Year |
Citation |
Score |
2014 |
Ghisaidoobe AT, van den Berg RJ, Butt SS, Strijland A, Donker-Koopman WE, Scheij S, van den Nieuwendijk AM, Koomen GJ, van Loevezijn A, Leemhuis M, Wennekes T, van der Stelt M, van der Marel GA, van Boeckel CA, Aerts JM, et al. Identification and development of biphenyl substituted iminosugars as improved dual glucosylceramide synthase/neutral glucosylceramidase inhibitors. Journal of Medicinal Chemistry. 57: 9096-104. PMID 25250725 DOI: 10.1021/jm501181z |
0.462 |
|
2001 |
Burm BEA, Blokker P, Jongmans E, Van Kampen E, Wanner MJ, Koomen GJ. Synthesis of xestomanzamines a and b Heterocycles. 55: 495-503. DOI: 10.3987/Com-00-9107 |
0.364 |
|
2000 |
Deghati PYF, Wanner MJ, Koomen GJ. Regioselective nitration of purine nucleosides: Synthesis of 2- nitroadenosine and 2-nitroinosine Tetrahedron Letters. 41: 1291-1295. DOI: 10.1016/S0040-4039(99)02271-6 |
0.334 |
|
1999 |
Madre M, Panchenko N, Golbraikh A, Zhuk R, Pandit UK, Geenevasen J, Koomen GJ. Purine nucleoside analogues. 11. An alternative synthesis of N- and O-alkyl derivatives of 9- and 7-[(2-acetoxyethoxy)methyl]-N2-acetylguanine Collection of Czechoslovak Chemical Communications. 64: 685-695. DOI: 10.1135/Cccc19990685 |
0.56 |
|
1999 |
Barends J, Van Der Linden JB, Van Delft FL, Koomen GJ. Palladium-catalyzed amination of 6-chloropurine. Synthesis of N6- substituted adenosine analogues Nucleosides and Nucleotides. 18: 2121-2126. |
0.364 |
|
1998 |
Overkleeft HS, Renkema GH, Neele J, Vianello P, Hung IO, Strijland A, van der Burg AM, Koomen GJ, Pandit UK, Aerts JM. Generation of specific deoxynojirimycin-type inhibitors of the non-lysosomal glucosylceramidase. The Journal of Biological Chemistry. 273: 26522-7. PMID 9756888 DOI: 10.1074/jbc.273.41.26522 |
0.567 |
|
1998 |
Burm BEA, Meijler MM, Korver J, Wanner MJ, Koomen GJ. Synthesis of the brominated marine alkaloids (±)-arborescidine A, B and C Tetrahedron. 54: 6135-6146. DOI: 10.1016/S0040-4020(98)00306-8 |
0.307 |
|
1997 |
Wanner MJ, Koomen GJ. Biomimetic synthesis of racemic alkaloids Pharmacochemistry Library. 28: 179-187. DOI: 10.1016/S0165-7208(97)80064-5 |
0.317 |
|
1997 |
Wanner MJ, Koomen GJ. Biomimetic Synthesis of Nitraria Alkaloids, based on Tetrahydropyridine Synthons Journal of the Indian Chemical Society. 74: 891-895. |
0.302 |
|
1996 |
Petra DGI, De Boer RF, Koomen GJ, Meeuwenoord NJ, Kuyl-Yeheskiely E, Van Der Marel GA, Van Boom JH. Synthesis and properties of a fluorescent nucleotide derivative Recueil Des Travaux Chimiques Des Pays-Bas-Journal of the Royal Netherlands. 115: 99-102. DOI: 10.1002/Recl.19961150117 |
0.39 |
|
1995 |
Wanner MJ, Koomen GJ. Biomimetic synthesis of nitraramine The Journal of Organic Chemistry. 60: 5634-5637. |
0.301 |
|
1995 |
Madre M, Geita L, Zhuk R, Koomen GJ. Purine nucleoside analogues. 7. 9-[2-(Alkylthio)ethoxymethyl] derivatives of adenine, hypoxanthine and guanine Chinese Pharmaceutical Journal. 47: 469-481. |
0.308 |
|
1994 |
Wanner MJ, Koomen GJ. Biomimetic synthesis of nazlinin and nitrarine Pure and Applied Chemistry. 66: 2239-2242. DOI: 10.1351/pac199466102239 |
0.301 |
|
1994 |
Boogaard AT, Pandit UK, Koomen GJ. Ring D modifications of ellipticine. Part 2. Chlorination of ellipticine via its N-oxide and synthesis and selective acetylation of 5,6,11-trimethyl-5H-benzo[b]carbazole. Tetrahedron. 50: 4811-4828. DOI: 10.1016/S0040-4020(01)85018-3 |
0.539 |
|
1992 |
Hartgers WA, De Boer RF, Wanner MJ, Koomen GJ. A potential suicide inhibitor of adenylosuccinate lyase Nucleosides and Nucleotides. 11: 1325-1332. DOI: 10.1080/07328319208021176 |
0.319 |
|
1992 |
Koomen GJ, Provoost LM, Van Maarschalkerwaart DAH, Willard NP. Synthesis of an acyclic analogue of azidothymidine Nucleosides and Nucleotides. 11: 1297-1303. DOI: 10.1080/07328319208021174 |
0.337 |
|
1992 |
Plug JPM, Koomen GJ, Pandit UK. An expedient synthesis of 9-hydroxyellipticine Synthesis. 1221-1222. DOI: 10.1055/S-1992-26342 |
0.517 |
|
1992 |
