Jerome Charles Bressi, Ph.D.
Affiliations: | 2000 | University of Washington, Seattle, Seattle, WA |
Area:
medicinal enzymologyGoogle:
"Jerome Bressi"Mean distance: 9.11 | S | N | B | C | P |
Parents
Sign in to add mentor| Michael H. Gelb | grad student | 2000 | University of Washington | |
| (Structure-based design of glycolysis inhibitors as anti -parasite drugs.) | ||||
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Publications
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| Bressi JC, Jennings AJ, Skene R, et al. (2010) Exploration of the HDAC2 foot pocket: Synthesis and SAR of substituted N-(2-aminophenyl)benzamides. Bioorganic & Medicinal Chemistry Letters. 20: 3142-5 |
| Verlinde C, Bressi J, Choe J, et al. (2002) Protein structure-based design of anti-protozoal drugs Journal of the Brazilian Chemical Society. 13: 843-844 |
| Verlinde CLMJ, Bressi JC, Choe J, et al. (2002) Protein structure-based design of anti-protozoal drugs Journal of the Brazilian Chemical Society. 13: 843-848 |
| Bressi JC, Verlinde CL, Aronov AM, et al. (2001) Adenosine analogues as selective inhibitors of glyceraldehyde-3-phosphate dehydrogenase of Trypanosomatidae via structure-based drug design. Journal of Medicinal Chemistry. 44: 2080-93 |
| Suresh S, Bressi JC, Kennedy KJ, et al. (2001) Conformational changes in Leishmania mexicana glyceraldehyde-3-phosphate dehydrogenase induced by designed inhibitors. Journal of Molecular Biology. 309: 423-35 |
| Kennedy KJ, Bressi JC, Gelb MH. (2001) A disubstituted NAD+ analogue is a nanomolar inhibitor of trypanosomal glyceraldehyde-3-phosphate dehydrogenase. Bioorganic & Medicinal Chemistry Letters. 11: 95-8 |
| Bressi JC, Choe J, Hough MT, et al. (2000) Adenosine analogues as inhibitors of Trypanosoma brucei phosphoglycerate kinase: elucidation of a novel binding mode for a 2-amino-N(6)-substituted adenosine. Journal of Medicinal Chemistry. 43: 4135-50 |
| Golisade A, Bressi JC, Van Calenbergh S, et al. (2000) Polymer-assisted solution-phase synthesis of 2'-amido-2'-deoxyadenosine derivatives targeted at the NAD(+)-binding sites of parasite enzymes. Journal of Combinatorial Chemistry. 2: 537-44 |
| Bernstein BE, Williams DM, Bressi JC, et al. (1998) A bisubstrate analog induces unexpected conformational changes in phosphoglycerate kinase from Trypanosoma brucei. Journal of Molecular Biology. 279: 1137-48 |