1995 |
Miles RW, Samano V, Robins MJ. Nucleic Acid Related Compounds. 86. Nucleophilic Functionalization of Adenine, Adenosine, Tubercidin, and Formycin Derivatives via Elaboration of the Heterocyclic Amino Group into a Readily Displaced 1,2,4-Triazol-4-yl Substituent Journal of the American Chemical Society. 117: 5951-5957. DOI: 10.1021/Ja00127A007 |
0.414 |
|
| 1994 |
Cory AH, Samano V, Robins MJ, Cory JG. 2'-Deoxy-2'-methylene derivatives of adenosine, guanosine, tubercidin, cytidine and uridine as inhibitors of L1210 cell growth in culture. Biochemical Pharmacology. 47: 365-71. PMID 8304981 DOI: 10.1016/0006-2952(94)90028-0 |
0.322 |
|
| 1994 |
Wnuk SF, Yuan CS, Borchardt RT, Balzarini J, De Clercq E, Robins MJ. Nucleic acid related compounds. 84. Synthesis of 6'-(E and Z)-halohomovinyl derivatives of adenosine, inactivation of S-adenosyl-L-homocysteine hydrolase, and correlation of anticancer and antiviral potencies with enzyme inhibition. Journal of Medicinal Chemistry. 37: 3579-87. PMID 7932585 DOI: 10.1021/Jm00047A015 |
0.361 |
|
| 1994 |
Wnuk SF, Stoeckler JD, Robins MJ. Nucleic Acid Related Compounds. 82. Conversions of Adenosine to Inosine 5′-Thioether Derivatives withAspergillus oryzaeAdenosine Deaminase or Alkyl Nitrites. Substrate and Inhibitory Activities of Inosine 5′-Thioether Derivatives with Purine Nucleoside Phosphorylase Nucleosides and Nucleotides. 13: 389-403. DOI: 10.1080/15257779408013249 |
0.439 |
|
| 1994 |
Robins MJ, Asakura J, Kaneko M, Shibuya S, Jakobs ES, Agbanyo FR, Cass CE, Paterson ARP. Synthesis of Substituted-Benzyl and Sugar-Modified Analogues of 6-N-(4-Nitrobenzyl)adenosine and Their Interactions with “ES” Nucleoside Transport Systems Nucleosides and Nucleotides. 13: 1627-1646. DOI: 10.1080/15257779408012177 |
0.352 |
|
| 1994 |
Robins MJ, Wnuk SF. Selected Aspects of the Chemistry and Biochemistry of Sulfur-Containing Nucleosides Phosphorus, Sulfur, and Silicon and the Related Elements. 95: 71-88. DOI: 10.1080/10426509408034202 |
0.455 |
|
| 1994 |
Robins MJ, Wnuk SF, Mullah KB, Dalley NK, Yuan C, Lee Y, Borchardt RT. Nucleic Acid Related Compounds. 80. Synthesis of 5'-S-(Alkyl and aryl)-5'-fluoro-5'-thioadenosines with Xenon Difluoride or (Diethylamido)sulfur Trifluoride, Hydrolysis in Aqueous Buffer, and Inhibition of S-Adenosyl-L-homocysteine hydrolase by derived "Adenosine 5'-Aldehyde" Species The Journal of Organic Chemistry. 59: 544-555. DOI: 10.1021/Jo00082A010 |
0.421 |
|
| 1994 |
Samano V, Miles RW, Robins MJ. Efficient Conversion of 6-Aminopurines and Nucleosides into 6-Substituted Analogs via Novel 6-(1,2,4-Triazol-4-yl)purine Derivatives. Journal of the American Chemical Society. 116: 9331-9332. DOI: 10.1021/Ja00099A061 |
0.396 |
|
| 1994 |
Samano V, Robins MJ. Synthesis of 3′-deoxyadenosine-3′-spirocyclopropane, 3′-deoxy-uridine-3′-spirocyclopropane, and 5′-deoxy-4′,5′-methanoadenosine Tetrahedron Letters. 35: 3445-3448. DOI: 10.1016/S0040-4039(00)73206-0 |
0.408 |
|
| 1993 |
Wnuk SF, Robins MJ. Nucleic acid related compounds. 78. Stereocontrolled syntheses of 6′(E and Z)-halovinyl analogues from uridine-derived vinylsulfones via vinyltin intermediates Canadian Journal of Chemistry. 71: 192-198. DOI: 10.1139/V93-028 |
0.355 |
|
| 1993 |
Samano V, Robins MJ. Nucleic acid related compounds. 77. 2′,3′-Didehydro-2′,3′-dideoxy-2′(and 3′)-methylnucleosides via [3,3]-sigmatropic rearrangements of 2′(and 3′)-methylene-3′(and 2′)-O-thiocarbonyl derivatives and radical reduction of a 2′-chloro-3′-methylene analogue Canadian Journal of Chemistry. 71: 186-191. DOI: 10.1139/V93-027 |
0.409 |
|
| 1993 |
Robins MJ, Wnuk SF. Nucleic acid related compounds. 79. Efficient conversions of thioethers to .alpha.-fluoro thioethers with DAST or DAST/antimony(III) chloride The Journal of Organic Chemistry. 58: 3800-3801. DOI: 10.1021/Jo00067A009 |
0.376 |
|
| 1993 |
Baraldi PG, Bazzanini R, Manfredini S, Simoni D, Robins MJ. Facile access to 2′-O-acyl prodrugs of 1- (β-d-arabinofuranosyl)-5(E)-(2-bromovinyl)uracil (BVAraU) via regioselective esterase-catalyzed hydrolysis of 2′ 3′, 5′-triesters1 Tetrahedron Letters. 34: 3177-3180. DOI: 10.1016/S0040-4039(00)93411-7 |
0.376 |
|
| 1992 |
Robins MJ, Samano V, Zhang W, Balzarini J, De Clercq E, Borchardt RT, Lee Y, Yuan CS. Nucleic acid related compounds. 74. Synthesis and biological activity of 2'(and 3')-deoxy-2'(and 3')-methylenenucleoside analogues that function as mechanism-based inhibitors of S-adenosyl-L-homocysteine hydrolase and/or ribonucleotide reductase. Journal of Medicinal Chemistry. 35: 2283-93. PMID 1613752 DOI: 10.1021/Jm00090A020 |
0.429 |
|
| 1992 |
Robins MJ, Hawrelak SD, Hernández AE, Wnuk SF. Nucleic Acid Related Compounds. LXXXI. Efficient General Synthesis of Purine (Amino, Azido, and Triflate)-Sugar Nucleosides Nucleosides and Nucleotides. 11: 821-834. DOI: 10.1080/07328319208021743 |
0.456 |
|
| 1992 |
Fleming SA, Rawlins DB, Samano V, Robins MJ. Photochemistry of nucleoside transport inhibitor 6-S-benzylated thiopurine ribonucleosides. Implications for a new class of photoaffinity labels Journal of Organic Chemistry. 57: 5968-5976. DOI: 10.1021/Jo00048A034 |
0.345 |
|