Vloon WJ, van den Bos JC, Koomen GJ, Pandit UK. Synthesis of ring C modified sesbanimide analogues Tetrahedron. 48: 8317-8328. DOI: 10.1016/S0040-4020(01)80499-3 |
0.537 |
|
1992 |
Plug JPM, Koomen GJ, Pandit UK. Sythesis of novel annulated ellipticines via Claisen rearrangement reactions Tetrahedron Letters. 33: 2179-2182. DOI: 10.1016/0040-4039(92)88171-Z |
0.577 |
|
1991 |
Wanner MJ, Koomen GJ. Biomimetic synthesis of quinolizidine alkaloids Tetrahedron. 47: 8431-8442. DOI: 10.1016/S0040-4020(01)96184-8 |
0.314 |
|
1991 |
van den Bos JC, Vloon WJ, Koomen GJ, Pandit UK. Synthesis of acyclic analogues of sesbanimides A and B Tetrahedron. 47: 6787-6794. DOI: 10.1016/S0040-4020(01)82330-9 |
0.562 |
|
1990 |
Van Maarschalkerwaart DAH, Willard NP, Koomen GJ. Carbocyclic nucleoside analogues. Synthesis and properties of 1-(4-hydroxymethyl-2-cyclopenten-1-yl)-thymine Nucleosides and Nucleotides. 9: 787-791. DOI: 10.1080/15257779008043144 |
0.321 |
|
1989 |
Langendoen A, Plug JPM, Koomen GJ, Pandit UK. Regiospecific C-9 substitution of ellipticine derivatives Tetrahedron. 45: 1759-1762. DOI: 10.1016/S0040-4020(01)80040-5 |
0.514 |
|
1988 |
Wanner MJ, Koomen GJ. 2-Substituted Glutarimides via Preformed Wittig Reagents Synthesis. 1988: 325-327. DOI: 10.1055/S-1988-27558 |
0.304 |
|
1988 |
Langendoen A, Koomen GJ, Pandit UK. An approach to novel ellipticine glycosides Tetrahedron. 44: 3627-3631. DOI: 10.1016/S0040-4020(01)85992-5 |
0.546 |
|
1988 |
WANNER MJ, KOOMEN G. ChemInform Abstract: 2-Substituted Glutarimides via Preformed Wittig Reagents. Cheminform. 19. DOI: 10.1002/CHIN.198833239 |
0.303 |
|
1987 |
Langendoen A, Koomen GJ, Pandit UK. A new approach to C-9 hydroxylation of N(6)-substituted ellipticine Heterocycles. 26: 91-94. DOI: 10.3987/R-1987-01-0091 |
0.495 |
|
1987 |
Langendoen A, Koomen GJ, Pandit UK. Side-chain substitution of 6-methylellipticine approach to a new class of ellipticine derivatives Heterocycles. 26: 69-73. DOI: 10.3987/R-1987-01-0069 |
0.468 |
|
1987 |
Wanner MJ, Willard NP, Koomen GJ, Pandit UK. Stereospecific synthesis of (+)- and (-)-sesbanimide A Tetrahedron. 43: 2549-2556. DOI: 10.1016/S0040-4020(01)81662-8 |
0.541 |
|
1986 |
Wijsmuller WFA, Wanner MJ, Koomen GJ, Pandit UK. Pyridocarbazole alkaloids. Synthesis of olivacine and ellipticine analogues Heterocycles. 24: 1795-1797. DOI: 10.1002/Chin.198647359 |
0.566 |
|
1986 |
Koomen GJ, Wolschrijn H, van Rhijn JBM, Wanner MJ, Pandit UK. Synthesis of 5-fluoro-3-(2-tetrahydrofuryl)-6-vinyluracil. Design of a 5-fu-derivative with extended conjugation Heterocycles. 24: 939-941. DOI: 10.1002/Chin.198642214 |
0.519 |
|
1986 |
Wanner MJ, Willard NP, Koomen GJ, Pandit UK. Synthesis of (7R,8S,9R,10S,11S)-sesbanimide A Journal of the Chemical Society - Series Chemical Communications. 396-397. DOI: 10.1002/Chin.198634331 |
0.418 |
|
1985 |
Koomen GJ, van Rhijn JBMv, Pandit UK. Non-glycosidic derivatives of 5-fluorouracil Nucleosides and Nucleotides. 4: 215-216. DOI: 10.1080/07328318508077858 |
0.476 |
|
1985 |
Odijk WM, Koomen GJ. Fluorescent nucleoside analogues. Synthesis of fluorescent pyrido[2,1-i]purines, and their corresponding ribosides Tetrahedron. 41: 1893-1904. DOI: 10.1016/S0040-4020(01)96552-4 |
0.443 |
|
1984 |
WANNER MJ, KOOMEN G, PANDIT UK. ChemInform Abstract: STUDIES IN THE STEREOSPECIFIC SYNTHESIS OF SESBANIMIDE. SYNTHESIS OF 4-SACCHARIDALGLUTARIMIDES Chemischer Informationsdienst. 15. DOI: 10.1002/Chin.198448332 |
0.557 |
|
1983 |
Wanner MJ, Koomen GJ, Pandit UK. Inter- and intramolecular addition of ester anions to nicotinium salts. A facile approach to nauclefine and ellipticine derivatives Tetrahedron. 39: 3673-3681. DOI: 10.1016/S0040-4020(01)88606-3 |
0.62 |
|
1983 |
WANNER MJ, KOOMEN G, PANDIT UK. ChemInform Abstract: A CONVENIENT SYNTHESIS OF 6-METHYLELLIPTICINE AND 6-METHYLOLIVACINE Chemischer Informationsdienst. 14. DOI: 10.1002/Chin.198322343 |
0.559 |
|
1982 |