| 1992 |
Robins MJ, Mullah KB, Wnuk SF, Dalley NK. Nucleic acid related compounds. 73. Fluorination of uridine 2'-thioethers with xenon difluoride or (diethylamino)sulfur trifluoride. Synthesis of stable 2'-[alkyl(or aryl)sulfonyl]-2'-deoxy-2'-fluorouridines The Journal of Organic Chemistry. 57: 2357-2364. DOI: 10.1021/Jo00034A031 |
0.443 |
|
| 1992 |
Samano V, Robins MJ. Nucleic acid and related compounds. 75. Synthesis and radical-induced ring-opening reactions of 2'-deoxyadenosine-2'-spirocyclopropane and its uridine analogs. Mechanistic probes for ribonucleotide reductases Journal of the American Chemical Society. 114: 4007-4008. DOI: 10.1021/Ja00036A077 |
0.41 |
|
| 1991 |
Robins MJ, Manfredini S, Wood SG, Wanklin RJ, Rennie BA, Sacks SL. Nucleic acid related compounds. 65. New syntheses of 1-(beta-D-arabinofuranosyl)-5(E)-(2-iodovinyl)uracil (IVAraU) from vinylsilane precursors. Radioiodine uptake as a marker for thymidine kinase positive herpes viral infections. Journal of Medicinal Chemistry. 34: 2275-80. PMID 2067000 DOI: 10.1021/Jm00111A050 |
0.344 |
|
| 1991 |
Baker CH, Banzon J, Bollinger JM, Stubbe J, Samano V, Robins MJ, Lippert B, Jarvi E, Resvick R. 2'-Deoxy-2'-methylenecytidine and 2'-deoxy-2',2'-difluorocytidine 5'-diphosphates: potent mechanism-based inhibitors of ribonucleotide reductase. Journal of Medicinal Chemistry. 34: 1879-84. PMID 2061926 DOI: 10.1021/Jm00110A019 |
0.322 |
|
| 1991 |
Wnuk SF, Dalley NK, Robins MJ. Nucleic acid related compounds. 67. Synthesis of 5′-amino and 5′-methylthio chain-extended nucleosides from uridine Canadian Journal of Chemistry. 69: 2104-2111. DOI: 10.1139/V91-303 |
0.453 |
|
| 1991 |
Robins MJ, Hansske F, Wnuk SF, Kanai T. Nucleic acid related compounds. 66. Improved syntheses of 5′-chloro-5′-deoxy- and 5′-S-aryl(or alkyl)-5′-thionucleosides Canadian Journal of Chemistry. 69: 1468-1474. DOI: 10.1139/V91-217 |
0.438 |
|
| 1991 |
Wnuk SF, Robins MJ. Nucleic acid related compounds. 63. Synthesis of 5′-deoxy-5′-methyleneadenosine and related Wittig-extended nucleosides Canadian Journal of Chemistry. 69: 334-338. DOI: 10.1139/V91-051 |
0.395 |
|
| 1991 |
Samano V, Robins MJ. Stereoselective Addition of a Wittig Reagent To Give a Single Nucleoside Oxaphosphetane Diastereoisomer. Synthesis of 2′(and 3′)-Deoxy-2′(and 3′)-methyleneuridine (and cytidine) Derivatives from Uridine Ketonucleosides Synthesis. 1991: 283-288. DOI: 10.1055/S-1991-26774 |
0.468 |
|
| 1991 |
Samano V, Robins MJ. Nucleic acid related compounds. 70. Synthesis of 2'(and 3')-deoxy-2'(and 3')-methyleneadenosines and bis(methylene)furan 4',5'-didehydro-5'-deoxy-2'(and 3')-methyleneadenosines. Inhibitors of S-adenosyl-L-homocysteine hydrolase and ribonucleotide reductase The Journal of Organic Chemistry. 56: 7108-7113. DOI: 10.1021/Jo00025A029 |
0.409 |
|
| 1991 |
Robins MJ, Wnuk SF, Mullah KB, Dalley NK. Nucleic acid-related compounds. 68. Fluorination at C5' of nucleoside 5'-thioethers with DAST/antimony(III) chloride or xenon difluoride to give 5'-S-aryl-5'-fluoro-5'-thiouridines The Journal of Organic Chemistry. 56: 6878-6884. DOI: 10.1021/Jo00024A033 |
0.393 |
|
| 1991 |
Chen YCJ, Hansske F, Janda KD, Robins MJ. Nucleic acid related compounds. 64. Synthesis of 2',3'-diazido-2',3'-dideoxyadenosine and 2',3'-diamino-2',3'-dideoxyadenosine from 9-(.beta.-D-arabinofuranosyl)adenine The Journal of Organic Chemistry. 56: 3410-3413. DOI: 10.1021/Jo00010A042 |
0.367 |
|
| 1991 |
Samano MC, Robins MJ. Efficient reduction of azides to amines with tributylstannane. high-yield syntheses of amino and diamino deoxynucleosides Tetrahedron Letters. 32: 6293-6296. DOI: 10.1016/0040-4039(91)80150-5 |
0.405 |
|
| 1990 |
Samano V, Robins MJ. Nucleic acid related compounds. 60. Mild periodinane oxidation of protected nucleosides to give 2'- and 3'-ketonucleosides. The first isolation of a purine 2'-deoxy-3'-ketonucleoside derivative The Journal of Organic Chemistry. 55: 5186-5188. DOI: 10.1021/Jo00305A003 |
0.364 |
|
| 1990 |
Asakura J, Robins MJ. Cerium(IV)-mediated halogenation at C-5 of uracil derivatives The Journal of Organic Chemistry. 55: 4928-4933. DOI: 10.1021/Jo00303A033 |
0.3 |
|
| 1990 |
Robins MJ, Samano V, Johnson MD. Nucleic acid-related compounds. 58. Periodinane oxidation, selective primary deprotection, and remarkably stereoselective reduction of tert-butyldimethylsilyl-protected ribonucleosides. Synthesis of 9-(.beta.-D-xylofuranosyl)adenine or 3'-deuterioadenosine from adenosine The Journal of Organic Chemistry. 55: 410-412. DOI: 10.1021/Jo00289A004 |
0.424 |
|
| 1990 |
ROBINS MJ, SAMANO V, JOHNSON MD. ChemInform Abstract: Nucleic Acid Related Compounds. Part 58. Periodinane Oxidation, Selective Primary Deprotection, and Remarkably Stereoselective Reduction of tert-Butyldimethylsilyl-Protected Ribonucleosides. Synthesis of 9-(β-D-Xylofuranosyl)adenine o Cheminform. 21. DOI: 10.1002/chin.199024302 |
0.308 |
|
| 1989 |
Robins MJ, Wood SG, Dalley NK, Herdewijn P, Balzarini J, De Clercq E. Nucleic acid related compounds. 57. Synthesis, x-ray crystal structure, lipophilic partition properties, and antiretroviral activities of anomeric 3'-azido-2',3'-dideoxy-2,6-diaminopurine ribosides. Journal of Medicinal Chemistry. 32: 1763-8. PMID 2754702 DOI: 10.1021/Jm00128A017 |