Wanner MJ, Koomen GJ, Pandit UK. Synthesis of polynuclear heterocycles via the reaction of α-ester carbanions with quaternized nicotinamide salts. A facile stereoselective synthesis of sesbanine Tetrahedron. 38: 2741-2748. DOI: 10.1016/0040-4020(82)80032-X |
0.615 |
|
1982 |
WANNER MJ, KOOMEN G, PANDIT UK. ChemInform Abstract: A New Approach to Ellipticine Analogues; Synthesis of 11-Hydroxy-5,6-dimethyl-pyrido[4,3-b]carbazole. Chemischer Informationsdienst. 13. DOI: 10.1002/Chin.198233202 |
0.542 |
|
1980 |
Wanner MJ, Hageman JJ, Koomen GJ, Pandit UK. Potential carcinostatics. 4. Synthesis and biological properties of erythro- and threo-beta-fluoroaspartic acid and erythro-beta-fluoroasparagine. Journal of Medicinal Chemistry. 23: 85-7. PMID 7359517 DOI: 10.1021/Jm00175A017 |
0.548 |
|
1980 |
Wanner MJ, Van Wijk EM, Koomen GJ, Pandit UK. Potential carcinostatics. V. Synthesis and properties of potential inhibitors of the adenylosuccinate synthetase and adenylosuccinate lyase system Recueil Des Travaux Chimiques Des Pays Bas. 99: 20-23. DOI: 10.1002/Recl.19780970711 |
0.609 |
|
1980 |
Wanner MJ, Hageman JJM, Koomen GJ, Pandit UK. POTENTIAL CARCINOSTATICS. 4. SYNTHESIS AND BIOLOGICAL PROPERTIES OF ERYTHRO- AND THREO-β-FLUOROASPARTIC ACID AND ERYTHRO-β-FLUOROASPARAGINE Cheminform. 11. DOI: 10.1002/Chin.198024111 |
0.503 |
|
1979 |
ODIJK WM, WANNER MJ, KOOMEN GJ, PANDIT UK. ChemInform Abstract: POTENTIAL CARCINOSTATIC AGENTS. PART III. PSEUDO-GLYCOSIDIC DERIVATIVES OF 5-FLUOROURACIL Chemischer Informationsdienst. 10. DOI: 10.1002/Chin.197909223 |
0.515 |
|
1978 |
Wanner MJ, Hageman JJM, Koomen GJ, Pandit UK. Potential Carcinostatics. Part Ii. Synthesis And Properties Of Potential Inhibitors Of The Adenylosuccinate Synthetase And Adenylosuccinate Lyase Systems Cheminform. 11. DOI: 10.1002/Chin.197843246 |
0.521 |
|
1978 |
HAGEMAN JJM, WANNER MJ, KOOMEN GJ, PANDIT UK. ChemInform Abstract: POTENTIAL CARCINOSTATICS. SYNTHESIS AND BIOLOGICAL PROPERTIES OF D- AND L-β,β-DIFLUOROASPARTIC ACID AND β,β-DIFLUOROASPARAGINE Chemischer Informationsdienst. 9. DOI: 10.1002/Chin.197816128 |
0.489 |
|
1978 |
THIELLIER HPM, KOOMEN GJ, PANDIT UK. ChemInform Abstract: UNCONVENTIONAL NUCLEOTIDE ANALOGS. XVIII. RING EXPANSION OF URIDINE HALOCARBENE ADDUCTS. SYNTHESIS OF DIAZEPINE NUCLEOSIDES Chemischer Informationsdienst. 9. DOI: 10.1002/chin.197802343 |
0.341 |
|
1978 |
Wanner MJ, Hageman JJM, Koomen GJ, Pandit UK. Potential carcinostatics. Synthesis and properties of potential inhibitors of the adenylosuccinate synthetase and adenylosuccinate lyase systems Recueil Des Travaux Chimiques Des Pays Bas. 97: 211-214. |
0.479 |
|
1977 |
Hageman JJ, Wanner MJ, Koomen GJ, Pandit UK. Potential carcinostatics. Synthesis and biological properties of d- and 1-beta,beta-difluoroaspartic acid and beta,beta-difluoroasparagine. Journal of Medicinal Chemistry. 20: 1677-9. PMID 592334 DOI: 10.1021/Jm00222A029 |
0.471 |
|
1977 |
Thiellier HPM, Koomen GJ, Pandit UK. Unconventional nucleotide analogues1 1 Part XV. H.P.M Thiellier, G.J. Koomen and U.K. Pandit, Heterocycles 5, 19 (1976). Reaction of carbenes with uracil and uridine derivatives Tetrahedron. 33: 1493-1500. DOI: 10.1016/0040-4020(77)88011-3 |
0.587 |
|
1977 |
Thiellier HPM, Koomen GJ, Pandit UK. Unconventional nucleotide analogues-XVIII1 1 Part XVII. H.P.M. Thiellier, G.J. Koomen and U.K. Pandit, Tetrahedron 33, 2603 (1977). Ring expansion of uridine halocarbene adducts. Synthesis of diazepine nucleosides Tetrahedron. 33: 2609-2612. DOI: 10.1016/0040-4020(77)80087-2 |
0.603 |
|
1977 |
Thiellier HPM, Koomen GJ, Pandit UK. Unconventional nucleotide analogues-XVII1 1 Part XVI. H.P.M. Thiellier, G.J. Koomen and U.K. Pandit, Tetrahedron 33, 1493 (1977). Ring-transformations of uracil dihalocarbene adducts Tetrahedron. 33: 2603-2607. DOI: 10.1016/0040-4020(77)80086-0 |
0.585 |
|
1977 |
THIELLIER HPM, KOOMEN GJ, PANDIT UK. ChemInform Abstract: UNCONVENTIONAL NUCLEOTIDE ANALOGS. XV. NOVEL BASE-MODIFIED NUCLEOSIDES Chemischer Informationsdienst. 8: no-no. DOI: 10.1002/Chin.197717341 |