0.341 |
|
| 1989 |
SAMANO MC, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 56. High-Yield Synthesis of 3′-Amino-3′-deoxynucleosides. Conversion of Adenosine (I) to 3′-Amino-3′-deoxyadenosine (VII). Cheminform. 20. DOI: 10.1002/chin.198949302 |
0.327 |
|
| 1989 |
ROBINS MJ, WNUK SF. ChemInform Abstract: Nucleic Acid-Related Compounds. Part 54. Fluorination at C5′ of Nucleosides. Synthesis of the New Class of 5′-Fluoro-5′-S-aryl (Alkyl) Thionucleosides from Adenosine. Cheminform. 20. DOI: 10.1002/chin.198919302 |
0.329 |
|
| 1988 |
Robins MJ, Madej D, Hansske F, Wilson JS, Gosselin G, Bergogne M, Imbach J, Balzarini J, Clercq ED. Nucleic acid related compounds. 53. Synthesis and biological evaluation of 2′-deoxy-β-threo-pentofuranosyl nucleosides. "Reversion to starting alcohol" in Barton-type reductions of thionocarbonates Canadian Journal of Chemistry. 66: 1258-1262. DOI: 10.1139/V88-204 |
0.424 |
|
| 1988 |
Robins MJ, Stanislaw WF. Fluorination at C5′ of nucleosides. Synthesis of the new class of 5′-fluoro-5′-S-aryl (alkyl) thionucleosides from adenosine. Tetrahedron Letters. 29: 5729-5732. DOI: 10.1016/S0040-4039(00)82174-7 |
0.404 |
|
| 1988 |
Asakura J, Robins MJ. Cerium(iv) catalyzed iodination at C5 of uracil nucleosides Tetrahedron Letters. 29: 2855-2858. DOI: 10.1016/0040-4039(88)85229-8 |
0.361 |
|
| 1987 |
De Clercq E, Balzarini J, Madej D, Hansske F, Robins MJ. Nucleic acid related compounds. 51. Synthesis and biological properties of sugar-modified analogues of the nucleoside antibiotics tubercidin, toyocamycin, sangivamycin, and formycin. Journal of Medicinal Chemistry. 30: 481-6. PMID 3820218 DOI: 10.1021/Jm00386A007 |
0.415 |
|
| 1987 |
Zou R, Robins MJ. High-yield regioselective synthesis of 9-glycosyl guanine nucleosides and analogues via coupling with 2-N-acetyl-6-O-diphenylcarbamoylguanine Canadian Journal of Chemistry. 65: 1436-1437. DOI: 10.1139/V87-243 |
0.405 |
|
| 1987 |
ZOU R, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 52. High-Yield Regioselective Synthesis of 9-Glycosyl Guanine Nucleosides and Analogues via Coupling with 2-N-Acetyl-6-O-diphenylcarbamoylguanine. Cheminform. 18. DOI: 10.1002/chin.198751354 |
0.353 |
|
| 1987 |
BIRNBAUM GI, DE CLERCQ E, HATFIELD PW, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 50. Synthesis and Conformational Studies of 4-Carbamoyl-1-((2-hydroxyethoxy)methyl)-5-(methylamino)imidazole and Derivatives as New Acyclonucleoside Analogues. Cheminform. 18. DOI: 10.1002/chin.198726170 |
0.32 |
|
| 1986 |
De Clercq E, Bernaerts R, Bergstrom DE, Robins MJ, Montgomery JA, Holy A. Antirhinovirus activity of purine nucleoside analogs. Antimicrobial Agents and Chemotherapy. 29: 482-7. PMID 3013084 DOI: 10.1128/Aac.29.3.482 |
0.328 |
|
| 1986 |
BUFFEL DK, MCGUIGAN C, ROBINS MJ. ChemInform Abstract: Nucleic Acid Related Compounds. Part 48. Photoaddition of Methanol to 9-(β-D- Ribofuranosyl)purine (Nebularine) to give Inhibitors of Adenosine Deaminase. Chemischer Informationsdienst. 17. DOI: 10.1002/Chin.198602322 |
0.58 |
|
| 1985 |
Buffel DK, McGuigan C, Robins MJ. Nucleic acid related compounds. 48. Photoaddition of methanol to 9-(.beta.-D-ribofuranosyl) purine (nebularine) to give inhibitors of adenosine deaminase. The Journal of Organic Chemistry. 50: 2664-2667. DOI: 10.1021/Jo00215A014 |
0.567 |
|
| 1985 |
Robins MJ, Hatfield PW, Balzarini J, Clercq ED. Nucleic Acid Related Compounds. 47. Synthesis And Biological Activities Of Pyrimidine And Purine “Acyclic” Nucleoside Analogs Cheminform. 16. DOI: 10.1002/Chin.198512237 |
0.406 |
|
| 1984 |
Robins MJ, Hatfield PW, Balzarini J, De Clercq E. Nucleic acid related compounds. 47. Synthesis and biological activities of pyrimidine and purine "acyclic" nucleoside analogues. Journal of Medicinal Chemistry. 27: 1486-92. PMID 6092636 DOI: 10.1021/Jm00377A018 |
0.388 |
|
| 1984 |
ROBINS MJ, HANSSKE F, LOW NH, PARK JI. ChemInform Abstract: NUCLEIC ACID-RELATED COMPOUNDS. 46. A MILD CONVERSION OF VICINAL DIOLS TO ALKENES. EFFICIENT TRANSFORMATION OF RIBONUCLEOSIDES INTO 2′-ENE AND 2′,3′-DIDEOXYNUCLEOSIDES Chemischer Informationsdienst. 15. DOI: 10.1002/chin.198421336 |
0.302 |
|
| 1983 |
De Clercq E, Descamps J, Balzarini J, Giziewicz J, Barr PJ, Robins MJ. Nucleic acid related compounds. 40. Synthesis and biological activities of 5-alkynyluracil nucleosides. Journal of Medicinal Chemistry. 26: 661-6. PMID 6302254 DOI: 10.1002/Chin.198338357 |
0.425 |
|
| 1983 |
Robins MJ, Wilson JS, Sawyer L, James MNG. Nucleic acid related compounds. 41. Restricted furanose conformations of 3′,5′-O-(1,1,3,3-tetraisopropyldisilox-1,3-diyl)nucleosides provide a convenient evaluation of anomeric configuration Canadian Journal of Chemistry. 61: 1911-1920. DOI: 10.1139/V83-328 |
0.412 |
|
| 1983 |
Robins MJ, Parker JMR. Chiral transformations of D-ribose to 2(S)-amino-2-[2,5-dihydro-5(R)-methylfuran-2(R)-yl]ethanoic acid, a diastereomer of the antibiotic (+)-furanomycin Canadian Journal of Chemistry. 61: 317-322. DOI: 10.1139/V83-057 |
0.383 |
|
| 1983 |
Robins MJ, Parker JMR. Chiral transformations of D-ribose to 2-(β-D-ribofuranosyl)-L and D-glycine and an anhydroallose hemiacetal used in C-nucleoside synthesis Canadian Journal of Chemistry. 61: 312-316. DOI: 10.1139/V83-056 |
0.367 |
|
| 1983 |
Robins MJ, Barr PJ. Nucleic acid related compounds. 39. Efficient conversion of 5-iodo to 5-alkynyl and derived 5-substituted uracil bases and nucleosides The Journal of Organic Chemistry. 48: 1854-1862. DOI: 10.1021/Jo00159A012 |
0.409 |
|
| 1983 |
Hansske F, Robins MJ. Nucleic acid related compounds. 45. A deoxygenative [1,2]-hydride shift rearrangement converting cyclic cis-diol monotosylates to inverted secondary alcohols Journal of the American Chemical Society. 105: 6736-6737. DOI: 10.1021/Ja00360A044 |
0.303 |
|
| 1983 |
Robins MJ, Wilson JS, Hansske F. Nucleic acid related compounds. 42. A general procedure for the efficient deoxygenation of secondary alcohols. Regiospecific and stereoselective conversion of ribonucleosides to 2'-deoxynucleosides Journal of the American Chemical Society. 105: 4059-4065. DOI: 10.1021/Ja00350A052 |
0.319 |
|
| 1983 |
ROBINS MJ, BARR PJ. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS. 39. EFFICIENT CONVERSION OF 5-IODO TO 5-ALKYNYL AND DERIVED 5-SUBSTITUTED URACIL BASES AND NUCLEOSIDES Chemischer Informationsdienst. 14. DOI: 10.1002/chin.198348328 |
0.313 |
|
| 1983 |
HANSSKE F, ROBINS MJ. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS. 43. A CONVENIENT PROCEDURE FOR THE SYNTHESIS OF 2′- AND 3′-KETONUCLEOSIDES Chemischer Informationsdienst. 14. DOI: 10.1002/chin.198331322 |
0.3 |
|
| 1982 |
Robins MJ, Hatfield PW. Nucleic acid related compounds. 37. Convenient and high-yield syntheses of N-[(2-hydroxyethoxy)methyl] heterocycles as "acyclic nucleoside" analogues Canadian Journal of Chemistry. 60: 547-553. DOI: 10.1139/V82-081 |
0.416 |
|
| 1982 |
ROBINS MJ, HATFIELD PW. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS. 37. CONVENIENT AND HIGH-YIELD SYNTHESES OF N-((2-HYDROXYETHOXY)METHYL)HETEROCYCLES AS “ACYCLIC NUCLEOSIDE” ANALOGS Chemischer Informationsdienst. 13. DOI: 10.1002/chin.198229302 |
0.319 |
|
| 1982 |
Robins MJ, Barr PJ, Giziewicz J. Nucleic acid related compounds. 38. Smooth and high-yield iodination and chlorination at C-5 of uracil bases and p-toluyl-protected nucleosides Canadian Journal of Chemistry. 60: 554-557. DOI: 10.1002/Chin.198228322 |
0.383 |
|
| 1982 |
ROBINS MJ, UZNANSKI B. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS. 33. CONVERSIONS OF ADENOSINE AND GUANOSINE TO O 2,6-DICHLORO, 2-AMINO-6-CHLORO, AND DERIVED PURINE NUCLEOSIDES Chemischer Informationsdienst. 13. DOI: 10.1002/chin.198204322 |
0.313 |
|
| 1981 |
Robins MJ, Uznański B. Nucleic acid related compounds. 34. Non-aqueous diazotization with tert-butyl nitrite. Introduction of fluorine, chlorine, and bromine at C-2 of purine nucleosides Canadian Journal of Chemistry. 59: 2608-2611. DOI: 10.1139/V81-375 |
0.344 |
|
| 1981 |
Robins MJ, Uznański B. Nucleic acid related compounds. 33. Conversions of adenosine and guanosine to 2,6-dichloro, 2-amino-6-chloro, and derived purine nucleosides Canadian Journal of Chemistry. 59: 2601-2607. DOI: 10.1139/V81-374 |
0.414 |
|
| 1981 |
Robins MJ, Hansske F, Bernier SE. Nucleic acid related compounds. 36. Synthesis of the 2′-O-methyl and 3′-O-methyl ethers of guanosine and 2-aminoadenosine and correlation of O′-methylnucleoside 13C nmr spectral shifts Canadian Journal of Chemistry. 59: 3360-3364. DOI: 10.1002/Chin.198218338 |
0.411 |
|
| 1981 |
Robins MJ, Kaneko C, Kaneko M. Nucleic acid related compounds. 35. Synthesis of 5-bromo- and 5-deuterio-3-deazauridine Canadian Journal of Chemistry. 59: 3356-3359. DOI: 10.1002/Chin.198218337 |
0.413 |
|
| 1979 |
Robins MJ, Hawrelak SD, Kanai T, Siefert JM, Mengel R. Nucleic acid related compounds. 30. Transformations of adenosine to the first 2',3'-aziridine-fused nucleosides, 9-(2,3-epimino-2,3-dideoxy-.beta.-D-ribofuranosyl)adenine and 9-(2,3-epimino-2,3-dideoxy-.beta.-D-lyxofuranosyl)adenine The Journal of Organic Chemistry. 44: 1317-1322. DOI: 10.1021/Jo01322A026 |
0.319 |
|
| 1979 |
Robins MJ, Sporns P, Muhs WH. Nucleic acid related compounds. 29. Thionyl chloride reactions with adenine nucleosides. Course of nucleophilic displacements and a preferential route to the 2′-chloro-arabino isomer Canadian Journal of Chemistry. 57: 274-282. DOI: 10.1002/Chin.197923296 |
0.432 |
|
| 1979 |
ROBINS MJ, SPORNS P, MUHS WH. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS. 29. THIONYL CHLORIDE REACTIONS WITH ADENINE NUCLEOSIDES. COURSE OF NUCLEOPHILIC DISPLACEMENTS AND A PREFERENTIAL ROUTE TO THE 2′-CHLORO-ARABINO ISOMER Chemischer Informationsdienst. 10. DOI: 10.1002/chin.197923296 |
0.311 |
|
| 1979 |
ROBINS MJ, HAWRELAK SD. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS. 28. 2′-AMINO-ARAA (9-(2-AMINO-2-DEOXY-β-D-ARABINOFURANOSYL)ADENINE). SYNTHESIS VIA NUCLEOSIDE-AZIRIDINE OR AZIDO INTERMEDIATES AND BIOLOGICAL EFFECTS Chemischer Informationsdienst. 10. DOI: 10.1002/chin.197903315 |
0.316 |
|
| 1978 |