0.539 |
|
1976 |
THIELLIER HPM, KOOMEN GJ, PANDIT UK. ChemInform Abstract: TRANSFORMATIONS OF 1,3-DISUBSTITUTED URACIL-CARBENE ADDUCTS. RING EXPANSION TO 1,3-DIAZEPINE DERIVATIVES Chemischer Informationsdienst. 7: no-no. DOI: 10.1002/Chin.197603227 |
0.559 |
|
1974 |
THIELLIER HPM, BURG AMVD, KOOMEN GJ, PANDIT UK. ChemInform Abstract: REACTION OF CARBENES WITH 1,3-DISUBSTITUTED URACIL DERIVATIVES Chemischer Informationsdienst. 5: no-no. DOI: 10.1002/Chin.197451349 |
0.55 |
|
1973 |
Koomen GJ, Pandit UK. Unconventional nucleotide analogues. IX. N-substituted 3-(pyrimidin-1-yl) pyrrolidin-2-ones. Journal of the Chemical Society. Perkin Transactions 1. 17: 1929-33. PMID 4799178 DOI: 10.1039/P19730001929 |
0.57 |
|
1973 |
Koomen GJ, Kroon AP, Mas Cabré FR, Goores AP, Peereboom R, Pandit UK. Unconventional nucleotide analogues. Part X. Synthesis of N-substituted 3-(Adenin-9-yl)pyrrolidin-2-ones Journal of the Chemical Society, Perkin Transactions 1. 1934-1940. PMID 4363162 DOI: 10.1039/P19730001934 |
0.599 |
|
1973 |
KOOMEN GJ, PANDIT UK. ChemInform Abstract: UNCONVENTIONAL NUCLEOTIDE ANALOGUES PART 9, N-SUBSTITUTED 3-(PYRIMIDIN-1-YL)-PYRROLIDIN-2-ONES Chemischer Informationsdienst. 4: no-no. DOI: 10.1002/chin.197349468 |
0.546 |
|
1971 |
Koomen GJ, Kroon AP, Goores AP, Pandit UK. Non-Sacccfaridal Nucleoside and Hucleotide Analocuses Synthetic Communications. 1: 41-45. DOI: 10.1080/00397917108081615 |
0.421 |
|
1971 |
KOOMEN GJ, KROON AP, GOORES AP, PANDIT UK. ChemInform Abstract: ZUCKERFREIE NUCLEOSID- UND NUCLEOTID-ANALOGA Chemischer Informationsdienst. Organische Chemie. 2: no-no. DOI: 10.1002/Chin.197139334 |
0.519 |
|
1969 |
Nollet AJH, Koomen GJ, Grose WFA, Pandit UK. Application of NMR spectroscopy in distinguishing between N1- and N3-substituted 2,4-dioxo-1,2,3,4,-tetrahydropyrimidines. Tetrahedron Letters. 10: 4607-4608. DOI: 10.1016/S0040-4039(01)88762-1 |
0.467 |
|
1967 |
Pandit UK, de Jonge K, Koomen GJ, Huisman HO. Heterocyclic steroids IX. A Convenient Synthesis of 14-Aza-11-Keto Steroids Tetrahedron Letters. 8: 3529-3533. |
0.688 |
|
Low-probability matches (unlikely to be authored by this person) |
2008 |
Läppchen T, Pinas VA, Hartog AF, Koomen GJ, Schaffner-Barbero C, Andreu JM, Trambaiolo D, Löwe J, Juhem A, Popov AV, den Blaauwen T. Probing FtsZ and tubulin with C8-substituted GTP analogs reveals differences in their nucleotide binding sites. Chemistry & Biology. 15: 189-99. PMID 18291323 DOI: 10.1016/J.Chembiol.2007.12.013 |
0.299 |
|
1998 |
Madre M, Zhuk R, Panchenko N, Geenevasen J, Van Den Burg A, Koomen GJ. Purine nucleoside analogues. 10. A new synthetic route to 8-substituted-7(9)-alkoxyalkylguanines Heterocyclic Communications. 4: 581-586. |
0.293 |
|
1994 |
Wanner MJ, Koomen GJ. Stereoselective synthesis of the indole alkaloids nitrarine, nitramidine, and isomers. A biomimetic approach Journal of Organic Chemistry. 59: 7479-7484. |
0.293 |
|
2004 |
Wanner MJ, Rodenko B, Koch M, Koomen GJ. New (1-deaza)purine derivatives via efficient C-2 nitration of the (1-deaza)purine ring. Nucleosides, Nucleotides & Nucleic Acids. 23: 1313-20. PMID 15571251 DOI: 10.1081/NCN-200027566 |
0.292 |
|
1990 |
Wanner MJ, Koomen GJ. Glutarimide nucleosides synthesis and properties of analogs of 1-deaza-thymidine Tetrahedron Letters. 31: 907-910. DOI: 10.1016/S0040-4039(00)94660-4 |
0.288 |
|
2010 |
BURM BEA, MEIJLER MM, KORVER J, WANNER MJ, KOOMEN G. ChemInform Abstract: Synthesis of the Brominated Marine Alkaloids (.+-.)-Arborescidine A (IV), B (VIII), and C (VI). Cheminform. 29: no-no. DOI: 10.1002/CHIN.199835262 |
0.279 |
|
1992 |
Wanner MJ, Koomen GJ. Biomimetic synthesis of nitraria alkaloids: stereoselective spirocyclization reactions Tetrahedron. 48: 3935-3944. DOI: 10.1016/S0040-4020(01)88473-8 |
0.272 |
|
2000 |
Deghati PYF, Bieräugel H, Wanner MJ, Koomen GJ. Mild and regioselective nitration of 1-deazapurine nucleosides using TBAN/TFAA Tetrahedron Letters. 41: 569-573. DOI: 10.1016/S0040-4039(99)02073-0 |
0.261 |
|
2000 |
Wanner MJ, Deghati PYF, Rodenko B, Koomen GJ. New nucleoside analogs, synthesis, and biological properties Pure and Applied Chemistry. 72: 1705-1708. |
0.26 |
|
2005 |
Rodenko B, Koch M, van der Burg AM, Wanner MJ, Koomen GJ. The mechanism of selective purine C-nitration revealed: NMR studies demonstrate formation and radical rearrangement of an N7-nitramine intermediate. Journal of the American Chemical Society. 127: 5957-63. PMID 15839695 DOI: 10.1021/ja042590x |
0.26 |
|
2010 |
Koomen GJ. Selective Fluorination in Organic and Bioorganic Chemistry. John T. Welch, ed. ACS, Washington D. C. 1991. VIII + 215 pp., $57.95. ISBN 0-8412-1948-6 Recueil Des Travaux Chimiques Des Pays-Bas. 110: 392-392. DOI: 10.1002/Recl.19911100914 |
0.259 |
|
1998 |
Gremmen C, Burm BEA, Wanner MJ, Koomen GJ. The synthesis of new heterocyclic bridged ring systems. Analogs of tetrahydro-β-carbolines Tetrahedron Letters. 39: 1441-1444. DOI: 10.1016/S0040-4039(97)10823-1 |
0.254 |
|
1993 |
Koomen GJ. Synthesis and biological properties of selected nucleoside analogues Recueil Des Travaux Chimiques Des Pays-Bas. 112: 51-65. |
0.252 |
|
1977 |
THIELLIER HPM, KOOMEN GJ, PANDIT UK. ChemInform Abstract: UNCONVENTIONAL NUCLEOTIDE ANALOGS. PART XV. REACTION OF CARBENES WITH URACIL AND URIDINE DERIVATIVES Chemischer Informationsdienst. 8: no-no. DOI: 10.1002/chin.197738358 |
0.251 |
|
2001 |
Wanner MJ, Koomen GJ. Synthesis and properties of 2-nitrosoadenosine Journal of the Chemical Society. Perkin Transactions 1. 1908-1915. |
0.25 |
|
2002 |
Wanner MJ, Koomen GJ. A new synthesis of temozolomide Journal of the Chemical Society. Perkin Transactions 1. 1877-1880. |
0.248 |
|
1987 |
Odijk WM, Koomen GJ. Pyrido[2,1-i]-purines: a new class of fluorescent stains. The Journal of Histochemistry and Cytochemistry : Official Journal of the Histochemistry Society. 35: 1161-3. PMID 3624854 DOI: 10.1177/35.10.3624854 |
0.248 |
|
2002 |
Rodenko B, Wanner MJ, Koomen GJ. Solid phase synthesis of C2,N6-disubstituted adenosine analogues Journal of the Chemical Society. Perkin Transactions 1. 1247-1252. |
0.24 |
|
1993 |
Veloo RA, Koomen GJ. Synthesis of enantiomerically pure (S)-(-)-propranolol from sorbitol Tetrahedron: Asymmetry. 4: 2401-2404. DOI: 10.1016/S0957-4166(00)82209-0 |
0.236 |
|
1995 |
de Boer RF, Petra DGI, Wanner MJ, Boesaart A, Koomen GJ. Mechanism of formation of fluorescent adenosine analogues Heterocycles. 41: 1197-1206. DOI: 10.3987/Com-94-7007 |
0.235 |
|
2005 |
Ozvegy-Laczka C, Várady G, Köblös G, Ujhelly O, Cervenak J, Schuetz JD, Sorrentino BP, Koomen GJ, Váradi A, Német K, Sarkadi B. Function-dependent conformational changes of the ABCG2 multidrug transporter modify its interaction with a monoclonal antibody on the cell surface. The Journal of Biological Chemistry. 280: 4219-27. PMID 15557326 DOI: 10.1074/Jbc.M411338200 |
0.233 |
|
2010 |
Koomen GJ. Fluorine in Bioorganic Chemistry. J. T. Welch and S. Eswarakrishnan. John Wiley & Sons, Chichester, 1991. XVIII + 261 pp., £47.50. ISBN 0-471-50649-4 Recueil Des Travaux Chimiques Des Pays-Bas. 110: 391-391. DOI: 10.1002/Recl.19911100913 |
0.229 |
|
1996 |
Wanner MJ, Koomen GJ. Biomimetic syntheses of alkaloids based on tetrahydropyridine Pure and Applied Chemistry. 68: 2051-2056. |
0.227 |
|
1987 |
Odijk WM, Koomen GJ. Aminolysis of pyrido[2,1-i]purines Journal of the Chemical Society, Perkin Transactions 2. 733-737. DOI: 10.1039/P29870000733 |
0.224 |
|
1978 |
THIELLIER HPM, KOOMEN GJ, PANDIT UK. ChemInform Abstract: UNCONVENTIONAL NUCLEOTIDE ANALOGS. XVII. RING-TRANSFORMATIONS OF URACIL DIHALOCARBENE ADDUCTS Chemischer Informationsdienst. 9. DOI: 10.1002/chin.197802260 |
0.223 |
|
1993 |
Koomen GJ. Progress in Heterocyclic Chemistry vol. 3 H. Suschitzky and E.F.V. Scriven, eds. Pergamon Press, UK 1991 ISBN 008 0405894 hard £55.00/$95.00 ISBN 008 0405886 soft £28.00/$50.00 Recueil Des Travaux Chimiques Des Pays-Bas. 112: 315-315. DOI: 10.1002/Recl.19931120508 |