ROBINS MJ, MUHS WH. ChemInform Abstract: PSEUDOURIDINE TRANSFORMATIONS. FORMATION OF 2′- AND 3′-DEOXYPSEUDOURIDINES VIA HALOGEN INTERMEDIATES USING α-ACETOXYISOBUTYRYL CHLORIDE Chemischer Informationsdienst. 9. DOI: 10.1002/Chin.197848216 |
0.316 |
|
| 1977 |
Robins MJ, MacCoss M, Wilson JS. Nucleic acid related compounds. 27. "Virtual coupling" of the anomeric proton of cyclic 2'-deoxynucleoside 3',5'-monophosphates. Reassessment of conformation using praseodymium shifts and assignment of H-2',2'' signals by biomimetic deuteration at C-2'. Journal of the American Chemical Society. 99: 4660-6. PMID 874229 DOI: 10.1021/Ja00456A023 |
0.354 |
|
| 1977 |
Robins MJ, MacCoss M. Nucleic acid related compounds. 26. A "geometry-only" method for determining the anomeric configuration of nucleosides based on the H-1' NMR signal of cyclic alpha and beta 3',5'-mononucleotides1. Journal of the American Chemical Society. 99: 4654-60. PMID 874228 DOI: 10.1021/Ja00456A022 |
0.321 |
|
| 1977 |
MacCoss M, Robins MJ, Rayner B, Imbach J. A new aspect of the use of 2′,3′-O-isopropylidene ribonucleosides for investigation of anomeric configuration Carbohydrate Research. 59: 575-579. DOI: 10.1016/S0008-6215(00)83197-3 |
0.32 |
|
| 1977 |
ROBINS MJ, MACCOSS M, WILSON JS. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS. 27. ′VIRTUAL COUPLING′ OF THE ANOMERIC PROTON N OF CYCLIC 2′-DEOXYNUCLEOSIDE 3′,5′-MONOPHOSPHATES. REASSESSMENT OF CONFORMATION USING PRASEODYMIUM SHIFTS AND ASSIGNMENT OF H-2′,2 SIGNALS BY BIOMIMETIC D Chemischer Informationsdienst. 8: no-no. DOI: 10.1002/Chin.197741065 |
0.414 |
|
| 1977 |
Robins MJ, Fouron Y, Muhs WH. Nucleic acid related compounds. 25. Syntheses of arabino, xylo, and lyxo-anhydro sugar nucleosides from tubercidin ribo-epoxide Canadian Journal of Chemistry. 55: 1260-1267. DOI: 10.1002/Chin.197727343 |
0.436 |
|
| 1977 |
Robins MJ, Jones RA, Mengel R. Nucleic acid related compounds. 24. Transformation of tubercidin 2′,3′-O-orthoacetate into halo, deoxy, epoxide, and unsaturated sugar nucleosides Canadian Journal of Chemistry. 55: 1251-1259. DOI: 10.1002/Chin.197727342 |
0.572 |
|
| 1977 |
ROBINS MJ, JONES RA, MENGEL R. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS. 24. TRANSFORMATION OF TUBERCIDIN 2′,3′-O-ORTHOACETATE INTO HALO, DEOXY, EPOXIDE, AND UNSATURATED SUGAR NUCLEOSIDES Chemischer Informationsdienst. 8: no-no. DOI: 10.1002/chin.197727342 |
0.5 |
|
| 1976 |
Robins MJ, Kanai T. Nucleic acid related compounds. 19. Concerning the mechanism of formation of "2,3′-imino-1-(β-D-lyxofuranosyl)uracil" [2-amino-1-(3-deoxy-β-D-lyxofuranosyl)-4-pyrimidinone-N 2→3′-anhydronucleoside] from O2→2′ cyclonucleosides and "ammonium azide" Journal of Organic Chemistry. 41: 1886-1887. PMID 1262996 DOI: 10.1021/Jo00872A051 |
0.368 |
|
| 1976 |
Robins MJ, Jones RA, Mengel R. Nucleic acid related compounds. 23. Transformation of ribonucleoside 2',3'-O-ortho esters into unsaturated and deoxy sugar nucleosides via enol ester-substituted iodo intermediates. Journal of the American Chemical Society. 98: 8213-7. PMID 993520 DOI: 10.1002/Chin.197711363 |
0.568 |
|
| 1976 |
Robins MJ, Mengel R, Jones RA, Fouron Y. Nucleic acid related compounds.22. Transformation of ribonucleoside 2,3'-O-ortho esters into halo, deoxy, and epoxy sugar nucleosides using acyl halides. Mechanism and structure of products. Journal of the American Chemical Society. 98: 8204-13. PMID 993519 DOI: 10.1002/Chin.197710371 |
0.532 |
|
| 1976 |
Robins MJ, MacCoss M, Naik SR, Ramani G. Nucleic acid related compounds. 21. Direct fluorination of uracil and cytosine bases and nucleosides using trifluoromethyl hypofluorite. Mechanism, stereochemistry, and synthetic applications. Journal of the American Chemical Society. 98: 7381-90. PMID 977870 DOI: 10.1002/Chin.197706320 |
0.369 |
|
| 1976 |
Robins MJ, Muhs WH. Synthesis of 2′-deoxytubercidin {4-amino-7-(2-deoxy-β-D-erythro-pentofuranosyl)pyrrolo[2,3-d]pyrimidine} from the parent antibiotic Journal of the Chemical Society, Chemical Communications. 269-269. DOI: 10.1039/C39760000269 |
0.401 |
|
| 1976 |
ROBINS MJ, MUHS WH. ChemInform Abstract: SYNTHESIS OF 2′-DEOXYTUBERCIDIN (4-AMINO-7-(2-DEOXY-β-D-ERYTHRO-PENTOFURANOSYL)PYRROLO(2,3-D)PYRIMIDINE) FROM THE PARENT ANTIBIOTIC Chemischer Informationsdienst. 7: no-no. DOI: 10.1002/Chin.197631332 |
0.338 |
|
| 1975 |
Robins MJ, Lee AS. Nucleic acid related compounds. 17.3-Deazuridine. Stannous chloride catalysis of cis-diol vs. phenolic base methylation with diazomethane. Journal of Medicinal Chemistry. 18: 1070-4. PMID 809580 DOI: 10.1002/Chin.197608346 |
0.361 |
|
| 1975 |
Robins MJ, Ramani G, MacCoss M. Nucleic Acid Related Compounds. 16. Direct Fluorination Of Uracil Nucleotides Using Trifluoromethyl Hypofluorite Canadian Journal of Chemistry. 53: 1302-1306. DOI: 10.1139/V75-178 |
0.351 |
|
| 1975 |
ROBINS MJ, RAMANI G, MACCOSS M. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS PART 16, DIRECT FLUORINATION OF URACIL NUCLEOTIDES USING TRIFLUOROMETHYL HYPOFLUORITE Chemischer Informationsdienst. 6: no-no. DOI: 10.1002/Chin.197535396 |
0.377 |
|
| 1975 |
ROBINS MJ, MACCOSS M, RAMANI G. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS PART 14, 3′-O-AMINOACYL-2′-O-METHYLADENOSINES AND 2′-O-AMINOACYL-3′-O-METHYLADENOSINES RELATED TO CHARGED TRNA TERMINI Chemischer Informationsdienst. 6: no-no. DOI: 10.1002/Chin.197507473 |