0.221 |
|
1988 |
Wanner MJ, Koomen GJ. Potential antiviral agents. Synthesis and properties of glutarimide-nucleosides Nucleosides and Nucleotides. 7: 511-517. DOI: 10.1080/07328318808075393 |
0.22 |
|
2007 |
Rodenko B, van der Burg AM, Wanner MJ, Kaiser M, Brun R, Gould M, de Koning HP, Koomen GJ. 2,N6-disubstituted adenosine analogs with antitrypanosomal and antimalarial activities. Antimicrobial Agents and Chemotherapy. 51: 3796-802. PMID 17698622 DOI: 10.1128/AAC.00425-07 |
0.217 |
|
2007 |
Glavinas H, Kis E, Pál A, Kovács R, Jani M, Vági E, Molnár E, Bánsághi S, Kele Z, Janáky T, Báthori G, von Richter O, Koomen GJ, Krajcsi P. ABCG2 (breast cancer resistance protein/mitoxantrone resistance-associated protein) ATPase assay: a useful tool to detect drug-transporter interactions. Drug Metabolism and Disposition: the Biological Fate of Chemicals. 35: 1533-42. PMID 17537873 DOI: 10.1124/Dmd.106.014605 |
0.213 |
|
2010 |
Koomen GJ. Progress in Heterocyclic Chemistry, vol. 2. H. Suschitzky and E. F. V. Scriven. Pergamon press, Oxford, U.K. 1990. VIII + 295 pp., £42.00 hard, £21.00 soft. ISBN 008 0370691 hard. ISBN 008 0370705 soft Recueil Des Travaux Chimiques Des Pays-Bas. 111: 198-198. DOI: 10.1002/Recl.19921110408 |
0.21 |
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1998 |
Van Loevezijn A, Van Maarseveen JH, Stegman K, Visser GM, Koomen GJ. Solid phase synthesis of fumitremorgin, verruculogen and tryprostatin analogs based on a cyclization/cleavage strategy Tetrahedron Letters. 39: 4737-4740. DOI: 10.1016/S0040-4039(98)00931-9 |
0.204 |
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1999 |
Madre M, Panchenko N, Zhuk R, Geenevasen JA, Van Den Burg A, Koomen GJ. Purine nucleoside analogues; 9: Benzylation of N2-acetyl-8- bromoguanine Synthesis. 775-778. |
0.204 |
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1995 |
De Boer RF, Petra DGI, Wanner MJ, Boesaart A, Koomen GJ. Synthesis of fluorescent adenosine analogues Nucleosides and Nucleotides. 14: 349-352. |
0.204 |
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2010 |
Verhoeven JW, Koomen GJ, van der Kerk SM. Resonant tunnelling as a possible source of catalysis by energy-matched enzymes Recueil Des Travaux Chimiques Des Pays-Bas. 105: 343-344. DOI: 10.1002/Recl.19861050920 |
0.202 |
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2000 |
Wanner MJ, Von Frijtag Drabbe Künzel JK, Ijzerman AP, Koomen GJ. 2-Nitro analogues of adenosine and 1-deazaadenosine: synthesis and binding studies at the adenosine A1, A2A and A3 receptor subtypes. Bioorganic & Medicinal Chemistry Letters. 10: 2141-4. PMID 10999489 DOI: 10.1016/S0960-894X(00)00415-7 |
0.201 |
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1993 |
Wanner MJ, Velzel AW, Koomen GJ. Biomimetic synthesis of nazlinin: A structural revision Journal of the Chemical Society - Series Chemical Communications. 174-175. DOI: 10.1039/C39930000174 |
0.2 |
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2001 |
Burm BEA, Gremmen C, Wanner MJ, Koomen GJ. Synthesis of new bridged tetrahydro-β-carbolines and spiro-fused quinuclidines Tetrahedron. 57: 2039-2049. DOI: 10.1016/S0040-4020(01)00023-0 |
0.199 |
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2000 |
Gremmen C, Willemse B, Wanner MJ, Koomen GJ. Enantiopure Tetrahydro-beta-carbolines via Pictet-Spengler Reactions with N-Sulfinyl Tryptamines. Organic Letters. 2: 1955-1958. PMID 10891200 |
0.193 |
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2006 |
Rodenko B, Detz RJ, Pinas VA, Lambertucci C, Brun R, Wanner MJ, Koomen GJ. Solid phase synthesis and antiprotozoal evaluation of di- and trisubstituted 5'-carboxamidoadenosine analogues. Bioorganic & Medicinal Chemistry. 14: 1618-29. PMID 16249090 DOI: 10.1016/j.bmc.2005.10.011 |
0.177 |
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1993 |