0.348 |
|
| 1974 |
Robins MJ, Naik SR, Lee AS. Nucleic acid related compounds. 12. The facile and high-yield stannous chloride catalyzed monomethylation of the cis-glycol system of nucleosides by diazomethane. The Journal of Organic Chemistry. 39: 1891-9. PMID 4853388 DOI: 10.1021/Jo00927A022 |
0.381 |
|
| 1974 |
Robins MJ, Fouron Y, Mengel R. Nucleic acid related compounds. 11. Adenosine 2',3'-ribo-epoxide. Synthesis, intramolecular degradation, and transformation into 3'-substituted xylofuranosyl nucleosides and the lyxo-epoxide. The Journal of Organic Chemistry. 39: 1564-70. PMID 4833508 DOI: 10.1021/Jo00924A025 |
0.423 |
|
| 1974 |
Robins MJ, Jones RA, MacCoss M. 3'-O-aminoacyl-2'-deoxyadenosines and 2'-O-aminoacyl-3'-deoxyadenosines related to charged transfer ribonucleic acid termini. Biochemistry. 13: 553-9. PMID 4543925 DOI: 10.1021/Bi00700A023 |
0.459 |
|
| 1974 |
Robins MJ, MacCoss M, Ramani G. Nucleic Acid Related Compounds. 14. 3′-O-Aminoacyl-2′-O-methyladenosines and 2′-O-Aminoacyl-3′-O-methyladenosines Related to Charged tRNA Termini Canadian Journal of Chemistry. 52: 3803-3813. DOI: 10.1139/V74-570 |
0.386 |
|
| 1974 |
Robins MJ, Jones RA. Nucleic acid related compounds. 9. Synthesis of 6-amino-9-(2-deoxy-D-erythro-pent-1-enofuranosyl)purine, the first 1', 2'-unsaturated purine nucleoside The Journal of Organic Chemistry. 39: 113-115. DOI: 10.1021/Jo00915A031 |
0.556 |
|
| 1974 |
ROBINS MJ, TRIP EM. ChemInform Abstract: NUCLEID ACID RELATED COMPOUNDS PART 13, 1-(2-DEOXY-D-ERYTHRO-PENT-1-ENOFURANOSYL) URACIL, SYNTHESIS OF THE FIRST 1′-2′-UNSATURATED PYRIMIDINE NUCLEOSIDE, A FURANOID N,O-KETENE ACETAL Chemischer Informationsdienst. 5: no-no. DOI: 10.1002/chin.197452470 |
0.371 |
|
| 1974 |
ROBINS MJ, FOURON Y, MENGEL R. ChemInform Abstract: NUCLEID ACID RELATED COMPOUNDS PART 11, ADENOSINE 2′,3′-RIBO-EPOXIDE, SYNTHESIS, INTRAMOLECULAR DEGRADATION, AND TRANSFORMATION INTO 3′-SUBSTITUTED XYLOFURANOSYL NUCLEOSIDES AND THE LYXO-EPOXIDE Chemischer Informationsdienst. 5: no-no. DOI: 10.1002/Chin.197441441 |
0.453 |
|
| 1974 |
ROBINS MJ, JONES RA. ChemInform Abstract: NUCLEID ACID RELATED COMPOUNDS PART 9, THE SYNTHESIS OF 6-AMINO-9-(2-DEOXY-D-ERYTHRO-PENT-1-ENOFURANOSYL)-PURINE, THE FIRST 1′,2′-UNSATURATED PURINE NUCLEOSIDE Chemischer Informationsdienst. 5: no-no. DOI: 10.1002/chin.197415485 |
0.526 |
|
| 1974 |
ROBINS MJ, BASOM GL. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS PART 8, DIRECT CONVERSION OF 2′-DEOXYINOSINE TO 6-CHLOROPURINE 2′-DEOXYRIBOSIDE AND SELECTED 6-SUBSTITUTED DEOXYNUCLEOSIDES AND THEIR EVALUATION AS SUBSTRATES OF ADENOSINE DEAMINASE Chemischer Informationsdienst. 5: no-no. DOI: 10.1002/chin.197403416 |
0.304 |
|
| 1973 |
Robins MJ, Trip EM. Sugar-modified N 6 -(3-methyl-2-butenyl)adenosine derivatives, N 6 -benzyl analogs, and cytokinin-related nucleosides containing sulfur or formycin. Biochemistry. 12: 2179-87. PMID 4710578 DOI: 10.1021/Bi00736A001 |
0.346 |
|
| 1973 |
Bloch A, Dutschman G, Currie BL, Robins RK, Robins MJ. Preparation and biological activity of various 3-deazapyrimidines and related nucleosides. Journal of Medicinal Chemistry. 16: 294-7. PMID 4200222 DOI: 10.1021/Jm00261A032 |
0.463 |
|
| 1973 |
Robins MJ, McCarthy Jr. JR, Jones RA, Mengel R. Nucleic Acid Related Compounds. 5. The Transformation of Formycin and Tubercidin into 2′- and 3′-Deoxynucleosides Canadian Journal of Chemistry. 51: 1313-1321. DOI: 10.1139/V73-198 |
0.559 |
|
| 1973 |
Robins MJ, Mengel R, Jone RA. Nucleic acid related compounds. VII. Conversion of ribonucleoside 2',3'-ortho esters into deoxy, epoxy, and unsaturated nucleosides Journal of the American Chemical Society. 95: 4074-4076. DOI: 10.1021/Ja00793A056 |
0.453 |
|
| 1973 |
Robins MJ, Basom GL. Nucleic Acid Related Compounds. 8. Direct Conversion of 2′-Deoxyinosine to 6-Chloropurine 2′-Deoxyriboside and Selected 6-Substituted Deoxynucleosides and Their Evaluation As Substrates of Adenosine Deaminase Canadian Journal of Chemistry. 51: 3161-3169. DOI: 10.1002/Chin.197403416 |
0.444 |
|
| 1973 |
ROBINS MJ, MENGEL R, JONES RA. ChemInform Abstract: NUCLEIC ACID RELATED COMPOUNDS PART 7, CONVERSION OF RIBONUCLEOSIDE 2′,3′-ORTHO ESTERS INTO DEOXY, EPOXY, AND UNSATURED NUCLEOSIDES Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/chin.197333433 |
0.516 |
|
| 1973 |
BLOCH A, DUTSCHMAN G, CURRIE BL, ROBINS RK, ROBINS MJ. ChemInform Abstract: HERST. UND BIOLOGISCHE AKTIVITAET EINIGER 3-DESAZA-PYRIMIDINE UND VERWANDTER NUCLEOSIDE Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/Chin.197329309 |
0.514 |
|
| 1973 |
ROBINS MJ, MCCARTHY JR, JONES RA, MENGEL R. ChemInform Abstract: NUCLEINSAEURE-VERWANDTE VERBINDUNGEN 5. MITT. UMWANDLUNG VON FORMYCIN UND TUBERCIDIN IN 2′- UND 3′-DESOXYNUCLEOSIDE Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/Chin.197328453 |
0.506 |
|
| 1972 |
Robins MJ, Naik SR. Nucleic acid related compounds. 1. Methylation and transformation of 4-methoxy-2-pyrimidinone 1- -D-ribofuranoside into 2'-O-methyl nucleoside components of ribonucleic acid, their analogs, and derivatives. Biochemistry. 10: 3591-7. PMID 5146572 DOI: 10.1021/Bi00795A017 |