Trang NT, Wanner MJ, Koomen GJ, Dung NX. New Acetophenone and Thymol Derivatives from Eupatorium stoechadosmum. Planta Medica. 59: 480-1. PMID 17236013 DOI: 10.1055/s-2006-959741 |
0.176 |
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1998 |
Deghati PYF, Wanner MJ, Koomen GJ. An efficient hetero Diels-Alder approach to imidazo[4,5-c]pyridazines as purine analogues Tetrahedron Letters. 39: 4561-4564. DOI: 10.1016/S0040-4039(98)00806-5 |
0.174 |
|
2001 |
Gremmen C, Wanner MJ, Koomen GJ. Enantiopure tetrahydroisoquinolines via N-sulfinyl Pictet-Spengler reactions Tetrahedron Letters. 42: 8885-8888. DOI: 10.1016/S0040-4039(01)01854-8 |
0.174 |
|
2004 |
Wanner MJ, Koch M, Koomen GJ. Synthesis and antitumor activity of methyltriazene prodrugs simultaneously releasing DNA-methylating agents and the antiresistance drug O(6)-benzylguanine. Journal of Medicinal Chemistry. 47: 6875-83. PMID 15615536 DOI: 10.1021/jm049556d |
0.169 |
|
2000 |
Gremmen C, Willemse B, Wanner MJ, Koomen GJ. Enantiopure tetrahydro-β-carbolines via Pictet-Spengler reactions with N-sulfinyl tryptamines Organic Letters. 2: 1955-1958. |
0.169 |
|
1996 |
Madre M, Zhuk R, Panchenko N, Geenevasen JAJ, van den Burg AM, Koomen G. Some peculiarities of N2-acetyl-8-bromoguanine alkylation Collection of Czechoslovak Chemical Communications. 61: 20-22. DOI: 10.1135/CCCC1996S020 |
0.168 |
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1995 |
Cheng E, Dekker HL, van Gelder BF, Koomen GJ. Inhibition of pig kidney diamine oxidase by nazlinin and nazlinin derivatives. Biochimica Et Biophysica Acta. 1253: 189-92. PMID 8519801 DOI: 10.1016/0167-4838(95)00169-5 |
0.168 |
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1997 |
Mohar B, Kobe J, Koomen GJ. Approach to carbocyclic 4-deoxypyrazofurin through asymmetrisation of a meso-norbornene derivative Synlett. 1467-1468. |
0.166 |
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1998 |
Wanner MJ, Koomen GJ. Synthesis of the Cyclostellettamines A-F and Related Bis(3-alkylpyridinium) Macrocycles European Journal of Organic Chemistry. 889-895. |
0.162 |
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1975 |
KOOMEN GJ, PANDIT UK. ChemInform Abstract: THE ′HILBERT-JOHNSON′ REACTION OF 3,5-DIETHOXY-1,2,4-THIADIAZOLE Chemischer Informationsdienst. 6. DOI: 10.1002/chin.197548301 |
0.159 |
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2011 |
Rodenko B, Al-Salabi MI, Teka IA, Ho W, El-Sabbagh N, Ali JA, Ibrahim HM, Wanner MJ, Koomen GJ, de Koning HP. Synthesis of marine-derived 3-alkylpyridinium alkaloids with potent antiprotozoal activity. Acs Medicinal Chemistry Letters. 2: 901-6. PMID 24900279 DOI: 10.1021/ml200160k |
0.155 |
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1996 |
Cheng E, Botzem J, Wanner MJ, Burnt BEA, Koomen GJ. Enzyme catalysed oxidation of nazlinin and nazlinin derivatives. Characterisation of the reaction products Tetrahedron. 52: 6725-6732. DOI: 10.1016/0040-4020(96)00286-4 |
0.153 |
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1992 |
Veloo RA, Wanner MJ, Koomen GJ. Stereoselective formation of tetrahydrofurans during allyltrimethylsilane additions to L-xylose derivatives Tetrahedron. 48: 5301-5316. DOI: 10.1016/S0040-4020(01)89027-X |
0.151 |
|
1997 |
Madre M, Zhuk R, Koomen GJ. Addition of 2,3-dihydrofuran to N2-acetyl-8-bromoguanine Nucleosides and Nucleotides. 16: 1107-1110. |
0.14 |
|
2003 |
Beukers MW, Wanner MJ, Von Frijtag Drabbe Künzel JK, Klaasse EC, IJzerman AP, Koomen GJ. N6-cyclopentyl-2-(3-phenylaminocarbonyltriazene-1-yl)adenosine (TCPA), a very selective agonist with high affinity for the human adenosine A1 receptor. Journal of Medicinal Chemistry. 46: 1492-503. PMID 12672250 DOI: 10.1021/jm021074j |
0.136 |
|
2005 |
Läppchen T, Hartog AF, Pinas VA, Koomen GJ, den Blaauwen T. GTP analogue inhibits polymerization and GTPase activity of the bacterial protein FtsZ without affecting its eukaryotic homologue tubulin. Biochemistry. 44: 7879-84. PMID 15910002 DOI: 10.1021/bi047297o |
0.133 |
|
2001 |
van Loevezijn A, Allen JD, Schinkel AH, Koomen GJ. Inhibition of BCRP-mediated drug efflux by fumitremorgin-type indolyl diketopiperazines. Bioorganic & Medicinal Chemistry Letters. 11: 29-32. PMID 11140726 DOI: 10.1016/S0960-894X(00)00588-6 |
0.122 |
|
1996 |
Kroon AR, Hoff WD, Fennema HP, Gijzen J, Koomen GJ, Verhoeven JW, Crielaard W, Hellingwerf KJ. Spectral tuning, fluorescence, and photoactivity in hybrids of photoactive yellow protein, reconstituted with native or modified chromophores. The Journal of Biological Chemistry. 271: 31949-56. PMID 8943241 DOI: 10.1074/Jbc.271.50.31949 |
0.12 |
|
1998 |
Cordfunke R, Kort R, Pierik A, Gobets B, Koomen GJ, Verhoeven JW, Hellingwerf KJ. Trans/cis (Z/E) photoisomerization of the chromophore of photoactive yellow protein is not a prerequisite for the initiation of the photocycle of this photoreceptor protein. Proceedings of the National Academy of Sciences of the United States of America. 95: 7396-401. PMID 9636160 DOI: 10.1073/Pnas.95.13.7396 |
0.115 |
|
2015 |
Rodenko B, Wanner MJ, Alkhaldi AA, Ebiloma GU, Barnes RL, Kaiser M, Brun R, McCulloch R, Koomen GJ, de Koning HP. Targeting the Parasite's DNA with Methyltriazenyl Purine Analogs Is a Safe, Selective, and Efficacious Antitrypanosomal Strategy. Antimicrobial Agents and Chemotherapy. 59: 6708-16. PMID 26282430 DOI: 10.1128/AAC.00596-15 |
0.109 |
|
2002 |
Allen JD, van Loevezijn A, Lakhai JM, van der Valk M, van Tellingen O, Reid G, Schellens JH, Koomen GJ, Schinkel AH. Potent and specific inhibition of the breast cancer resistance protein multidrug transporter in vitro and in mouse intestine by a novel analogue of fumitremorgin C. Molecular Cancer Therapeutics. 1: 417-25. PMID 12477054 |
0.101 |
|
1997 |
Jonker SA, Nkunya MHH, Mwamtobe L, Geenevasen J, Koomen GJ. A new coumarin and polyhydroxysqualenes from Ekebergia benguelensis Natural Product Letters. 10: 245-248. |
0.072 |
|
1992 |
Wanner MJ, Koomen GJ. New phosphonium ylides by functionalization of triphenylphosphoranylideneacetamide Tetrahedron Letters. 33: 1513-1516. DOI: 10.1016/S0040-4039(00)91662-9 |
0.071 |
|
1989 |
Compernolle F, Saleh A, Hoornaert G, Damianos N, Galons H, Miocque M, Ouero AM, Cntto J, De Clercq E, Schols D, Baba M, Pauwels R, De Meyer N, Pandey HK, Mishra L, ... ... Koomen GJ, et al. Abstracts of papers Symposium “new therapeutic developments in human infectious diseases” Pharmaceutisch Weekblad. 11: C3-C9. DOI: 10.1007/BF02196043 |
0.07 |
|
1989 |
Wanner MJ, Koomen GJ. Synthesis of (±)-nitramine, (±)-isonitramine and (±)-sibirine via Diels-Alder reactions Tetrahedron Letters. 30: 2301-2304. DOI: 10.1016/S0040-4039(00)99677-1 |
0.07 |
|
2013 |
Wielsma S, Gerrits AM, Koomen GJ, Witteman B. Pancreatitis and a sudden loss of sight. The Netherlands Journal of Medicine. 71: 137-141. PMID 23712810 |
0.058 |
|
1986 |
Odijk WM, Koomen GJ. Photophysical properties of fluorescent pyrido[2,1-i]purines Journal of the Chemical Society, Perkin Transactions 2. 1561-1565. DOI: 10.1039/P29860001561 |
0.044 |
|
1996 |
Wanner MJ, Koomen GJ. Oxidative deamination of tetrahydroanabasine with o-quinones: An easy entry to lupinine, sparteine, and anabasine Journal of Organic Chemistry. 61: 5581-5586. DOI: 10.1021/jo9602130 |
0.038 |
|
1993 |
Trang NT, Wanner MJ, Phuong le VN, Koomen GJ, Dung NX. Thymoquinone from Eupatorium ayapana. Planta Medica. 59: 99. PMID 17230346 DOI: 10.1055/s-2006-959619 |
0.019 |
|
1977 |
Koomen GJ, Thijssen GM, Kruizinga R. Possibilities of tissue diagnosis in ophthalmologic echography [proceedings]. Ophthalmologica. Journal International D'Ophtalmologie. International Journal of Ophthalmology. Zeitschrift FüR Augenheilkunde. 175: 45-6. PMID 904905 |
0.018 |
|
1985 |
Nielen MWF, Koomen G, Frei RW, Brinkman UAT. Electrochemical detection of phenylurea herbicides in liquid chromatography Journal of Liquid Chromatography. 8: 315-332. DOI: 10.1080/01483918508067080 |
0.016 |
|
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