0.394 |
|
| 1972 |
Christensen LF, Broom AD, Robins MJ, Bloch A. Synthesis and biological activity of selected 2,6-disubstituted-(2-deoxy- -and- -D-erythro-pentofuranosyl)purines. Journal of Medicinal Chemistry. 15: 735-9. PMID 4625489 DOI: 10.1021/Jm00277A010 |
0.338 |
|
| 1972 |
Robins MJ, Naik SR. Nucleic acid related compounds. 3. A facile synthesis of 5-fluorouracil bases and nucleosides by direct fluorination. Journal of the American Chemical Society. 93: 5277-8. PMID 4257572 DOI: 10.1021/Ja00749A063 |
0.403 |
|
| 1972 |
Robins M, Naik S. Additions and Corrections - Nucleic Acid Related Compounds. III. A Facile Synthesis of 5-Fluorouracil Bases and Nucleosides by Direct Fluorination Journal of the American Chemical Society. 94: 2158-2158. DOI: 10.1021/Ja00761A604 |
0.401 |
|
| 1971 |
Miles DW, Townsend LB, Robins MJ, Robins RK, Inskeep WH, Eyring H. Circular dichroism of nucleoside derivatives. X. Influence of solvents and substituents upon the Cotton effects of guanosine derivatives. Journal of the American Chemical Society. 93: 1600-8. PMID 5550248 |
0.555 |
|
| 1971 |
Robins MJ, Simon LN, Stout MG, Ivanovics GA, Schweizer MP, Rousseau RJ, Robins RK. Nucleoside peptides. I. The synthesis of 5'-deoxy-5'-amino-5'-N-aminoacyl peptide derivatives of guanosine, adenosine, and 2'-deoxyadenosine and their effect on cell-free protein synthesis. Journal of the American Chemical Society. 93: 1474-80. PMID 5548345 DOI: 10.1021/Ja00735A025 |
0.464 |
|
| 1971 |
Robins MJ, Currie BL, Robins RK, Broom AD. A Novel Nucleophilic Displacement of Benzoate by Sulfur During Thiation of 3-Deazauridine Tribenzoate Canadian Journal of Chemistry. 49: 3067-3068. DOI: 10.1139/V71-513 |
0.498 |
|
| 1971 |
Currie BL, Robins MJ, Robins RK. The synthesis of 3-deazaorotidine and related nucleoside derivatives of 4-hydroxy-2-pyridone Journal of Heterocyclic Chemistry. 8: 221-224. DOI: 10.1002/Jhet.5570080207 |
0.517 |
|
| 1971 |
ROBINS MJ, CURRIE BL, ROBINS RK, BROOM AD. ChemInform Abstract: NEUE SUBSTITUTION VON BENZOAT DURCH SCHWEFEL BEI DER THIIERUNG VON 3-DESAZAURIDINTRIBENZOAT Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/Chin.197151392 |
0.525 |
|
| 1971 |
CURRIE BL, ROBINS MJ, ROBINS RK. ChemInform Abstract: DIE SYNTHESE VON 3-DESAZAOROTIDIN UND AEHNLICHEN NUCLEOSIDEN DES 4-HYDROXY-2-PYRIDONS Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/Chin.197135385 |
0.51 |
|
| 1971 |
PUGMIRE RJ, GRANT DM, ROBINS MJ, ROBINS RK. ChemInform Abstract: (13)C-NMR 19. MITT. BENZIMIDAZOL, PURIM UND DEREN ANION- UND KATION-SPEZIES 20. MITT. 4-AZA-INDEN (PYRROCOLIN) UND VERWANDTE N-BRUECKENKOPF-HETEROCYCLEN Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/Chin.197128077 |
0.498 |
|
| 1971 |
ROBINS MJ, SIMON LN, STOUT MG, IVANOVICS GA, SCHWEIZER MP, ROUSSEAU RJ, ROBINS RK. ChemInform Abstract: NUCLEOSIDPEPTIDE 1. MITT. SYNTHESE VON 5′-N-AMINOACYL-5′-DESOXY-5′-AMINO-DERIVATEN VON GUANOSIN, ADENOSIN UND 2′-DESOXY-ADENOSIN UND IHR EINFLUSS AUF DIE ZELLFREIE PROTEIN-SYNTHESE Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/Chin.197125377 |
0.541 |
|
| 1971 |
MILES DW, TOWNSEND LB, ROBINS MJ, ROBINS RK, INSKEEP WH, EYRING H. ChemInform Abstract: CIRCULARDICHROISMUS VON NUCLEOSIDDERIVATIVEN 10. MITT. LOESUNGSMITTEL- UND SUBSTITUENTENEINFLUSS AUF DIE COTTON-EFFEKTE VON GUANOSINDERIVATEN Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/Chin.197125072 |
0.566 |
|
| 1970 |
Shuman DA, Robins MJ, Robins RK. The synthesis of nucleos9de sulfamates related to nucleocidin. Journal of the American Chemical Society. 92: 3434-40. PMID 5422764 DOI: 10.1021/Ja00714A035 |
0.49 |
|
| 1970 |
Miles DW, Inskeep WH, Robins MJ, Winkley MW, Robins RK, Eyring H. Circular dichroism of nucleoside derivatives. IX. Vicinal effects on the circular dichroism of pyrimidine nucleosides. Journal of the American Chemical Society. 92: 3872-81. PMID 5419044 DOI: 10.1021/Ja00716A007 |
0.513 |
|
| 1970 |
Robins MJ, Khwaja TA, Robins RK. Purine nucleosides. XXIX. The synthesis of 2'-deoxy-L-adenosine and 2'-deoxy-L-guanosine and their alpha anomers. The Journal of Organic Chemistry. 35: 636-9. PMID 5416936 DOI: 10.1021/Jo00828A019 |
0.447 |
|
| 1970 |
Currie BL, Robins RK, Robins MJ. The synthesis of 3-deazapyrimidine nucleosides related to uridine and cytidine and their derivatives Journal of Heterocyclic Chemistry. 7: 323-329. DOI: 10.1002/Jhet.5570070211 |
0.457 |
|
| 1970 |
MILES DW, INSKEEP WH, ROBINS MJ, WINKLEY MW, ROBINS RK, EYRING H. ChemInform Abstract: CIRCULARDICHROISMUS VON NUCLEOSIDDERIVATEN 9. MITT. VICINALE EFFEKTE AUF DEN CIRCULARDICHROISMUS VON PYRIMIDIN-NUCLEOSIDEN Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/Chin.197040068 |
0.487 |
|
| 1970 |
SHUMAN DA, ROBINS MJ, ROBINS RK. ChemInform Abstract: SYNTH. VON NUCLEOCIDIN-AEHNLICHEN NUCLEOSID-SULFAMATEN Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/Chin.197034413 |
0.491 |
|
| 1970 |
CURRIE BL, ROBINS RK, ROBINS MJ. ChemInform Abstract: SYNTH. VON 3-DESAZAPYRIMIDIN-NUCLEOSIDEN ANALOG DEM URIDIN UND CYTIDIN SOWIE IHRER DERIVATE Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/Chin.197032440 |
0.531 |
|
| 1970 |
ROBINS MJ, KHWAJA TA, ROBINS RK. ChemInform Abstract: PURIN-NUCLEOSIDE 29. MITT. SYNTH. VON 2′-DESOXY-L-ADENOSIN UND 2′-DESOXY-L-GUANOSIN UND IHREN ALPHA-ANOMEREN Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/Chin.197025377 |
0.451 |
|
| 1970 |
PUGMIRE RJ, GRANT DM, ROBINS MJ, ROBINS RK. ChemInform Abstract: C(13)-NMR 14. MITT. AZAANALOGA POLYCYCLISCHER AROMATISCHER KOHLENWASSERSTOFFE Chemischer Informationsdienst. Organische Chemie. 1: no-no. DOI: 10.1002/Chin.197006011 |
0.459 |
|
| 1969 |
Robins MJ, Robins RK. Purine nucleosides. XXIV. A new method for the synthesis of guanine nucleosides. The preparation of 2'-deoxy-alpha and beta-guanosines and the corresponding N2-methyl derivatives. The Journal of Physical Chemistry. 34: 2160-3. PMID 5788210 DOI: 10.1021/Jo01259A029 |
0.503 |
|
| 1969 |
Miles DW, Robins MJ, Robins RK, Winkley MW, Eyring H. Circular dichroism of nucleoside derivatives. IV. Uracil derivatives. Journal of the American Chemical Society. 91: 824-31. PMID 5781567 DOI: 10.1021/Ja01032A005 |
0.508 |
|
| 1969 |
Miles DW, Robins MJ, Robins RK, Winkley MW, Eyring H. Circular dichroism of nucleoside derivatives. V. Cytosine derivatives. Journal of the American Chemical Society. 91: 831-8. PMID 5778273 DOI: 10.1021/Ja01032A006 |
0.474 |
|
| 1969 |
Miles DW, Robins MJ, Robins RK, Eyring H. Circular dichroism of nucleoside derivatives. VI. The optically active bands of adenine nucleoside derivatives. Proceedings of the National Academy of Sciences of the United States of America. 62: 22-9. PMID 5253660 DOI: 10.1073/Pnas.62.1.22 |
0.413 |
|
| 1969 |
Stout MG, Robins MJ, Olsen RK, Robins RK. Purine nucleosides. XXV. The synthesis of certain derivatives of 5'-amino-5'-deoxy- and 5'-amino-2',5'-dideoxy-beta-d-ribofuranosylpurines as purine nucleotide analogs. Journal of Medicinal Chemistry. 12: 658-62. PMID 4893464 DOI: 10.1021/Jm00304A022 |
0.523 |
|
| 1969 |
Shuman DA, Bloch A, Robins RK, Robins MJ. Synthesis and biological activity of certain 8-mercaptopurine and 6-mercaptopyrimidine S-nucleosides. Journal of Medicinal Chemistry. 12: 653-7. PMID 4893463 DOI: 10.1021/Jm00304A021 |
0.476 |
|
| 1969 |
Pugmire RJ, Grant DM, Robins MJ, Robins RK. Carbon-13 magnetic resonance. XIV. Aza-analogs of polycyclic aromatic hydrocarbons Journal of the American Chemical Society. 91: 6381-6389. DOI: 10.1021/Ja01051A034 |
0.401 |
|
| 1968 |
McCarthy JR, Robins RK, Robins MJ. Purine nucleosides. XXII. The synthesis of angustmycin A (decoyinine) and related unsaturated nucleosides. Journal of the American Chemical Society. 90: 4993-9. PMID 5665542 DOI: 10.1021/Ja01020A038 |
0.527 |
|
| 1968 |
Miles DW, Hahn SJ, Robins RK, Robins MJ, Eyring H. Vicinal effects on the optical activity of some adenine nucleosides. The Journal of Physical Chemistry. 72: 1483-91. PMID 5648867 DOI: 10.1021/J100851A015 |
0.399 |
|
| 1968 |
Robins MJ, Currie BL. The synthesis of 3-deazauridine ‘4-hydroxy-1-(β-D-ribo-pentofuranosyl)-2-pyridone] Chemical Communications (London). DOI: 10.1039/C1968001547B |
0.324 |
|
| 1967 |
McCarthy JR, Robins MJ, Robins RK. The synthesis of unsaturated adenine nucleosides related to angustmycin A Chemical Communications (London). 536-537. DOI: 10.1039/C19670000536 |
0.52 |
|
| 1967 |
Robins MJ, Mccarthy JR, Robins RK. The chemical transformation of uridine to an α-L-lyxo nucleoside via a 4′-unsaturated intermediate Journal of Heterocyclic Chemistry. 4: 313-314. DOI: 10.1002/Jhet.5570040229 |
0.387 |
|
| 1966 |
Robins MJ, McCarthy JR, Robins RK. Purine nucleosides. XII. The preparation of 2',3'-dideoxyadenosine, 2',5'-dideoxyadenosine, and 2',3',5'-trideoxyadenosine from 2'-deoxyadenosine. Biochemistry. 5: 224-31. PMID 5938940 DOI: 10.1021/Bi00865A029 |
0.514 |
|
| 1966 |
McCarthy JR, Robins MJ, Townsend LB, Robins RK. Purine nucleosides. XIV. Unsaturated furanosyl adenine nucleosides prepared via base-catalyzed elimination reactions of 2'-deoxyadenosine derivatives. Journal of the American Chemical Society. 88: 1549-53. PMID 5914527 DOI: 10.1021/Ja00959A043 |
0.624 |
|
| 1966 |
Hall RH, Robins MJ, Stasiuk L, Thedford R. Isolation of N6-(γ,γ-Dimethylallyl)adenosine from Soluble Ribonucleic Acid1 Journal of the American Chemical Society. 88: 2614-2615. DOI: 10.1021/Ja00963A061 |
0.306 |
|
| 1965 |
Robins MJ, Robins RK. Purine nucleosides. XI. The synthesis of 2'-deoxy-9-alpha- and-beta-D-ribofuranosylpurines and the correlation of their anomeric structure with proton magnetic resonance spectra. Journal of the American Chemical Society. 87: 4934-40. PMID 5844465 DOI: 10.1021/Ja00949A042 |
0.375 |
|
| 1964 |
Robins MJ, Robins RK. The Synthesis of 2′,3′-Dideoxyadenosine from 2′-Deoxyadenosine Journal of the American Chemical Society. 86: 3585-3586. DOI: 10.1021/Ja01071A055 |
0.46 |
|
| 1964 |
Robins MJ, Bowles WA, Robins RK. Purine Deoxynucleosides. Synthesis of 9-(2′-deoxy-α and -β-D-ribofuranosyl and 2′-deoxy-α- and -β-D-ribopyranosyl)purines by the Fusion Method Journal of the American Chemical Society. 86: 1251-1252. DOI: 10.1021/Ja01060A063 |
0.395 |
|
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